In vivo pharmacological profile of novel, potent, stable BK antagonists at B1 and B2 receptors

Immunopharmacology

Volumn 33, Issue 1-3, 1996, Pages 191-193

  Hanson, Wendy L ^a   McCullough, Rosann G ^a   Selig, William M ^a   Wieczorek, Maciej ^a   Ross, Sherman ^a   Whalley, Eric T ^a   Stewart, John M ^b   Gera, Lajos ^b  

^a Departments of New Leads Chemistry and Pharmacology   (United States)

^b Dept Biochemistry   (United States)

Author keywords

bradykinin; bradykinin antagonists; des Arg9 bradykinin; dog blood pressure; kinin receptors

Indexed keywords

ACETYLCHOLINE; ANGIOTENSIN; B 9340; B 9430; BRADYKININ; BRADYKININ ANTAGONIST; BRADYKININ B1 RECEPTOR ANTAGONIST; BRADYKININ B2 RECEPTOR ANTAGONIST; BRADYKININ[1-8]; CP 0298; CP 0364; CP 0597; ICATIBANT; LYSYLLYSYLARGINYLPROLYL(4 HYDROXYPROLYL)GLYCYL 2 (2,3 DIHYDRO 1H INDEN 2 YL)GLYCYLSERYL 2 (2,3 DIHYDRO 1H INDEN 2 YL)GLYCYLOCTAHYDRO 1H INDOLE 2 CARBOXYLIC ACID; NORADRENALIN; SUBSTANCE P; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; BLOOD PRESSURE; CONFERENCE PAPER; CONTROLLED STUDY; DEPRESSOR RESPONSE; DOG; DRUG ANTAGONISM; DRUG HALF LIFE; DRUG POTENCY; DRUG SELECTIVITY; DRUG STABILITY; FEMALE; HUMAN; INTRAVENOUS DRUG ADMINISTRATION; KIDNEY TUBULE EPITHELIUM; LUNG; MALE; NONHUMAN; PLASMA; PRIORITY JOURNAL; RAT;

EID: 0030176099     PISSN: 01623109     EISSN: None     Source Type: Journal    
DOI: 10.1016/0162-3109(96)00037-9     Document Type: Conference Paper

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