Differences in active site gorge dimensions of cholinesterases revealed by binding of inhibitors to human butyrylcholinesterase

Biochemistry

Volumn 36, Issue 48, 1997, Pages 14642-14651

  Saxena, Ashima ^a   Redman, Ann M G ^a   Jiang, Xuliang ^b   Lockridge, Oksana ^c   Doctor, B P ^a  

^a WALTER REED ARMY INSTITUTE OF RESEARCH   (United States)

^b The New York Presbyterian Hospital   (United States)

^c UNIVERSITY OF NEBRASKA MEDICAL CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1,5 BIS(4 ALLYLDIMETHYLAMMONIUMPHENYL)PENTAN 3 ONE DIBROMIDE; ACETYLCHOLINESTERASE; CHOLINESTERASE; CHOLINESTERASE INHIBITOR; DECAMETHONIUM; EDROPHONIUM; HUPERZINE A; PROFENAMINE; PROPIDIUM IODIDE; TACRINE;

ARTICLE; CRYSTAL STRUCTURE; ENZYME ACTIVE SITE; ENZYME BINDING; ENZYME INHIBITION; ENZYME INHIBITOR COMPLEX; MOLECULAR MODEL; PRIORITY JOURNAL;

ANIMALS; BINDING SITES; BUTYRYLCHOLINESTERASE; BUTYRYLTHIOCHOLINE; CHOLINESTERASE INHIBITORS; CHOLINESTERASES; COMPUTER SIMULATION; ENZYME ACTIVATION; HUMANS; MODELS, CHEMICAL; MODELS, MOLECULAR; MUTAGENESIS; PROTEIN CONFORMATION; SPECIES SPECIFICITY; TORPEDO;

MAMMALIA;

EID: 0030780763     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi971425+     Document Type: Article

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