The expanded hansen approach to solubility parameters. Paracetamol and citric acid in individual solvents

Journal of Pharmacy and Pharmacology

Volumn 49, Issue 7, 1997, Pages 644-651

  Barra, Jerome ^a,b   Lescure, François ^b   Doelker, Eric ^a   Bustamante, Pilar ^c  

^a UNIVERSITY OF GENEVA   (Switzerland)

^b UPSA Laboratories   (France)

^c UNIVERSITY OF ALCALÁ   (Spain)

Author keywords

[No Author keywords available]

Indexed keywords

CITRIC ACID; PARACETAMOL; PROTON; SOLVENT;

ARTICLE; CONTROLLED STUDY; DIFFERENTIAL SCANNING CALORIMETRY; DRUG SOLUBILITY; HYDROGEN BOND; MULTIPLE REGRESSION; PH; TECHNIQUE;

EID: 0030757139     PISSN: 00223573     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.2042-7158.1997.tb06086.x     Document Type: Article

References (30)

1. Barton, A. F. M. (1991) Handbook of Solubility Parameters and Other Cohesion Parameters. 2nd edn, CRC Press, Boca Raton, FL
2. Beerbower, A., Wu, P. L., Martin, A. (1984) Expanded solubility parameter approach I. Naphthalene and benzoic acid in individual solvents. J. Pharm. Sci. 73: 179-188
3. Bogardus, J. (1983) Crystalline anhydrous-hydrate phase changes of caffeine and theophylline in solvent-water mixtures. J. Pharm. Sci. 72: 837-838
4. Burrell, H. (1975) Pigment wetting parameter. Am. Chem. Soc. Div. Org. Coat. Plast. 35: 18-24
5. Bustamante, P., Escalera, B., Martin, A., Selles, E. (1989) Predicting the solubility of sulfamethoxypyridazine in individual solvents I: calculating partial solubility parameters. J. Pharm. Sci. 78: 567-573
6. Bustamante, P., Hinkley, D. V., Martin, A., Shi, S. W. (1991) Statistical analysis of the extended Hansen method using the bootstrap technique. J. Pharm. Sci. 80: 971-977
7. Bustamante, P., Martin, A., Gonzalez-Guisandez, M. A. (1993) Partial-solubility parameters and solvatochromic parameters for predicting the solubility of single and multiple drugs in individual solvents. J. Pharm. Sci. 82: 635-640
8. Bustamante, P., Romero, S., Reillo, A. (1995) Thermodynamics of paracetamol in amphiprotic and amphiprotic-aprotic solvent mixtures. Pharm. Sci. 1: 505-507
9. Fedors, R. F. (1974) A method for estimating both the solubility parameters and molar volumes of liquids. Polym. Eng. Sci. 14: 147-154
10. Fokkens, J. G., Van Amelsfoort, J. G. M., De Blaey, C. J., De Kruif, C. G., Wilting, J. (1983) A thermodynamic study of the solubility of theophylline and its hydrate. Int. J. Pharm. 14: 79-93
11. Gardon, J. L. (1966) The influence of polarity upon the solubility parameter concept. J. Paint Technol. 38: 43-57
12. Ghosal, S. K., Gupta, B. K. (1979) Determination of the solubility parameters of several barbiturates: their significance in drug activity. J. Inst. Chem. (India) 51: 117-123
13. Hansen, C. M. (1967) The three-dimensional solubility parameters. Key to paint component affinities. II. Dyes, emulsifiers, mutual solubility and compatibility and pigments. J. Paint Technol. 39: 505-511
14. Hansen, C. M. (1970) Characterization of surfaces by spreading liquids. J. Paint Technol. 42: 660-664
15. Hansen, C. M., Beerbower, A. (1971) Solubility parameters. In: Herman, F. M., McKetta, J. J., Othmer, D. F., Standen, A. (eds) Kirk-Othmer Encyclopedia of Chemical Technology, Interscience, New York, pp 889
16. Hildebrand, J. H., Prausnitz, J. M., Scott, R. L. (1970) Regular and Related Solutions. Van Nostrand Reinhold, New York
17. Hintze, J. L. (1990) Number Cruncher Statistical System. Kaysville, Utah, pp 147-148, 152-154, 179-181, 184
18. Hoy, K. L. (1970) New values of the solubility parameters from vapor pressure data. J. Paint Technol. 42: 76-118
19. Karger, B. L., Snyder, L. R., Eon, C. (1976) An expanded solubility parameter treatment for classification and use of chromatographic solvents and adsorbents. Parameters for dispersion, dipole and hydrogen-bonding interactions. J. Chromatogr. 125: 71-88
20. Keller, R. A., Karger, B. L., Snyder, L. R. (1971) Use of the solubility parameter in predicting chromatographic retention and eluotropic strength. In: Stock, R., Perry S. E. (eds) Gas Chromatography. Institute of Petroleum, London, pp 125-144
21. Khalil, S. A., Moustafa, M. A., Abdallah, O. Y. (1976) The use of the solubility parameter as an index of drug activity. Can. J. Pharm. Sci. 11: 121-126
22. Martin, A., Bustamante, P. (1989) Solubility parameters applied to the pharmaceutical sciences. An. Real Acad. Farm. 55: 175-202
23. Martin, A., Wu, P. L., Adjei, A., Beerbower, A., Prausnitz, J. M. (1981) Extended Hansen solubility approach: naphthalene in individual solvents. J. Pharm. Sci. 70: 1260-1264
24. Martin, A., Wu, P. L., Beerbower, A. (1984) Expanded solubility parameter approach. II. p-Hydroxybenzoic acid and methyl p-hydroxybenzoate in individual solvents. J. Pharm. Sci. 73: 188-194
25. Martin, A., Bustamante, P., Escalera, B., Selles, E. (1989) Predicting the solubility of sulfamethoxypyridazine in individual solvents II. Relationship between solute-solvent interaction terms and partial-solubility parameters. J. Pharm. Sci. 78: 672-678
26. Moldenhauer, M. G., Nairn, J. G. (1994) Solubility parameter effects on microencapsulation in the presence of polyisobutylene. J. Contr. Rel. 31: 151-162
27. Romero, S., Reillo, A., Escalera, B., Bustamante, P. (1996) The behavior of paracetamol in mixtures of amphiprotic and amphiprotic-aprotic solvents. Relationship of solubility curves to specific and nonspecific interactions. Chem. Pharm. Bull. 44: 1061-1064
28. Small, P. A. (1953) Some factors affecting the solubility of polymers. J. Appl. Chem. 3: 71-80
29. Subrahmanyam, C. V., Sreenivasa Reddy, M., Venkata Rao, J., Gundu Rao, P. (1992) Irregular solution behavior of paracetamol in binary solvents. Int. J. Pharm. 78: 17-24
30. Van Krevelen, D. W. (1976) Properties of Polymers: Their Estimation and Correlation with Chemical Structure. 2nd edn, Elsevier, Amsterdam