Evaluation of carbon-11 labeled KF15372 and its ethyl and methyl derivatives as a potential CNS adenosine A1 receptor ligand

Nuclear Medicine and Biology

Volumn 24, Issue 1, 1997, Pages 53-59

  Noguchi, Junko ^a,b   Ishiwata, Kiichi ^a   Furuta, Riko ^a,b   Simada, Jun Ichi ^c   Kiyosawa, Motohiro ^d   Ishii, Shin Ichi ^a   Endo, Kazutoyo ^b   Suzuki, Fumio ^c   Senda, Michio ^a  

^a TOKYO METROPOLITAN INSTITUTE OF GERONTOLOGY   (Japan)

^b SHOWA PHARMACEUTICAL UNIVERSITY   (Japan)

^c KYOWA HAKKO KOGYO CO LTD   (Japan)

^d TOKYO MEDICAL AND DENTAL UNIVERSITY   (Japan)

Author keywords

11C KF15372; adenosine A1 ligand; CNS; PET; receptor

Indexed keywords

8 DICYCLOPROPYLMETHYL 1,3 DIPROPYLXANTHINE; ADENOSINE DERIVATIVE; ADENOSINE RECEPTOR BLOCKING AGENT;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CENTRAL NERVOUS SYSTEM; CONTROLLED STUDY; MOUSE; POSITRON EMISSION TOMOGRAPHY; RAT;

ANIMALS; AUTORADIOGRAPHY; BRAIN; CARBON RADIOISOTOPES; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; DIURETICS; LIGANDS; MALE; MICE; RADIOLIGAND ASSAY; RATS; RECEPTORS, PURINERGIC P1; STRUCTURE-ACTIVITY RELATIONSHIP; TISSUE DISTRIBUTION; TOMOGRAPHY, EMISSION-COMPUTED; XANTHINES;

EID: 0030909033     PISSN: 09698051     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0969-8051(96)00161-8     Document Type: Article

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