메뉴 건너뛰기




Volumn 7, Issue 5, 1996, Pages 568-578

Ranking of P-glycoprotein substrates and inhibitors by a calcein-AM fluorometry screening assay

Author keywords

calcein AM; multidrug resistance; P glycoprotein; SDZ PSC 833

Indexed keywords

ACETOXYMETHYL CALCEIN; AMIODARONE; BETA LUMICOLCHICINE; CHLOROQUINE; COLCHICINE; CYCLOSPORIN A; DOXORUBICIN; ETOPOSIDE; GLYCOPROTEIN P; MEPACRINE; QUINIDINE; SDZ 280446; SUBSTRATE; UNCLASSIFIED DRUG; VALSPODAR; VERAPAMIL; VINBLASTINE; VINCRISTINE;

EID: 0029793039     PISSN: 09594973     EISSN: None     Source Type: Journal    
DOI: 10.1097/00001813-199607000-00012     Document Type: Article
Times cited : (177)

References (27)
  • 2
    • 0010367313 scopus 로고
    • Reversal of multidrug-resistance in CHO cells by Cyclosporin A and other resistance modifying agents
    • Boesch D, Gavériaux C, Loor F. Reversal of multidrug-resistance in CHO cells by Cyclosporin A and other resistance modifying agents. J Cell Pharmacol 1991; 2: 92-8.
    • (1991) J Cell Pharmacol , vol.2 , pp. 92-98
    • Boesch, D.1    Gavériaux, C.2    Loor, F.3
  • 3
    • 0000185678 scopus 로고
    • SDZ PSC 833, a non-immunosuppressive cyclosporin analog, is a very potent multidrug-resistance modifier
    • Gavériaux C, Boesch D, Jachez B, Bollinger P, Payne T, Loor F. SDZ PSC 833, a non-immunosuppressive cyclosporin analog, is a very potent multidrug-resistance modifier. J Cell Pharmacol 1991; 2: 225-34.
    • (1991) J Cell Pharmacol , vol.2 , pp. 225-234
    • Gavériaux, C.1    Boesch, D.2    Jachez, B.3    Bollinger, P.4    Payne, T.5    Loor, F.6
  • 5
    • 0022622036 scopus 로고
    • Non-antitumor vinca alkaloids reverse multidrug resistance in P388 leukemia cells in vitro
    • Inaba M, Nagashima K. Non-antitumor vinca alkaloids reverse multidrug resistance in P388 leukemia cells in vitro. Jpn J Cancer Res (Gann) 1986; 77: 197-204.
    • (1986) Jpn J Cancer Res (Gann) , vol.77 , pp. 197-204
    • Inaba, M.1    Nagashima, K.2
  • 7
    • 0023100505 scopus 로고
    • Effects of microtubule inhibitors on etoposide accumulation and DNA damage in human K562 cells in vitro
    • Yalowich JC. Effects of microtubule inhibitors on etoposide accumulation and DNA damage in human K562 cells in vitro. Cancer Res 1987; 47: 1010-5.
    • (1987) Cancer Res , vol.47 , pp. 1010-1015
    • Yalowich, J.C.1
  • 8
    • 0023748077 scopus 로고
    • Effects of indole alkaloids on multidrug resistance and labeling of P-glycoprotein by a photoaffinity analog of vinblastine
    • Beck WT, Cirtain MC, Look AT, Ashmun TA. Effects of indole alkaloids on multidrug resistance and labeling of P-glycoprotein by a photoaffinity analog of vinblastine. Biochem Biophys Res Commun 1988; 153: 959-66.
    • (1988) Biochem Biophys Res Commun , vol.153 , pp. 959-966
    • Beck, W.T.1    Cirtain, M.C.2    Look, A.T.3    Ashmun, T.A.4
  • 9
    • 0025007511 scopus 로고
    • Pharmacology of drugs that alter multidrug resistance in cancer
    • Ford JM, Hait WN, Pharmacology of drugs that alter multidrug resistance in cancer. Pharmacol Rev 1990; 42: 155-99.
    • (1990) Pharmacol Rev , vol.42 , pp. 155-199
    • Ford, J.M.1    Hait, W.N.2
  • 10
    • 0025935235 scopus 로고
    • Restoration of daunomycin retention in multidrug-resistant P388 cells by submicromolar concentrations of SDZ PSC 833, a nonimmunosuppressive cyclosporin derivative
    • Boesch D, Muller K, Pourtier-Manzanedo A, Loor F. Restoration of daunomycin retention in multidrug-resistant P388 cells by submicromolar concentrations of SDZ PSC 833, a nonimmunosuppressive cyclosporin derivative. Exp Cell Res 1991; 196: 26-32.
    • (1991) Exp Cell Res , vol.196 , pp. 26-32
    • Boesch, D.1    Muller, K.2    Pourtier-Manzanedo, A.3    Loor, F.4
  • 11
    • 0026699007 scopus 로고
    • SDZ PSC 833 and SDZ 280-446 are the most active of various resistance-modifying agents in restoring rhodamine-123 retention within multidrug resistant P388 cells
    • Pourtier-Manzanedo A, Didier AD, Muller CD, Loor F. SDZ PSC 833 and SDZ 280-446 are the most active of various resistance-modifying agents in restoring rhodamine-123 retention within multidrug resistant P388 cells. Anti-Cancer Drugs 1992; 3: 419-25.
    • (1992) Anti-Cancer Drugs , vol.3 , pp. 419-425
    • Pourtier-Manzanedo, A.1    Didier, A.D.2    Muller, C.D.3    Loor, F.4
  • 12
    • 0028272044 scopus 로고
    • Extent and persistance of P-glycoprotein inhibition in multidrug-resistant P388 cells after exposure to resistance-modifying agents
    • Boesch D, Loor F. Extent and persistance of P-glycoprotein inhibition in multidrug-resistant P388 cells after exposure to resistance-modifying agents. Anti-Cancer Drugs 1994; 5: 229-38.
    • (1994) Anti-Cancer Drugs , vol.5 , pp. 229-238
    • Boesch, D.1    Loor, F.2
  • 13
    • 0028030228 scopus 로고
    • Rhodamine efflux pattern predict P-glycoprotein substrates in the National Cancer Institute Drug Screen
    • Lee J-S, Paull K, Alvarez M, et al. Rhodamine efflux pattern predict P-glycoprotein substrates in the National Cancer Institute Drug Screen. Mol Pharmacol 1994; 46: 627-38.
    • (1994) Mol Pharmacol , vol.46 , pp. 627-638
    • Lee, J.-S.1    Paull, K.2    Alvarez, M.3
  • 14
    • 0028871929 scopus 로고
    • Decreased uptake of cyclosporin A by P-glycoprotein (Pgp) expressing CEM leukemia cells and restoration of normal retention by Pgp blockers
    • Didier A, Wenger J, Loor F. Decreased uptake of cyclosporin A by P-glycoprotein (Pgp) expressing CEM leukemia cells and restoration of normal retention by Pgp blockers. Anti-Cancer Drugs 1995; 6: 669-80.
    • (1995) Anti-Cancer Drugs , vol.6 , pp. 669-680
    • Didier, A.1    Wenger, J.2    Loor, F.3
  • 15
  • 16
    • 0028332661 scopus 로고
    • Calcein accumulation as a fluorometric functional assay of the multidrug transporter
    • Hollo Zs, Homolya L, Davis CW, Sarkadi B. Calcein accumulation as a fluorometric functional assay of the multidrug transporter. Biochim Biophys Acta 1994; 1191: 384-8.
    • (1994) Biochim Biophys Acta , vol.1191 , pp. 384-388
    • Hollo, Zs.1    Homolya, L.2    Davis, C.W.3    Sarkadi, B.4
  • 17
    • 0028365179 scopus 로고
    • Microfluorometric evaluation of calcein acetoxymethyl ester as a probe for P-glycoprotein-mediated resistance: Effects of cyclosporin A and its nonimmunosuppressive analogue SDZ PSC 833
    • Liminga G, Nygren P, Larsson R. Microfluorometric evaluation of calcein acetoxymethyl ester as a probe for P-glycoprotein-mediated resistance: effects of cyclosporin A and its nonimmunosuppressive analogue SDZ PSC 833. Exp Cell Res 1994; 212: 291-6.
    • (1994) Exp Cell Res , vol.212 , pp. 291-296
    • Liminga, G.1    Nygren, P.2    Larsson, R.3
  • 18
    • 0029658974 scopus 로고    scopus 로고
    • Detection of P-glycoprotein expression by tumoral cells with NBDL-CsA, a fluorescent derivative of cyclosporin A
    • Didier A, Tiberghien F, Wenger R, Loor F. Detection of P-glycoprotein expression by tumoral cells with NBDL-CsA, a fluorescent derivative of cyclosporin A. Anti-Cancer Drugs 1996; 7: 257-65.
    • (1996) Anti-Cancer Drugs , vol.7 , pp. 257-265
    • Didier, A.1    Tiberghien, F.2    Wenger, R.3    Loor, F.4
  • 19
    • 0026558762 scopus 로고
    • SDZ 280-446, a novel semi-synthetic cyclopeptolide:in vitro and in vivo circumvention of the P-glycoprotein-mediated tumour cell multidrug-resistance
    • Loor F, Boesch D, Gavériaux C, Jachez B, Pourtier-Manzanedo A, Emmer G. SDZ 280-446, a novel semi-synthetic cyclopeptolide:in vitro and in vivo circumvention of the P-glycoprotein-mediated tumour cell multidrug-resistance. Br J Cancer 1992; 65: 11-8.
    • (1992) Br J Cancer , vol.65 , pp. 11-18
    • Loor, F.1    Boesch, D.2    Gavériaux, C.3    Jachez, B.4    Pourtier-Manzanedo, A.5    Emmer, G.6
  • 20
    • 0027533571 scopus 로고
    • Restoration of taxol sensitivity of multidrug-resistant cells by the cyclosporin SDZ PSC 833 und the cyclopeptolide SDZ 280-446
    • Jachez B, Nordmann R, Loor F. Restoration of taxol sensitivity of multidrug-resistant cells by the cyclosporin SDZ PSC 833 und the cyclopeptolide SDZ 280-446. J Natl Cancer Inst 1993; 85: 478-83.
    • (1993) J Natl Cancer Inst , vol.85 , pp. 478-483
    • Jachez, B.1    Nordmann, R.2    Loor, F.3
  • 21
    • 0022632544 scopus 로고
    • Amiodarone-induced enhancement of doxorubicin and 4′-deoxyrubicin cytotoxicity to rat colon cancer cells in vitro and in vivo
    • Chauffert B, Martin M, Hamman A, Michel MF, Martin F. Amiodarone-induced enhancement of doxorubicin and 4′-deoxyrubicin cytotoxicity to rat colon cancer cells in vitro and in vivo. Cancer Res 1986; 46: 825-30.
    • (1986) Cancer Res , vol.46 , pp. 825-830
    • Chauffert, B.1    Martin, M.2    Hamman, A.3    Michel, M.F.4    Martin, F.5
  • 22
    • 0021180629 scopus 로고
    • Effects of quinidine and related compounds on cytotoxicity and cellular accumulation of vincristine and adryamicin in drug-resistant tumor cells
    • Tsuruo T, Iida H, Kitatani Y, Yokota K, Tsukagoshi S, Yakurai Y. Effects of quinidine and related compounds on cytotoxicity and cellular accumulation of vincristine and adryamicin in drug-resistant tumor cells. Cancer Res 1984; 44: 4303-7.
    • (1984) Cancer Res , vol.44 , pp. 4303-4307
    • Tsuruo, T.1    Iida, H.2    Kitatani, Y.3    Yokota, K.4    Tsukagoshi, S.5    Yakurai, Y.6
  • 23
    • 0021149466 scopus 로고
    • Restoration of doxorubicin responsiveness in doxorubicin-resistant P388 murine leukemia cells
    • Ramu A, Spanier R, Rahaminoff H, Fuks Z. Restoration of doxorubicin responsiveness in doxorubicin-resistant P388 murine leukemia cells. Br J Cancer 1984; 50: 501-7.
    • (1984) Br J Cancer , vol.50 , pp. 501-507
    • Ramu, A.1    Spanier, R.2    Rahaminoff, H.3    Fuks, Z.4
  • 24
    • 0022612462 scopus 로고
    • Lysosomotropic agents reverse multiple drug resistance in human cancer cells
    • Shiraishi N, Akiyama S, Kobayashi M, Kuwano M. Lysosomotropic agents reverse multiple drug resistance in human cancer cells. Cancer Lett 1986; 30: 251-9.
    • (1986) Cancer Lett , vol.30 , pp. 251-259
    • Shiraishi, N.1    Akiyama, S.2    Kobayashi, M.3    Kuwano, M.4
  • 25
    • 0022971454 scopus 로고
    • Chloroquine enhancement of anticancer drug cytotoxicity in multiple drug resistant human leukemic cells
    • Zamora JM, Beck WT. Chloroquine enhancement of anticancer drug cytotoxicity in multiple drug resistant human leukemic cells. Biochem Pharmacol 1986; 35: 4303-10.
    • (1986) Biochem Pharmacol , vol.35 , pp. 4303-4310
    • Zamora, J.M.1    Beck, W.T.2
  • 26
    • 0023926589 scopus 로고
    • Reversal of resistance to vincristine in P388 leukemia by various polycyclic clinical drugs, with a special emphasis on quinacrine
    • Inaba M, Maruyama E. Reversal of resistance to vincristine in P388 leukemia by various polycyclic clinical drugs, with a special emphasis on quinacrine. Cancer Res 1988; 48: 2064-7.
    • (1988) Cancer Res , vol.48 , pp. 2064-2067
    • Inaba, M.1    Maruyama, E.2
  • 27
    • 0023898749 scopus 로고
    • Physical-chemical properties shared by compounds that modulate multidrug resistance in human leukemic cells
    • Zamora JM, Pearce HL, Beck WT. Physical-chemical properties shared by compounds that modulate multidrug resistance in human leukemic cells. Mol Pharmacol 1988; 33: 454-62.
    • (1988) Mol Pharmacol , vol.33 , pp. 454-462
    • Zamora, J.M.1    Pearce, H.L.2    Beck, W.T.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.