SCOPUS 정보 검색 플랫폼

Journal of the American Chemical Society

Volumn 118, Issue 37, 1996, Pages 8860-8870

Synthesis, X-ray structure, and properties of fluorocyclopropane analogs of the duocarmycins incorporating the 9,9-difluoro-1,2,9,9a-tetrahydrocyclopropa[c]benzo[e]indol-4-one (F2CBI) alkylation subunit

(2) Boger, Dale L a Jenkins, Tracy J a

a SCRIPPS RESEARCH INSTITUTE (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTINEOPLASTIC AGENT; INDOLE DERIVATIVE; ORGANOFLUORINE DERIVATIVE; RACHELMYCIN DERIVATIVE;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; REACTION ANALYSIS; ULTRAVIOLET SPECTROPHOTOMETRY; X RAY ANALYSIS;

EID: 0029813588 PISSN: 00027863 EISSN: None Source Type: Journal
DOI: 10.1021/ja961888n Document Type: Article

Times cited : (62)

References (141)

1
- 0019779478
- Chidester, C. G.; Krueger, W. C.; Mizsak, S. A.; Duchamp, D. J.; Martin, D. G. J. Am. Chem. Soc. 1981, 103, 7629.
- (1981) J. Am. Chem. Soc. , vol.103 , pp. 7629
- Chidester, C.G.¹ Krueger, W.C.² Mizsak, S.A.³ Duchamp, D.J.⁴ Martin, D.G.⁵

2
- 0024996602
- Ichimura, M.; Ogawa, T.; Takahashi, K.; Kobayashi, E.; Kawamoto, I.; Yasuzawa, T.; Takahashi, I.; Nakano, H. J. Antibiot. 1990, 43, 1037. Ichimura, M.; Ogawa, T.; Katsumata, S.; Takahashi, K.; Takahashi, I.; Nakano, H. J. Antibiot. 1991, 44, 1045.
- (1990) J. Antibiot. , vol.43 , pp. 1037
- Ichimura, M.¹ Ogawa, T.² Takahashi, K.³ Kobayashi, E.⁴ Kawamoto, I.⁵ Yasuzawa, T.⁶ Takahashi, I.⁷ Nakano, H.⁸

3
- 0026069784
- Ichimura, M.; Ogawa, T.; Takahashi, K.; Kobayashi, E.; Kawamoto, I.; Yasuzawa, T.; Takahashi, I.; Nakano, H. J. Antibiot. 1990, 43, 1037. Ichimura, M.; Ogawa, T.; Katsumata, S.; Takahashi, K.; Takahashi, I.; Nakano, H. J. Antibiot. 1991, 44, 1045.
- (1991) J. Antibiot. , vol.44 , pp. 1045
- Ichimura, M.¹ Ogawa, T.² Katsumata, S.³ Takahashi, K.⁴ Takahashi, I.⁵ Nakano, H.⁶

4
- 0024261683
- Takahashi, I.; Takahashi, K.; Ichimura, M.; Morimoto, M.; Asano, K.; Kawamoto, I.; Tomita, F.; Nakano, H. J. Antibiot. 1988, 41, 1915. Yasuzawa, T.; Iida, T.; Muroi, K.; Ichimura, M.; Takahashi, K.; Sano, H. Chem. Pharm. Bull. 1988, 36, 3728.
- (1988) J. Antibiot. , vol.41 , pp. 1915
- Takahashi, I.¹ Takahashi, K.² Ichimura, M.³ Morimoto, M.⁴ Asano, K.⁵ Kawamoto, I.⁶ Tomita, F.⁷ Nakano, H.⁸

5
- 0023748655
- Takahashi, I.; Takahashi, K.; Ichimura, M.; Morimoto, M.; Asano, K.; Kawamoto, I.; Tomita, F.; Nakano, H. J. Antibiot. 1988, 41, 1915. Yasuzawa, T.; Iida, T.; Muroi, K.; Ichimura, M.; Takahashi, K.; Sano, H. Chem. Pharm. Bull. 1988, 36, 3728.
- (1988) Chem. Pharm. Bull. , vol.36 , pp. 3728
- Yasuzawa, T.¹ Iida, T.² Muroi, K.³ Ichimura, M.⁴ Takahashi, K.⁵ Sano, H.⁶

6
- 0028937557
- Yasuzawa, T.; Muroi, K.; Ichimura, M.; Takahashi, I.; Ogawa, T.; Takahashi, K.; Sano, H.; Saitoh, Y. Chem. Pharm. Bull. 1995, 43, 378.
- (1995) Chem. Pharm. Bull. , vol.43 , pp. 378
- Yasuzawa, T.¹ Muroi, K.² Ichimura, M.³ Takahashi, I.⁴ Ogawa, T.⁵ Takahashi, K.⁶ Sano, H.⁷ Saitoh, Y.⁸

7
- 0023707447
- Ichimura, M.; Muroi, K.; Asano, K.; Kawamoto, I.; Tomita, F.; Morimoto, M.; Nakano, H. J. Antibiot. 1988, 41, 1285.
- (1988) J. Antibiot. , vol.41 , pp. 1285
- Ichimura, M.¹ Muroi, K.² Asano, K.³ Kawamoto, I.⁴ Tomita, F.⁵ Morimoto, M.⁶ Nakano, H.⁷

8
- 0024400866
- Ogawa, T.; Ichimura, M.; Katsumata, S.; Morimoto, M.; Takahashi, K. J. Antibiot. 1989, 42, 1299.
- (1989) J. Antibiot. , vol.42 , pp. 1299
- Ogawa, T.¹ Ichimura, M.² Katsumata, S.³ Morimoto, M.⁴ Takahashi, K.⁵

9
- 0023700046
- Ohba, K.; Watabe, H.; Saski, T.; Takeuchi, Y.; Kodama, Y.; Nakazawa, T.; Yamamoto, H.; Shomura, T.; Sezaki, M.; Kondo, S. J. Antibiot. 1988, 41, 1515. Ishii, S.; Nagasawa, M.; Kariya, Y.; Yamamoto, H.; Inouye, S.; Kondo, S. J. Antibiot. 1989, 42, 1713.
- (1988) J. Antibiot. , vol.41 , pp. 1515
- Ohba, K.¹ Watabe, H.² Saski, T.³ Takeuchi, Y.⁴ Kodama, Y.⁵ Nakazawa, T.⁶ Yamamoto, H.⁷ Shomura, T.⁸ Sezaki, M.⁹ Kondo, S.¹⁰

10
- 0024388410
- Ohba, K.; Watabe, H.; Saski, T.; Takeuchi, Y.; Kodama, Y.; Nakazawa, T.; Yamamoto, H.; Shomura, T.; Sezaki, M.; Kondo, S. J. Antibiot. 1988, 41, 1515. Ishii, S.; Nagasawa, M.; Kariya, Y.; Yamamoto, H.; Inouye, S.; Kondo, S. J. Antibiot. 1989, 42, 1713.
- (1989) J. Antibiot. , vol.42 , pp. 1713
- Ishii, S.¹ Nagasawa, M.² Kariya, Y.³ Yamamoto, H.⁴ Inouye, S.⁵ Kondo, S.⁶

11
- 0024240366
- Warpehoski, M. A.; Hurley, L. H. Chem. Res. Toxicol. 1988, 1, 315. Warpehoski, M. A. In Advances in DNA Sequence Specific Agents; Hurley, L. H., Ed.; JAI: Greenwich, CT, 1992; Vol. 1, 217.
- (1988) Chem. Res. Toxicol. , vol.1 , pp. 315
- Warpehoski, M.A.¹ Hurley, L.H.²

12
- 0001124924
- Hurley, L. H., Ed.; JAI: Greenwich, CT
- Warpehoski, M. A.; Hurley, L. H. Chem. Res. Toxicol. 1988, 1, 315. Warpehoski, M. A. In Advances in DNA Sequence Specific Agents; Hurley, L. H., Ed.; JAI: Greenwich, CT, 1992; Vol. 1, 217.
- (1992) Advances in DNA Sequence Specific Agents , vol.1 , pp. 217
- Warpehoski, M.A.¹

13
- 33845376321
- Hurley, L. H.; Needham-VanDevanter, D. R. Ace. Chem. Res. 1986, 19, 230. Hurley, L. H.; Draves, P. H. In Molecular Aspects of Anticancer Drug-DNA Interactions; Neidle, S., Waring, M., Eds.; CRC Press: Ann Arbor, MI, 1993; Vol. 1, 89.
- (1986) Ace. Chem. Res. , vol.19 , pp. 230
- Hurley, L.H.¹ Needham-VanDevanter, D.R.²

14
- 0001911789
- Neidle, S., Waring, M., Eds.; CRC Press: Ann Arbor, MI
- Hurley, L. H.; Needham-VanDevanter, D. R. Ace. Chem. Res. 1986, 19, 230. Hurley, L. H.; Draves, P. H. In Molecular Aspects of Anticancer Drug-DNA Interactions; Neidle, S., Waring, M., Eds.; CRC Press: Ann Arbor, MI, 1993; Vol. 1, 89.
- (1993) Molecular Aspects of Anticancer Drug-DNA Interactions , vol.1 , pp. 89
- Hurley, L.H.¹ Draves, P.H.²

15
- 0000819601
- Rahman, A.-u., Ed.; Elsevier: Amsterdam
- Coleman, R. S.; Boger, D. L. In Studies in Natural Product Chemistry: Rahman, A.-u., Ed.; Elsevier: Amsterdam, 1989; Vol. 3, 301. Boger, D. L. In Heterocycles in Bioorganic Chemistry; Bergman, J., van der Plas, H. C., Simonyl, M., Eds.; Royal Soc. of Chem.; Cambridge, 1991; p 103. Boger, D. L. In Advances in Heterocylic Natural Product Synthesis; Pearson, W. H., Ed.; JAI: Greenwich, CT, 1992; Vol. 2, 1.
- (1989) Studies in Natural Product Chemistry , vol.3 , pp. 301
- Coleman, R.S.¹ Boger, D.L.²

16
- 0002195060
- Bergman, J., van der Plas, H. C., Simonyl, M., Eds.; Royal Soc. of Chem.; Cambridge
- Coleman, R. S.; Boger, D. L. In Studies in Natural Product Chemistry: Rahman, A.-u., Ed.; Elsevier: Amsterdam, 1989; Vol. 3, 301. Boger, D. L. In Heterocycles in Bioorganic Chemistry; Bergman, J., van der Plas, H. C., Simonyl, M., Eds.; Royal Soc. of Chem.; Cambridge, 1991; p 103. Boger, D. L. In Advances in Heterocylic Natural Product Synthesis; Pearson, W. H., Ed.; JAI: Greenwich, CT, 1992; Vol. 2, 1.
- (1991) Heterocycles in Bioorganic Chemistry , pp. 103
- Boger, D.L.¹

17
- 0002872624
- Pearson, W. H., Ed.; JAI: Greenwich, CT
- Coleman, R. S.; Boger, D. L. In Studies in Natural Product Chemistry: Rahman, A.-u., Ed.; Elsevier: Amsterdam, 1989; Vol. 3, 301. Boger, D. L. In Heterocycles in Bioorganic Chemistry; Bergman, J., van der Plas, H. C., Simonyl, M., Eds.; Royal Soc. of Chem.; Cambridge, 1991; p 103. Boger, D. L. In Advances in Heterocylic Natural Product Synthesis; Pearson, W. H., Ed.; JAI: Greenwich, CT, 1992; Vol. 2, 1.
- (1992) Advances in Heterocylic Natural Product Synthesis , vol.2 , pp. 1
- Boger, D.L.¹

18
- 0029782488
- Boger, D. L.; Johnson, D. S. Angew Chem., Int. Ed. Engl. 1996, 35, 1439. Boger, D. L.; Johnson, D. S. Proc. Natl Acad. Sci. U.S.A. 1995, 92, 3642. Boger, D. L. Acc. Chem. Res. 1995, 28, 20. Boger, D. L. Chemtracts: Org. Chem. 1991, 4, 329. Boger, D. L. In Proc. R. A. Welch Found. Conf. Chem. Res., XXXV., Chem. Frontiers Med. 1991, 35, 137.
- (1996) Angew Chem., Int. Ed. Engl. , vol.35 , pp. 1439
- Boger, D.L.¹ Johnson, D.S.²

19
- 0029053550
- Boger, D. L.; Johnson, D. S. Angew Chem., Int. Ed. Engl. 1996, 35, 1439. Boger, D. L.; Johnson, D. S. Proc. Natl Acad. Sci. U.S.A. 1995, 92, 3642. Boger, D. L. Acc. Chem. Res. 1995, 28, 20. Boger, D. L. Chemtracts: Org. Chem. 1991, 4, 329. Boger, D. L. In Proc. R. A. Welch Found. Conf. Chem. Res., XXXV., Chem. Frontiers Med. 1991, 35, 137.
- (1995) Proc. Natl Acad. Sci. U.S.A. , vol.92 , pp. 3642
- Boger, D.L.¹ Johnson, D.S.²

20
- 0002631330
- Boger, D. L.; Johnson, D. S. Angew Chem., Int. Ed. Engl. 1996, 35, 1439. Boger, D. L.; Johnson, D. S. Proc. Natl Acad. Sci. U.S.A. 1995, 92, 3642. Boger, D. L. Acc. Chem. Res. 1995, 28, 20. Boger, D. L. Chemtracts: Org. Chem. 1991, 4, 329. Boger, D. L. In Proc. R. A. Welch Found. Conf. Chem. Res., XXXV., Chem. Frontiers Med. 1991, 35, 137.
- (1995) Acc. Chem. Res. , vol.28 , pp. 20
- Boger, D.L.¹

21
- 0000923199
- Boger, D. L.; Johnson, D. S. Angew Chem., Int. Ed. Engl. 1996, 35, 1439. Boger, D. L.; Johnson, D. S. Proc. Natl Acad. Sci. U.S.A. 1995, 92, 3642. Boger, D. L. Acc. Chem. Res. 1995, 28, 20. Boger, D. L. Chemtracts: Org. Chem. 1991, 4, 329. Boger, D. L. In Proc. R. A. Welch Found. Conf. Chem. Res., XXXV., Chem. Frontiers Med. 1991, 35, 137.
- (1991) Chemtracts: Org. Chem. , vol.4 , pp. 329
- Boger, D.L.¹

22
- 0001112837
- Boger, D. L.; Johnson, D. S. Angew Chem., Int. Ed. Engl. 1996, 35, 1439. Boger, D. L.; Johnson, D. S. Proc. Natl Acad. Sci. U.S.A. 1995, 92, 3642. Boger, D. L. Acc. Chem. Res. 1995, 28, 20. Boger, D. L. Chemtracts: Org. Chem. 1991, 4, 329. Boger, D. L. In Proc. R. A. Welch Found. Conf. Chem. Res., XXXV., Chem. Frontiers Med. 1991, 35, 137.
- (1991) Proc. R. A. Welch Found. Conf. Chem. Res., XXXV., Chem. Frontiers Med. , vol.35 , pp. 137
- Boger, D.L.¹

23
- 0021715394
- Hurley, L. H.; Reynolds, V. L.; Swenson, D. H.; Petzold, G. L.; Scahill, T. A. Science 1984, 226, 843. Reynolds, V. L.; Molineux, I. J.; Kaplan, D. J.; Swedson, D. H.; Hurley, L. H. Biochemistry 1985, 24, 6228. Hurley. L. H.; Lee, C-S.; McGovren, J. P.; Warpehoski, M. A.; Mitchell, M. A.; Kelly, R. C.; Aristoff, P. A. Biochemistry 1988, 27, 3886. Scahill, T. A.; Jensen, R. M.; Swenson, D. H.; Hatzenbuhler, N. T.; Petzold, G.; Wierenga, W.; Brahme, N. D. Biochemistry 1990, 29, 2852. Hurley, L. H.; Warpehoski, M. A.; Lee, C-S.; McGovren, J. P.; Scahill, T. A.; Kelly, R. C.; Mitchell, M. A.; Wicnienski, N. A.; Gebhard, I.; Johnson, P. D.; Bradford, V. S. J. Am. Chem. Soc. 1990, 112, 4633. Warpehoski, M. A.; Harper, D. E.; Mitchell, M. A.; Monroe, T. J. Biochemistry 1992, 31, 2502.
- (1984) Science , vol.226 , pp. 843
- Hurley, L.H.¹ Reynolds, V.L.² Swenson, D.H.³ Petzold, G.L.⁴ Scahill, T.A.⁵

24
- 0022358966
- Hurley, L. H.; Reynolds, V. L.; Swenson, D. H.; Petzold, G. L.; Scahill, T. A. Science 1984, 226, 843. Reynolds, V. L.; Molineux, I. J.; Kaplan, D. J.; Swedson, D. H.; Hurley, L. H. Biochemistry 1985, 24, 6228. Hurley. L. H.; Lee, C-S.; McGovren, J. P.; Warpehoski, M. A.; Mitchell, M. A.; Kelly, R. C.; Aristoff, P. A. Biochemistry 1988, 27, 3886. Scahill, T. A.; Jensen, R. M.; Swenson, D. H.; Hatzenbuhler, N. T.; Petzold, G.; Wierenga, W.; Brahme, N. D. Biochemistry 1990, 29, 2852. Hurley, L. H.; Warpehoski, M. A.; Lee, C-S.; McGovren, J. P.; Scahill, T. A.; Kelly, R. C.; Mitchell, M. A.; Wicnienski, N. A.; Gebhard, I.; Johnson, P. D.; Bradford, V. S. J. Am. Chem. Soc. 1990, 112, 4633. Warpehoski, M. A.; Harper, D. E.; Mitchell, M. A.; Monroe, T. J. Biochemistry 1992, 31, 2502.
- (1985) Biochemistry , vol.24 , pp. 6228
- Reynolds, V.L.¹ Molineux, I.J.² Kaplan, D.J.³ Swedson, D.H.⁴ Hurley, L.H.⁵

25
- 0024290406
- Hurley, L. H.; Reynolds, V. L.; Swenson, D. H.; Petzold, G. L.; Scahill, T. A. Science 1984, 226, 843. Reynolds, V. L.; Molineux, I. J.; Kaplan, D. J.; Swedson, D. H.; Hurley, L. H. Biochemistry 1985, 24, 6228. Hurley. L. H.; Lee, C-S.; McGovren, J. P.; Warpehoski, M. A.; Mitchell, M. A.; Kelly, R. C.; Aristoff, P. A. Biochemistry 1988, 27, 3886. Scahill, T. A.; Jensen, R. M.; Swenson, D. H.; Hatzenbuhler, N. T.; Petzold, G.; Wierenga, W.; Brahme, N. D. Biochemistry 1990, 29, 2852. Hurley, L. H.; Warpehoski, M. A.; Lee, C-S.; McGovren, J. P.; Scahill, T. A.; Kelly, R. C.; Mitchell, M. A.; Wicnienski, N. A.; Gebhard, I.; Johnson, P. D.; Bradford, V. S. J. Am. Chem. Soc. 1990, 112, 4633. Warpehoski, M. A.; Harper, D. E.; Mitchell, M. A.; Monroe, T. J. Biochemistry 1992, 31, 2502.
- (1988) Biochemistry , vol.27 , pp. 3886
- Hurley, L.H.¹ Lee, C.-S.² McGovren, J.P.³ Warpehoski, M.A.⁴ Mitchell, M.A.⁵ Kelly, R.C.⁶ Aristoff, P.A.⁷

26
- 0025269611
- Hurley, L. H.; Reynolds, V. L.; Swenson, D. H.; Petzold, G. L.; Scahill, T. A. Science 1984, 226, 843. Reynolds, V. L.; Molineux, I. J.; Kaplan, D. J.; Swedson, D. H.; Hurley, L. H. Biochemistry 1985, 24, 6228. Hurley. L. H.; Lee, C-S.; McGovren, J. P.; Warpehoski, M. A.; Mitchell, M. A.; Kelly, R. C.; Aristoff, P. A. Biochemistry 1988, 27, 3886. Scahill, T. A.; Jensen, R. M.; Swenson, D. H.; Hatzenbuhler, N. T.; Petzold, G.; Wierenga, W.; Brahme, N. D. Biochemistry 1990, 29, 2852. Hurley, L. H.; Warpehoski, M. A.; Lee, C-S.; McGovren, J. P.; Scahill, T. A.; Kelly, R. C.; Mitchell, M. A.; Wicnienski, N. A.; Gebhard, I.; Johnson, P. D.; Bradford, V. S. J. Am. Chem. Soc. 1990, 112, 4633. Warpehoski, M. A.; Harper, D. E.; Mitchell, M. A.; Monroe, T. J. Biochemistry 1992, 31, 2502.
- (1990) Biochemistry , vol.29 , pp. 2852
- Scahill, T.A.¹ Jensen, R.M.² Swenson, D.H.³ Hatzenbuhler, N.T.⁴ Petzold, G.⁵ Wierenga, W.⁶ Brahme, N.D.⁷

27
- 0025148364
- Hurley, L. H.; Reynolds, V. L.; Swenson, D. H.; Petzold, G. L.; Scahill, T. A. Science 1984, 226, 843. Reynolds, V. L.; Molineux, I. J.; Kaplan, D. J.; Swedson, D. H.; Hurley, L. H. Biochemistry 1985, 24, 6228. Hurley. L. H.; Lee, C-S.; McGovren, J. P.; Warpehoski, M. A.; Mitchell, M. A.; Kelly, R. C.; Aristoff, P. A. Biochemistry 1988, 27, 3886. Scahill, T. A.; Jensen, R. M.; Swenson, D. H.; Hatzenbuhler, N. T.; Petzold, G.; Wierenga, W.; Brahme, N. D. Biochemistry 1990, 29, 2852. Hurley, L. H.; Warpehoski, M. A.; Lee, C-S.; McGovren, J. P.; Scahill, T. A.; Kelly, R. C.; Mitchell, M. A.; Wicnienski, N. A.; Gebhard, I.; Johnson, P. D.; Bradford, V. S. J. Am. Chem. Soc. 1990, 112, 4633. Warpehoski, M. A.; Harper, D. E.; Mitchell, M. A.; Monroe, T. J. Biochemistry 1992, 31, 2502.
- (1990) J. Am. Chem. Soc. , vol.112 , pp. 4633
- Hurley, L.H.¹ Warpehoski, M.A.² Lee, C.-S.³ McGovren, J.P.⁴ Scahill, T.A.⁵ Kelly, R.C.⁶ Mitchell, M.A.⁷ Wicnienski, N.A.⁸ Gebhard, I.⁹ Johnson, P.D.¹⁰ Bradford, V.S.¹¹

28
- 0026511431
- Hurley, L. H.; Reynolds, V. L.; Swenson, D. H.; Petzold, G. L.; Scahill, T. A. Science 1984, 226, 843. Reynolds, V. L.; Molineux, I. J.; Kaplan, D. J.; Swedson, D. H.; Hurley, L. H. Biochemistry 1985, 24, 6228. Hurley. L. H.; Lee, C-S.; McGovren, J. P.; Warpehoski, M. A.; Mitchell, M. A.; Kelly, R. C.; Aristoff, P. A. Biochemistry 1988, 27, 3886. Scahill, T. A.; Jensen, R. M.; Swenson, D. H.; Hatzenbuhler, N. T.; Petzold, G.; Wierenga, W.; Brahme, N. D. Biochemistry 1990, 29, 2852. Hurley, L. H.; Warpehoski, M. A.; Lee, C-S.; McGovren, J. P.; Scahill, T. A.; Kelly, R. C.; Mitchell, M. A.; Wicnienski, N. A.; Gebhard, I.; Johnson, P. D.; Bradford, V. S. J. Am. Chem. Soc. 1990, 112, 4633. Warpehoski, M. A.; Harper, D. E.; Mitchell, M. A.; Monroe, T. J. Biochemistry 1992, 31, 2502.
- (1992) Biochemistry , vol.31 , pp. 2502
- Warpehoski, M.A.¹ Harper, D.E.² Mitchell, M.A.³ Monroe, T.J.⁴

29
- 0028376605
- Boger, D. L.; Johnson, D. S.; Yun, W.; Tarby, C. M. Bioorg. Med. Chem. 1994, 2, 115. Boger, D. L.; Munk, S. A.; Zarrinmayeh, H.; Ishizaki, T.; Haught, J.; Bina, M. Tetrahedron 1991, 47, 2661. Boger, D. L.; Coleman, R. S.; Invergo, B. J.; Sakya, S. M.; Ishizaki, T.; Munk, S. A.; Zarrinmayeh, H.; Kitos, P. A.; Thompson, S. C. J. Am. Chem. Soc. 1990, 112, 4623. Boger, D. L.; Coleman, R. S. J. Am. Chem. Soc. 1988, 110, 4796 and 1321.
- (1994) Bioorg. Med. Chem. , vol.2 , pp. 115
- Boger, D.L.¹ Johnson, D.S.² Yun, W.³ Tarby, C.M.⁴

30
- 0025980193
- Boger, D. L.; Johnson, D. S.; Yun, W.; Tarby, C. M. Bioorg. Med. Chem. 1994, 2, 115. Boger, D. L.; Munk, S. A.; Zarrinmayeh, H.; Ishizaki, T.; Haught, J.; Bina, M. Tetrahedron 1991, 47, 2661. Boger, D. L.; Coleman, R. S.; Invergo, B. J.; Sakya, S. M.; Ishizaki, T.; Munk, S. A.; Zarrinmayeh, H.; Kitos, P. A.; Thompson, S. C. J. Am. Chem. Soc. 1990, 112, 4623. Boger, D. L.; Coleman, R. S. J. Am. Chem. Soc. 1988, 110, 4796 and 1321.
- (1991) Tetrahedron , vol.47 , pp. 2661
- Boger, D.L.¹ Munk, S.A.² Zarrinmayeh, H.³ Ishizaki, T.⁴ Haught, J.⁵ Bina, M.⁶

31
- 0025111222
- Boger, D. L.; Johnson, D. S.; Yun, W.; Tarby, C. M. Bioorg. Med. Chem. 1994, 2, 115. Boger, D. L.; Munk, S. A.; Zarrinmayeh, H.; Ishizaki, T.; Haught, J.; Bina, M. Tetrahedron 1991, 47, 2661. Boger, D. L.; Coleman, R. S.; Invergo, B. J.; Sakya, S. M.; Ishizaki, T.; Munk, S. A.; Zarrinmayeh, H.; Kitos, P. A.; Thompson, S. C. J. Am. Chem. Soc. 1990, 112, 4623. Boger, D. L.; Coleman, R. S. J. Am. Chem. Soc. 1988, 110, 4796 and 1321.
- (1990) J. Am. Chem. Soc. , vol.112 , pp. 4623
- Boger, D.L.¹ Coleman, R.S.² Invergo, B.J.³ Sakya, S.M.⁴ Ishizaki, T.⁵ Munk, S.A.⁶ Zarrinmayeh, H.⁷ Kitos, P.A.⁸ Thompson, S.C.⁹

32
- 0001607781
- Boger, D. L.; Johnson, D. S.; Yun, W.; Tarby, C. M. Bioorg. Med. Chem. 1994, 2, 115. Boger, D. L.; Munk, S. A.; Zarrinmayeh, H.; Ishizaki, T.; Haught, J.; Bina, M. Tetrahedron 1991, 47, 2661. Boger, D. L.; Coleman, R. S.; Invergo, B. J.; Sakya, S. M.; Ishizaki, T.; Munk, S. A.; Zarrinmayeh, H.; Kitos, P. A.; Thompson, S. C. J. Am. Chem. Soc. 1990, 112, 4623. Boger, D. L.; Coleman, R. S. J. Am. Chem. Soc. 1988, 110, 4796 and 1321.
- (1988) J. Am. Chem. Soc. , vol.110 , pp. 4796
- Boger, D.L.¹ Coleman, R.S.²

33
- 0025143478
- Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 4499. Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H.; Munk, S. A.; Kitos, P. A.; Suntornwat, O. J. Am. Chem. Soc. 1990, 112, 8961. Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H. J. Am. Chem. Soc. 1991, 113, 6645. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1993, 115, 9872. Boger, D. L.; Yun, W.; Terashima, S.; Fukuda, Y.; Nakatani, K.; Kitos, P. A.; Jin, Q. Bioorg. Med. Chem. Lett. 1992, 2, 759.
- (1990) J. Org. Chem. , vol.55 , pp. 4499
- Boger, D.L.¹ Ishizaki, T.² Zarrinmayeh, H.³ Kitos, P.A.⁴ Suntornwat, O.⁵

34
- 0025644317
- Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 4499. Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H.; Munk, S. A.; Kitos, P. A.; Suntornwat, O. J. Am. Chem. Soc. 1990, 112, 8961. Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H. J. Am. Chem. Soc. 1991, 113, 6645. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1993, 115, 9872. Boger, D. L.; Yun, W.; Terashima, S.; Fukuda, Y.; Nakatani, K.; Kitos, P. A.; Jin, Q. Bioorg. Med. Chem. Lett. 1992, 2, 759.
- (1990) J. Am. Chem. Soc. , vol.112 , pp. 8961
- Boger, D.L.¹ Ishizaki, T.² Zarrinmayeh, H.³ Munk, S.A.⁴ Kitos, P.A.⁵ Suntornwat, O.⁶

35
- 0025773799
- Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 4499. Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H.; Munk, S. A.; Kitos, P. A.; Suntornwat, O. J. Am. Chem. Soc. 1990, 112, 8961. Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H. J. Am. Chem. Soc. 1991, 113, 6645. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1993, 115, 9872. Boger, D. L.; Yun, W.; Terashima, S.; Fukuda, Y.; Nakatani, K.; Kitos, P. A.; Jin, Q. Bioorg. Med. Chem. Lett. 1992, 2, 759.
- (1991) J. Am. Chem. Soc. , vol.113 , pp. 6645
- Boger, D.L.¹ Ishizaki, T.² Zarrinmayeh, H.³

36
- 0027367893
- Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 4499. Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H.; Munk, S. A.; Kitos, P. A.; Suntornwat, O. J. Am. Chem. Soc. 1990, 112, 8961. Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H. J. Am. Chem. Soc. 1991, 113, 6645. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1993, 115, 9872. Boger, D. L.; Yun, W.; Terashima, S.; Fukuda, Y.; Nakatani, K.; Kitos, P. A.; Jin, Q. Bioorg. Med. Chem. Lett. 1992, 2, 759.
- (1993) J. Am. Chem. Soc. , vol.115 , pp. 9872
- Boger, D.L.¹ Yun, W.²

37
- 0026646153
- Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 4499. Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H.; Munk, S. A.; Kitos, P. A.; Suntornwat, O. J. Am. Chem. Soc. 1990, 112, 8961. Boger, D. L.; Ishizaki, T.; Zarrinmayeh, H. J. Am. Chem. Soc. 1991, 113, 6645. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1993, 115, 9872. Boger, D. L.; Yun, W.; Terashima, S.; Fukuda, Y.; Nakatani, K.; Kitos, P. A.; Jin, Q. Bioorg. Med. Chem. Lett. 1992, 2, 759.
- (1992) Bioorg. Med. Chem. Lett. , vol.2 , pp. 759
- Boger, D.L.¹ Yun, W.² Terashima, S.³ Fukuda, Y.⁴ Nakatani, K.⁵ Kitos, P.A.⁶ Jin, Q.⁷

38
- 0028095610
- Boger, D. L.; Johnson, D. S.; Yun, W. J. Am. Chem. Soc. 1994, 116, 1635.
- (1994) J. Am. Chem. Soc. , vol.116 , pp. 1635
- Boger, D.L.¹ Johnson, D.S.² Yun, W.³

39
- 0025600433
- Sugiyama, H.; Hosoda, M.; Saito, I.; Asai, A.; Saito, H. Tetrahedron Lett. 1990, 31, 7197. Lin, C. H.; Patel, D. J. J. Am. Chem. Soc. 1992, 114, 10658. Sugiyama, H.; Ohmori, K.; Chan, K. L.; Hosoda, M.; Asai, A.; Saito, H.; Saito, I. Tetrahedron Lett. 1993, 34, 2179. Yamamoto, K.; Sugiyama, H.; Kawanishi, S. Biochemistry 1993, 32, 1059. Asai, A.; Nagamura, S.; Saito, H. J. Am. Chem. Soc. 1994, 116, 4171.
- (1990) Tetrahedron Lett. , vol.31 , pp. 7197
- Sugiyama, H.¹ Hosoda, M.² Saito, I.³ Asai, A.⁴ Saito, H.⁵

40
- 0027051914
- Sugiyama, H.; Hosoda, M.; Saito, I.; Asai, A.; Saito, H. Tetrahedron Lett. 1990, 31, 7197. Lin, C. H.; Patel, D. J. J. Am. Chem. Soc. 1992, 114, 10658. Sugiyama, H.; Ohmori, K.; Chan, K. L.; Hosoda, M.; Asai, A.; Saito, H.; Saito, I. Tetrahedron Lett. 1993, 34, 2179. Yamamoto, K.; Sugiyama, H.; Kawanishi, S. Biochemistry 1993, 32, 1059. Asai, A.; Nagamura, S.; Saito, H. J. Am. Chem. Soc. 1994, 116, 4171.
- (1992) J. Am. Chem. Soc. , vol.114 , pp. 10658
- Lin, C.H.¹ Patel, D.J.²

41
- 0027528626
- Sugiyama, H.; Hosoda, M.; Saito, I.; Asai, A.; Saito, H. Tetrahedron Lett. 1990, 31, 7197. Lin, C. H.; Patel, D. J. J. Am. Chem. Soc. 1992, 114, 10658. Sugiyama, H.; Ohmori, K.; Chan, K. L.; Hosoda, M.; Asai, A.; Saito, H.; Saito, I. Tetrahedron Lett. 1993, 34, 2179. Yamamoto, K.; Sugiyama, H.; Kawanishi, S. Biochemistry 1993, 32, 1059. Asai, A.; Nagamura, S.; Saito, H. J. Am. Chem. Soc. 1994, 116, 4171.
- (1993) Tetrahedron Lett. , vol.34 , pp. 2179
- Sugiyama, H.¹ Ohmori, K.² Chan, K.L.³ Hosoda, M.⁴ Asai, A.⁵ Saito, H.⁶ Saito, I.⁷

42
- 0027466247
- Sugiyama, H.; Hosoda, M.; Saito, I.; Asai, A.; Saito, H. Tetrahedron Lett. 1990, 31, 7197. Lin, C. H.; Patel, D. J. J. Am. Chem. Soc. 1992, 114, 10658. Sugiyama, H.; Ohmori, K.; Chan, K. L.; Hosoda, M.; Asai, A.; Saito, H.; Saito, I. Tetrahedron Lett. 1993, 34, 2179. Yamamoto, K.; Sugiyama, H.; Kawanishi, S. Biochemistry 1993, 32, 1059. Asai, A.; Nagamura, S.; Saito, H. J. Am. Chem. Soc. 1994, 116, 4171.
- (1993) Biochemistry , vol.32 , pp. 1059
- Yamamoto, K.¹ Sugiyama, H.² Kawanishi, S.³

43
- 0028338850
- Sugiyama, H.; Hosoda, M.; Saito, I.; Asai, A.; Saito, H. Tetrahedron Lett. 1990, 31, 7197. Lin, C. H.; Patel, D. J. J. Am. Chem. Soc. 1992, 114, 10658. Sugiyama, H.; Ohmori, K.; Chan, K. L.; Hosoda, M.; Asai, A.; Saito, H.; Saito, I. Tetrahedron Lett. 1993, 34, 2179. Yamamoto, K.; Sugiyama, H.; Kawanishi, S. Biochemistry 1993, 32, 1059. Asai, A.; Nagamura, S.; Saito, H. J. Am. Chem. Soc. 1994, 116, 4171.
- (1994) J. Am. Chem. Soc. , vol.116 , pp. 4171
- Asai, A.¹ Nagamura, S.² Saito, H.³

44
- 0001631789
- Dolbier, W. R., Jr. Ace. Chem. Res. 1981, 14, 195. Dolbier, W. R., Jr. Adv. Strain Org. Chem. 1993, 2, 1.
- (1981) Ace. Chem. Res. , vol.14 , pp. 195
- Dolbier Jr., W.R.¹

45
- 0001631789
- Dolbier, W. R., Jr. Ace. Chem. Res. 1981, 14, 195. Dolbier, W. R., Jr. Adv. Strain Org. Chem. 1993, 2, 1.
- (1993) Adv. Strain Org. Chem. , vol.2 , pp. 1
- Dolbier Jr., W.R.¹

46
- 2742568845
- O'Neal, H. E.; Benson, S. W. J. Phys. Chem. 1968, 72, 1866. Roth, W. R.; Kirmse, W.; Hoffmann, W.; Lennartz, H.-W. Chem. Ber. 1982, 115, 2508.
- (1968) J. Phys. Chem. , vol.72 , pp. 1866
- O'Neal, H.E.¹ Benson, S.W.²

47
- 0000922207
- O'Neal, H. E.; Benson, S. W. J. Phys. Chem. 1968, 72, 1866. Roth, W. R.; Kirmse, W.; Hoffmann, W.; Lennartz, H.-W. Chem. Ber. 1982, 115, 2508.
- (1982) Chem. Ber. , vol.115 , pp. 2508
- Roth, W.R.¹ Kirmse, W.² Hoffmann, W.³ Lennartz, H.-W.⁴

48
- 0000254656
- Hoffmann, R.; Stohrer, N. P. J. Am. Chem. Soc. 1971, 93, 6941. Hoffmann, R. Tetrahedron Lett. 1970, 2907. Gunter, H. Tetrahedron Lett. 1970, 5173.
- (1971) J. Am. Chem. Soc. , vol.93 , pp. 6941
- Hoffmann, R.¹ Stohrer, N.P.²

49
- 0001466851
- Hoffmann, R.; Stohrer, N. P. J. Am. Chem. Soc. 1971, 93, 6941. Hoffmann, R. Tetrahedron Lett. 1970, 2907. Gunter, H. Tetrahedron Lett. 1970, 5173.
- (1970) Tetrahedron Lett. , pp. 2907
- Hoffmann, R.¹

50
- 0002114302
- Hoffmann, R.; Stohrer, N. P. J. Am. Chem. Soc. 1971, 93, 6941. Hoffmann, R. Tetrahedron Lett. 1970, 2907. Gunter, H. Tetrahedron Lett. 1970, 5173.
- (1970) Tetrahedron Lett. , pp. 5173
- Gunter, H.¹

51
- 0038471978
- Dolbier, W. R., Jr.; Fielder, T. H., Jr. J. Am. Chem. Soc. 1978, 100, 5577. Dolbier, W. R., Jr.; Sellers, S. F.; Al-Sader, B. H.; Elsheimer, S. J. Am. Chem. Soc. 1981, 103, 715.
- (1978) J. Am. Chem. Soc. , vol.100 , pp. 5577
- Dolbier Jr., W.R.¹ Fielder Jr., T.H.²

52
- 0038559753
- Dolbier, W. R., Jr.; Fielder, T. H., Jr. J. Am. Chem. Soc. 1978, 100, 5577. Dolbier, W. R., Jr.; Sellers, S. F.; Al-Sader, B. H.; Elsheimer, S. J. Am. Chem. Soc. 1981, 103, 715.
- (1981) J. Am. Chem. Soc. , vol.103 , pp. 715
- Dolbier Jr., W.R.¹ Sellers, S.F.² Al-Sader, B.H.³ Elsheimer, S.⁴

53
- 0008931078
- Dolbier, W. R., Jr.; Enoch, H. O. J. Am. Chem. Soc. 1977, 99, 4532. Sellers, S. F.; Dolbier, W. R., Jr.; Koroniak, H.; Al-Fekri, D. M. J. Org. Chem. 1984, 49, 1033. See also: Jefford, C. W.; Mareda, J.; Gehret, J.-C. E.; Karbengele, nT.; Graham, W. D.; Burger, U. J. Am. Chem. Soc. 1976, 98, 2585.
- (1977) J. Am. Chem. Soc. , vol.99 , pp. 4532
- Dolbier Jr., W.R.¹ Enoch, H.O.²

54
- 0037545669
- Dolbier, W. R., Jr.; Enoch, H. O. J. Am. Chem. Soc. 1977, 99, 4532. Sellers, S. F.; Dolbier, W. R., Jr.; Koroniak, H.; Al-Fekri, D. M. J. Org. Chem. 1984, 49, 1033. See also: Jefford, C. W.; Mareda, J.; Gehret, J.-C. E.; Karbengele, nT.; Graham, W. D.; Burger, U. J. Am. Chem. Soc. 1976, 98, 2585.
- (1984) J. Org. Chem. , vol.49 , pp. 1033
- Sellers, S.F.¹ Dolbier Jr., W.R.² Koroniak, H.³ Al-Fekri, D.M.⁴

55
- 0038559703
- Dolbier, W. R., Jr.; Enoch, H. O. J. Am. Chem. Soc. 1977, 99, 4532. Sellers, S. F.; Dolbier, W. R., Jr.; Koroniak, H.; Al-Fekri, D. M. J. Org. Chem. 1984, 49, 1033. See also: Jefford, C. W.; Mareda, J.; Gehret, J.-C. E.; Karbengele, nT.; Graham, W. D.; Burger, U. J. Am. Chem. Soc. 1976, 98, 2585.
- (1976) J. Am. Chem. Soc. , vol.98 , pp. 2585
- Jefford, C.W.¹ Mareda, J.² Gehret, J.-C.E.³ Karbengele, N.T.⁴ Graham, W.D.⁵ Burger, U.⁶

56
- 0025806550
- Sundberg, R. J.; Pitts, W. J. J. Org. Chem. 1991, 56, 3048. Sundberg, R. J.; Baxter, E. W.; Pitts, W. J.; Ahmed-Schofield, R.; Nishiguchi, T. J. Org. Chem. 1988, 53, 5097. Sundberg, R. J.; Baxter, E. W. Tetrahedron Lett. 1986, 27, 2687. Sundberg, R. J.; Nishiguchi, T. Tetrahedron Lett. 1983, 24, 4773.
- (1991) J. Org. Chem. , vol.56 , pp. 3048
- Sundberg, R.J.¹ Pitts, W.J.²

57
- 0023742849
- Sundberg, R. J.; Pitts, W. J. J. Org. Chem. 1991, 56, 3048. Sundberg, R. J.; Baxter, E. W.; Pitts, W. J.; Ahmed-Schofield, R.; Nishiguchi, T. J. Org. Chem. 1988, 53, 5097. Sundberg, R. J.; Baxter, E. W. Tetrahedron Lett. 1986, 27, 2687. Sundberg, R. J.; Nishiguchi, T. Tetrahedron Lett. 1983, 24, 4773.
- (1988) J. Org. Chem. , vol.53 , pp. 5097
- Sundberg, R.J.¹ Baxter, E.W.² Pitts, W.J.³ Ahmed-Schofield, R.⁴ Nishiguchi, T.⁵

58
- 0342577177
- Sundberg, R. J.; Pitts, W. J. J. Org. Chem. 1991, 56, 3048. Sundberg, R. J.; Baxter, E. W.; Pitts, W. J.; Ahmed-Schofield, R.; Nishiguchi, T. J. Org. Chem. 1988, 53, 5097. Sundberg, R. J.; Baxter, E. W. Tetrahedron Lett. 1986, 27, 2687. Sundberg, R. J.; Nishiguchi, T. Tetrahedron Lett. 1983, 24, 4773.
- (1986) Tetrahedron Lett. , vol.27 , pp. 2687
- Sundberg, R.J.¹ Baxter, E.W.²

59
- 8344250562
- Sundberg, R. J.; Pitts, W. J. J. Org. Chem. 1991, 56, 3048. Sundberg, R. J.; Baxter, E. W.; Pitts, W. J.; Ahmed-Schofield, R.; Nishiguchi, T. J. Org. Chem. 1988, 53, 5097. Sundberg, R. J.; Baxter, E. W. Tetrahedron Lett. 1986, 27, 2687. Sundberg, R. J.; Nishiguchi, T. Tetrahedron Lett. 1983, 24, 4773.
- (1983) Tetrahedron Lett. , vol.24 , pp. 4773
- Sundberg, R.J.¹ Nishiguchi, T.²

60
- 0003940950
- Elsevier: Amsterdam
- Ershov, V. V.; Nikiforov, G. A.; de Jonge, C. R. H. I, Quinonediazide; Elsevier: Amsterdam, 1981.
- (1981) Quinonediazide
- Ershov, V.V.¹ Nikiforov, G.A.² De Jonge, C.R.H.I.³

61
- 0026638104
- Boger, D. L.; Yun, W.; Teegarden, B. R. J. Org. Chem. 1992, 57, 2873.
- (1992) J. Org. Chem. , vol.57 , pp. 2873
- Boger, D.L.¹ Yun, W.² Teegarden, B.R.³

62
- 0026690441
- Sabol, J. S.; McCarthy, J. R. Tetrahedron Lett. 1992, 33, 3101.
- (1992) Tetrahedron Lett. , vol.33 , pp. 3101
- Sabol, J.S.¹ McCarthy, J.R.²

63
- 0011791477
- Stahly, G. P. J. Fluorine Chem. 1989, 43, 53. Miller, T. G.; Thanassi, J. W. J. Org. Chem. 1960, 25, 2009.
- (1989) J. Fluorine Chem. , vol.43 , pp. 53
- Stahly, G.P.¹

64
- 0005599532
- Stahly, G. P. J. Fluorine Chem. 1989, 43, 53. Miller, T. G.; Thanassi, J. W. J. Org. Chem. 1960, 25, 2009.
- (1960) J. Org. Chem. , vol.25 , pp. 2009
- Miller, T.G.¹ Thanassi, J.W.²

65
- 10144244116
- Diagnostic characterization is supplied in the supporting information
- Diagnostic characterization is supplied in the supporting information.

66
- 10144264687
- note
- 27 (9%).

67
- 0001161350
- Obayashi, M.; Ito, E.; Matsui, K.; Kondo, K. Tetrahedron Lett. 1982, 23, 2323. Obayasi, M.; Kondo, K. Tetrahedron Lett. 1982, 23, 2327.
- (1982) Tetrahedron Lett. , vol.23 , pp. 2323
- Obayashi, M.¹ Ito, E.² Matsui, K.³ Kondo, K.⁴

68
- 0001148194
- Obayashi, M.; Ito, E.; Matsui, K.; Kondo, K. Tetrahedron Lett. 1982, 23, 2323. Obayasi, M.; Kondo, K. Tetrahedron Lett. 1982, 23, 2327.
- (1982) Tetrahedron Lett. , vol.23 , pp. 2327
- Obayasi, M.¹ Kondo, K.²

69
- 0024998965
- Edwards, M. L.; Stemerick, D. M.; Jarvi, E. T.; Mattews, D. P.; McCarthy, J. R. Tetrahedron Lett. 1990, 31, 5571. Moore, W. R.; Sehatzman, G. L.; Jarvi, E. T.; Gross, R. S.; McCarthy, J. R. J. Am. Chem. Soc. 1992, 114, 360.
- (1990) Tetrahedron Lett. , vol.31 , pp. 5571
- Edwards, M.L.¹ Stemerick, D.M.² Jarvi, E.T.³ Mattews, D.P.⁴ McCarthy, J.R.⁵

70
- 85022502051
- Edwards, M. L.; Stemerick, D. M.; Jarvi, E. T.; Mattews, D. P.; McCarthy, J. R. Tetrahedron Lett. 1990, 31, 5571. Moore, W. R.; Sehatzman, G. L.; Jarvi, E. T.; Gross, R. S.; McCarthy, J. R. J. Am. Chem. Soc. 1992, 114, 360.
- (1992) J. Am. Chem. Soc. , vol.114 , pp. 360
- Moore, W.R.¹ Sehatzman, G.L.² Jarvi, E.T.³ Gross, R.S.⁴ McCarthy, J.R.⁵

71
- 0001664203
- Fuqua, S. A.; Duncan, W. G.; Silverstein, R. M. J. Org. Chem. 1965, 30, 1027. Naae, D. G.; Kesling, H. S.; Burton, D. J. Tetrahedron Lett. 1975, 3789. Naae, D. G.; Burton, D. J. J. Fluorine Chem. 1971, 1, 123. Naae, D. G.; Burton, D. J. Synth, Commun. 1973, 3, 197. Burton, D. J. J. Fluorine Chem. 1983, 18, 339. Burton, D. J.; Kesling, H. S.; Naae, D. G. J. Fluorine Chem. 1981, 18, 293. Wheaton, G. A.; Burton, D. J. J. Org. Chem. 1983, 48, 917. Matsuda, A.; Itoh, H.; Takenishi, K.; Susuki, T.; Ueda, T. Chem. Pharm. Bull. 1988, 36, 945. Fried, J.; Kittisopikul, S.; Hallinan, E. A. Tetrahedron Lett. 1984, 25, 4329. For recent and potentially useful alternatives: Dolbier, W. R., Jr.; Ocampo, R. J. Org. Chem. 1995, 60, 5378. Kim, K.-I.; McCarthy, J. R. Tetrahedron Lett. 1996, 37, 3223.
- (1965) Org. Chem. , vol.30 , pp. 1027
- Fuqua, S.A.¹ Duncan, W.G.² Silverstein, R.M.J.³

72
- 0343726998
- Fuqua, S. A.; Duncan, W. G.; Silverstein, R. M. J. Org. Chem. 1965, 30, 1027. Naae, D. G.; Kesling, H. S.; Burton, D. J. Tetrahedron Lett. 1975, 3789. Naae, D. G.; Burton, D. J. J. Fluorine Chem. 1971, 1, 123. Naae, D. G.; Burton, D. J. Synth, Commun. 1973, 3, 197. Burton, D. J. J. Fluorine Chem. 1983, 18, 339. Burton, D. J.; Kesling, H. S.; Naae, D. G. J. Fluorine Chem. 1981, 18, 293. Wheaton, G. A.; Burton, D. J. J. Org. Chem. 1983, 48, 917. Matsuda, A.; Itoh, H.; Takenishi, K.; Susuki, T.; Ueda, T. Chem. Pharm. Bull. 1988, 36, 945. Fried, J.; Kittisopikul, S.; Hallinan, E. A. Tetrahedron Lett. 1984, 25, 4329. For recent and potentially useful alternatives: Dolbier, W. R., Jr.; Ocampo, R. J. Org. Chem. 1995, 60, 5378. Kim, K.-I.; McCarthy, J. R. Tetrahedron Lett. 1996, 37, 3223.
- (1975) Tetrahedron Lett. , pp. 3789
- Naae, D.G.¹ Kesling, H.S.² Burton, D.J.³

73
- 49649155494
- Fuqua, S. A.; Duncan, W. G.; Silverstein, R. M. J. Org. Chem. 1965, 30, 1027. Naae, D. G.; Kesling, H. S.; Burton, D. J. Tetrahedron Lett. 1975, 3789. Naae, D. G.; Burton, D. J. J. Fluorine Chem. 1971, 1, 123. Naae, D. G.; Burton, D. J. Synth, Commun. 1973, 3, 197. Burton, D. J. J. Fluorine Chem. 1983, 18, 339. Burton, D. J.; Kesling, H. S.; Naae, D. G. J. Fluorine Chem. 1981, 18, 293. Wheaton, G. A.; Burton, D. J. J. Org. Chem. 1983, 48, 917. Matsuda, A.; Itoh, H.; Takenishi, K.; Susuki, T.; Ueda, T. Chem. Pharm. Bull. 1988, 36, 945. Fried, J.; Kittisopikul, S.; Hallinan, E. A. Tetrahedron Lett. 1984, 25, 4329. For recent and potentially useful alternatives: Dolbier, W. R., Jr.; Ocampo, R. J. Org. Chem. 1995, 60, 5378. Kim, K.-I.; McCarthy, J. R. Tetrahedron Lett. 1996, 37, 3223.
- (1971) J. Fluorine Chem. , vol.1 , pp. 123
- Naae, D.G.¹ Burton, D.J.²

74
- 84948510143
- Fuqua, S. A.; Duncan, W. G.; Silverstein, R. M. J. Org. Chem. 1965, 30, 1027. Naae, D. G.; Kesling, H. S.; Burton, D. J. Tetrahedron Lett. 1975, 3789. Naae, D. G.; Burton, D. J. J. Fluorine Chem. 1971, 1, 123. Naae, D. G.; Burton, D. J. Synth, Commun. 1973, 3, 197. Burton, D. J. J. Fluorine Chem. 1983, 18, 339. Burton, D. J.; Kesling, H. S.; Naae, D. G. J. Fluorine Chem. 1981, 18, 293. Wheaton, G. A.; Burton, D. J. J. Org. Chem. 1983, 48, 917. Matsuda, A.; Itoh, H.; Takenishi, K.; Susuki, T.; Ueda, T. Chem. Pharm. Bull. 1988, 36, 945. Fried, J.; Kittisopikul, S.; Hallinan, E. A. Tetrahedron Lett. 1984, 25, 4329. For recent and potentially useful alternatives: Dolbier, W. R., Jr.; Ocampo, R. J. Org. Chem. 1995, 60, 5378. Kim, K.-I.; McCarthy, J. R. Tetrahedron Lett. 1996, 37, 3223.
- (1973) Synth, Commun. , vol.3 , pp. 197
- Naae, D.G.¹ Burton, D.J.²

75
- 0000564055
- Fuqua, S. A.; Duncan, W. G.; Silverstein, R. M. J. Org. Chem. 1965, 30, 1027. Naae, D. G.; Kesling, H. S.; Burton, D. J. Tetrahedron Lett. 1975, 3789. Naae, D. G.; Burton, D. J. J. Fluorine Chem. 1971, 1, 123. Naae, D. G.; Burton, D. J. Synth, Commun. 1973, 3, 197. Burton, D. J. J. Fluorine Chem. 1983, 18, 339. Burton, D. J.; Kesling, H. S.; Naae, D. G. J. Fluorine Chem. 1981, 18, 293. Wheaton, G. A.; Burton, D. J. J. Org. Chem. 1983, 48, 917. Matsuda, A.; Itoh, H.; Takenishi, K.; Susuki, T.; Ueda, T. Chem. Pharm. Bull. 1988, 36, 945. Fried, J.; Kittisopikul, S.; Hallinan, E. A. Tetrahedron Lett. 1984, 25, 4329. For recent and potentially useful alternatives: Dolbier, W. R., Jr.; Ocampo, R. J. Org. Chem. 1995, 60, 5378. Kim, K.-I.; McCarthy, J. R. Tetrahedron Lett. 1996, 37, 3223.
- (1983) J. Fluorine Chem. , vol.18 , pp. 339
- Burton, D.J.¹

76
- 0000071861
- Fuqua, S. A.; Duncan, W. G.; Silverstein, R. M. J. Org. Chem. 1965, 30, 1027. Naae, D. G.; Kesling, H. S.; Burton, D. J. Tetrahedron Lett. 1975, 3789. Naae, D. G.; Burton, D. J. J. Fluorine Chem. 1971, 1, 123. Naae, D. G.; Burton, D. J. Synth, Commun. 1973, 3, 197. Burton, D. J. J. Fluorine Chem. 1983, 18, 339. Burton, D. J.; Kesling, H. S.; Naae, D. G. J. Fluorine Chem. 1981, 18, 293. Wheaton, G. A.; Burton, D. J. J. Org. Chem. 1983, 48, 917. Matsuda, A.; Itoh, H.; Takenishi, K.; Susuki, T.; Ueda, T. Chem. Pharm. Bull. 1988, 36, 945. Fried, J.; Kittisopikul, S.; Hallinan, E. A. Tetrahedron Lett. 1984, 25, 4329. For recent and potentially useful alternatives: Dolbier, W. R., Jr.; Ocampo, R. J. Org. Chem. 1995, 60, 5378. Kim, K.-I.; McCarthy, J. R. Tetrahedron Lett. 1996, 37, 3223.
- (1981) J. Fluorine Chem. , vol.18 , pp. 293
- Burton, D.J.¹ Kesling, H.S.² Naae, D.G.³

77
- 0001272864
- Fuqua, S. A.; Duncan, W. G.; Silverstein, R. M. J. Org. Chem. 1965, 30, 1027. Naae, D. G.; Kesling, H. S.; Burton, D. J. Tetrahedron Lett. 1975, 3789. Naae, D. G.; Burton, D. J. J. Fluorine Chem. 1971, 1, 123. Naae, D. G.; Burton, D. J. Synth, Commun. 1973, 3, 197. Burton, D. J. J. Fluorine Chem. 1983, 18, 339. Burton, D. J.; Kesling, H. S.; Naae, D. G. J. Fluorine Chem. 1981, 18, 293. Wheaton, G. A.; Burton, D. J. J. Org. Chem. 1983, 48, 917. Matsuda, A.; Itoh, H.; Takenishi, K.; Susuki, T.; Ueda, T. Chem. Pharm. Bull. 1988, 36, 945. Fried, J.; Kittisopikul, S.; Hallinan, E. A. Tetrahedron Lett. 1984, 25, 4329. For recent and potentially useful alternatives: Dolbier, W. R., Jr.; Ocampo, R. J. Org. Chem. 1995, 60, 5378. Kim, K.-I.; McCarthy, J. R. Tetrahedron Lett. 1996, 37, 3223.
- (1983) J. Org. Chem. , vol.48 , pp. 917
- Wheaton, G.A.¹ Burton, D.J.²

78
- 0023952556
- Fuqua, S. A.; Duncan, W. G.; Silverstein, R. M. J. Org. Chem. 1965, 30, 1027. Naae, D. G.; Kesling, H. S.; Burton, D. J. Tetrahedron Lett. 1975, 3789. Naae, D. G.; Burton, D. J. J. Fluorine Chem. 1971, 1, 123. Naae, D. G.; Burton, D. J. Synth, Commun. 1973, 3, 197. Burton, D. J. J. Fluorine Chem. 1983, 18, 339. Burton, D. J.; Kesling, H. S.; Naae, D. G. J. Fluorine Chem. 1981, 18, 293. Wheaton, G. A.; Burton, D. J. J. Org. Chem. 1983, 48, 917. Matsuda, A.; Itoh, H.; Takenishi, K.; Susuki, T.; Ueda, T. Chem. Pharm. Bull. 1988, 36, 945. Fried, J.; Kittisopikul, S.; Hallinan, E. A. Tetrahedron Lett. 1984, 25, 4329. For recent and potentially useful alternatives: Dolbier, W. R., Jr.; Ocampo, R. J. Org. Chem. 1995, 60, 5378. Kim, K.-I.; McCarthy, J. R. Tetrahedron Lett. 1996, 37, 3223.
- (1988) Chem. Pharm. Bull. , vol.36 , pp. 945
- Matsuda, A.¹ Itoh, H.² Takenishi, K.³ Susuki, T.⁴ Ueda, T.⁵

79
- 0021173134
- Fuqua, S. A.; Duncan, W. G.; Silverstein, R. M. J. Org. Chem. 1965, 30, 1027. Naae, D. G.; Kesling, H. S.; Burton, D. J. Tetrahedron Lett. 1975, 3789. Naae, D. G.; Burton, D. J. J. Fluorine Chem. 1971, 1, 123. Naae, D. G.; Burton, D. J. Synth, Commun. 1973, 3, 197. Burton, D. J. J. Fluorine Chem. 1983, 18, 339. Burton, D. J.; Kesling, H. S.; Naae, D. G. J. Fluorine Chem. 1981, 18, 293. Wheaton, G. A.; Burton, D. J. J. Org. Chem. 1983, 48, 917. Matsuda, A.; Itoh, H.; Takenishi, K.; Susuki, T.; Ueda, T. Chem. Pharm. Bull. 1988, 36, 945. Fried, J.; Kittisopikul, S.; Hallinan, E. A. Tetrahedron Lett. 1984, 25, 4329. For recent and potentially useful alternatives: Dolbier, W. R., Jr.; Ocampo, R. J. Org. Chem. 1995, 60, 5378. Kim, K.-I.; McCarthy, J. R. Tetrahedron Lett. 1996, 37, 3223.
- (1984) Tetrahedron Lett. , vol.25 , pp. 4329
- Fried, J.¹ Kittisopikul, S.² Hallinan, E.A.³

80
- 0000776033
- Fuqua, S. A.; Duncan, W. G.; Silverstein, R. M. J. Org. Chem. 1965, 30, 1027. Naae, D. G.; Kesling, H. S.; Burton, D. J. Tetrahedron Lett. 1975, 3789. Naae, D. G.; Burton, D. J. J. Fluorine Chem. 1971, 1, 123. Naae, D. G.; Burton, D. J. Synth, Commun. 1973, 3, 197. Burton, D. J. J. Fluorine Chem. 1983, 18, 339. Burton, D. J.; Kesling, H. S.; Naae, D. G. J. Fluorine Chem. 1981, 18, 293. Wheaton, G. A.; Burton, D. J. J. Org. Chem. 1983, 48, 917. Matsuda, A.; Itoh, H.; Takenishi, K.; Susuki, T.; Ueda, T. Chem. Pharm. Bull. 1988, 36, 945. Fried, J.; Kittisopikul, S.; Hallinan, E. A. Tetrahedron Lett. 1984, 25, 4329. For recent and potentially useful alternatives: Dolbier, W. R., Jr.; Ocampo, R. J. Org. Chem. 1995, 60, 5378. Kim, K.-I.; McCarthy, J. R. Tetrahedron Lett. 1996, 37, 3223.
- (1995) J. Org. Chem. , vol.60 , pp. 5378
- Dolbier Jr., W.R.¹ Ocampo, R.²

81
- 0029947242
- Fuqua, S. A.; Duncan, W. G.; Silverstein, R. M. J. Org. Chem. 1965, 30, 1027. Naae, D. G.; Kesling, H. S.; Burton, D. J. Tetrahedron Lett. 1975, 3789. Naae, D. G.; Burton, D. J. J. Fluorine Chem. 1971, 1, 123. Naae, D. G.; Burton, D. J. Synth, Commun. 1973, 3, 197. Burton, D. J. J. Fluorine Chem. 1983, 18, 339. Burton, D. J.; Kesling, H. S.; Naae, D. G. J. Fluorine Chem. 1981, 18, 293. Wheaton, G. A.; Burton, D. J. J. Org. Chem. 1983, 48, 917. Matsuda, A.; Itoh, H.; Takenishi, K.; Susuki, T.; Ueda, T. Chem. Pharm. Bull. 1988, 36, 945. Fried, J.; Kittisopikul, S.; Hallinan, E. A. Tetrahedron Lett. 1984, 25, 4329. For recent and potentially useful alternatives: Dolbier, W. R., Jr.; Ocampo, R. J. Org. Chem. 1995, 60, 5378. Kim, K.-I.; McCarthy, J. R. Tetrahedron Lett. 1996, 37, 3223.
- (1996) Tetrahedron Lett. , vol.37 , pp. 3223
- Kim, K.-I.¹ McCarthy, J.R.²

82
- 0012932159
- Kendrick, D. A.; Kolb, M. J. Fluorine Chem. 1989, 45, 265. Begue, J.-P.; Bonnet-Delpon, D.; Rock, M. H. Tetrahedron Lett. 1995, 36, 5003.
- (1989) J. Fluorine Chem. , vol.45 , pp. 265
- Kendrick, D.A.¹ Kolb, M.²

83
- 0028998675
- Kendrick, D. A.; Kolb, M. J. Fluorine Chem. 1989, 45, 265. Begue, J.-P.; Bonnet-Delpon, D.; Rock, M. H. Tetrahedron Lett. 1995, 36, 5003.
- (1995) Tetrahedron Lett. , vol.36 , pp. 5003
- Begue, J.-P.¹ Bonnet-Delpon, D.² Rock, M.H.³

84
- 0010420577
- Fuji, K.; Ichikawa, K.; Node, M.; Fujita, E. J. Org. Chem. 1979, 44, 1661.
- (1979) J. Org. Chem. , vol.44 , pp. 1661
- Fuji, K.¹ Ichikawa, K.² Node, M.³ Fujita, E.⁴

85
- 84986468501
- Smith, W. B. J. Heterocycl. Chem. 1987, 24, 745. Petrini, M.; Ballini, Rosini, G. Synthesis 1987, 713.
- (1987) J. Heterocycl. Chem. , vol.24 , pp. 745
- Smith, W.B.¹

86
- 84986468501
- Smith, W. B. J. Heterocycl. Chem. 1987, 24, 745. Petrini, M.; Ballini, Rosini, G. Synthesis 1987, 713.
- (1987) Synthesis , pp. 713
- Petrini, M.¹ Ballini Rosini, G.²

87
- 0347868119
- Kraus, G. A.; Nagy, J. O.; Delano, J. Tetrahedron 1985, 41, 2337.
- (1985) Tetrahedron , vol.41 , pp. 2337
- Kraus, G.A.¹ Nagy, J.O.² Delano, J.³

88
- 0028296957
- Muratake, H.; Abe, I.; Natsume, M. Tetrahedron Lett. 1994, 35, 2573.
- (1994) Tetrahedron Lett. , vol.35 , pp. 2573
- Muratake, H.¹ Abe, I.² Natsume, M.³

89
- 0025119357
- Boger, D. L.; Ishizaki, T.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 5823. Boger, D. L.; Ishizaki, T.; Wysocki, R. J., Jr.; Munk, S. A.; Kitos, P. A.; Sumornwat, O. J. Am. Chem. Soc. 1989, 111, 6461. Boger, D. L.; Ishizaki, T. Tetrahedron Lett. 1990, 31, 793. Boger, D. L.; Ishizaki, T.; Sakya, S. M.; Munk, S. A.; Kitos, P. A.; Jin, Q.; Besterman, J. M. Bioorg. Med. Chem. Lett. 1991, 1, 115. Boger, D. L.; Munk, S. A.; Ishizaki, T. J. Am. Chem. Soc. 1991, 113, 2779. Boger, D. L.; Munk, S. A. J. Am. Chem. Soc. 1992, 114, 5487. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1994, 116, 7996. Boger, D. L.; Yun, W.; Han, N. Bioorg. Med. Chem. 1995, 3, 1429.
- (1990) J. Org. Chem. , vol.55 , pp. 5823
- Boger, D.L.¹ Ishizaki, T.² Kitos, P.A.³ Suntornwat, O.⁴

90
- 0024393748
- Boger, D. L.; Ishizaki, T.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 5823. Boger, D. L.; Ishizaki, T.; Wysocki, R. J., Jr.; Munk, S. A.; Kitos, P. A.; Sumornwat, O. J. Am. Chem. Soc. 1989, 111, 6461. Boger, D. L.; Ishizaki, T. Tetrahedron Lett. 1990, 31, 793. Boger, D. L.; Ishizaki, T.; Sakya, S. M.; Munk, S. A.; Kitos, P. A.; Jin, Q.; Besterman, J. M. Bioorg. Med. Chem. Lett. 1991, 1, 115. Boger, D. L.; Munk, S. A.; Ishizaki, T. J. Am. Chem. Soc. 1991, 113, 2779. Boger, D. L.; Munk, S. A. J. Am. Chem. Soc. 1992, 114, 5487. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1994, 116, 7996. Boger, D. L.; Yun, W.; Han, N. Bioorg. Med. Chem. 1995, 3, 1429.
- (1989) J. Am. Chem. Soc. , vol.111 , pp. 6461
- Boger, D.L.¹ Ishizaki, T.² Wysocki Jr., R.J.³ Munk, S.A.⁴ Kitos, P.A.⁵ Sumornwat, O.⁶

91
- 0025099719
- Boger, D. L.; Ishizaki, T.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 5823. Boger, D. L.; Ishizaki, T.; Wysocki, R. J., Jr.; Munk, S. A.; Kitos, P. A.; Sumornwat, O. J. Am. Chem. Soc. 1989, 111, 6461. Boger, D. L.; Ishizaki, T. Tetrahedron Lett. 1990, 31, 793. Boger, D. L.; Ishizaki, T.; Sakya, S. M.; Munk, S. A.; Kitos, P. A.; Jin, Q.; Besterman, J. M. Bioorg. Med. Chem. Lett. 1991, 1, 115. Boger, D. L.; Munk, S. A.; Ishizaki, T. J. Am. Chem. Soc. 1991, 113, 2779. Boger, D. L.; Munk, S. A. J. Am. Chem. Soc. 1992, 114, 5487. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1994, 116, 7996. Boger, D. L.; Yun, W.; Han, N. Bioorg. Med. Chem. 1995, 3, 1429.
- (1990) Tetrahedron Lett. , vol.31 , pp. 793
- Boger, D.L.¹ Ishizaki, T.²

92
- 0025891696
- Boger, D. L.; Ishizaki, T.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 5823. Boger, D. L.; Ishizaki, T.; Wysocki, R. J., Jr.; Munk, S. A.; Kitos, P. A.; Sumornwat, O. J. Am. Chem. Soc. 1989, 111, 6461. Boger, D. L.; Ishizaki, T. Tetrahedron Lett. 1990, 31, 793. Boger, D. L.; Ishizaki, T.; Sakya, S. M.; Munk, S. A.; Kitos, P. A.; Jin, Q.; Besterman, J. M. Bioorg. Med. Chem. Lett. 1991, 1, 115. Boger, D. L.; Munk, S. A.; Ishizaki, T. J. Am. Chem. Soc. 1991, 113, 2779. Boger, D. L.; Munk, S. A. J. Am. Chem. Soc. 1992, 114, 5487. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1994, 116, 7996. Boger, D. L.; Yun, W.; Han, N. Bioorg. Med. Chem. 1995, 3, 1429.
- (1991) Bioorg. Med. Chem. Lett. , vol.1 , pp. 115
- Boger, D.L.¹ Ishizaki, T.² Sakya, S.M.³ Munk, S.A.⁴ Kitos, P.A.⁵ Jin, Q.⁶ Besterman, J.M.⁷

93
- 0025811775
- Boger, D. L.; Ishizaki, T.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 5823. Boger, D. L.; Ishizaki, T.; Wysocki, R. J., Jr.; Munk, S. A.; Kitos, P. A.; Sumornwat, O. J. Am. Chem. Soc. 1989, 111, 6461. Boger, D. L.; Ishizaki, T. Tetrahedron Lett. 1990, 31, 793. Boger, D. L.; Ishizaki, T.; Sakya, S. M.; Munk, S. A.; Kitos, P. A.; Jin, Q.; Besterman, J. M. Bioorg. Med. Chem. Lett. 1991, 1, 115. Boger, D. L.; Munk, S. A.; Ishizaki, T. J. Am. Chem. Soc. 1991, 113, 2779. Boger, D. L.; Munk, S. A. J. Am. Chem. Soc. 1992, 114, 5487. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1994, 116, 7996. Boger, D. L.; Yun, W.; Han, N. Bioorg. Med. Chem. 1995, 3, 1429.
- (1991) J. Am. Chem. Soc. , vol.113 , pp. 2779
- Boger, D.L.¹ Munk, S.A.² Ishizaki, T.³

94
- 84994476837
- Boger, D. L.; Ishizaki, T.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 5823. Boger, D. L.; Ishizaki, T.; Wysocki, R. J., Jr.; Munk, S. A.; Kitos, P. A.; Sumornwat, O. J. Am. Chem. Soc. 1989, 111, 6461. Boger, D. L.; Ishizaki, T. Tetrahedron Lett. 1990, 31, 793. Boger, D. L.; Ishizaki, T.; Sakya, S. M.; Munk, S. A.; Kitos, P. A.; Jin, Q.; Besterman, J. M. Bioorg. Med. Chem. Lett. 1991, 1, 115. Boger, D. L.; Munk, S. A.; Ishizaki, T. J. Am. Chem. Soc. 1991, 113, 2779. Boger, D. L.; Munk, S. A. J. Am. Chem. Soc. 1992, 114, 5487. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1994, 116, 7996. Boger, D. L.; Yun, W.; Han, N. Bioorg. Med. Chem. 1995, 3, 1429.
- (1992) J. Am. Chem. Soc. , vol.114 , pp. 5487
- Boger, D.L.¹ Munk, S.A.²

95
- 0028036453
- Boger, D. L.; Ishizaki, T.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 5823. Boger, D. L.; Ishizaki, T.; Wysocki, R. J., Jr.; Munk, S. A.; Kitos, P. A.; Sumornwat, O. J. Am. Chem. Soc. 1989, 111, 6461. Boger, D. L.; Ishizaki, T. Tetrahedron Lett. 1990, 31, 793. Boger, D. L.; Ishizaki, T.; Sakya, S. M.; Munk, S. A.; Kitos, P. A.; Jin, Q.; Besterman, J. M. Bioorg. Med. Chem. Lett. 1991, 1, 115. Boger, D. L.; Munk, S. A.; Ishizaki, T. J. Am. Chem. Soc. 1991, 113, 2779. Boger, D. L.; Munk, S. A. J. Am. Chem. Soc. 1992, 114, 5487. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1994, 116, 7996. Boger, D. L.; Yun, W.; Han, N. Bioorg. Med. Chem. 1995, 3, 1429.
- (1994) J. Am. Chem. Soc. , vol.116 , pp. 7996
- Boger, D.L.¹ Yun, W.²

96
- 0028790373
- Boger, D. L.; Ishizaki, T.; Kitos, P. A.; Suntornwat, O. J. Org. Chem. 1990, 55, 5823. Boger, D. L.; Ishizaki, T.; Wysocki, R. J., Jr.; Munk, S. A.; Kitos, P. A.; Sumornwat, O. J. Am. Chem. Soc. 1989, 111, 6461. Boger, D. L.; Ishizaki, T. Tetrahedron Lett. 1990, 31, 793. Boger, D. L.; Ishizaki, T.; Sakya, S. M.; Munk, S. A.; Kitos, P. A.; Jin, Q.; Besterman, J. M. Bioorg. Med. Chem. Lett. 1991, 1, 115. Boger, D. L.; Munk, S. A.; Ishizaki, T. J. Am. Chem. Soc. 1991, 113, 2779. Boger, D. L.; Munk, S. A. J. Am. Chem. Soc. 1992, 114, 5487. Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1994, 116, 7996. Boger, D. L.; Yun, W.; Han, N. Bioorg. Med. Chem. 1995, 3, 1429.
- (1995) Bioorg. Med. Chem. , vol.3 , pp. 1429
- Boger, D.L.¹ Yun, W.² Han, N.³

97
- 0029980340
- Boger, D. L.; McKie, J. A.; Cai, H.; Cacciari, B.; Baraldi, P. G. J. Org. Chem. 1996, 61, 1710.
- (1996) J. Org. Chem. , vol.61 , pp. 1710
- Boger, D.L.¹ McKie, J.A.² Cai, H.³ Cacciari, B.⁴ Baraldi, P.G.⁵

98
- 0030036747
- Boger, D. L.; Han, N.; Tarby, C. M.; Boyce, C. W.; Cai, H.; Jing, Q.; Kitos, P. A. J. Org. Chem. 1996, 61, 4894. Boger, D. L.; McKie, J. A.; Han, N.; Tarby, C. M.; Riggs, H. W.; Kitos, P. A. Bioorg. Med. Chem. Lett. 1996, 6, 659.
- (1996) J. Org. Chem. , vol.61 , pp. 4894
- Boger, D.L.¹ Han, N.² Tarby, C.M.³ Boyce, C.W.⁴ Cai, H.⁵ Jing, Q.⁶ Kitos, P.A.⁷

99
- 0029872086
- Boger, D. L.; Han, N.; Tarby, C. M.; Boyce, C. W.; Cai, H.; Jing, Q.; Kitos, P. A. J. Org. Chem. 1996, 61, 4894. Boger, D. L.; McKie, J. A.; Han, N.; Tarby, C. M.; Riggs, H. W.; Kitos, P. A. Bioorg. Med. Chem. Lett. 1996, 6, 659.
- (1996) Bioorg. Med. Chem. Lett. , vol.6 , pp. 659
- Boger, D.L.¹ McKie, J.A.² Han, N.³ Tarby, C.M.⁴ Riggs, H.W.⁵ Kitos, P.A.⁶

100
- 0028100406
- Boger, D. L.; Yun, W. J. Am. Chem. Soc. 1994, 116, 5523.
- (1994) J. Am. Chem. Soc. , vol.116 , pp. 5523
- Boger, D.L.¹ Yun, W.²

101
- 0028592579
- Boger, D. L.; Mésini, P.J. Am. Chem. Soc. 1994, 116, 11335. Boger, D. L.; Mésini, P. J. Am. Chem. Soc. 1995, 117, 11647. Boger, D. L.; Mésini, P.; Tarby, C. M. J. Am. Chem. Soc. 1994, 116, 6461.
- (1994) J. Am. Chem. Soc. , vol.116 , pp. 11335
- Boger, D.L.¹ Mésini, P.²

102
- 0028806129
- Boger, D. L.; Mésini, P.J. Am. Chem. Soc. 1994, 116, 11335. Boger, D. L.; Mésini, P. J. Am. Chem. Soc. 1995, 117, 11647. Boger, D. L.; Mésini, P.; Tarby, C. M. J. Am. Chem. Soc. 1994, 116, 6461.
- (1995) J. Am. Chem. Soc. , vol.117 , pp. 11647
- Boger, D.L.¹ Mésini, P.²

103
- 0028024034
- Boger, D. L.; Mésini, P.J. Am. Chem. Soc. 1994, 116, 11335. Boger, D. L.; Mésini, P. J. Am. Chem. Soc. 1995, 117, 11647. Boger, D. L.; Mésini, P.; Tarby, C. M. J. Am. Chem. Soc. 1994, 116, 6461.
- (1994) J. Am. Chem. Soc. , vol.116 , pp. 6461
- Boger, D.L.¹ Mésini, P.² Tarby, C.M.³

104
- 0024559965
- Boger, D. L.; Wysocki, R. J., Jr. J. Org. Chem. 1989, 54, 1238. Boger, D. L.; Wysocki, R. J., Jr.; Ishizaki, T. J. Am. Chem. Soc. 1990, 112, 5230. Boger, D. L.; Munk, S. A.; Zarrinmayeh, H. J. Am. Chem. Soc. 1991, 113, 3980. Boger, D. L.; Zarrinmayeh, H.; Munk, S. A.; Kitos. P. A.; Suntornwat, O. Proc. Natl. Acad. Sci. U.S.A. 1991, 88, 1431.
- (1989) J. Org. Chem. , vol.54 , pp. 1238
- Boger, D.L.¹ Wysocki Jr., R.J.²

105
- 0025045711
- Boger, D. L.; Wysocki, R. J., Jr. J. Org. Chem. 1989, 54, 1238. Boger, D. L.; Wysocki, R. J., Jr.; Ishizaki, T. J. Am. Chem. Soc. 1990, 112, 5230. Boger, D. L.; Munk, S. A.; Zarrinmayeh, H. J. Am. Chem. Soc. 1991, 113, 3980. Boger, D. L.; Zarrinmayeh, H.; Munk, S. A.; Kitos. P. A.; Suntornwat, O. Proc. Natl. Acad. Sci. U.S.A. 1991, 88, 1431.
- (1990) J. Am. Chem. Soc. , vol.112 , pp. 5230
- Boger, D.L.¹ Wysocki Jr., R.J.² Ishizaki, T.³

106
- 0025900895
- Boger, D. L.; Wysocki, R. J., Jr. J. Org. Chem. 1989, 54, 1238. Boger, D. L.; Wysocki, R. J., Jr.; Ishizaki, T. J. Am. Chem. Soc. 1990, 112, 5230. Boger, D. L.; Munk, S. A.; Zarrinmayeh, H. J. Am. Chem. Soc. 1991, 113, 3980. Boger, D. L.; Zarrinmayeh, H.; Munk, S. A.; Kitos. P. A.; Suntornwat, O. Proc. Natl. Acad. Sci. U.S.A. 1991, 88, 1431.
- (1991) J. Am. Chem. Soc. , vol.113 , pp. 3980
- Boger, D.L.¹ Munk, S.A.² Zarrinmayeh, H.³

107
- 0026092765
- Boger, D. L.; Wysocki, R. J., Jr. J. Org. Chem. 1989, 54, 1238. Boger, D. L.; Wysocki, R. J., Jr.; Ishizaki, T. J. Am. Chem. Soc. 1990, 112, 5230. Boger, D. L.; Munk, S. A.; Zarrinmayeh, H. J. Am. Chem. Soc. 1991, 113, 3980. Boger, D. L.; Zarrinmayeh, H.; Munk, S. A.; Kitos. P. A.; Suntornwat, O. Proc. Natl. Acad. Sci. U.S.A. 1991, 88, 1431.
- (1991) Proc. Natl. Acad. Sci. U.S.A. , vol.88 , pp. 1431
- Boger, D.L.¹ Zarrinmayeh, H.² Munk, S.A.³ Kitos, P.A.⁴ Suntornwat, O.⁵

108
- 0028085388
- Warpehoski, M. A.; Harper, D. E. J. Am. Chem. Soc. 1994, 116, 7573. Warpehoski, M. A.; Harper, D. E. J. Am. Chem. Soc. 1995, 117, 2951.
- (1994) J. Am. Chem. Soc. , vol.116 , pp. 7573
- Warpehoski, M.A.¹ Harper, D.E.²

109
- 0028958933
- Warpehoski, M. A.; Harper, D. E. J. Am. Chem. Soc. 1994, 116, 7573. Warpehoski, M. A.; Harper, D. E. J. Am. Chem. Soc. 1995, 117, 2951.
- (1995) J. Am. Chem. Soc. , vol.117 , pp. 2951
- Warpehoski, M.A.¹ Harper, D.E.²

110
- 10144244115
- in press
- Boger, D. L.; Goldberg, J. A.; McKie, J. A. Bioorg. Med. Chem. Lett., in press. Boger, D. L.; McKie, J. A.; Nishi, T.; Ogiku, T. J. Am. Chem. Soc. Submitted.
- Bioorg. Med. Chem. Lett.
- Boger, D.L.¹ Goldberg, J.A.² McKie, J.A.³

111
- 10144220794
- Submitted
- Boger, D. L.; Goldberg, J. A.; McKie, J. A. Bioorg. Med. Chem. Lett., in press. Boger, D. L.; McKie, J. A.; Nishi, T.; Ogiku, T. J. Am. Chem. Soc. Submitted.
- J. Am. Chem. Soc.
- Boger, D.L.¹ McKie, J.A.² Nishi, T.³ Ogiku, T.⁴

112
- 10144260779
- note
- 44 and suggests that the ambiguous experimental basis for this proposal be reexamined.

113
- 10144231576
- note
- The author has deposited the atomic coordinates for this structure with the Cambridge Crystallographic Data Centre, and the coordinates may be obtained upon request from the Director, Cambridge Crystallographic Data Centre, 12 Union Road, Cambridge, CB2 1EZ, UK.

114
- 0000063791
- Martin, D. G.; Kelly, R. C.; Watt, W.; Wienienski, N.; Mizsak, S. A.; Nielsen, J. W.; Prairie, M. D. J. Org. Chem. 1988, 53, 4610.
- (1988) J. Org. Chem. , vol.53 , pp. 4610
- Martin, D.G.¹ Kelly, R.C.² Watt, W.³ Wienienski, N.⁴ Mizsak, S.A.⁵ Nielsen, J.W.⁶ Prairie, M.D.⁷

115
- 2942583333
- Bond lengths of 1.464-1.447 and 1.553-1.552 Å for the adjacent and opposite bonds have been established for symmetrical difluorocyclopropanes by microwave spectroscopy or X-ray versus cyclopropane itself (1.514 Å). X-ray: Dolbier, W. R., Jr.; Odaniec, M.: Gomulka, E.; Jaskolski, M.; Koroniak, H. Tetrahedron 1984, 40, 3945. Dolbier, W. R., Jr.; Odaniec, M.; Jaskolski, M.; Koroniak, H. J. Mol. Struct. 1986, 147, 155. Microwave spectroscopy: Parretta, A. T.; Laurie, V. W. J. Chem. Phys. 1975, 62, 2463. Computational studies: Deakyne, C. A.; Allen, L. C.; Craig, N. C. J. Am. Chem. Soc. 1977, 99, 3845. Durmaz, S.; Kollmar. H. J. Am. Chem. Soc. 1980, 102, 6942. Clark, T.; Spitznagel, G. W.; Klose, R.; Schleyer, P. von R. J. Am. Chem. Soc. 1984, 106, 4412. Boggs, J. E.; Fan, K. Acta Chem. Scand. 1988, A42, 595.
- (1984) Tetrahedron , vol.40 , pp. 3945
- Dolbier Jr., W.R.¹ Odaniec, M.² Gomulka, E.³ Jaskolski, M.⁴ Koroniak, H.⁵

116
- 10144229485
- Bond lengths of 1.464-1.447 and 1.553-1.552 Å for the adjacent and opposite bonds have been established for symmetrical difluorocyclopropanes by microwave spectroscopy or X-ray versus cyclopropane itself (1.514 Å). X-ray: Dolbier, W. R., Jr.; Odaniec, M.: Gomulka, E.; Jaskolski, M.; Koroniak, H. Tetrahedron 1984, 40, 3945. Dolbier, W. R., Jr.; Odaniec, M.; Jaskolski, M.; Koroniak, H. J. Mol. Struct. 1986, 147, 155. Microwave spectroscopy: Parretta, A. T.; Laurie, V. W. J. Chem. Phys. 1975, 62, 2463. Computational studies: Deakyne, C. A.; Allen, L. C.; Craig, N. C. J. Am. Chem. Soc. 1977, 99, 3845. Durmaz, S.; Kollmar. H. J. Am. Chem. Soc. 1980, 102, 6942. Clark, T.; Spitznagel, G. W.; Klose, R.; Schleyer, P. von R. J. Am. Chem. Soc. 1984, 106, 4412. Boggs, J. E.; Fan, K. Acta Chem. Scand. 1988, A42, 595.
- (1986) J. Mol. Struct. , vol.147 , pp. 155
- Dolbier Jr., W.R.¹ Odaniec, M.² Jaskolski, M.³ Koroniak, H.⁴

117
- 10144255344
- Bond lengths of 1.464-1.447 and 1.553-1.552 Å for the adjacent and opposite bonds have been established for symmetrical difluorocyclopropanes by microwave spectroscopy or X-ray versus cyclopropane itself (1.514 Å). X-ray: Dolbier, W. R., Jr.; Odaniec, M.: Gomulka, E.; Jaskolski, M.; Koroniak, H. Tetrahedron 1984, 40, 3945. Dolbier, W. R., Jr.; Odaniec, M.; Jaskolski, M.; Koroniak, H. J. Mol. Struct. 1986, 147, 155. Microwave spectroscopy: Parretta, A. T.; Laurie, V. W. J. Chem. Phys. 1975, 62, 2463. Computational studies: Deakyne, C. A.; Allen, L. C.; Craig, N. C. J. Am. Chem. Soc. 1977, 99, 3845. Durmaz, S.; Kollmar. H. J. Am. Chem. Soc. 1980, 102, 6942. Clark, T.; Spitznagel, G. W.; Klose, R.; Schleyer, P. von R. J. Am. Chem. Soc. 1984, 106, 4412. Boggs, J. E.; Fan, K. Acta Chem. Scand. 1988, A42, 595.
- (1975) J. Chem. Phys. , vol.62 , pp. 2463
- Parretta, A.T.¹ Laurie, V.W.²

118
- 10144260156
- Bond lengths of 1.464-1.447 and 1.553-1.552 Å for the adjacent and opposite bonds have been established for symmetrical difluorocyclopropanes by microwave spectroscopy or X-ray versus cyclopropane itself (1.514 Å). X-ray: Dolbier, W. R., Jr.; Odaniec, M.: Gomulka, E.; Jaskolski, M.; Koroniak, H. Tetrahedron 1984, 40, 3945. Dolbier, W. R., Jr.; Odaniec, M.; Jaskolski, M.; Koroniak, H. J. Mol. Struct. 1986, 147, 155. Microwave spectroscopy: Parretta, A. T.; Laurie, V. W. J. Chem. Phys. 1975, 62, 2463. Computational studies: Deakyne, C. A.; Allen, L. C.; Craig, N. C. J. Am. Chem. Soc. 1977, 99, 3845. Durmaz, S.; Kollmar. H. J. Am. Chem. Soc. 1980, 102, 6942. Clark, T.; Spitznagel, G. W.; Klose, R.; Schleyer, P. von R. J. Am. Chem. Soc. 1984, 106, 4412. Boggs, J. E.; Fan, K. Acta Chem. Scand. 1988, A42, 595.
- (1977) J. Am. Chem. Soc. , vol.99 , pp. 3845
- Deakyne, C.A.¹ Allen, L.C.² Craig, N.C.³

119
- 33847085990
- Bond lengths of 1.464-1.447 and 1.553-1.552 Å for the adjacent and opposite bonds have been established for symmetrical difluorocyclopropanes by microwave spectroscopy or X-ray versus cyclopropane itself (1.514 Å). X-ray: Dolbier, W. R., Jr.; Odaniec, M.: Gomulka, E.; Jaskolski, M.; Koroniak, H. Tetrahedron 1984, 40, 3945. Dolbier, W. R., Jr.; Odaniec, M.; Jaskolski, M.; Koroniak, H. J. Mol. Struct. 1986, 147, 155. Microwave spectroscopy: Parretta, A. T.; Laurie, V. W. J. Chem. Phys. 1975, 62, 2463. Computational studies: Deakyne, C. A.; Allen, L. C.; Craig, N. C. J. Am. Chem. Soc. 1977, 99, 3845. Durmaz, S.; Kollmar. H. J. Am. Chem. Soc. 1980, 102, 6942. Clark, T.; Spitznagel, G. W.; Klose, R.; Schleyer, P. von R. J. Am. Chem. Soc. 1984, 106, 4412. Boggs, J. E.; Fan, K. Acta Chem. Scand. 1988, A42, 595.
- (1980) J. Am. Chem. Soc. , vol.102 , pp. 6942
- Durmaz, S.¹ Kollmar, H.²

120
- 1842601941
- Bond lengths of 1.464-1.447 and 1.553-1.552 Å for the adjacent and opposite bonds have been established for symmetrical difluorocyclopropanes by microwave spectroscopy or X-ray versus cyclopropane itself (1.514 Å). X-ray: Dolbier, W. R., Jr.; Odaniec, M.: Gomulka, E.; Jaskolski, M.; Koroniak, H. Tetrahedron 1984, 40, 3945. Dolbier, W. R., Jr.; Odaniec, M.; Jaskolski, M.; Koroniak, H. J. Mol. Struct. 1986, 147, 155. Microwave spectroscopy: Parretta, A. T.; Laurie, V. W. J. Chem. Phys. 1975, 62, 2463. Computational studies: Deakyne, C. A.; Allen, L. C.; Craig, N. C. J. Am. Chem. Soc. 1977, 99, 3845. Durmaz, S.; Kollmar. H. J. Am. Chem. Soc. 1980, 102, 6942. Clark, T.; Spitznagel, G. W.; Klose, R.; Schleyer, P. von R. J. Am. Chem. Soc. 1984, 106, 4412. Boggs, J. E.; Fan, K. Acta Chem. Scand. 1988, A42, 595.
- (1984) J. Am. Chem. Soc. , vol.106 , pp. 4412
- Clark, T.¹ Spitznagel, G.W.² Klose, R.³ Von Schleyer, P.R.⁴

121
- 0037883523
- Bond lengths of 1.464-1.447 and 1.553-1.552 Å for the adjacent and opposite bonds have been established for symmetrical difluorocyclopropanes by microwave spectroscopy or X-ray versus cyclopropane itself (1.514 Å). X-ray: Dolbier, W. R., Jr.; Odaniec, M.: Gomulka, E.; Jaskolski, M.; Koroniak, H. Tetrahedron 1984, 40, 3945. Dolbier, W. R., Jr.; Odaniec, M.; Jaskolski, M.; Koroniak, H. J. Mol. Struct. 1986, 147, 155. Microwave spectroscopy: Parretta, A. T.; Laurie, V. W. J. Chem. Phys. 1975, 62, 2463. Computational studies: Deakyne, C. A.; Allen, L. C.; Craig, N. C. J. Am. Chem. Soc. 1977, 99, 3845. Durmaz, S.; Kollmar. H. J. Am. Chem. Soc. 1980, 102, 6942. Clark, T.; Spitznagel, G. W.; Klose, R.; Schleyer, P. von R. J. Am. Chem. Soc. 1984, 106, 4412. Boggs, J. E.; Fan, K. Acta Chem. Scand. 1988, A42, 595.
- (1988) Acta Chem. Scand. , vol.A42 , pp. 595
- Boggs, J.E.¹ Fan, K.²

122
- 84985560982
- Schwager, H.; Kruger, C.; Neidlein, R.; Wilke, G. Angew. Chem., Int. Ed. Engl. 1987, 26, 65. Thom, E.; Christensen, A, T. Acta Crystallogr., Sect. B: Struct. Sci. 1971, 27, 573. Christensen, A. T. Acta Crystallogr., Sect. B.; Struct. Sci. 1970, 26, 1519. Diaz, E.; Barrios, H.; Villena, R.; Toscano, R. A. Acta Crystallogr., Sect. C: Cryst. Struct. Commun. 1991, 47, 2720 and 2723. Irngartinger, H.; Gries, S.; Klaus, P.; Gleiter, R. Chem. Ber. 1992, 125, 2503. Taguchi, T.; Shibuya, A.; Sasaki, H.; Endo, J.; Morikawa, T.; Shiro, M. Tetrahedron: Asymmetry 1994, 5, 1423.
- (1987) Angew. Chem., Int. Ed. Engl. , vol.26 , pp. 65
- Schwager, H.¹ Kruger, C.² Neidlein, R.³ Wilke, G.⁴

123
- 10144244114
- Schwager, H.; Kruger, C.; Neidlein, R.; Wilke, G. Angew. Chem., Int. Ed. Engl. 1987, 26, 65. Thom, E.; Christensen, A, T. Acta Crystallogr., Sect. B: Struct. Sci. 1971, 27, 573. Christensen, A. T. Acta Crystallogr., Sect. B.; Struct. Sci. 1970, 26, 1519. Diaz, E.; Barrios, H.; Villena, R.; Toscano, R. A. Acta Crystallogr., Sect. C: Cryst. Struct. Commun. 1991, 47, 2720 and 2723. Irngartinger, H.; Gries, S.; Klaus, P.; Gleiter, R. Chem. Ber. 1992, 125, 2503. Taguchi, T.; Shibuya, A.; Sasaki, H.; Endo, J.; Morikawa, T.; Shiro, M. Tetrahedron: Asymmetry 1994, 5, 1423.
- (1971) Acta Crystallogr., Sect. B: Struct. Sci. , vol.27 , pp. 573
- Thom, E.¹ Christensen, A.T.²

124
- 0014949907
- Schwager, H.; Kruger, C.; Neidlein, R.; Wilke, G. Angew. Chem., Int. Ed. Engl. 1987, 26, 65. Thom, E.; Christensen, A, T. Acta Crystallogr., Sect. B: Struct. Sci. 1971, 27, 573. Christensen, A. T. Acta Crystallogr., Sect. B.; Struct. Sci. 1970, 26, 1519. Diaz, E.; Barrios, H.; Villena, R.; Toscano, R. A. Acta Crystallogr., Sect. C: Cryst. Struct. Commun. 1991, 47, 2720 and 2723. Irngartinger, H.; Gries, S.; Klaus, P.; Gleiter, R. Chem. Ber. 1992, 125, 2503. Taguchi, T.; Shibuya, A.; Sasaki, H.; Endo, J.; Morikawa, T.; Shiro, M. Tetrahedron: Asymmetry 1994, 5, 1423.
- (1970) Acta Crystallogr., Sect. B.; Struct. Sci. , vol.26 , pp. 1519
- Christensen, A.T.¹

125
- 10144261396
- Schwager, H.; Kruger, C.; Neidlein, R.; Wilke, G. Angew. Chem., Int. Ed. Engl. 1987, 26, 65. Thom, E.; Christensen, A, T. Acta Crystallogr., Sect. B: Struct. Sci. 1971, 27, 573. Christensen, A. T. Acta Crystallogr., Sect. B.; Struct. Sci. 1970, 26, 1519. Diaz, E.; Barrios, H.; Villena, R.; Toscano, R. A. Acta Crystallogr., Sect. C: Cryst. Struct. Commun. 1991, 47, 2720 and 2723. Irngartinger, H.; Gries, S.; Klaus, P.; Gleiter, R. Chem. Ber. 1992, 125, 2503. Taguchi, T.; Shibuya, A.; Sasaki, H.; Endo, J.; Morikawa, T.; Shiro, M. Tetrahedron: Asymmetry 1994, 5, 1423.
- (1991) Acta Crystallogr., Sect. C: Cryst. Struct. Commun. , vol.47 , pp. 2720
- Diaz, E.¹ Barrios, H.² Villena, R.³ Toscano, R.A.⁴

126
- 0001474229
- Schwager, H.; Kruger, C.; Neidlein, R.; Wilke, G. Angew. Chem., Int. Ed. Engl. 1987, 26, 65. Thom, E.; Christensen, A, T. Acta Crystallogr., Sect. B: Struct. Sci. 1971, 27, 573. Christensen, A. T. Acta Crystallogr., Sect. B.; Struct. Sci. 1970, 26, 1519. Diaz, E.; Barrios, H.; Villena, R.; Toscano, R. A. Acta Crystallogr., Sect. C: Cryst. Struct. Commun. 1991, 47, 2720 and 2723. Irngartinger, H.; Gries, S.; Klaus, P.; Gleiter, R. Chem. Ber. 1992, 125, 2503. Taguchi, T.; Shibuya, A.; Sasaki, H.; Endo, J.; Morikawa, T.; Shiro, M. Tetrahedron: Asymmetry 1994, 5, 1423.
- (1992) Chem. Ber. , vol.125 , pp. 2503
- Irngartinger, H.¹ Gries, S.² Klaus, P.³ Gleiter, R.⁴

127
- 0027965577
- Schwager, H.; Kruger, C.; Neidlein, R.; Wilke, G. Angew. Chem., Int. Ed. Engl. 1987, 26, 65. Thom, E.; Christensen, A, T. Acta Crystallogr., Sect. B: Struct. Sci. 1971, 27, 573. Christensen, A. T. Acta Crystallogr., Sect. B.; Struct. Sci. 1970, 26, 1519. Diaz, E.; Barrios, H.; Villena, R.; Toscano, R. A. Acta Crystallogr., Sect. C: Cryst. Struct. Commun. 1991, 47, 2720 and 2723. Irngartinger, H.; Gries, S.; Klaus, P.; Gleiter, R. Chem. Ber. 1992, 125, 2503. Taguchi, T.; Shibuya, A.; Sasaki, H.; Endo, J.; Morikawa, T.; Shiro, M. Tetrahedron: Asymmetry 1994, 5, 1423.
- (1994) Tetrahedron: Asymmetry , vol.5 , pp. 1423
- Taguchi, T.¹ Shibuya, A.² Sasaki, H.³ Endo, J.⁴ Morikawa, T.⁵ Shiro, M.⁶

128
- 0026088954
- Bessard, Y.; Schlosser, M. Tetrahedron 1991, 47, 1231.
- (1991) Tetrahedron , vol.47 , pp. 1231
- Bessard, Y.¹ Schlosser, M.²

129
- 0038559821
- Bernett, W. A. J. Org. Chem. 1969, 34, 1772. For relevant discussions, see: Jason, M. E.; Ibers, J. A. J. Am. Chem. Soc. 1977, 99, 6012. Bernett, W. A. J. Chem. Educ. 1967, 44, 17.
- (1969) J. Org. Chem. , vol.34 , pp. 1772
- Bernett, W.A.¹

130
- 0347183507
- Bernett, W. A. J. Org. Chem. 1969, 34, 1772. For relevant discussions, see: Jason, M. E.; Ibers, J. A. J. Am. Chem. Soc. 1977, 99, 6012. Bernett, W. A. J. Chem. Educ. 1967, 44, 17.
- (1977) J. Am. Chem. Soc. , vol.99 , pp. 6012
- Jason, M.E.¹ Ibers, J.A.²

131
- 33947334946
- Bernett, W. A. J. Org. Chem. 1969, 34, 1772. For relevant discussions, see: Jason, M. E.; Ibers, J. A. J. Am. Chem. Soc. 1977, 99, 6012. Bernett, W. A. J. Chem. Educ. 1967, 44, 17.
- (1967) J. Chem. Educ. , vol.44 , pp. 17
- Bernett, W.A.¹

132
- 33947479158
- Bent, H. A. Chem. Ber. 1961, 61, 275. Bent, H. A. J. Chem. Phys. 1960, 33, 1258, 1259-1260.
- (1961) Chem. Ber. , vol.61 , pp. 275
- Bent, H.A.¹

133
- 36849140696
- Bent, H. A. Chem. Ber. 1961, 61, 275. Bent, H. A. J. Chem. Phys. 1960, 33, 1258, 1259-1260.
- (1960) J. Chem. Phys. , vol.33 , pp. 1258
- Bent, H.A.¹

134
- 0000534419
- Walsh, A. D. Nature (London) 1947, 159, 712. Walsh, A. D. Trans. Faraday Soc. 1949, 45, 179.
- (1947) Nature (London) , vol.159 , pp. 712
- Walsh, A.D.¹

135
- 37049157774
- Walsh, A. D. Nature (London) 1947, 159, 712. Walsh, A. D. Trans. Faraday Soc. 1949, 45, 179.
- (1949) Trans. Faraday Soc. , vol.45 , pp. 179
- Walsh, A.D.¹

136
- 0141507287
- Goldish, E. J. Chem. Educ. 1959, 36, 408.
- (1959) J. Chem. Educ. , vol.36 , pp. 408
- Goldish, E.¹

137
- 84985072237
- Dunitz, J. D.; Schweizer, W. B.; Seiler, B. Helv. Chim. Acta 1983, 66, 134.
- (1983) Helv. Chim. Acta , vol.66 , pp. 134
- Dunitz, J.D.¹ Schweizer, W.B.² Seiler, B.³

138
- 10144226529
- note
- Direct resolution of 17-19 on an HPLC ChiralCel OD column (0.46 × 25 cm, flow rate 0.7-1.0 mL/min) was examined and provides access to the optically active materials: 17, α = 1.18 (10-20% i-PrOH-hexane); 18, α = 1.09-1.05 (10-25% i-PrOH-hexane); 19. α = 1.12 (50% i-PrOH-hexane). However, the recovery was expected to be diminished due to the reactivity of the agents and consequently the preparative resolution of the agents was not pursued.

139
- 10144251916
- note
- 50 values for the natural enantiomers of 17-19 and 24 are 30, 70, 55 μM, and 18 nM, respectively, and consequently follow the trends between reactivity and cytotoxic potency even more closely.

140
- 0025980193
- Boger, D. L.; Munk, S. A.; Zarrinmayeh, H.; Ishizaki, T.; Haught, J.; Bina, M. Tetrahedron 1991, 47, 2661.
- (1991) Tetrahedron , vol.47 , pp. 2661
- Boger, D.L.¹ Munk, S.A.² Zarrinmayeh, H.³ Ishizaki, T.⁴ Haught, J.⁵ Bina, M.⁶

141
- 10144263414
- Full experimental and characterization for 5-12 is provided in supporting information
- Full experimental and characterization for 5-12 is provided in supporting information.

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