Pyrazolo[3,4-d]pyrimidines: C4, C6 substitution leads to adenosine A1 receptor selectivity

Bioorganic and Medicinal Chemistry Letters

Volumn 6, Issue 4, 1996, Pages 357-360

  Poulsen, Sally Ann ^a   Quinn, Ronald J ^a  

^a GRIFFITH UNIVERSITY   (Australia)

Author keywords

[No Author keywords available]

Indexed keywords

8 (2 NOR 1 ADAMANTYL) 1,3 DIPROPYLXANTHINE; ADENOSINE A1 RECEPTOR; ADENOSINE A2 RECEPTOR; ALPHA (1 PHENYL 4 PROPYLTHIOPYRAZOLO[3,4 D]PYRIMIDIN 6 YLTHIO)BUTANAMIDE; ALPHA (4 METHYLAMINO 1 PHENYLPYRAZOLO[3,4 D]PYRIMIDIN 6 YLTHIO)HEXANAMIDE; PYRAZOLO[3,4 D]PYRIMIDINE DERIVATIVE; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BRAIN; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; NONHUMAN; RAT; STRUCTURE ACTIVITY RELATION;

EID: 0029947382     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0960-894X(96)00027-3     Document Type: Article

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