Competitive, non-competitive and cooperative interactions between substrates of P-glycoproteins as measured by ATPase activity

Biochimica et Biophysica Acta - Molecular Basis of Disease

Volumn 1361, Issue 2, 1997, Pages 169-176

  Litman, Thomas ^a,b   Zeuthen, Thomas ^b   Skovsgaard, Torben ^a   Stein, Wilfred D ^c  

^a UNIVERSITY OF COPENHAGEN   (Denmark)

^b UNIVERSITY OF COPENHAGEN   (Denmark)

^c HEBREW UNIVERSITY OF JERUSALEM   (Israel)

Author keywords

ATPase; Chinese Hamster ovary cell; Drug interactions; Multidrug resistance; P glycoprotein

Indexed keywords

ADENOSINE TRIPHOSPHATASE; AMIODARONE; AMITRIPTYLINE; COLCHICINE; CYCLOSPORIN A; DAUNORUBICIN; DILTIAZEM; EPIRUBICIN; GLYCOPROTEIN P; GRAMICIDIN D; GRAMICIDIN S; PROGESTERONE; PROPRANOLOL; VANADIC ACID; VERAPAMIL; VINBLASTINE;

ANIMAL CELL; ARTICLE; BINDING SITE; CELL MEMBRANE; CHO CELL; COMPETITIVE INHIBITION; CONTROLLED STUDY; ENZYME ACTIVITY; IN VITRO STUDY; MULTIDRUG RESISTANCE; NONHUMAN; PRIORITY JOURNAL; PROTEIN BINDING; STRUCTURE ACTIVITY RELATION;

ADENOSINE TRIPHOSPHATASES; ANIMALS; BINDING SITES; CHO CELLS; COLCHICINE; CRICETINAE; DAUNORUBICIN; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG INTERACTIONS; DRUG RESISTANCE, MULTIPLE; ENZYME ACTIVATION; GRAMICIDIN; KINETICS; MICROSOMES; P-GLYCOPROTEIN; PROGESTERONE; VANADATES; VERAPAMIL; VINBLASTINE;

ANIMALIA; CRICETINAE; CRICETULUS GRISEUS;

EID: 0030743356     PISSN: 09254439     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0925-4439(97)00027-6     Document Type: Article

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