Synthesis of 3-[(1-[11C]Methyl-2(S)-pyrrolidinyl) methoxy]pyridine and 3-[(1-[11C]methyl-2(R)-pyrrolidinyl) methoxylpyridine: Radioligands for in vivo studies of neuronal nicotinic acetylcholine receptors

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 39, Issue 5, 1997, Pages 425-431

  Kassiou, Michael ^a   Ravert, Hayden T ^b   Mathews, William B ^b   Musachio, John L ^b   London, Edythe D ^a   Dannals, Robert F ^b  

^a NATIONAL INSTITUTE ON DRUG ABUSE   (United States)

^b DEPARTMENT OF PATHOLOGY   (United States)

Author keywords

3 Pyridyl ethers; Carbon 11; Nicotinic acetylcholine receptors; Positron emission tomography

Indexed keywords

CARBON; POSITRON EMISSION TOMOGRAPHY; RADIOACTIVITY; SYNTHESIS (CHEMICAL);

3-PYRIDYL ETHER; ACETYLCHOLINE RECEPTOR; CARBON-11; IN-VIVO; METHOXY; NICOTINIC ACETYLCHOLINE; NICOTINIC ACETYLCHOLINE RECEPTOR; PYRIDYL; RADIOLIGANDS; SPECIFIC RADIOACTIVITY;

PYRIDINE;

CARBON 11; NICOTINIC RECEPTOR; RADIOLIGAND;

ARTICLE; DRUG PURIFICATION; DRUG SYNTHESIS; ENANTIOMER; IN VITRO STUDY; ISOTOPE LABELING; RADIOCHEMISTRY; REVERSED PHASE HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; ULTRAVIOLET SPECTROPHOTOMETRY;

EOS;

EID: 0030954216     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(199705)39:5<425::AID-JLCR984>3.0.CO;2-R     Document Type: Article

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