메뉴 건너뛰기




Volumn 20, Issue 6, 1997, Pages 348-367

Molecular pharmacology of somatastatin receptor subtypes

Author keywords

Somatostatin; Somatostatin receptor; SSTR subtypes

Indexed keywords

ADENYLATE CYCLASE; CALCIUM CHANNEL; CYCLIC AMP; GUANINE NUCLEOTIDE BINDING PROTEIN; MESSENGER RNA; MITOGEN ACTIVATED PROTEIN KINASE; PHOSPHOPROTEIN PHOSPHATASE; POTASSIUM CHANNEL; RECEPTOR SUBTYPE; SOMATOSTATIN; SOMATOSTATIN RECEPTOR;

EID: 0030612281     PISSN: 03914097     EISSN: None     Source Type: Journal    
DOI: 10.1007/BF03350317     Document Type: Review
Times cited : (277)

References (159)
  • 1
    • 0015914428 scopus 로고
    • Hypothalamic polypeptide that inhibits the secretion of immunoreactive pituitary growth hormone
    • Brazeau P., Vale W., Burgus R., Ling N., Butcher M., Rivier J., Guillemin R. Hypothalamic polypeptide that inhibits the secretion of immunoreactive pituitary growth hormone. Science 179:77, 1973.
    • (1973) Science , vol.179 , pp. 77
    • Brazeau, P.1    Vale, W.2    Burgus, R.3    Ling, N.4    Butcher, M.5    Rivier, J.6    Guillemin, R.7
  • 2
    • 0018837330 scopus 로고
    • N-terminally extended somatostatin: The primary structure of somatostatin 28
    • Pradayrol L., Jornvall H., Mutt V., Ribet A. N-terminally extended somatostatin: the primary structure of somatostatin 28. FEBS Lett. 109: 55, 1980.
    • (1980) FEBS Lett , vol.109 , pp. 55
    • Pradayrol, L.1    Jornvall, H.2    Mutt, V.3    Ribet, A.4
  • 3
    • 0002722115 scopus 로고
    • General aspects of the biology and function of somatostatin
    • Müller, E.E., Thorner, M.O., Weil, C. (Eds.), Springer-Verlag, Berlin
    • Patel Y.C. General aspects of the biology and function of somatostatin. In: Müller, E.E., Thorner, M.O., Weil, C. (Eds.), The role of somatostatin: basic and clinical aspects of neuroscience series. Springer-Verlag, Berlin, Vol. 4, 1992, pp. 1-16.
    • (1992) The Role of Somatostatin: Basic and Clinical Aspects of Neuroscience Series , vol.4 , pp. 1-16
    • Patel, Y.C.1
  • 4
    • 3042601444 scopus 로고    scopus 로고
    • Galanopoulou, D.N. Papachristou. Production, action, and degradation of somatostatin
    • Jefferson L.S., Cherrington A.D. (Eds.), Oxford University Press, N.Y. (in press)
    • Patel Y.C., J-L Liu A.S. Galanopoulou, D.N. Papachristou. Production, action, and degradation of somatostatin. In: Jefferson L.S., Cherrington A.D. (Eds.), The Handbook of Physiology, The endocrine pancreas and regulation of metabolism, Oxford University Press, N.Y. 1997 (in press).
    • (1997) The Handbook of Physiology, The Endocrine Pancreas and Regulation of Metabolism
    • Patel, Y.C.1    J-L Liu, A.S.2
  • 5
    • 0023835514 scopus 로고
    • Peptides derived from cleavage of prosomatostatin at carboxy and amino terminal segments: Characterization of tissue and secreted forms in the rat
    • Patel Y.C., O'Neil W. Peptides derived from cleavage of prosomatostatin at carboxy and amino terminal segments: characterization of tissue and secreted forms in the rat. J. Biol. Chem. 263: 745, 1988.
    • (1988) J. Biol. Chem. , vol.263 , pp. 745
    • Patel, Y.C.1    O'Neil, W.2
  • 6
    • 0021105680 scopus 로고
    • Somatostatin
    • Reichlin S. Somatostatin. N. Engl. J. Med. 309: 1495, 1556, 1983.
    • (1983) N. Engl. J. Med. , vol.309 , pp. 1495
    • Reichlin, S.1
  • 7
    • 0026347208 scopus 로고
    • Evidence that somatostatin is localized and synthesized in lymphoid organs
    • (USA)
    • Aguila M.C., Dees W.L., Haensly W.E., McCann S.M. Evidence that somatostatin is localized and synthesized in lymphoid organs. Proc. Natl. Acad. Sci. (USA) 88: 11485, 1991.
    • (1991) Proc. Natl. Acad. Sci. , vol.88 , pp. 11485
    • Aguila, M.C.1    Dees, W.L.2    Haensly, W.E.3    McCann, S.M.4
  • 11
    • 0022501337 scopus 로고
    • Cyclic AMP regulates somatostatin mRNA accumulation in primary diencephalic cultures and in transfected fibroblast cells
    • Montminy M.R., Low M.J., Tapia-Arancibia L., Reichlin S., Mandel G., Goodman R.H. Cyclic AMP regulates somatostatin mRNA accumulation in primary diencephalic cultures and in transfected fibroblast cells. J. Neurosci. 6: 1171, 1986.
    • (1986) J. Neurosci. , vol.6 , pp. 1171
    • Montminy, M.R.1    Low, M.J.2    Tapia-Arancibia, L.3    Reichlin, S.4    Mandel, G.5    Goodman, R.H.6
  • 12
    • 0025733310 scopus 로고
    • Regulation of islet somatostatin secretion and gene expression: Selective effects of adenosine 3′, 5′ monophosphate and phorbol esters in normal islets of Langerhans and in a somatostatin producing rat islet clonal cell line 1027B2
    • Patel Y.C., Papachristou D.N., Zingg H.H., Farkas E.M. Regulation of islet somatostatin secretion and gene expression: selective effects of adenosine 3′, 5′ monophosphate and phorbol esters in normal islets of Langerhans and in a somatostatin producing rat islet clonal cell line 1027B2. Endocrinology 128: 1754, 1991.
    • (1991) Endocrinology , vol.128 , pp. 1754
    • Patel, Y.C.1    Papachristou, D.N.2    Zingg, H.H.3    Farkas, E.M.4
  • 13
    • 0028009750 scopus 로고
    • Growth hormone-releasing factor increases somatostatin release and mRNA levels in the rat periventricular nucleus via nitric oxide by activation of guanylate cyclase
    • (USA)
    • Aguila M.C. Growth hormone-releasing factor increases somatostatin release and mRNA levels in the rat periventricular nucleus via nitric oxide by activation of guanylate cyclase. Proc. Natl. Acad. Sci. (USA) 91: 782, 1994.
    • (1994) Proc. Natl. Acad. Sci. , vol.91 , pp. 782
    • Aguila, M.C.1
  • 15
    • 0029114410 scopus 로고
    • Molecular biology of somatostatin receptors
    • Reisine T., Bell G.I. Molecular biology of somatostatin receptors. Endocrinol. Rev. 16: 427, 1995.
    • (1995) Endocrinol. Rev. , vol.16 , pp. 427
    • Reisine, T.1    Bell, G.I.2
  • 18
    • 0028901533 scopus 로고
    • An early increase in somatostatin mRNA expression in the frontal cortex of Rhesus monkeys infected with simian immunodeficiency virus
    • (USA)
    • Da Cunha A., Rausch D.M., Eiden L.E. An early increase in somatostatin mRNA expression in the frontal cortex of Rhesus monkeys infected with simian immunodeficiency virus. Proc. Natl. Acad. Sci. (USA) 92: 1371, 1995.
    • (1995) Proc. Natl. Acad. Sci. , vol.92 , pp. 1371
    • Da Cunha, A.1    Rausch, D.M.2    Eiden, L.E.3
  • 19
    • 0028032277 scopus 로고
    • Molecular pharmacology of somatostatin receptors
    • Hoyer D., Lubbert H., Bruns C. Molecular pharmacology of somatostatin receptors. Arch. Pharmacol. 350: 441, 1994.
    • (1994) Arch. Pharmacol. , vol.350 , pp. 441
    • Hoyer, D.1    Lubbert, H.2    Bruns, C.3
  • 22
    • 0025030059 scopus 로고
    • Mechanism of action of somatostatin: An overview of receptor function and studies of the molecular characterization and purification of somatostatin receptor proteins
    • Patel Y.C., Murthy K.K., Escher E., Banville D., Spiess J., Srikant C.B. Mechanism of action of somatostatin: an overview of receptor function and studies of the molecular characterization and purification of somatostatin receptor proteins. Metabolism 39 (Suppl. 2): 63, 1990.
    • (1990) Metabolism , vol.39 , Issue.2 SUPPL. , pp. 63
    • Patel, Y.C.1    Murthy, K.K.2    Escher, E.3    Banville, D.4    Spiess, J.5    Srikant, C.B.6
  • 23
    • 0018073907 scopus 로고
    • Characterization of functional receptors for somatostatin in rat pituitary cells in culture
    • Schonbrunn A., Tashjian A.M. Jr. Characterization of functional receptors for somatostatin in rat pituitary cells in culture. J. Biol. Chem. 253: 6473, 1978.
    • (1978) J. Biol. Chem. , vol.253 , pp. 6473
    • Schonbrunn, A.1    Tashjian Jr., A.M.2
  • 24
    • 0000127560 scopus 로고
    • Somatostatin receptors: Identification and characterization in rat brain membranes
    • (USA)
    • Srikant C.B., Patel Y.C. Somatostatin receptors: identification and characterization in rat brain membranes. Proc. Natl. Acad. Sci. (USA) 78: 3930, 1981.
    • (1981) Proc. Natl. Acad. Sci. , vol.78 , pp. 3930
    • Srikant, C.B.1    Patel, Y.C.2
  • 25
    • 0019884587 scopus 로고
    • Receptor binding of somatostatin-28 is tissue specific
    • Srikant C.B., Patel Y.C. Receptor binding of somatostatin-28 is tissue specific. Nature 294: 259, 1981.
    • (1981) Nature , vol.294 , pp. 259
    • Srikant, C.B.1    Patel, Y.C.2
  • 26
    • 0022548218 scopus 로고
    • Distribution of somatostatin receptors in the human brain: An autoradiographic study
    • Reubi J-C., Cortes R., Maurer R., Probst A., Palacios J.M. Distribution of somatostatin receptors in the human brain: an autoradiographic study. Neuroscience. 18: 329, 1986.
    • (1986) Neuroscience , vol.18 , pp. 329
    • Reubi, J.-C.1    Cortes, R.2    Maurer, R.3    Probst, A.4    Palacios, J.M.5
  • 27
    • 0023928070 scopus 로고
    • Somatostatin receptor subtypes in the clonal anterior pituitary cell lines AtT-20 and GH3
    • Thermos, K., Reisine T. Somatostatin receptor subtypes in the clonal anterior pituitary cell lines AtT-20 and GH3. Mol. Pharmacol. 33: 370, 1988.
    • (1988) Mol. Pharmacol. , vol.33 , pp. 370
    • Thermos, K.1    Reisine, T.2
  • 28
    • 0026724150 scopus 로고
    • Photoaffinity labelling of the somatostatin receptor: Identification of molecular subtypes
    • Srikant C.B., Murthy K.K., Escher E., Patel Y.C. Photoaffinity labelling of the somatostatin receptor: Identification of molecular subtypes. Endocrinology 130: 2937, 1992.
    • (1992) Endocrinology , vol.130 , pp. 2937
    • Srikant, C.B.1    Murthy, K.K.2    Escher, E.3    Patel, Y.C.4
  • 29
    • 0025144963 scopus 로고
    • Identification of somatostatin receptors by covalent labeling with a novel photoreactive somatostatin analog
    • Brown P.J., Lee A.B., Norman M.G., Presky D.H., Schonbrunn A. Identification of somatostatin receptors by covalent labeling with a novel photoreactive somatostatin analog. J. Biol. Chem. 265: 17995, 1990.
    • (1990) J. Biol. Chem. , vol.265 , pp. 17995
    • Brown, P.J.1    Lee, A.B.2    Norman, M.G.3    Presky, D.H.4    Schonbrunn, A.5
  • 31
    • 0026710669 scopus 로고
    • Purification of a pituitary receptor for somatostatin. the utility of biotinylated somatostatin analogs
    • Eppler C.M., Zysk J.R., Corbett M., Shieh H-M. Purification of a pituitary receptor for somatostatin. The utility of biotinylated somatostatin analogs. J. Biol. Chem. 267: 15603, 1992.
    • (1992) J. Biol. Chem. , vol.267 , pp. 15603
    • Eppler, C.M.1    Zysk, J.R.2    Corbett, M.3    Shieh, H.-M.4
  • 32
    • 0026729131 scopus 로고
    • Solubilization and partial purification of somatostatin-28 preferring receptors from hamster pancreatic beta cells
    • Maletti M., Andersson M., Marie J-C., Rosselin G., Mutt V. Solubilization and partial purification of somatostatin-28 preferring receptors from hamster pancreatic beta cells. J. Biol. Chem. 267: 15620, 1992.
    • (1992) J. Biol. Chem. , vol.267 , pp. 15620
    • Maletti, M.1    Andersson, M.2    Marie, J.-C.3    Rosselin, G.4    Mutt, V.5
  • 33
    • 0023907127 scopus 로고
    • Distribution of somatostatin receptors in RINm5F insulinoma cells
    • Sullivan S.J., Schonbrunn A. Distribution of somatostatin receptors in RINm5F insulinoma cells. Endocrinology 122: 1137, 1988.
    • (1988) Endocrinology , vol.122 , pp. 1137
    • Schonbrunn A, S.S.J.1
  • 34
    • 0024600650 scopus 로고
    • Somatostatin analogues inhibit growth of pancreatic cancer by stimulating tyrosine phosphatase
    • (USA)
    • Liebow C., Reilly C., Serrano M., Schally A.V. Somatostatin analogues inhibit growth of pancreatic cancer by stimulating tyrosine phosphatase. Proc. Natl. Acad. Sci. (USA) 86: 2003, 1989.
    • (1989) Proc. Natl. Acad. Sci. , vol.86 , pp. 2003
    • Liebow, C.1    Reilly, C.2    Serrano, M.3    Schally, A.V.4
  • 36
    • 0025719564 scopus 로고
    • Inhibition of human breast cancer cell (MCF-7) growth in vitro by the somatostatin analog SMS201-995: Effects on cell cycle parameters and apoptotic cell death
    • Pagliacci M.C., Tognellinin R., Grignani F., Nicoletti F. Inhibition of human breast cancer cell (MCF-7) growth in vitro by the somatostatin analog SMS201-995: effects on cell cycle parameters and apoptotic cell death. Endocrinology 129: 2555, 1991.
    • (1991) Endocrinology , vol.129 , pp. 2555
    • Pagliacci, M.C.1    Tognellinin, R.2    Grignani, F.3    Nicoletti, F.4
  • 37
    • 0031023467 scopus 로고    scopus 로고
    • Coexistence of somatostatin receptor subtypes in the human neuroblastoma cell line LA-N-2
    • Nilsson L., Folkesson R. Coexistence of somatostatin receptor subtypes in the human neuroblastoma cell line LA-N-2. FEBS Lett. 401: 838, 1997.
    • (1997) FEBS Lett , vol.401 , pp. 838
    • Nilsson, L.1    Folkesson, R.2
  • 39
    • 0024509206 scopus 로고
    • Distinct subsets of somatostatin receptors on cultured human lymphocytes
    • Sreedharan S.P., Kodama K.T., Peterson K.E., Goetzl E.J. Distinct subsets of somatostatin receptors on cultured human lymphocytes. J. Biol. Chem. 264: 949, 1989.
    • (1989) J. Biol. Chem. , vol.264 , pp. 949
    • Sreedharan, S.P.1    Kodama, K.T.2    Peterson, K.E.3    Goetzl, E.J.4
  • 40
    • 0026544424 scopus 로고
    • Cloning and functional characterization of a family of human and mouse somatostatin receptors expressed in brain, gastrointestinal tract, and kidney
    • (USA)
    • Yamada Y., Post S.R., Wang K., Tager H.S., Bell G.I., Seine S. Cloning and functional characterization of a family of human and mouse somatostatin receptors expressed in brain, gastrointestinal tract, and kidney. Proc. Natl. Acad. Sci. (USA) 89: 251, 1992.
    • (1992) Proc. Natl. Acad. Sci. , vol.89 , pp. 251
    • Yamada, Y.1    Post, S.R.2    Wang, K.3    Tager, H.S.4    Bell, G.I.5    Seine, S.6
  • 41
    • 0026551305 scopus 로고
    • Expression cloning of a rat brain somatostatin receptor cDNA
    • (USA)
    • Kluxen F.W., Bruns C.H., Lubbert H. Expression cloning of a rat brain somatostatin receptor cDNA. Proc. Natl. Acad. Sci. (USA) 89: 4618, 1992.
    • (1992) Proc. Natl. Acad. Sci. , vol.89 , pp. 4618
    • Kluxen, F.W.1    Bruns, C.H.2    Lubbert, H.3
  • 42
    • 0026802434 scopus 로고
    • Cloning and expression of a rat somatostatin receptor enriched in brain
    • Li X-J., Forte M., North R.A., Ross C.A., Snyder S.H. Cloning and expression of a rat somatostatin receptor enriched in brain. J. Biol. Chem. 267: 21307, 1992.
    • (1992) J. Biol. Chem. , vol.267 , pp. 21307
    • Li, X.-J.1    Forte, M.2    North, R.A.3    Ross, C.A.4    Snyder, S.H.5
  • 44
    • 0026489450 scopus 로고
    • Molecular cloning of a somatostatin-28 receptor and comparison of its expression pattern with that of a somatostatin 14 receptor in rat brain
    • (USA)
    • Meyerhof W., Wulfsen I., Schonrock C., Fehr S., Richter D. Molecular cloning of a somatostatin-28 receptor and comparison of its expression pattern with that of a somatostatin 14 receptor in rat brain. Proc. Natl. Acad. Sci. (USA) 89: 10267, 1992.
    • (1992) Proc. Natl. Acad. Sci. , vol.89 , pp. 10267
    • Meyerhof, W.1    Wulfsen, I.2    Schonrock, C.3    Fehr, S.4    Richter, D.5
  • 45
    • 0027055232 scopus 로고
    • Somatostatin receptors, an expanding gene family: Cloning and functional characterization of human SSTR3, a protein coupled to adenylate cyclase
    • Yamada Y., Reisine T., Law S.F., Ihara Y., Kubota A., Kagimoto S., Seino M., Seino Y., Bell G.I., Seino S. Somatostatin receptors, an expanding gene family: cloning and functional characterization of human SSTR3, a protein coupled to adenylate cyclase. Mol. Endocrinol. 6: 2136, 1992.
    • (1992) Mol. Endocrinol. , vol.6 , pp. 2136
    • Yamada, Y.1    Reisine, T.2    Law, S.F.3    Ihara, Y.4    Kubota, A.5    Kagimoto, S.6    Seino, M.7    Seino, Y.8    Bell, G.I.9    Seino, S.10
  • 46
    • 0026453393 scopus 로고
    • Molecular cloning and functional expression of a brain-specific somatostatin receptor
    • (USA)
    • Bruno J.F., Xu Y., Song J., Berelowitz M. Molecular cloning and functional expression of a brain-specific somatostatin receptor. Proc. Natl. Acad. Sci. (USA) 89: 11151, 1992.
    • (1992) Proc. Natl. Acad. Sci. , vol.89 , pp. 11151
    • Bruno, J.F.1    Xu, Y.2    Song, J.3    Berelowitz, M.4
  • 49
    • 0027536220 scopus 로고
    • A human somatostatin receptor (SSTR3), located on chromosome 22, displays preferential affinity for somatostatin-14 like peptides
    • Corness J.D., Demchyshyn L.L., Seeman P., Van Tol H.H.M., Srikant C.B., Kent G., Patel Y.C., Niznik H.B. A human somatostatin receptor (SSTR3), located on chromosome 22, displays preferential affinity for somatostatin-14 like peptides. FEBS Lett. 321: 279, 1993.
    • (1993) FEBS Lett , vol.321 , pp. 279
    • Corness, J.D.1    Demchyshyn, L.L.2    Seeman, P.3    Van Tol, H.H.M.4    Srikant, C.B.5    Kent, G.6    Patel, Y.C.7    Niznik, H.B.8
  • 50
    • 0027086821 scopus 로고
    • Molecular cloning and expression of a pituitary somatostatin receptor with preferential affinity for somatostatin-28
    • O'Carroll A.M., Lolait S.J., Konig M., Mahan L.C. Molecular cloning and expression of a pituitary somatostatin receptor with preferential affinity for somatostatin-28. Mol. Pharmacol. 42: 939, 1992.
    • (1992) Mol. Pharmacol. , vol.42 , pp. 939
    • O'Carroll, A.M.1    Lolait, S.J.2    Konig, M.3    Mahan, L.C.4
  • 51
    • 0028210475 scopus 로고
    • Molecular cloning, functional characterization, and chromosomal localization of a human somatostatin receptor (somatostatin receptor type 5) with preferential affinity for somatostatin-28
    • Panetta R., Greenwood M.T., Warszynska A., Demchyshyn L.L, Day R., Niznik H.B., Srikant C.B., Patel Y.C. Molecular cloning, functional characterization, and chromosomal localization of a human somatostatin receptor (somatostatin receptor type 5) with preferential affinity for somatostatin-28. Mol. Pharmacol. 45: 417, 1994.
    • (1994) Mol. Pharmacol. , vol.45 , pp. 417
    • Panetta, R.1    Greenwood, M.T.2    Warszynska, A.3    Demchyshyn, L.L.4    Day, R.5    Niznik, H.B.6    Srikant, C.B.7    Patel, Y.C.8
  • 52
    • 0026673028 scopus 로고
    • Cloning and expression of a novel mouse somatostatin receptor (SSTR2B)
    • Vanetti M., Kouba M., Wang X., Vogt G., Hollt V. Cloning and expression of a novel mouse somatostatin receptor (SSTR2B). FEBS Lett. 311: 290, 1992.
    • (1992) FEBS Lett , vol.311 , pp. 290
    • Vanetti, M.1    Kouba, M.2    Wang, X.3    Vogt, G.4    Hollt, V.5
  • 53
    • 0027302917 scopus 로고
    • Multiple gene transcripts of the somatostatin receptor SSTR2: Tissue selective distribution and cAMP regulation
    • Patel Y.C., Greenwood M.T., Kent G., Panetta R., Srikant C.B. Multiple gene transcripts of the somatostatin receptor SSTR2: tissue selective distribution and cAMP regulation. Biochem. Biophys. Res. Commun. 192: 28, 1993.
    • (1993) Biochem. Biophys. Res. Commun. , vol.192 , pp. 28
    • Patel, Y.C.1    Greenwood, M.T.2    Kent, G.3    Panetta, R.4    Srikant, C.B.5
  • 60
    • 0023893674 scopus 로고
    • In vitro and in vivo inhibition of human small cell lung carcinoma (NCI-H69) growth by a somatostatin analogue
    • Taylor J.E., Bogden A.E., Moreau J.-P., Coy D.H. In vitro and in vivo inhibition of human small cell lung carcinoma (NCI-H69) growth by a somatostatin analogue. Biochem. Biophys. Res. Commun. 153: 81, 1988.
    • (1988) Biochem. Biophys. Res. Commun. , vol.153 , pp. 81
    • Taylor, J.E.1    Bogden, A.E.2    Moreau, J.-P.3    Coy, D.H.4
  • 61
    • 0027287377 scopus 로고
    • Cloned somatostatin receptors: Identification of subtype-selective peptides and demonstration of high affinity binding of linea peptides
    • Raynor K., Murphy W.A., Coy D.H., Taylor J.E., Moreau J.-P., Yasuda K., Bell G.I., Reisine T. Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding of linea peptides. Mol. Pharmacol. 43: 838, 1993
    • (1993) Mol. Pharmacol. , vol.43 , pp. 838
    • Raynor, K.1    Murphy, W.A.2    Coy, D.H.3    Taylor, J.E.4    Moreau, J.-P.5    Yasuda, K.6    Bell, G.I.7    Reisine, T.8
  • 62
    • 0028020115 scopus 로고
    • Subtype selectivity of peptide analogs for all five cloned human somatostatin receptors (hsstrl-5)
    • Patel Y.C., Srikant C.B. Subtype selectivity of peptide analogs for all five cloned human somatostatin receptors (hsstrl-5). Endocrinology 135: 2814, 1994.
    • (1994) Endocrinology , vol.135 , pp. 2814
    • Patel, Y.C.1    Srikant, C.B.2
  • 65
    • 0030111425 scopus 로고    scopus 로고
    • Development of a selective agonist at the somatostatin receptor subtype SSTR1
    • Liapakis G., Haeger C., Rivier J., Reisine T. Development of a selective agonist at the somatostatin receptor subtype SSTR1. J. PET 276: 1089, 1996.
    • (1996) J. PET , vol.276 , pp. 1089
    • Liapakis, G.1    Haeger, C.2    Rivier, J.3    Reisine, T.4
  • 67
    • 0028227013 scopus 로고
    • Structure and function of receptors coupled to G proteins
    • Baldwin J.M. Structure and function of receptors coupled to G proteins. Curr. Opin. Cell Biol. 6: 180, 1994.
    • (1994) Curr. Opin. Cell Biol. , vol.6 , pp. 180
    • Baldwin, J.M.1
  • 69
    • 0029898348 scopus 로고    scopus 로고
    • Is there a lock for all agonist keys in 7 TM receptors
    • Schwartz T.W., Rosenkilde M.M. Is there a lock for all agonist keys in 7 TM receptors. TIPS 17: 213, 1996.
    • (1996) TIPS , vol.17 , pp. 213
    • Schwartz, T.W.1    Rosenkilde, M.M.2
  • 71
    • 0027988149 scopus 로고
    • Identification of peptide binding residues in the extracellular domains of the AT1 receptor
    • Hjorth S.A., Schambye H.T., Greenlee W.J., Schwartz T.W. Identification of peptide binding residues in the extracellular domains of the AT1 receptor. J. Biol. Chem. 269: 30953, 1994.
    • (1994) J. Biol. Chem. , vol.269 , pp. 30953
    • Hjorth, S.A.1    Schambye, H.T.2    Greenlee, W.J.3    Schwartz, T.W.4
  • 72
    • 0028100755 scopus 로고
    • Glutamate 301 of the mouse gonadotrophin releasing hormone receptor confers specificity for arginine 8 of mammalian gonadotrophin releasing hormone
    • Flanagan C.A., Becker I.I., Davidson J.S., Wakefield I.K., Zhou W., Sealfon S.C., Miller R.P. Glutamate 301 of the mouse gonadotrophin releasing hormone receptor confers specificity for arginine 8 of mammalian gonadotrophin releasing hormone. J. Biol. Chem. 269: 22636, 1994.
    • (1994) J. Biol. Chem. , vol.269 , pp. 22636
    • Flanagan, C.A.1    Becker, I.I.2    Davidson, J.S.3    Wakefield, I.K.4    Zhou, W.5    Sealfon, S.C.6    Miller, R.P.7
  • 73
    • 0028925786 scopus 로고
    • Two amino acids, located in transmembrane domains VI and VII, determine the selectivity of the peptide agonist SMS201-995 for the SSTR2 somatostatin receptor
    • Kaupman K., Bruns C., Raulf F., Weber H.P., Mattes H., Lubbert H. Two amino acids, located in transmembrane domains VI and VII, determine the selectivity of the peptide agonist SMS201-995 for the SSTR2 somatostatin receptor. EMBO J. 14: 727, 1995.
    • (1995) EMBO J , vol.14 , pp. 727
    • Kaupman, K.1    Bruns, C.2    Raulf, F.3    Weber, H.P.4    Mattes, H.5    Lubbert, H.6
  • 74
    • 0028850149 scopus 로고
    • Aspartic acid residue 124 in the third transmembrane domain of the somatostatin receptor subtype 3 is essential for somatostatin 14 binding
    • Nehring R.B., Meyerhof W., Richter D. Aspartic acid residue 124 in the third transmembrane domain of the somatostatin receptor subtype 3 is essential for somatostatin 14 binding. DNA and Cell Biol. 14: 939, 1995.
    • (1995) DNA and Cell Biol , vol.14 , pp. 939
    • Nehring, R.B.1    Meyerhof, W.2    Richter, D.3
  • 75
    • 0028787944 scopus 로고
    • Identification of a critical aspartate residue in transmembrane domain three necessary for the binding of somatostatin to the somatostatin receptor SSTR2
    • Strnad J., Hadcock J.R. Identification of a critical aspartate residue in transmembrane domain three necessary for the binding of somatostatin to the somatostatin receptor SSTR2. Biochem. Biophys. Res. Commun. 216: 913, 1995.
    • (1995) Biochem. Biophys. Res. Commun. , vol.216 , pp. 913
    • Strnad, J.1    Hadcock, J.R.2
  • 76
    • 0028170656 scopus 로고
    • 6 agonist selectivity determinants in somatostatin receptor subtypes I and II
    • Fitz-Patrick V.D., Vandlen R.L. 6 agonist selectivity determinants in somatostatin receptor subtypes I and II. J. Biol. Chem. 269: 24621, 1994.
    • (1994) J. Biol. Chem. , vol.269 , pp. 24621
    • Fitz-Patrick, V.D.1    Vandlen, R.L.2
  • 77
    • 0030817407 scopus 로고    scopus 로고
    • Ligand binding pocket of the human somatostatin receptor 5 (hsstr5): Mutational analysis of the extracellular domains
    • (in press)
    • Greenwood M.T., Hukovic N., Kumar U., Panetta R., Hjorth S.A., Srikant C.B., Patel Y.C. Ligand binding pocket of the human somatostatin receptor 5 (hsstr5): mutational analysis of the extracellular domains. Mol. Pharmacol. 1997 (in press).
    • (1997) Mol. Pharmacol.
    • Greenwood, M.T.1    Hukovic, N.2    Kumar, U.3    Panetta, R.4    Hjorth, S.A.5    Srikant, C.B.6    Patel, Y.C.7
  • 78
    • 0027339347 scopus 로고
    • Identification and quantification of Gi-type GTPbinding proteins that copurify with a pituitary somatostatin receptor
    • Luthin D.R., Eppler C.M., Linden J. Identification and quantification of Gi-type GTPbinding proteins that copurify with a pituitary somatostatin receptor. J. Biol. Chem. 268: 5990, 1993.
    • (1993) J. Biol. Chem. , vol.268 , pp. 5990
    • Luthin, D.R.1    Eppler, C.M.2    Linden, J.3
  • 79
    • 0027336786 scopus 로고
    • Gi alpha 3 and G (o) alpha selectively associate with cloned somatostatin in receptor subtypes SSTR2
    • Law S.F., Yasuda K., Bell G.I., Reisine T. Gi alpha 3 and G (o) alpha selectively associate with cloned somatostatin in receptor subtypes SSTR2. J. Biol. Chem. 268: 10721, 1993.
    • (1993) J. Biol. Chem. , vol.268 , pp. 10721
    • Law, S.F.1    Yasuda, K.2    Bell, G.I.3    Reisine, T.4
  • 80
    • 0026612461 scopus 로고
    • Gi alpha 1 selectively couples somatostatin receptors to adenylyl cyclase in pituitary-derived AtT-20 cells
    • Tallent M., and Reisine T. Gi alpha 1 selectively couples somatostatin receptors to adenylyl cyclase in pituitary-derived AtT-20 cells. Mol. Pharmacol. 41: 452, 1992.
    • (1992) Mol. Pharmacol. , vol.41 , pp. 452
    • Tallent, M.1    Reisine, T.2
  • 81
    • 0028359453 scopus 로고
    • G protein specificity in receptor effector coupling: Analysis of the roles of Go and Gi in GH4CI pituitary cells
    • Liu Y.F., Jacobs K.H., Rosewick M.M., Albert P.R. G protein specificity in receptor effector coupling: analysis of the roles of Go and Gi in GH4CI pituitary cells. J. Biol. Chem. 269: 13880, 1994.
    • (1994) J. Biol. Chem. , vol.269 , pp. 13880
    • Liu, Y.F.1    Jacobs, K.H.2    Rosewick, M.M.3    Albert, P.R.4
  • 82
    • 0028128734 scopus 로고
    • The D2 dopamine receptor isoforms signal through distinct Gi alpha proteins to inhibit adenylyl cyclase. A study with site-directed mutant Gi alpha proteins
    • Senogles S.E. The D2 dopamine receptor isoforms signal through distinct Gi alpha proteins to inhibit adenylyl cyclase. A study with site-directed mutant Gi alpha proteins. J. Biol. Chem. 269: 23120, 1994.
    • (1994) J. Biol. Chem. , vol.269 , pp. 23120
    • Senogles, S.E.1
  • 83
    • 0024308853 scopus 로고
    • Somatostatin-14 and somatostatin-28 induce opposite effects on potassium currents in rat neocortical neurons
    • (USA)
    • Wang H.L., Bogen C., Reisine T., Dichter M. Somatostatin-14 and somatostatin-28 induce opposite effects on potassium currents in rat neocortical neurons. Proc. Natl. Acad. Sci. (USA) 86: 9616, 1989.
    • (1989) Proc. Natl. Acad. Sci. , vol.86 , pp. 9616
    • Wang, H.L.1    Bogen, C.2    Reisine, T.3    Dichter, M.4
  • 84
    • 0025741172 scopus 로고
    • Somatostatin activates an inwardly rectifying K+ conductance in freshly dispersed rat somatotrophs
    • Sims S.M., Lussier B.T., Kraicer J. Somatostatin activates an inwardly rectifying K+ conductance in freshly dispersed rat somatotrophs. J. Physiol. 441: 615, 1991.
    • (1991) J. Physiol. , vol.441 , pp. 615
    • Sims, S.M.1    Lussier, B.T.2    Kraicer, J.3
  • 88
    • 0023879290 scopus 로고
    • Characterization of the cyclic AMP-independent actions of somatostatin in GH cells
    • Koch B.D., Schonbrunn A. Characterization of the cyclic AMP-independent actions of somatostatin in GH cells. J. Biol. Chem. 263: 226, 1988.
    • (1988) J. Biol. Chem. , vol.263 , pp. 226
    • Koch, B.D.1    Schonbrunn, A.2
  • 89
    • 0024578585 scopus 로고
    • Somatostatin blocks a calcium current in rat sympathetic ganglion neurons
    • Ikeda S.R., Schofield G.G. Somatostatin blocks a calcium current in rat sympathetic ganglion neurons. J. Physiol. 409: 221, 1989.
    • (1989) J. Physiol. , vol.409 , pp. 221
    • Ikeda, S.R.1    Schofield, G.G.2
  • 90
    • 0025880464 scopus 로고
    • Assignment of G protein subtypes to specific receptors inducing inhibition of calcium currents
    • Kleuss C., Heschefeler J., Ewel C., Rosenthal W., Schultz G., Wittig B. Assignment of G protein subtypes to specific receptors inducing inhibition of calcium currents. Nature 353: 43, 1991.
    • (1991) Nature , vol.353 , pp. 43
    • Kleuss, C.1    Heschefeler, J.2    Ewel, C.3    Rosenthal, W.4    Schultz, G.5    Wittig, B.6
  • 91
    • 0028365950 scopus 로고
    • 2+ current modulated by cGMP-dependent protein kinase
    • 2+ current modulated by cGMP-dependent protein kinase. Nature 369: 336, 1994.
    • (1994) Nature , vol.369 , pp. 336
    • Meriney, S.D.1    Gray, D.B.2    Pilar, G.R.3
  • 92
    • 0030245732 scopus 로고    scopus 로고
    • Neurotransmitter-induced inhibition of exocytosis in insulin-secreting β cells by activation of calcineurin
    • Renstrom E., Ding W-G., Bokvist K., Rorsman P. Neurotransmitter-induced inhibition of exocytosis in insulin-secreting β cells by activation of calcineurin. Neuron 17: 513, 1996.
    • (1996) Neuron , vol.17 , pp. 513
    • Renstrom, E.1    Ding, W.-G.2    Bokvist, K.3    Rorsman, P.4
  • 93
    • 0024801629 scopus 로고
    • Beta-adrenergic and somatostatin receptors regulate Na-H exchange independent of cAMP
    • Barber, D.L., M.E. McGuire, M.B. Ganz. Beta-adrenergic and somatostatin receptors regulate Na-H exchange independent of cAMP. J. Biol. Chem. 264: 21038, 1989.
    • (1989) J. Biol. Chem. , vol.264 , pp. 21038
    • Barber, D.L.1    McGuire, M.E.2    Ganz, M.B.3
  • 94
    • 0025050521 scopus 로고
    • Arachidonic acid metabolites as mediators of somatostatin-induced increase of neuronal M-current
    • Schweitzer R., Madamba S., Siggins G.R. Arachidonic acid metabolites as mediators of somatostatin-induced increase of neuronal M-current. Nature 346: 464, 1990.
    • (1990) Nature , vol.346 , pp. 464
    • Schweitzer, R.1    Madamba, S.2    Siggins, G.R.3
  • 95
    • 0025168456 scopus 로고
    • Somatostatin action in pituitary cells involves two independent transduction mechanisms
    • Schonbrunn A. Somatostatin action in pituitary cells involves two independent transduction mechanisms. Metabolism 39 (Suppl. 2): 96, 1990.
    • (1990) Metabolism , vol.39 , Issue.2 SUPPL. , pp. 96
    • Schonbrunn, A.1
  • 96
    • 0027469601 scopus 로고
    • Affinity purification of a somatostatin receptor-G-protein complex demonstrates specificity in receptor-G-protein coupling
    • Brown P., Schonbrunn A. Affinity purification of a somatostatin receptor-G-protein complex demonstrates specificity in receptor-G-protein coupling J. Biol. Chem. 268: 6668, 1993.
    • (1993) J. Biol. Chem. , vol.268 , pp. 6668
    • Brown, P.1    Schonbrunn, A.2
  • 98
    • 0028134705 scopus 로고
    • The somatostatin receptor SSTR1 is coupled to phosphotyrosine phosphatase activity in CHO-K1 cells
    • Florio T., Rim C., Hershberger R.E., Loda M., Stork P.J. The somatostatin receptor SSTR1 is coupled to phosphotyrosine phosphatase activity in CHO-K1 cells. Mol. Endocrinol. 8: 1289, 1994.
    • (1994) Mol. Endocrinol. , vol.8 , pp. 1289
    • Florio, T.1    Rim, C.2    Hershberger, R.E.3    Loda, M.4    Stork, P.J.5
  • 101
    • 0029939159 scopus 로고    scopus 로고
    • Somatostatin inhibits PC C13 thyroid cell proliferation through the modulation of phosphotyrosine phosphatase activity-impairment of the somatostatinergic effects by stable expression of EIA viral oncogene
    • Florio T., Scarziello A., Fattore M., Dalto V., Salzano S., Rossi G., Berlingieri M.T., Fusco A., Schettini G. Somatostatin inhibits PC C13 thyroid cell proliferation through the modulation of phosphotyrosine phosphatase activity-impairment of the somatostatinergic effects by stable expression of EIA viral oncogene. J. Biol. Chem. 271: 6129, 1996.
    • (1996) J. Biol. Chem. , vol.271 , pp. 6129
    • Florio, T.1    Scarziello, A.2    Fattore, M.3    Dalto, V.4    Salzano, S.5    Rossi, G.6    Berlingieri, M.T.7    Fusco, A.8    Schettini, G.9
  • 102
    • 1842324483 scopus 로고    scopus 로고
    • Subtype selective human somatostatin receptor (hSSTR) mediated cytostatin and cytotoxic actions involve different signalling mechanisms
    • Minneapolis, June (abstract)
    • Sharma K., Patel Y.C., Srikant C.B. Subtype selective human somatostatin receptor (hSSTR) mediated cytostatin and cytotoxic actions involve different signalling mechanisms. Program Annual Meeting US Endocrine Society, Minneapolis, June 1997 (abstract).
    • (1997) Program Annual Meeting US Endocrine Society
    • Sharma, K.1    Patel, Y.C.2    Srikant, C.B.3
  • 103
    • 0028246882 scopus 로고
    • Subtype-specific signalling mechanisms of somatostatin receptors SSTR1 and SSTR2
    • Hou C., Gilbert R.L., Barber D.L. Subtype-specific signalling mechanisms of somatostatin receptors SSTR1 and SSTR2. J. Biol. Chem. 269: 10357, 1994.
    • (1994) J. Biol. Chem. , vol.269 , pp. 10357
    • Hou, C.1    Gilbert, R.L.2    Barber, D.L.3
  • 104
    • 0027943354 scopus 로고
    • Somatostatin receptor subtype SSTR2 mediates the inhibition of high voltage activated calcium channels by somatostatin and its analogue SMS201-995
    • Fujii Y., Gonoi T., Yamada Y., Chihara K., Inagaki N., Seino S. Somatostatin receptor subtype SSTR2 mediates the inhibition of high voltage activated calcium channels by somatostatin and its analogue SMS201-995. FEBS Lett. 355: 117, 1994.
    • (1994) FEBS Lett , vol.355 , pp. 117
    • Fujii, Y.1    Gonoi, T.2    Yamada, Y.3    Chihara, K.4    Inagaki, N.5    Seino, S.6
  • 105
    • 0029812770 scopus 로고    scopus 로고
    • Modulation of high voltage-activated calcium channels by somatostatin in acutely isolated rat amygdaloid neurons
    • Viana F., Hille B. Modulation of high voltage-activated calcium channels by somatostatin in acutely isolated rat amygdaloid neurons. J. Neurosci. 16: 6000, 1996.
    • (1996) J. Neurosci. , vol.16 , pp. 6000
    • Viana, F.1    Hille, B.2
  • 106
    • 0028336973 scopus 로고
    • Functional coupling of SSTR4, a major hippocampal somatostatin receptor, to adenylate cyclase inhibition, arachidonate release and activation of the mitogen-activated protein kinase cascade
    • Bito H., Mori M., Sakanaka C., Takano T., Honda Z., Gotoh Y., Nishida E., Shimizu T. Functional coupling of SSTR4, a major hippocampal somatostatin receptor, to adenylate cyclase inhibition, arachidonate release and activation of the mitogen-activated protein kinase cascade. J. Biol. Chem. 269: 12722, 1994.
    • (1994) J. Biol. Chem. , vol.269 , pp. 12722
    • Bito, H.1    Mori, M.2    Sakanaka, C.3    Takano, T.4    Honda, Z.5    Gotoh, Y.6    Nishida, E.7    Shimizu, T.8
  • 108
    • 0025117441 scopus 로고
    • Evidence that receptor-linked G protein inhibits exocytosis by a post-second messenger mechanism in AtT-20 cells
    • Luini A., de Matteis M.A. Evidence that receptor-linked G protein inhibits exocytosis by a post-second messenger mechanism in AtT-20 cells. J. Neurochem. 54: 30, 1990.
    • (1990) J. Neurochem. , vol.54 , pp. 30
    • Luini, A.1    De Matteis, M.A.2
  • 109
    • 0025061707 scopus 로고
    • Somatostatin inhibition of hormone release: Effects on cytosolic Cal' and interference with distal secretory events
    • Wollheim C.B., Winiger B.P., Ullrich S., Wuarin F. Schlegel W. Somatostatin inhibition of hormone release: effects on cytosolic Cal' and interference with distal secretory events. Metabolism (Suppl. 11) 39: 101, 1990.
    • (1990) Metabolism , vol.39 , Issue.11 SUPPL. , pp. 101
    • Wollheim, C.B.1    Winiger, B.P.2    Ullrich, S.3    Schlegel W, W.F.4
  • 110
    • 0026682699 scopus 로고
    • G protein activation of a hormone-stimulated phosphatase in human tumor cells
    • Pan M.G., Florio T., Stork P.J.S. G protein activation of a hormone-stimulated phosphatase in human tumor cells. Science 256: 1215, 1992.
    • (1992) Science , vol.256 , pp. 1215
    • Pan, M.G.1    Florio, T.2    Stork, P.J.S.3
  • 111
    • 0029937024 scopus 로고    scopus 로고
    • Octapeptide somatostatin analog SMS 201-995 induces translocation of intracellular PTPIC to membranes in MCF-7 human breast cancer adenocarcinoma cells
    • Srikant C.B., Shen S.H. Octapeptide somatostatin analog SMS 201-995 induces translocation of intracellular PTPIC to membranes in MCF-7 human breast cancer adenocarcinoma cells. Endocrinology 137: 3461, 1996.
    • (1996) Endocrinology , vol.137 , pp. 3461
    • Srikant, C.B.1    Shen, S.H.2
  • 112
    • 0028933059 scopus 로고
    • Cell cycle dependent induction of apoptosis by somatostatin analog SMS201995 in AtT-20 mouse pituitary tumor cells
    • Srikant C.B. Cell cycle dependent induction of apoptosis by somatostatin analog SMS201995 in AtT-20 mouse pituitary tumor cells. Biochem. Biophys. Res. Commun. 209: 400, 1995.
    • (1995) Biochem. Biophys. Res. Commun. , vol.209 , pp. 400
    • Srikant, C.B.1
  • 113
    • 0029959644 scopus 로고    scopus 로고
    • Subtype selective induction of p53-dependent apoptosis but not bell cycle arrest by human somatostatin receptor 3
    • Sharma K., Patel Y.C., Srikant C.B. Subtype selective induction of p53-dependent apoptosis but not bell cycle arrest by human somatostatin receptor 3. Mol. Endocrinol. 10: 1688, 1996.
    • (1996) Mol. Endocrinol. , vol.10 , pp. 1688
    • Sharma, K.1    Patel, Y.C.2    Srikant, C.B.3
  • 114
    • 0027142895 scopus 로고
    • Tissue distribution of somatostatin receptor subtype messenger ribonucleic acid in the rat
    • Bruno J.F., Xu Y., Song J., Berelowitz M. Tissue distribution of somatostatin receptor subtype messenger ribonucleic acid in the rat. Endocrinology 133: 2561, 1993.
    • (1993) Endocrinology , vol.133 , pp. 2561
    • Bruno, J.F.1    Xu, Y.2    Song, J.3    Berelowitz, M.4
  • 116
    • 0028295877 scopus 로고
    • Differential expression of messenger RNAs for somatostatin receptor subtypes SSTR1, SSTR2, and SSTR3 in adult rat brain: Analysis by RNA blotting and in situ hybridization histochemistry
    • Kong H., DePaoli A.M., Breder C.D., Yasuda K., Bell G.I., Reisine T. Differential expression of messenger RNAs for somatostatin receptor subtypes SSTR1, SSTR2, and SSTR3 in adult rat brain: analysis by RNA blotting and in situ hybridization histochemistry. Neuroscience 59: 175, 1994.
    • (1994) Neuroscience , vol.59 , pp. 175
    • Kong, H.1    DePaoli, A.M.2    Breder, C.D.3    Yasuda, K.4    Bell, G.I.5    Reisine, T.6
  • 117
    • 0029617807 scopus 로고
    • Embryonic and postnatal mRNA distribution of five somatostatin receptor subtypes in the rat brain
    • Thoss V.S., Perez J., Due D., Hoyer D. Embryonic and postnatal mRNA distribution of five somatostatin receptor subtypes in the rat brain. Neuropharmacology 34: 1673, 1995.
    • (1995) Neuropharmacology , vol.34 , pp. 1673
    • Thoss, V.S.1    Perez, J.2    Due, D.3    Hoyer, D.4
  • 118
    • 0030254426 scopus 로고    scopus 로고
    • Expression of five somatostatin receptor mRNAs in the human brain and pituitary
    • Thoss V.S., Perez J., Probat A., Hoyer D. Expression of five somatostatin receptor mRNAs in the human brain and pituitary. Arch. Pharmacol. 354: 411-419, 1996.
    • (1996) Arch. Pharmacol. , vol.354 , pp. 411-419
    • Thoss, V.S.1    Perez, J.2    Probat, A.3    Hoyer, D.4
  • 119
    • 0029947693 scopus 로고    scopus 로고
    • Localization of the somatostatin receptor SST2a in rat brain using a specific antipeptide antibody
    • Dournaud P., Gu Y.Z., Schonbrunn A., Mazella J., Tannenbaum G.S., Beaudet A. Localization of the somatostatin receptor SST2A in rat brain using a specific antipeptide antibody. J. Neurosci. 16: 4468, 1996.
    • (1996) J. Neurosci. , vol.16 , pp. 4468
    • Dournaud, P.1    Gu, Y.Z.2    Schonbrunn, A.3    Mazella, J.4    Tannenbaum, G.S.5    Beaudet, A.6
  • 120
    • 0028153733 scopus 로고
    • Expression of multiple somatostatin receptor genes in AtT-20 cells: Evidence for a novel somatostatin-28 selective receptor subtype
    • Patel Y.C., Panetta R., Escher E., Greenwood M., Srikant C.B. Expression of multiple somatostatin receptor genes in AtT-20 cells: evidence for a novel somatostatin-28 selective receptor subtype. J. Biol. Chem. 269: 1506, 1994.
    • (1994) J. Biol. Chem. , vol.269 , pp. 1506
    • Patel, Y.C.1    Panetta, R.2    Escher, E.3    Greenwood, M.4    Srikant, C.B.5
  • 121
    • 0028823431 scopus 로고
    • Expression of mRNA for somatostatin receptor (sstr) types 2 and 5 in individual rat pituitary cells. A double labeling in situ hybridization analysis
    • Day R., Dong W., Panetta R., Kraicer J., Greenwood M.T., Patel Y.C. Expression of mRNA for somatostatin receptor (sstr) types 2 and 5 in individual rat pituitary cells. A double labeling in situ hybridization analysis. Endocrinology 136: 5232, 1995.
    • (1995) Endocrinology , vol.136 , pp. 5232
    • Day, R.1    Dong, W.2    Panetta, R.3    Kraicer, J.4    Greenwood, M.T.5    Patel, Y.C.6
  • 122
    • 0028789364 scopus 로고
    • Widespread distribution of somatostatin receptor messenger ribonucleic acids in rat pituitary
    • O'Carroll A., Krempels K. Widespread distribution of somatostatin receptor messenger ribonucleic acids in rat pituitary. Endocrinology 136: 5224, 1995.
    • (1995) Endocrinology , vol.136 , pp. 5224
    • O'Carroll, A.1    Krempels, K.2
  • 123
    • 0028888586 scopus 로고
    • Expression of mRNA for all 5 human somatostatin receptor (hSSTR1-5) in pituitary tumors
    • Panetta R., Patel Y.C. Expression of mRNA for all 5 human somatostatin receptor (hSSTR1-5) in pituitary tumors. Life Sci. 56: 333, 1994.
    • (1994) Life Sci. , vol.56 , pp. 333
    • Panetta, R.1    Patel, Y.C.2
  • 124
    • 0011274397 scopus 로고
    • Expression of mRNA for somatostatin receptor (sstr) subtypes 1-5 in islets and differential downregulation of sstr2 mRNA by SST agonists
    • June 10-13, Atlanta, Georgia, Abstr. no. 485
    • Grigorakis S.I., Panetta R., Patel Y.C. Expression of mRNA for somatostatin receptor (sstr) subtypes 1-5 in islets and differential downregulation of sstr2 mRNA by SST agonists. Program Annual Meeting American Diabetes Association, June 10-13, 1995, Atlanta, Georgia, Abstr. no. 485, p. 132A.
    • (1995) Program Annual Meeting American Diabetes Association
    • Grigorakis, S.I.1    Panetta, R.2    Patel, Y.C.3
  • 125
    • 0023547202 scopus 로고
    • Selective binding of somatostatin-14 and somatostatin -28 to islet cells revealed by quantitative electron microscopic autoradiography
    • Amherdt M., Patel Y.C., Orci L. Selective binding of somatostatin-14 and somatostatin -28 to islet cells revealed by quantitative electron microscopic autoradiography. J. Clin. Invest. 80: 1455, 1987.
    • (1987) J. Clin. Invest. , vol.80 , pp. 1455
    • Amherdt, M.1    Patel, Y.C.2    Orci, L.3
  • 127
    • 0026041670 scopus 로고
    • The role of somatostatin and its analogs in the diagnosis and treatment of tumors
    • Lamberts S.W.J., Krenning E.P., and Reubi J.-C. The role of somatostatin and its analogs in the diagnosis and treatment of tumors. Endocr. Rev. 12: 450, 1991.
    • (1991) Endocr. Rev. , vol.12 , pp. 450
    • Lamberts, S.W.J.1    Krenning, E.P.2    Reubi, J.-C.3
  • 128
    • 0028044677 scopus 로고
    • Heterogeneous expression of two somatostatin receptor subtypes in pituitary tumors
    • Greenman Y., Melmed S. Heterogeneous expression of two somatostatin receptor subtypes in pituitary tumors. J. Clin. Endocrinol. Metab. 78: 398, 1994.
    • (1994) J. Clin. Endocrinol. Metab. , vol.78 , pp. 398
    • Greenman, Y.1    Melmed, S.2
  • 129
    • 0027980885 scopus 로고
    • Expression of three somatostatin receptor subtypes in pituitary adenomas: Evidence for preferential SSTR5 expression in the mammosomatotroph lineage
    • Greenman Y., Melmed S. Expression of three somatostatin receptor subtypes in pituitary adenomas: evidence for preferential SSTR5 expression in the mammosomatotroph lineage. J. Clin. Endocrinol. Metab. 79: 724, 1994.
    • (1994) J. Clin. Endocrinol. Metab. , vol.79 , pp. 724
    • Greenman, Y.1    Melmed, S.2
  • 131
    • 0028820057 scopus 로고
    • Expression of somatostatin receptor subtypes in breast carcinoma, carcinoid tumor, and renal cell carcinoma
    • Vikic-Topic S., Reisch K.P., Kvols L.K., Vuk-Pavlovic S. Expression of somatostatin receptor subtypes in breast carcinoma, carcinoid tumor, and renal cell carcinoma. J. Clin. Endocrinol. Metab. 80: 2974, 1995.
    • (1995) J. Clin. Endocrinol. Metab. , vol.80 , pp. 2974
    • Vikic-Topic, S.1    Reisch, K.P.2    Kvols, L.K.3    Vuk-Pavlovic, S.4
  • 132
    • 0028280635 scopus 로고
    • Identification of somatostatin receptor subtypes and an implication for the efficacy of somatostatin analogue SMS201-995 in treatment of human endocrine tumors
    • Kubota A., Yamada Y., Kagimoto S., Shimatsu A., Imamura M., Tsuda K., Imura H., Seino S., Seino Y. Identification of somatostatin receptor subtypes and an implication for the efficacy of somatostatin analogue SMS201-995 in treatment of human endocrine tumors. J. Clin. Invest. 93: 1321, 1994.
    • (1994) J. Clin. Invest. , vol.93 , pp. 1321
    • Kubota, A.1    Yamada, Y.2    Kagimoto, S.3    Shimatsu, A.4    Imamura, M.5    Tsuda, K.6    Imura, H.7    Seino, S.8    Seino, Y.9
  • 136
    • 0009792609 scopus 로고
    • Model systems for the study of seven transmembrane segment receptors
    • Dohlman H.G., Thorner J., Caron M.G., Lelkowitz R.J. Model systems for the study of seven transmembrane segment receptors. J. Biol. Chem. 268: 337, 1991.
    • (1991) J. Biol. Chem. , vol.268 , pp. 337
    • Dohlman, H.G.1    Thorner, J.2    Caron, M.G.3    Lelkowitz, R.J.4
  • 137
    • 0020573238 scopus 로고
    • Prolonged somatostatin treatment desensitizes somatostatin's inhibition of receptor-mediated release of adrenocorticotropin hormone and sensitizes adenylate cyclase
    • Reisine T.D., Axelrod J. Prolonged somatostatin treatment desensitizes somatostatin's inhibition of receptor-mediated release of adrenocorticotropin hormone and sensitizes adenylate cyclase. Endocrinology 113: 811, 1983.
    • (1983) Endocrinology , vol.113 , pp. 811
    • Reisine, T.D.1    Axelrod, J.2
  • 138
    • 0021839891 scopus 로고
    • Ultrastructural autoradiographic localization of somatostatin-28 in the rat pituitary gland
    • Morel G., Leroux P., Pelletier G. Ultrastructural autoradiographic localization of somatostatin-28 in the rat pituitary gland. Endocrinology 116: 1615, 1985.
    • (1985) Endocrinology , vol.116 , pp. 1615
    • Morel, G.1    Leroux, P.2    Pelletier, G.3
  • 139
    • 0024307980 scopus 로고
    • Binding and internalization of somatostatin, insulin, and glucagon by cultured rat islet cells
    • Amherdt M., Patel Y.C., Orci L. Binding and internalization of somatostatin, insulin, and glucagon by cultured rat islet cells. J. Clin. Invest. 84: 412, 1989.
    • (1989) J. Clin. Invest. , vol.84 , pp. 412
    • Amherdt, M.1    Patel, Y.C.2    Orci, L.3
  • 141
    • 0023871632 scopus 로고
    • Somatostatin pretreatment increases the number of somatostatin receptors in GH4C1 pituitary cells and does not reduce cellular responsiveness to somatostatin
    • Presky D.H., Schonbrunn A. Somatostatin pretreatment increases the number of somatostatin receptors in GH4C1 pituitary cells and does not reduce cellular responsiveness to somatostatin. J. Biol. Chem. 263: 714, 1988
    • (1988) J. Biol. Chem. , vol.263 , pp. 714
    • Presky, D.H.1    Schonbrunn, A.2
  • 142
    • 0029791822 scopus 로고    scopus 로고
    • Agonist-dependent regulation of cloned human somatostatin receptor types 1-5 (hSSTR1-5): Subtype selective internalization or upregulation
    • Hukovic N., Panetta R., Kumar U., Patel Y.C. Agonist-dependent regulation of cloned human somatostatin receptor types 1-5 (hSSTR1-5): subtype selective internalization or upregulation. Endocrinology 137: 4046, 1996.
    • (1996) Endocrinology , vol.137 , pp. 4046
    • Hukovic, N.1    Panetta, R.2    Kumar, U.3    Patel, Y.C.4
  • 143
    • 0031032344 scopus 로고    scopus 로고
    • Differential internalization of somatostatin in COS-7 cells transfected with SST1 and SST2 receptor subtypes: A confocal microscopic study using novel fluorescent somatostatin derivatives
    • Nouel D., Gaudriault G., Houle M., Reisine T., Vincent J-P., Mazella J., Beaudet A. Differential internalization of somatostatin in COS-7 cells transfected with SST1 and SST2 receptor subtypes: a confocal microscopic study using novel fluorescent somatostatin derivatives. Endocrinology 138: 296, 1997.
    • (1997) Endocrinology , vol.138 , pp. 296
    • Nouel, D.1    Gaudriault, G.2    Houle, M.3    Reisine, T.4    Vincent, J.-P.5    Mazella, J.6    Beaudet, A.7
  • 144
    • 0031025989 scopus 로고    scopus 로고
    • Endocytosis of the rat somatostatin receptors - Subtype discrimination, ligand specificity and delineation of carboxyterminal positive and negative sequence motifs
    • Roth A., Kreienkamp H.J., Nehring R.B., Roosterman D., Meyerhof W., Richter D. Endocytosis of the rat somatostatin receptors - subtype discrimination, ligand specificity and delineation of carboxyterminal positive and negative sequence motifs. DNA and Cell Biology 16: 111, 1997.
    • (1997) DNA and Cell Biology , vol.16 , pp. 111
    • Roth, A.1    Kreienkamp, H.J.2    Nehring, R.B.3    Roosterman, D.4    Meyerhof, W.5    Richter, D.6
  • 148
    • 0022514580 scopus 로고
    • 17β estradiol induces somatostatin (SRIF) inhibition of prolactin release and regulates SRIF receptors in rat anterior pituitary cells
    • Kimura N., Hayafiji C., Konagaye H., Takahashi K. 17β estradiol induces somatostatin (SRIF) inhibition of prolactin release and regulates SRIF receptors in rat anterior pituitary cells. Endocrinology 119: 1028, 1986.
    • (1986) Endocrinology , vol.119 , pp. 1028
    • Kimura, N.1    Hayafiji, C.2    Konagaye, H.3    Takahashi, K.4
  • 149
    • 0030474240 scopus 로고    scopus 로고
    • Estrogen regulates somatostatin receptor subtype 2 messenger ribonucleic acid expression in human breast cancer cells
    • Xu Y.X., Song J., Berelowitz M., Bruno J.F. Estrogen regulates somatostatin receptor subtype 2 messenger ribonucleic acid expression in human breast cancer cells. Endocrinology 5634, 1996.
    • (1996) Endocrinology , pp. 5634
    • Xu, Y.X.1    Song, J.2    Berelowitz, M.3    Bruno, J.F.4
  • 151
    • 0031047393 scopus 로고    scopus 로고
    • Thyroid hormone induced expression of specific somatostatin receptor subtypes correlates with involution of the TtT-97 murine thyrotrope tumor
    • James R.A., Sarapura V.D., Bruns C., Raulf F., Dowding J.M., Gordon D.F., Wood W.M., Ridgway E.G. Thyroid hormone induced expression of specific somatostatin receptor subtypes correlates with involution of the TtT-97 murine thyrotrope tumor. Endocrinology 138: 719, 1997.
    • (1997) Endocrinology , vol.138 , pp. 719
    • James, R.A.1    Sarapura, V.D.2    Bruns, C.3    Raulf, F.4    Dowding, J.M.5    Gordon, D.F.6    Wood, W.M.7    Ridgway, E.G.8
  • 152
    • 0027985614 scopus 로고
    • Pituitary and hypothalamic somatostatin receptor subtype messenger ribonucleic acid expression in the food-deprived and diabetic rat
    • Bruno J.F., Xu Y., Song J., Berelowitz M. Pituitary and hypothalamic somatostatin receptor subtype messenger ribonucleic acid expression in the food-deprived and diabetic rat. Endocrinology 135: 1787, 1994.
    • (1994) Endocrinology , vol.135 , pp. 1787
    • Bruno, J.F.1    Xu, Y.2    Song, J.3    Berelowitz, M.4
  • 153
    • 0028321929 scopus 로고
    • Sequence analysis of the promoter region of the rat somatostatin receptor subtype 1 gene
    • Hauser F., Meyerhof W., Wulfsen I., Schonrock C., Richter D. Sequence analysis of the promoter region of the rat somatostatin receptor subtype 1 gene. FEBS Lett. 345: 225, 1994.
    • (1994) FEBS Lett , vol.345 , pp. 225
    • Hauser, F.1    Meyerhof, W.2    Wulfsen, I.3    Schonrock, C.4    Richter, D.5
  • 154
    • 0029077967 scopus 로고
    • Cloning of the gene encoding the human somatostatin receptor 2: Sequence analysis of the 5′ flanking promoter region
    • Greenwood M.T., Robertson L.-A., Patel Y.C. Cloning of the gene encoding the human somatostatin receptor 2: sequence analysis of the 5′ flanking promoter region. Gene 159: 291, 1995.
    • (1995) Gene , vol.159 , pp. 291
    • Greenwood, M.T.1    Robertson, L.-A.2    Patel, Y.C.3
  • 155
    • 0029850996 scopus 로고    scopus 로고
    • The helix-loop-helix transcription factor SEF2 regulates the activity of a novel initiator element in the promoter of the human somatostatin receptor II gene
    • Pscherer A., Dorflinger U., Kirfel J., Gawlas K., Ruschoff J., Buettner R., Schule R. The helix-loop-helix transcription factor SEF2 regulates the activity of a novel initiator element in the promoter of the human somatostatin receptor II gene. EMBO J. 15: 6680, 1996.
    • (1996) EMBO J , vol.15 , pp. 6680
    • Pscherer, A.1    Dorflinger, U.2    Kirfel, J.3    Gawlas, K.4    Ruschoff, J.5    Buettner, R.6    Schule, R.7
  • 156
    • 0028890214 scopus 로고
    • Characterization of the proximal region of the rat somatostatin receptor gene, SSTR4
    • Xu Y., Bruno J.F., Berelowitz M. Characterization of the proximal region of the rat somatostatin receptor gene, SSTR4. Biochem. Biophys. Res. Commun. 206: 935, 1995.
    • (1995) Biochem. Biophys. Res. Commun. , vol.206 , pp. 935
    • Xu, Y.1    Bruno, J.F.2    Berelowitz, M.3
  • 158
    • 0030588656 scopus 로고    scopus 로고
    • The tuberin (TSC2) autosomal dominant polycystic kidney disease (PKD1) and somatostatin type V receptor (SSTR5) genes form a synteny group in the fugu genome
    • Sanford R., Sgotto B., Burn T., Brenner S. The tuberin (TSC2) autosomal dominant polycystic kidney disease (PKD1) and somatostatin type V receptor (SSTR5) genes form a synteny group in the fugu genome. Genomics 38: 84, 1996.
    • (1996) Genomics , vol.38 , pp. 84
    • Sanford, R.1    Sgotto, B.2    Burn, T.3    Brenner, S.4
  • 159
    • 0031035050 scopus 로고    scopus 로고
    • Loss of the polycystic kidney (PKD 1) region of chromosome 1 6pl 3 in renal cyst cells support a loss of function model for cyst pathogenesis
    • Brassier J., Henske E.P. Loss of the polycystic kidney (PKD 1) region of chromosome 1 6pl 3 in renal cyst cells support a loss of function model for cyst pathogenesis. J. Clin. Invest. 99. 194, 1997.
    • (1997) J. Clin. Invest. , vol.99 , pp. 194
    • Brassier, J.1    Henske, E.P.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.