P2-purinoceptor antagonists: I. Blockade of P2-purinoceptor subtypes and ecto-nucleotidases by small aromatic isothiocyanato-sulphonates

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 354, Issue 4, 1996, Pages 481-490

  Bültmann, Ralph ^a   Pause, Birgit ^a,c   Wittenburg, Henning ^a   Kurz, Gerhad ^b   Starke, Klaus ^a  

^a UNIVERSITY OF FREIBURG   (Germany)

^b UNIVERSITY OF FREIBURG   (Germany)

^c Institut fur Biochemie I   (Germany)

Author keywords

DIDS; Ecto nucleotidases; Guinea pig taenia coli; Isothiocyanates; P(2X) purinoceptor; P(2Y) purinoceptor; P2 purinoceptor antagonists; Rat vas deferens

Indexed keywords

ADENOSINE 5' O (2 THIODIPHOSPHATE); ADENOSINE TRIPHOSPHATE; ALPHA,BETA METHYLENEADENOSINE TRIPHOSPHATE; ISOTHIOCYANIC ACID DERIVATIVE; NUCLEOTIDASE; PURINE P2 RECEPTOR; RECEPTOR SUBTYPE; SULFONIC ACID DERIVATIVE; ADENOSINE 5'-O-(2-THIODIPHOSPHATE); ADENOSINE DIPHOSPHATE; ADENOSINE TRIPHOSPHATASE; ALPHA,BETA-METHYLENEADENOSINE 5'-TRIPHOSPHATE; DRUG DERIVATIVE; ECTOATPASE; NUCLEOTIDE;

ANIMAL TISSUE; ARTICLE; COLON TENIA; CONTROLLED STUDY; ENZYME ACTIVITY; FEMALE; GUINEA PIG; MALE; NONHUMAN; RAT; STRUCTURE ACTIVITY RELATION; VAS DEFERENS; VASODILATATION; ANIMAL; COLON; COMPARATIVE STUDY; DRUG ANTAGONISM; DRUG EFFECT; METABOLISM; MUSCLE CONTRACTION; SMOOTH MUSCLE; WISTAR RAT;

ADENOSINE DIPHOSPHATE; ADENOSINE TRIPHOSPHATASES; ADENOSINE TRIPHOSPHATE; ANIMALS; COLON; FEMALE; GUINEA PIGS; ISOTHIOCYANATES; MALE; MUSCLE CONTRACTION; MUSCLE, SMOOTH; RATS; RATS, WISTAR; RECEPTORS, PURINERGIC P2; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONIC ACIDS; THIONUCLEOTIDES; VAS DEFERENS;

EID: 0029658867     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/BF00168440     Document Type: Article

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