Synthesis and structure-activity relationship of pyrazolo[3,4- d]pyrimidines: Potent and selective adenosine A1 receptor antagonists

Journal of Medicinal Chemistry

Volumn 39, Issue 21, 1996, Pages 4156-4161

  Poulsen, Sally Ann ^a   Quinn, Ronald J ^a  

^a GRIFFITH UNIVERSITY   (Australia)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINE A1 RECEPTOR; ADENOSINE A2 RECEPTOR; ADENOSINE RECEPTOR BLOCKING AGENT; PYRAZOLOPYRIMIDINE DERIVATIVE;

ARTICLE; BINDING AFFINITY; BINDING KINETICS; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; STRUCTURE ACTIVITY RELATION;

ADENOSINE; ANIMALS; BINDING, COMPETITIVE; BRAIN; MAGNETIC RESONANCE SPECTROSCOPY; PHENETHYLAMINES; PHENYLISOPROPYLADENOSINE; PYRAZOLES; PYRIMIDINES; RATS; RECEPTORS, PURINERGIC P1; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0029796714     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm960052s     Document Type: Article

References (12)

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