New bradykinin antagonists having very high potency at B1 receptors

Immunopharmacology

Volumn 33, Issue 1-3, 1996, Pages 183-185

  Gera, Lajos ^a   Stewart, John M ^a   Whalley, Eric T ^b   Burkard, Michael ^b   Zuzack, John S ^b  

^a Dept of Biochem Univ of C ^*  (United States)

^b Departments of New Leads Chemistry and Pharmacology   (United States)

Author keywords

bradykinin antagonist; receptors, B1

Indexed keywords

BRADYKININ ANTAGONIST; BRADYKININ B1 RECEPTOR; BRADYKININ B1 RECEPTOR ANTAGONIST; BRADYKININ B2 RECEPTOR; BRADYKININ[1-8]; CP 0298; NEW DRUG; UNCLASSIFIED DRUG;

AMINO ACID ANALYSIS; ANIMAL CELL; ANIMAL TISSUE; AORTA; CHO CELL; CONFERENCE PAPER; CONTROLLED STUDY; DRUG SYNTHESIS; GUINEA PIG; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HUMAN; HUMAN CELL; ILEUM; LUNG FIBROBLAST; MASS SPECTROMETRY; NONHUMAN; PEPTIDE SYNTHESIS; PRIORITY JOURNAL; RABBIT; RECEPTOR BINDING; SMOOTH MUSCLE CONTRACTILITY;

EID: 0030175857     PISSN: 01623109     EISSN: None     Source Type: Journal    
DOI: 10.1016/0162-3109(96)00100-2     Document Type: Conference Paper

References (9)

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