Inhibition by propofol of [3H]-batrachotoxinin-A, 20-α-benzoate binding to voltage-dependent sodium channels in rat cortical synaptosomes

British Journal of Pharmacology

Volumn 119, Issue 7, 1996, Pages 1498-1504

  Ratnakumari, L ^a   Hemmings Jr , H C ^a  

^a WEILL CORNELL MEDICAL COLLEGE   (United States)

Author keywords

Batrachotoxin; Brevetoxin; General anaesthesia; Na+ influx; Propofol; Saxitoxin; Scorpion toxin; Synaptosomes; Veratridine; Voltage dependent Na+ channel

Indexed keywords

ANESTHETIC AGENT; BATRACHOTOXININ A 20ALPHA BENZOATE; NEUROTOXIN; PROPOFOL; SAXITOXIN; SCORPION VENOM; SODIUM CHANNEL; SODIUM ION; TRITIUM; VERATRIDINE; BATRACHOTOXIN; BATRACHOTOXININ A 20 ALPHA BENZOATE; BATRACHOTOXININ A 20-ALPHA-BENZOATE; BREVETOXIN; INTRAVENOUS ANESTHETIC AGENT; MARINE TOXIN; OXOCIN DERIVATIVE; SODIUM;

ANIMAL TISSUE; ARTICLE; BINDING KINETICS; BRAIN CORTEX; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG MECHANISM; MALE; NONHUMAN; PRIORITY JOURNAL; RADIOASSAY; RAT; RECEPTOR BINDING; SCATCHARD PLOT; SODIUM TRANSPORT; SYNAPTOSOME; ANIMAL; CHANNEL GATING; DRUG EFFECT; IN VITRO STUDY; KINETICS; METABOLISM; SPRAGUE DAWLEY RAT;

ANESTHETICS, INTRAVENOUS; ANIMALS; BATRACHOTOXINS; CEREBRAL CORTEX; ION CHANNEL GATING; KINETICS; MALE; MARINE TOXINS; NEUROTOXINS; OXOCINS; PROPOFOL; RATS; RATS, SPRAGUE-DAWLEY; SAXITOXIN; SODIUM; SODIUM CHANNELS; SYNAPTOSOMES;

EID: 0029658265     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1476-5381.1996.tb16064.x     Document Type: Article

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