Dynorphin peptides: Antagonists of melanocortin receptors

Pharmaceutical Research

Volumn 14, Issue 6, 1997, Pages 713-719

  Quillan, J Mark ^a   Sadée, Wolfgang ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

Melanocyte stimulating hormone ( MSH); des Tyr dynorphin; Adrenocorticotropic hormone (ACTH); Dependence; Melanocortin peptides; Melanocortin receptors; Non opioid dynorphin effects; Opioid peptides; Receptor cross reactivity; Shock; Tolerance; Trauma

Indexed keywords

CORTICOTROPIN RECEPTOR; DYNORPHIN A; DYNORPHIN DERIVATIVE; DYNORPHIN[1-13]; DYNORPHIN[1-8]; DYNORPHIN[1-9]; ENKEPHALIN; ENKEPHALIN[2,5 DEXTRO PENICILLAMINE]; FORSKOLIN; HISTAMINE; HORMONE RECEPTOR; INTERMEDIN; LEUCINE ENKEPHALIN; LEUCINE ENKEPHALIN[2 DEXTRO SERINE 6 THREONINE]; MELANOCORTIN 1 RECEPTOR; MELANOCORTIN 2 RECEPTOR; MELANOCORTIN 3 RECEPTOR; MELANOCORTIN 4 RECEPTOR; MELANOCORTIN RECEPTOR; METENKEPHALIN; N,N DIALLYLTYROSYL 2 METHYLALANYL 2 METHYLALANYLPHENYLALANYLLEUCINE; NEUROPEPTIDE Y; OPIATE PEPTIDE; OPIATE RECEPTOR; PRODYNORPHIN; RECEPTOR SUBTYPE; SOMATOSTATIN; SOMATOSTATIN RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONCENTRATION RESPONSE; DISSOCIATION CONSTANT; DRUG RECEPTOR BINDING; EMBRYO; FIBROBLAST; HUMAN; HUMAN CELL; KIDNEY CELL; NONHUMAN; PRIORITY JOURNAL; XENOPUS;

ADRENOCORTICOTROPIC HORMONE; ALPHA-MSH; ANIMALS; COS CELLS; DYNORPHINS; HUMANS; MELANOPHORES; PEPTIDE FRAGMENTS; RECEPTOR, MELANOCORTIN, TYPE 2; RECEPTOR, MELANOCORTIN, TYPE 3; RECEPTOR, MELANOCORTIN, TYPE 4; RECEPTORS, CORTICOTROPIN; RECEPTORS, MELANOCORTIN; RECEPTORS, PEPTIDE; RECOMBINANT PROTEINS; XENOPUS LAEVIS;

EID: 0030916995     PISSN: 07248741     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1012185919153     Document Type: Article

References (30)

1. L. Stanfa, and A. Dickenson. Inflamm. Res. 44:231-41 (1995).
2. J. M. Walker, H. C. Moises, D. H. Coy, G. Baldrighi, and H. Akil. Science 218:1136-8 (1982).
3. H. Akil, S. J. Watson, E. Young, M. E. Lewis, H. Khachaturian, and J. M. Walker. Ann. Rev. Neurosci. 7:223-55 (1984).
4. R. Poggioli, A. V. Vergoni, and A. Bertolini. Peptides 7:843-8 (1986).
5. A. I. Faden. J. Neurosci. 12:425-9 (1992).
6. V. K. Shukla, and S. Lemaire. Trends Pharmacol. Sci. 15:420-4 (1994).
7. M. Dumont, and S. Lemaire J. Mol. Cell Cardiol. 25:983-91 (1993).
8. C. Chavkin, I. F. James, and A. Goldstein. Science 215:413-5 (1982).
9. S. Zhang, and L. Yu. J. Biol. Chem. 270:22772-6 (1995).
10. M. Miura, A. Inui, K. Sano, N. Ueno, A. Teranishi, Y. Hirosue, M. Nakajima, M. Okita, J. Togami, K. Koshiya, S. Baba, and M. Kasuga. Am. J. Physiol. 267:E702-9 (1994).
11. W. H. Gispen, J. Buitelaar, V. M. Wiegant, L. Terenius, and D. De Wied. Eur. J. Pharmacol. 39:393-7 (1976).
12. M. E. Hadley. The Melanotropic Peptides, Vols 1-3, CRC Press Inc., Boca Raton, Florida, 1988.
13. A. N. Eberle. The Melanotropins: Chemistry, Physiology and Mechanism of Action, Karger, Basel, Switzerland, 1988.
14. J. M. Walker, H. C. Moises, D. H. Coy, E. A. Young, S. J. Watson, and H. Akil. Life Sci. 31:1821-4 (1982).
15. A. E. Takemori, H. H. Loh, and N. M. Lee. J. Pharmacol. Exp. Ther. 266:121-4 (1993).
16. L. P. Hooke, L. He, and N. M. Lee. J. Pharmacol. Exp. Ther. 273:292-7 (1995).
17. P. C. Contreras and A. E. Takemori. J. Pharmacol. Exp. Ther. 229:21-6 (1984).
18. J. I. Szekely, E. Miglecz, Z. Dunai-Kovacs, I. Tarnawa, A. Z. Ronai, L. Graf, and S. Bajusz. Life Sci. 24:1931-8 (1979).
19. A. Bertolini, S. Guarini, E. Rompianesi, and W. Ferrari. Eur. J. Pharmacol. 130:19-26 (1986).
20. J. D. Alvaro, J. B. Tatro, J. M. Quillan, M. Fogliano, M. Eisenhard, M. R. Lerner, E. J. Nestler, and R. S. Duman. Mol. Pharm. 50:583-91 (1996).
21. A. Bertolini, S. Guarini, W. Ferrari, and E. Rompianesi. Life Sci. 39:1271-80 (1986).
22. J. M. Quillan and W. Sadée. Pharm. Res. 13:1622-28 (1996).
23. A. Daniolos, A. B. Lerner, and M. R. Lerner. Pigment Cell Res. 3:38-43 (1990).
24. J. M. Quillan, C. K. Jayawickreme, and M. R. Lerner. Proc. Natl. Acad. Sci. (USA) 92:2894-98 (1995).
25. J. M. Quillan. Development of a Combinatorial Diffusion Assay and Discovery of MSH Receptor Antagonists, UMI, Ann Arbour, Michigan, 1995.
26. G. Weng, F. Yee, P. Michl, D. Reis, and C. Wahlestedt. Mol. Pharmacol. 48:9-14 (1995).
27. W. E. Polgar, C. M. Bitler, and L. Toll. Life Sci. 58:1223-9 (1996).
28. L. Chen, Y. Gu, and L. Y. Huang. J. Neurosci. 15:4602-11 (1995).
29. J. M. Walker, G. G. Berntson, C. A. Sandman, A. J. Kastin, and H. Akil. Eur. J. Pharmacol. 69:71-9 (1981).
30. P. C. Datta, C. A. Sandman, and F. K. Hoehler. Peptides 3:433-7 (1982).