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Volumn 80, Issue 3, 1997, Pages 122-126

Binding of pinoline on the 5-hydroxytryptamine transporter: Competitive interaction with [3H] citalopram

Author keywords

[No Author keywords available]

Indexed keywords

4 ETHYL 6,7 DIMETHOXY BETA CARBOLINE 3 CARBOXYLIC ACID METHYL ESTER; CITALOPRAM; DESIPRAMINE; FLUOXETINE; HARMALOL; HARMAN; IMIPRAMINE; MELATONIN; PINOLINE; SEROTONIN; TRYPTAMINE; TRYPTOLINE; TRYPTOLINE DERIVATIVE; UNCLASSIFIED DRUG;

EID: 0030966365     PISSN: 09019928     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1600-0773.1997.tb00384.x     Document Type: Article
Times cited : (19)

References (25)
  • 1
    • 84993887070 scopus 로고
    • Pinoline, the natural ligand of serotonin transporter in retina and pineal gland
    • Airaksinen, M. M. & E. Kari: Pinoline, the natural ligand of serotonin transporter in retina and pineal gland. Adv. Biosci. 1991, 82, 239-240.
    • (1991) Adv. Biosci. , vol.82 , pp. 239-240
    • Airaksinen, M.M.1    Kari, E.2
  • 2
    • 0019377920 scopus 로고
    • Identification and quantification of 1,2,3,4-tetrahydro-β-carboline, 2-methyl-1,2,3,4-tetrahydro-β-carboline and 6-methoxy-1,2,3,4-tetrahydro-β-carboline as in vivo constituents of rat brain and adrenal gland
    • Barker, S. A., R. E. Harrison, J. A. Monti, G. B. Brown & S. T. Christian: Identification and quantification of 1,2,3,4-tetrahydro-β-carboline, 2-methyl-1,2,3,4-tetrahydro-β-carboline and 6-methoxy-1,2,3,4-tetrahydro-β-carboline as in vivo constituents of rat brain and adrenal gland. Biochem. Pharmacol. 1981, 30, 9-17.
    • (1981) Biochem. Pharmacol. , vol.30 , pp. 9-17
    • Barker, S.A.1    Harrison, R.E.2    Monti, J.A.3    Brown, G.B.4    Christian, S.T.5
  • 3
    • 0003089394 scopus 로고
    • Neurotransmitter, hormone, or drug receptor binding methods
    • Eds.: H. I. Yamamura, S. J. Enna and M. J. Kuhar. Raven Press, New York
    • Bennet, J. P. & H. I. Yamamura: Neurotransmitter, hormone, or drug receptor binding methods. In: Neurotransmitter receptor binding. Eds.: H. I. Yamamura, S. J. Enna and M. J. Kuhar. Raven Press, New York 1985, 61-95.
    • (1985) Neurotransmitter Receptor Binding , pp. 61-95
    • Bennet, J.P.1    Yamamura, H.I.2
  • 4
    • 0015861774 scopus 로고
    • Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50 per cent inhibition (IC50) on an enzymatic reaction
    • Cheng, Y. & W. H. Prusoff: Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50 per cent inhibition (IC50) on an enzymatic reaction. Biochem. Pharmacol. 1973, 27, 3099-3108.
    • (1973) Biochem. Pharmacol. , vol.27 , pp. 3099-3108
    • Cheng, Y.1    Prusoff, W.H.2
  • 5
    • 0023186425 scopus 로고
    • Selective labeling of serotonin uptake sites in rat brain by [3H]citalopram contrasted to labeling of multiple sites by [3H]imipramine
    • D'Amato, R. J., B. L. Largent, A. M. Snowman & S. H. Snyder: Selective labeling of serotonin uptake sites in rat brain by [3H]citalopram contrasted to labeling of multiple sites by [3H]imipramine. J. Pharmacol. Exp. Therap. 1987, 242, 364-371.
    • (1987) J. Pharmacol. Exp. Therap. , vol.242 , pp. 364-371
    • D'Amato, R.J.1    Largent, B.L.2    Snowman, A.M.3    Snyder, S.H.4
  • 7
    • 0019992996 scopus 로고
    • β-carbolines as selective monoamine oxidase inhibitors: In vivo implications
    • Glover, V, J. Liebowitz, I. Armando & M. Sandler:. β-carbolines as selective monoamine oxidase inhibitors: in vivo implications. J. Neural Transmission 1982, 54, 209-218.
    • (1982) J. Neural Transmission , vol.54 , pp. 209-218
    • Glover, V.1    Liebowitz, J.2    Armando, I.3    Sandler, M.4
  • 8
    • 0020416931 scopus 로고
    • Citalopram, pharmacological profile of a specific serotonin-uptake inhibitor with antidepressant activity
    • Hyttel, J.: Citalopram, pharmacological profile of a specific serotonin-uptake inhibitor with antidepressant activity. Prog. Neuro-psychopharmacol. Biol. Psychiatry 1982, 6, 277-295.
    • (1982) Prog. Neuro-psychopharmacol. Biol. Psychiatry , vol.6 , pp. 277-295
    • Hyttel, J.1
  • 9
    • 0011277404 scopus 로고
    • Mass spectrometric identification of 6-methoxy-1,2,3,4-tetrahydro-β-carboline in pineal gland
    • Ed,: A. Frigerio. Elsevier Scientific Publishing Company, Amsterdam
    • Kari, I., M. M. Airaksinen, J. Gynther & A. Huhtikangas: Mass spectrometric identification of 6-methoxy-1,2,3,4-tetrahydro-β-carboline in pineal gland. In: Recent developments in biochemistry, medicine and environmental research 8. Ed,: A. Frigerio. Elsevier Scientific Publishing Company, Amsterdam 1983, 19-24
    • (1983) Recent Developments in Biochemistry, Medicine and Environmental Research 8 , pp. 19-24
    • Kari, I.1    Airaksinen, M.M.2    Gynther, J.3    Huhtikangas, A.4
  • 10
    • 0018874128 scopus 로고
    • Tetrahydro-β-carbolines and corresponding tryptamines: In vitro inhibition of serotonin, dopamine and noradren-aline uptake in rat brain synaptosomes
    • Komulainen, H., J. Toumisto, M. M. Airaksinen, I. Kari, P. Peura & L. Pollari: Tetrahydro-β-carbolines and corresponding tryptamines: In vitro inhibition of serotonin, dopamine and noradren-aline uptake in rat brain synaptosomes. Acta pharmacol. et toxicol. 1980, 46, 299-307.
    • (1980) Acta Pharmacol. et Toxicol. , vol.46 , pp. 299-307
    • Komulainen, H.1    Toumisto, J.2    Airaksinen, M.M.3    Kari, I.4    Peura, P.5    Pollari, L.6
  • 11
    • 0021368931 scopus 로고
    • Substituted tetrahydro-β-carbolines are possible candidates as endogenous ligand of the [3H]imipramine recognition site
    • Langer, S. Z., R. Raisman, L. Tahraoui, B. Scatton, R. Niddam, C. R. Lee & Y. Claustre: Substituted tetrahydro-β-carbolines are possible candidates as endogenous ligand of the [3H]imipramine recognition site. Eur. J. Pharmacol. 1984a, 98, 153-154.
    • (1984) Eur. J. Pharmacol. , vol.98 , pp. 153-154
    • Langer, S.Z.1    Raisman, R.2    Tahraoui, L.3    Scatton, B.4    Niddam, R.5    Lee, C.R.6    Claustre, Y.7
  • 12
    • 0021261733 scopus 로고
    • Possible endocrine role of the pineal gland for 6-methoxytetrahydro-β-carboline, a putative endogenous neuromodulator of the [3H]imipramine recognition site
    • Langer, S. Z., C. R. Lee, A. Segonzac, T. Tateishi, H. Esnaud, H., Schoemaker & B. Winblad: Possible endocrine role of the pineal gland for 6-methoxytetrahydro-β-carboline, a putative endogenous neuromodulator of the [3H]imipramine recognition site. Ear. J. Pharmacol. 1984b, 102, 379-380.
    • (1984) Ear. J. Pharmacol. , vol.102 , pp. 379-380
    • Langer, S.Z.1    Lee, C.R.2    Segonzac, A.3    Tateishi, T.4    Esnaud, H.5    Schoemaker, H.6    Winblad, B.7
  • 15
    • 0020670602 scopus 로고
    • 6-Methoxytetrahydro-β-carboline in the retina of rabbits and pigs
    • Leino, M., I. Kari, M. M. Airaksinen & J. Gynther: 6-Methoxytetrahydro-β-carboline in the retina of rabbits and pigs. Exp. Eye Res. 1983, 36, 135-138.
    • (1983) Exp. Eye Res. , vol.36 , pp. 135-138
    • Leino, M.1    Kari, I.2    Airaksinen, M.M.3    Gynther, J.4
  • 17
    • 0025110895 scopus 로고
    • Binding of some antidepressants to the 5-hydroxytryptamine transporter in brain and platelets
    • Marcusson, J. O. & S. B. Ross: Binding of some antidepressants to the 5-hydroxytryptamine transporter in brain and platelets. Psychopharmacology 1990, 102, 144-155.
    • (1990) Psychopharmacology , vol.102 , pp. 144-155
    • Marcusson, J.O.1    Ross, S.B.2
  • 18
    • 0001165186 scopus 로고
    • Formation of 1-methyl-6-methoxy-1,2,3,4-tetrahydro-2-carboline under physiological conditions
    • McIsaac, W. M.: Formation of 1-methyl-6-methoxy-1,2,3,4-tetrahydro-2-carboline under physiological conditions. Biochem. Biophys. Acta 1961, 52, 607.
    • (1961) Biochem. Biophys. Acta , vol.52 , pp. 607
    • McIsaac, W.M.1
  • 19
    • 0030185038 scopus 로고    scopus 로고
    • Behavioural effects of pinoline in the rat forced swimming, open field and elevated plus-maze tests
    • in press
    • Pähkla, R., J. Harro & L. Rägo: Behavioural effects of pinoline in the rat forced swimming, open field and elevated plus-maze tests. Pharmacol. Res. 1996, in press.
    • (1996) Pharmacol. Res.
    • Pähkla, R.1    Harro, J.2    Rägo, L.3
  • 20
    • 0022400048 scopus 로고
    • Antidepressive drugs can change the affinity of [3H]imipramine and [3H]paroxetine binding to platelet and neuronal membranes
    • Plenge, P. & E. T. Mellerup: Antidepressive drugs can change the affinity of [3H]imipramine and [3H]paroxetine binding to platelet and neuronal membranes. Eur. J. Pharmacol. 1985, 119, 1-8.
    • (1985) Eur. J. Pharmacol. , vol.119 , pp. 1-8
    • Plenge, P.1    Mellerup, E.T.2
  • 21
    • 0024990025 scopus 로고
    • Inhibitory and regulatory binding sites on the rat brain serotonin transporter: Molecular weight of the [3H]paroxetine and [3H]citalopram binding proteins
    • Plenge, P., E. T. Mellerup & M. Nielsen: Inhibitory and regulatory binding sites on the rat brain serotonin transporter: molecular weight of the [3H]paroxetine and [3H]citalopram binding proteins. Eur. J. Pharmacol [Mol. Pharmacol. Sec.] 1990, 189, 129-134.
    • (1990) Eur. J. Pharmacol [Mol. Pharmacol. Sec.] , vol.189 , pp. 129-134
    • Plenge, P.1    Mellerup, E.T.2    Nielsen, M.3
  • 22
    • 0024587174 scopus 로고
    • Effect of different photoperiod exposure on [3H]imipramine binding and serotonin uptake in the rat brain
    • Rovescally, A. S., N. Brunello, M. Riva, R. Galimberti & G. Racagni: Effect of different photoperiod exposure on [3H]imipramine binding and serotonin uptake in the rat brain. J. Neurochem. 1989, 52, 507-514.
    • (1989) J. Neurochem. , vol.52 , pp. 507-514
    • Rovescally, A.S.1    Brunello, N.2    Riva, M.3    Galimberti, R.4    Racagni, G.5
  • 23
    • 0022262840 scopus 로고
    • High-performance liquid chromatography of telrahydro-β-carbolines extracted from plasma and platelets
    • Schouten, M. J. & J. Bruinvels: High-performance liquid chromatography of telrahydro-β-carbolines extracted from plasma and platelets. Anal. Biochem. 1985, 147, 401-409.
    • (1985) Anal. Biochem. , vol.147 , pp. 401-409
    • Schouten, M.J.1    Bruinvels, J.2
  • 24
    • 0021876677 scopus 로고
    • 5-methoxytryptoline, a competitive endocoid acting at [3H]imipramine recognition site in human platelets
    • Segonzac, A., H. Schoemaker, T. Tateishi & S. Z. Langer: 5-methoxytryptoline, a competitive endocoid acting at [3H]imipramine recognition site in human platelets. J. Neurochem. 1985, 45, 249-256.
    • (1985) J. Neurochem. , vol.45 , pp. 249-256
    • Segonzac, A.1    Schoemaker, H.2    Tateishi, T.3    Langer, S.Z.4
  • 25
    • 0021908064 scopus 로고
    • Serotonin uptake inhibitors differentially modulate high affinity imipramine dissociation in human platelet membranes
    • Wennogle, P. L. & L. R. Meyerson: Serotonin uptake inhibitors differentially modulate high affinity imipramine dissociation in human platelet membranes. Life Sci. 1985, 36, 1541-1550.
    • (1985) Life Sci. , vol.36 , pp. 1541-1550
    • Wennogle, P.L.1    Meyerson, L.R.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.