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Volumn 97, Issue 6, 1997, Pages 2243-2266

Chemical synthesis of natural product peptides: Coupling methods for the incorporation of noncoded amino acids into peptides

(2) Humphrey, John M a,b Chamberlin, A Richard a

a UNIVERSITY OF CALIFORNIA (United States)

b UNIVERSITY OF TEXAS AT AUSTIN (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0007193238 PISSN: 00092665 EISSN: None Source Type: Journal
DOI: 10.1021/cr950005s Document Type: Article

Times cited : (1131)

References (199)

1
- 0000915203
- Fusetani, N.; Matsunaga, S. Chem. Rev. 1993, 93, 1793.
- (1993) Chem. Rev. , vol.93 , pp. 1793
- Fusetani, N.¹ Matsunaga, S.²

2
- 0000853969
- Davidson, B. S. Chem. Rev. 1993, 93, 1771.
- (1993) Chem. Rev. , vol.93 , pp. 1771
- Davidson, B.S.¹

3
- 0000314051
- Wipf, P. Chem. Rev. 1995, 95, 2115.
- (1995) Chem. Rev. , vol.95 , pp. 2115
- Wipf, P.¹

4
- 0021047126
- Wenger, R. W. Helv. Chim. Acta 1983, 66, 2308.
- (1983) Helv. Chim. Acta , vol.66 , pp. 2308
- Wenger, R.W.¹

5
- 0023123986
- Tung, R. D.; Rich, D. H. Tetrahedron Lett. 1987, 28, 1139.
- (1987) Tetrahedron Lett. , vol.28 , pp. 1139
- Tung, R.D.¹ Rich, D.H.²

6
- 0022490196
- Evans, D. A.; Weber, A. E. J. Am. Chem. Soc. 1986, 108, 6757.
- (1986) J. Am. Chem. Soc. , vol.108 , pp. 6757
- Evans, D.A.¹ Weber, A.E.²

7
- 0001344734
- Moore, R. E.; Chen, J. L.; Moore, B. S.; Patterson, G. M. L. J. Am. Chem. Soc. 1991, 113, 5083.
- (1991) J. Am. Chem. Soc. , vol.113 , pp. 5083
- Moore, R.E.¹ Chen, J.L.² Moore, B.S.³ Patterson, G.M.L.⁴

8
- 33749709837
- Rinehart, K. L.; Harada, K.; Namikoshi, M.; Chen, C.; Harvis, C. A.; Munro, M. H. G.; Blunt, J. W.; Mulligan, P. E.; Beasley, V. R.; Dahlein, A. M.; Carmichael, W. W. J. Am. Chem. Soc. 1988, 110, 8557.
- (1988) J. Am. Chem. Soc. , vol.110 , pp. 8557
- Rinehart, K.L.¹ Harada, K.² Namikoshi, M.³ Chen, C.⁴ Harvis, C.A.⁵ Munro, M.H.G.⁶ Blunt, J.W.⁷ Mulligan, P.E.⁸ Beasley, V.R.⁹ Dahlein, A.M.¹⁰ Carmichael, W.W.¹¹

9
- 0026594555
- Tohdo, K.; Hamada, Y.; Shiori, T. Tetrahedron Lett. 1992, 33, 2031.
- (1992) Tetrahedron Lett. , vol.33 , pp. 2031
- Tohdo, K.¹ Hamada, Y.² Shiori, T.³

10
- 0024598229
- Matsunaga, S.; Fusetani, N.; Hashimoto, K.; Wälchli, M. J. Am. Chem. Soc. 1989, 111, 2582.
- (1989) J. Am. Chem. Soc. , vol.111 , pp. 2582
- Matsunaga, S.¹ Fusetani, N.² Hashimoto, K.³ Wälchli, M.⁴

11
- 0019263093
- Smith, J. A.; Pease, L. G. CRC Crit. Rev. Biochem. 1980, 8, 315.
- (1980) CRC Crit. Rev. Biochem. , vol.8 , pp. 315
- Smith, J.A.¹ Pease, L.G.²

12
- 0021064132
- Wenger, R. M. Helv. Chim. Acta 1983, 66, 2672.
- (1983) Helv. Chim. Acta , vol.66 , pp. 2672
- Wenger, R.M.¹

13
- 0021912607
- Wenger, R. M. Angew. Chem. Int. Ed. Engl. 1985, 24, 77.
- (1985) Angew. Chem. Int. Ed. Engl. , vol.24 , pp. 77
- Wenger, R.M.¹

14
- 0019519870
- Nagaraj, R.; Balaram, P. Tetrahedron 1981, 37, 1263.
- (1981) Tetrahedron , vol.37 , pp. 1263
- Nagaraj, R.¹ Balaram, P.²

15
- 0000930648
- Slomczynska, U.; Beusen, D. D.; Zabrocki, J.; Kociolek, K.; Redlinski, A.; Reusser, F.; Hutton, W. C.; Leplawy, M. T.; Marshall, G. R. J. Am. Chem. Soc. 1992, 114, 4095.
- (1992) J. Am. Chem. Soc. , vol.114 , pp. 4095
- Slomczynska, U.¹ Beusen, D.D.² Zabrocki, J.³ Kociolek, K.⁴ Redlinski, A.⁵ Reusser, F.⁶ Hutton, W.C.⁷ Leplawy, M.T.⁸ Marshall, G.R.⁹

16
- 0005157002
- Valle, G.; Crisma, M.; Toniolo, C.; Beisswenger, R.; Rieker, A.; Jung, G. J. Am. Chem. Soc. 1989, 111, 6128.
- (1989) J. Am. Chem. Soc. , vol.111 , pp. 6128
- Valle, G.¹ Crisma, M.² Toniolo, C.³ Beisswenger, R.⁴ Rieker, A.⁵ Jung, G.⁶

17
- 0005114091
- Wilkening, R. R.; Stevens, E. S.; Bonora, G. M.; Toniolo, C. J. Am. Chem. Soc. 1983, 105, 2560.
- (1983) J. Am. Chem. Soc. , vol.105 , pp. 2560
- Wilkening, R.R.¹ Stevens, E.S.² Bonora, G.M.³ Toniolo, C.⁴

18
- 8344260956
- Pandey, R. C.; Meng, H.; Cook, J. C., Jr. J. Am. Chem. Soc. 1977, 99, 5201.
- (1977) J. Am. Chem. Soc. , vol.99 , pp. 5201
- Pandey, R.C.¹ Meng, H.² Cook Jr., J.C.³

19
- 0028862474
- Wenschuh, H.; Beyermann, M.; Haber, H.; Seydel, J. K.; Krause, E.; Bienert, M.; Carpino, L. A.; El-Fahem, A.; Albericio, F. J. Org. Chem. 1995, 60, 405.
- (1995) J. Org. Chem. , vol.60 , pp. 405
- Wenschuh, H.¹ Beyermann, M.² Haber, H.³ Seydel, J.K.⁴ Krause, E.⁵ Bienert, M.⁶ Carpino, L.A.⁷ El-Fahem, A.⁸ Albericio, F.⁹

20
- 0000087077
- Bodo, B.; Rebuffat, S.; El Hajji, M.; Davoust, D. J. Am. Chem. 1985, 107, 6011.
- (1985) J. Am. Chem. , vol.107 , pp. 6011
- Bodo, B.¹ Rebuffat, S.² El Hajji, M.³ Davoust, D.⁴

21
- 0010692948
- Kenner, G. W.; Sheppard, R. C. Nature, London 1958, 181, 48.
- (1958) Nature, London , vol.181 , pp. 48
- Kenner, G.W.¹ Sheppard, R.C.²

22
- 0014428197
- Müller, P.; Rudin, D. O. Nature 1968, 277, 713.
- (1968) Nature , vol.277 , pp. 713
- Müller, P.¹ Rudin, D.O.²

23
- 0021255704
- Schmidt, U.; Lieberknecht, A.; Griesser, H.; Bartkowiak, F. Angew. Chem. Int. Ed. Engl. 1984, 23, 318.
- (1984) Angew. Chem. Int. Ed. Engl. , vol.23 , pp. 318
- Schmidt, U.¹ Lieberknecht, A.² Griesser, H.³ Bartkowiak, F.⁴

24
- 8344236280
- Testa, B., Ed.; Academic Press: London
- Fauchère, J. L. In Advances in Drug Research; Testa, B., Ed.; Academic Press: London, 1986; p 15.
- (1986) Advances in Drug Research , pp. 15
- Fauchère, J.L.¹

25
- 8344250491
- Ragnarsson, U., Ed.; Almqvist and Wiksell Int.: Stockholm, Sweden
- Cordopatis, P.; Gatos, D.; Theodoropoulos, D.; Mizrahi, J.; Regoli, D.; Escher, E. In Peptides 1984; Ragnarsson, U., Ed.; Almqvist and Wiksell Int.: Stockholm, Sweden, 1985; p 249.
- (1985) Peptides 1984 , pp. 249
- Cordopatis, P.¹ Gatos, D.² Theodoropoulos, D.³ Mizrahi, J.⁴ Regoli, D.⁵ Escher, E.⁶

26
- 0002893709
- John Wright and Sons Ltd.: London
- Stammer, C. H. In Chemistry and Biology of Amino Acids, Peptides and Proteins; John Wright and Sons Ltd.: London, 1982; Vol. 6, p 33.
- (1982) Chemistry and Biology of Amino Acids, Peptides and Proteins , vol.6 , pp. 33
- Stammer, C.H.¹

27
- 84985738595
- Agò, D.H.; Granozzi, G.; Tondello, E.; Del Prà, A. Biopolymers 1980, 19, 469.
- (1980) Biopolymers , vol.19 , pp. 469
- Agò, D.H.¹ Granozzi, G.² Tondello, E.³ Del Prà, A.⁴

28
- 0016162738
- Rich, D. H.; Mathiaparanam, P. Tetrahedron Lett. 1974, 46, 4037.
- (1974) Tetrahedron Lett. , vol.46 , pp. 4037
- Rich, D.H.¹ Mathiaparanam, P.²

29
- 85007932604
- Konno, S.; Stammer, C. H. Synthesis 1978, 598.
- (1978) Synthesis , pp. 598
- Konno, S.¹ Stammer, C.H.²

30
- 0014670910
- Givot, I. L.; Smith, T. A.; Abeles, R. H. J. Biol. Chem. 1969, 244, 6341.
- (1969) J. Biol. Chem. , vol.244 , pp. 6341
- Givot, I.L.¹ Smith, T.A.² Abeles, R.H.³

31
- 0014670950
- Wickner, R. B. J. Biol. Chem. 1969, 244, 6550.
- (1969) J. Biol. Chem. , vol.244 , pp. 6550
- Wickner, R.B.¹

32
- 0018195713
- English, M. L.; Stammer, C. H. Int. J. Peptide Protein Res. 1978, 85, 780.
- (1978) Int. J. Peptide Protein Res. , vol.85 , pp. 780
- English, M.L.¹ Stammer, C.H.²

33
- 8344260155
- Chipkin, R. E.; Stewart, J. M.; Stammer, C. H. Biochem. Biophys. Res. Commun. 1979, 87, 780.
- (1979) Biochem. Biophys. Res. Commun. , vol.87 , pp. 780
- Chipkin, R.E.¹ Stewart, J.M.² Stammer, C.H.³

34
- 0030061507
- Spatola, A. F.; Darlak, K.; Romanovskis, P. Tetrahedron Lett. 1996, 37, 591.
- (1996) Tetrahedron Lett. , vol.37 , pp. 591
- Spatola, A.F.¹ Darlak, K.² Romanovskis, P.³

35
- 0021169493
- Schmidt, U.; Schanbacher, U. Liebigs Ann. Chem. 1984, 1205.
- (1984) Liebigs Ann. Chem. , pp. 1205
- Schmidt, U.¹ Schanbacher, U.²

36
- 84985633295
- Schmidt, U.; Wild, J. Angew. Chem. Int. Ed. Engl. 1984, 23, 991.
- (1984) Angew. Chem. Int. Ed. Engl. , vol.23 , pp. 991
- Schmidt, U.¹ Wild, J.²

37
- 0003416748
- Pergamon Press: Oxford
- Williams, R. M. Synthesis of Optically Active α-Amino Acids; Pergamon Press: Oxford, 1989.
- (1989) Synthesis of Optically Active α-Amino Acids
- Williams, R.M.¹

38
- 8344233724
- Williams, R. M. Aldrichimica Acta 1992, 25, 1992.
- (1992) Aldrichimica Acta , vol.25 , pp. 1992
- Williams, R.M.¹

39
- 0001463392
- Ohfune, Y. Acc. Chem. Res. 1992, 25, 360.
- (1992) Acc. Chem. Res. , vol.25 , pp. 360
- Ohfune, Y.¹

40
- 0027082945
- Kamphius, J.; Meijer, E. M.; Boesten, W. H. J.; Sonke, T.; Van Den Tweel, W. J. J.; Schoemaker, H. E. A. New York Acad. Sci. 1992, 672, 510.
- (1992) New York Acad. Sci. , vol.672 , pp. 510
- Kamphius, J.¹ Meijer, E.M.² Boesten, W.H.J.³ Sonke, T.⁴ Van Den Tweel, W.J.J.⁵ Schoemaker, H.E.A.⁶

41
- 0001122927
- Williams, R. M.; Hendrix, J. A. Chem. Rev. 1992, 52, 889.
- (1992) Chem. Rev. , vol.52 , pp. 889
- Williams, R.M.¹ Hendrix, J.A.²

42
- 0001168887
- Verhovskaya, M. A.; Yamskov, I. A. Russ. Chem. Rev. 1991, 60, 1163.
- (1991) Russ. Chem. Rev. , vol.60 , pp. 1163
- Verhovskaya, M.A.¹ Yamskov, I.A.²

43
- 0000360708
- Havlicek, L.; Hanus, J. Collect. Czech. Chem. Commun. 1991, 56, 1365.
- (1991) Collect. Czech. Chem. Commun. , vol.56 , pp. 1365
- Havlicek, L.¹ Hanus, J.²

44
- 0000242199
- Arnold, L. D.; Drover, J. C.; Vederas, J. C. J. Am. Chem. Soc. 1987, 109, 4649.
- (1987) J. Am. Chem. Soc. , vol.109 , pp. 4649
- Arnold, L.D.¹ Drover, J.C.² Vederas, J.C.³

45
- 0000411342
- Gross, E., Meienhofer, J., Eds.; Academic Press, Inc.
- Roberts, D. C.; Vellaccio, F. In The Peptides; Gross, E., Meienhofer, J., Eds.; Academic Press, Inc.: 1983; Vol. 5, p 341.
- (1983) The Peptides , vol.5 , pp. 341
- Roberts, D.C.¹ Vellaccio, F.²

46
- 84985610072
- Schmidt, U.; Griesser, H.; Lieberknecht, A.; Talbiersky, J. Angew. Chem., Int. Ed. Engl. 1981, 20, 280.
- (1981) Angew. Chem., Int. Ed. Engl. , vol.20 , pp. 280
- Schmidt, U.¹ Griesser, H.² Lieberknecht, A.³ Talbiersky, J.⁴

47
- 0001087038
- Schmidt, U.; Lieberknecht, A.; Griesser, H.; Talbiersky, J. J. Org. Chem. 1982, 47, 3261.
- (1982) J. Org. Chem. , vol.47 , pp. 3261
- Schmidt, U.¹ Lieberknecht, A.² Griesser, H.³ Talbiersky, J.⁴

48
- 0001300170
- Schmidt, U.; Lieberknecht, A.; Bökens, H.; Griesser, H. J. Org. Chem. 1983, 48, 2680.
- (1983) J. Org. Chem. , vol.48 , pp. 2680
- Schmidt, U.¹ Lieberknecht, A.² Bökens, H.³ Griesser, H.⁴

49
- 0023901959
- Schmidt, U.; Weller, D.; Holder, A.; Lieberknecht, A. Tetrahedron Lett. 1988, 29, 3227.
- (1988) Tetrahedron Lett. , vol.29 , pp. 3227
- Schmidt, U.¹ Weller, D.² Holder, A.³ Lieberknecht, A.⁴

50
- 0024833960
- Heffner, R. J.; Joullié, M. M. Tetrahedron Lett. 1989, 30, 7021.
- (1989) Tetrahedron Lett. , vol.30 , pp. 7021
- Heffner, R.J.¹ Joullié, M.M.²

51
- 0024508264
- Evans, D. A.; Ellman, J. A. J. Am. Chem. Soc. 1989, 111, 1063.
- (1989) J. Am. Chem. Soc. , vol.111 , pp. 1063
- Evans, D.A.¹ Ellman, J.A.²

52
- 0028328499
- Aguilar, E.; Meyers, A. I. Tetrahedron Lett. 1994, 35, 2477.
- (1994) Tetrahedron Lett. , vol.35 , pp. 2477
- Aguilar, E.¹ Meyers, A.I.²

53
- 0028090132
- Boden, C.; Pattenden, G. Tetrahedron Lett. 1994, 35, 8271.
- (1994) Tetrahedron Lett. , vol.35 , pp. 8271
- Boden, C.¹ Pattenden, G.²

54
- 85082557998
- Schmidt, U.; Utz, R.; Lieberknecht, A.; Griesser, H.; Potzolli, B.; Bahr, J.; Wagner, K.; Fischer, P. Synthesis 1987, 236.
- (1987) Synthesis , vol.236
- Schmidt, U.¹ Utz, R.² Lieberknecht, A.³ Griesser, H.⁴ Potzolli, B.⁵ Bahr, J.⁶ Wagner, K.⁷ Fischer, P.⁸

55
- 0021799961
- Hamada, Y.; Kato, S.; Shiori, T. Tetrahedron Lett. 1985, 26, 3223.
- (1985) Tetrahedron Lett. , vol.26 , pp. 3223
- Hamada, Y.¹ Kato, S.² Shiori, T.³

56
- 0022640986
- Schmidt, U.; Griesser, H. Tetrahedron Lett. 1986, 27, 163.
- (1986) Tetrahedron Lett. , vol.27 , pp. 163
- Schmidt, U.¹ Griesser, H.²

57
- 0001640898
- Goff, D.; Lagarias, J. C.; Willy, C. S.; Klein, M. P.; Rapoport, H. J. Org. Chem. 1980, 45, 4813.
- (1980) J. Org. Chem. , vol.45 , pp. 4813
- Goff, D.¹ Lagarias, J.C.² Willy, C.S.³ Klein, M.P.⁴ Rapoport, H.⁵

58
- 0029847930
- Wipf, P.; Venkatraman, S. J. Org. Chem. 1996, 61, 6517.
- (1996) J. Org. Chem. , vol.61 , pp. 6517
- Wipf, P.¹ Venkatraman, S.²

59
- 0023872535
- Schmidt, U.; Lieberknecht, A.; Wild, J. Synthesis 1988, 159.
- (1988) Synthesis , pp. 159
- Schmidt, U.¹ Lieberknecht, A.² Wild, J.³

60
- 0003175687
- Gross, E. and J. Meienhofer, E.; Academic Press, Inc.: New York-London
- Noda, K.; Shimohigashi, Y.; Izumiya, N. In The Peptides; Gross, E. and J. Meienhofer, E.; Academic Press, Inc.: New York-London, 1983; Vol. 5, pp 285.
- (1983) The Peptides , vol.5 , pp. 285
- Noda, K.¹ Shimohigashi, Y.² Izumiya, N.³

61
- 85023346540
- Hagihara, M.; Anthony, N. J.; Stout, T. J.; Clardy, J.; Schreiber, S. L. J. Am. Chem. Soc. 1992, 114, 6568.
- (1992) J. Am. Chem. Soc. , vol.114 , pp. 6568
- Hagihara, M.¹ Anthony, N.J.² Stout, T.J.³ Clardy, J.⁴ Schreiber, S.L.⁵

62
- 0026795414
- Hagihara, M.; Schreiber, S. L. J. Am. Chem. Soc. 1992, 114, 6570.
- (1992) J. Am. Chem. Soc. , vol.114 , pp. 6570
- Hagihara, M.¹ Schreiber, S.L.²

63
- 0026716205
- Roth, P.; Metternich, R. Tetrahedron Lett. 1992, 33, 3993.
- (1992) Tetrahedron Lett. , vol.33 , pp. 3993
- Roth, P.¹ Metternich, R.²

64
- 0027487010
- Wipf, P.; Kim, H. J. Org. Chem 1993, 58, 5592.
- (1993) J. Org. Chem , vol.58 , pp. 5592
- Wipf, P.¹ Kim, H.²

65
- 33750259615
- Deng, J.; Hamada, Y.; Shioiri, T.; Matsunaga, S.; Fusetani, N. Angew. Chem., Int. Ed. Engl. 1994, 33, 1729.
- (1994) Angew. Chem., Int. Ed. Engl. , vol.33 , pp. 1729
- Deng, J.¹ Hamada, Y.² Shioiri, T.³ Matsunaga, S.⁴ Fusetani, N.⁵

66
- 85047671524
- Bastiaans, H. M. M.; van der Baan, J. L.; Ottenheijm, H. C. J. Tetrahedron Lett. 1995, 36, 5963.
- (1995) Tetrahedron Lett. , vol.36 , pp. 5963
- Bastiaans, H.M.M.¹ Van Der Baan, J.L.² Ottenheijm, H.C.J.³

67
- 0029880219
- Deng, J.; Hamada, Y.; Shioiri, T. Tetrahedron Lett. 1996, 37, 2261.
- (1996) Tetrahedron Lett. , vol.37 , pp. 2261
- Deng, J.¹ Hamada, Y.² Shioiri, T.³

68
- 0001001070
- For some N-alkylation methods, see: (a) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906. (b) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911. (c) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 916. (d) Freidinger, R. M.; Hinkle, J. S.; Perlow, D. S.; Arison, B. H. J. Org. Chem. 1983, 48, 77. (e) McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915. (f) Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991,56, 5196. (g) Grieco, P. A.; Bahsas, A. J. Org. Chem. 1987, 26, 5647. (h) Olsen, R. K. J. Org. Chem. 1970, 35, 1912. (i) Hansen, D. W.; Pilipauskas, D. J. Org. Chem. 1985, 50, 945. (j) Pine, S. H. J. Org. Chem. 1971, 36, 829. (k) Borch, R. F.; Hassid, A. I. J. Org. Chem. 1972, 37, 1673. (l) Coggins, J. R.; Benoiton, N. L. Can. J. Chem. 1971, 1, 1968.
- (1977) Can. J. Chem. , vol.55 , pp. 906
- Cheung, S.T.¹ Benoiton, N.L.²

69
- 0001001070
- For some N-alkylation methods, see: (a) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906. (b) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911. (c) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 916. (d) Freidinger, R. M.; Hinkle, J. S.; Perlow, D. S.; Arison, B. H. J. Org. Chem. 1983, 48, 77. (e) McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915. (f) Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991,56, 5196. (g) Grieco, P. A.; Bahsas, A. J. Org. Chem. 1987, 26, 5647. (h) Olsen, R. K. J. Org. Chem. 1970, 35, 1912. (i) Hansen, D. W.; Pilipauskas, D. J. Org. Chem. 1985, 50, 945. (j) Pine, S. H. J. Org. Chem. 1971, 36, 829. (k) Borch, R. F.; Hassid, A. I. J. Org. Chem. 1972, 37, 1673. (l) Coggins, J. R.; Benoiton, N. L. Can. J. Chem. 1971, 1, 1968.
- (1977) Can. J. Chem. , vol.55 , pp. 911
- Cheung, S.T.¹ Benoiton, N.L.²

70
- 0000878731
- For some N-alkylation methods, see: (a) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906. (b) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911. (c) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 916. (d) Freidinger, R. M.; Hinkle, J. S.; Perlow, D. S.; Arison, B. H. J. Org. Chem. 1983, 48, 77. (e) McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915. (f) Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991,56, 5196. (g) Grieco, P. A.; Bahsas, A. J. Org. Chem. 1987, 26, 5647. (h) Olsen, R. K. J. Org. Chem. 1970, 35, 1912. (i) Hansen, D. W.; Pilipauskas, D. J. Org. Chem. 1985, 50, 945. (j) Pine, S. H. J. Org. Chem. 1971, 36, 829. (k) Borch, R. F.; Hassid, A. I. J. Org. Chem. 1972, 37, 1673. (l) Coggins, J. R.; Benoiton, N. L. Can. J. Chem. 1971, 1, 1968.
- (1977) Can. J. Chem. , vol.55 , pp. 916
- Cheung, S.T.¹ Benoiton, N.L.²

71
- 0002840747
- For some N-alkylation methods, see: (a) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906. (b) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911. (c) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 916. (d) Freidinger, R. M.; Hinkle, J. S.; Perlow, D. S.; Arison, B. H. J. Org. Chem. 1983, 48, 77. (e) McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915. (f) Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991,56, 5196. (g) Grieco, P. A.; Bahsas, A. J. Org. Chem. 1987, 26, 5647. (h) Olsen, R. K. J. Org. Chem. 1970, 35, 1912. (i) Hansen, D. W.; Pilipauskas, D. J. Org. Chem. 1985, 50, 945. (j) Pine, S. H. J. Org. Chem. 1971, 36, 829. (k) Borch, R. F.; Hassid, A. I. J. Org. Chem. 1972, 37, 1673. (l) Coggins, J. R.; Benoiton, N. L. Can. J. Chem. 1971, 1, 1968.
- (1983) J. Org. Chem. , vol.48 , pp. 77
- Freidinger, R.M.¹ Hinkle, J.S.² Perlow, D.S.³ Arison, B.H.⁴

72
- 0001023731
- For some N-alkylation methods, see: (a) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906. (b) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911. (c) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 916. (d) Freidinger, R. M.; Hinkle, J. S.; Perlow, D. S.; Arison, B. H. J. Org. Chem. 1983, 48, 77. (e) McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915. (f) Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991,56, 5196. (g) Grieco, P. A.; Bahsas, A. J. Org. Chem. 1987, 26, 5647. (h) Olsen, R. K. J. Org. Chem. 1970, 35, 1912. (i) Hansen, D. W.; Pilipauskas, D. J. Org. Chem. 1985, 50, 945. (j) Pine, S. H. J. Org. Chem. 1971, 36, 829. (k) Borch, R. F.; Hassid, A. I. J. Org. Chem. 1972, 37, 1673. (l) Coggins, J. R.; Benoiton, N. L. Can. J. Chem. 1971, 1, 1968.
- (1973) Can. J. Chem. , vol.51 , pp. 1915
- McDermott, J.R.¹ Benoiton, N.L.²

73
- 0025819848
- For some N-alkylation methods, see: (a) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906. (b) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911. (c) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 916. (d) Freidinger, R. M.; Hinkle, J. S.; Perlow, D. S.; Arison, B. H. J. Org. Chem. 1983, 48, 77. (e) McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915. (f) Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991,56, 5196. (g) Grieco, P. A.; Bahsas, A. J. Org. Chem. 1987, 26, 5647. (h) Olsen, R. K. J. Org. Chem. 1970, 35, 1912. (i) Hansen, D. W.; Pilipauskas, D. J. Org. Chem. 1985, 50, 945. (j) Pine, S. H. J. Org. Chem. 1971, 36, 829. (k) Borch, R. F.; Hassid, A. I. J. Org. Chem. 1972, 37, 1673. (l) Coggins, J. R.; Benoiton, N. L. Can. J. Chem. 1971, 1, 1968.
- (1991) J. Org. Chem. , vol.56 , pp. 5196
- Chu, K.S.¹ Negrete, G.R.² Konopelski, J.P.³

74
- 8344253123
- For some N-alkylation methods, see: (a) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906. (b) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911. (c) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 916. (d) Freidinger, R. M.; Hinkle, J. S.; Perlow, D. S.; Arison, B. H. J. Org. Chem. 1983, 48, 77. (e) McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915. (f) Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991,56, 5196. (g) Grieco, P. A.; Bahsas, A. J. Org. Chem. 1987, 26, 5647. (h) Olsen, R. K. J. Org. Chem. 1970, 35, 1912. (i) Hansen, D. W.; Pilipauskas, D. J. Org. Chem. 1985, 50, 945. (j) Pine, S. H. J. Org. Chem. 1971, 36, 829. (k) Borch, R. F.; Hassid, A. I. J. Org. Chem. 1972, 37, 1673. (l) Coggins, J. R.; Benoiton, N. L. Can. J. Chem. 1971, 1, 1968.
- (1987) J. Org. Chem. , vol.26 , pp. 5647
- Grieco, P.A.¹ Bahsas, A.²

75
- 0014802891
- For some N-alkylation methods, see: (a) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906. (b) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911. (c) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 916. (d) Freidinger, R. M.; Hinkle, J. S.; Perlow, D. S.; Arison, B. H. J. Org. Chem. 1983, 48, 77. (e) McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915. (f) Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991,56, 5196. (g) Grieco, P. A.; Bahsas, A. J. Org. Chem. 1987, 26, 5647. (h) Olsen, R. K. J. Org. Chem. 1970, 35, 1912. (i) Hansen, D. W.; Pilipauskas, D. J. Org. Chem. 1985, 50, 945. (j) Pine, S. H. J. Org. Chem. 1971, 36, 829. (k) Borch, R. F.; Hassid, A. I. J. Org. Chem. 1972, 37, 1673. (l) Coggins, J. R.; Benoiton, N. L. Can. J. Chem. 1971, 1, 1968.
- (1970) J. Org. Chem. , vol.35 , pp. 1912
- Olsen, R.K.¹

76
- 0000763544
- For some N-alkylation methods, see: (a) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906. (b) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911. (c) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 916. (d) Freidinger, R. M.; Hinkle, J. S.; Perlow, D. S.; Arison, B. H. J. Org. Chem. 1983, 48, 77. (e) McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915. (f) Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991,56, 5196. (g) Grieco, P. A.; Bahsas, A. J. Org. Chem. 1987, 26, 5647. (h) Olsen, R. K. J. Org. Chem. 1970, 35, 1912. (i) Hansen, D. W.; Pilipauskas, D. J. Org. Chem. 1985, 50, 945. (j) Pine, S. H. J. Org. Chem. 1971, 36, 829. (k) Borch, R. F.; Hassid, A. I. J. Org. Chem. 1972, 37, 1673. (l) Coggins, J. R.; Benoiton, N. L. Can. J. Chem. 1971, 1, 1968.
- (1985) J. Org. Chem. , vol.50 , pp. 945
- Hansen, D.W.¹ Pilipauskas, D.²

77
- 0000235826
- For some N-alkylation methods, see: (a) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906. (b) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911. (c) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 916. (d) Freidinger, R. M.; Hinkle, J. S.; Perlow, D. S.; Arison, B. H. J. Org. Chem. 1983, 48, 77. (e) McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915. (f) Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991,56, 5196. (g) Grieco, P. A.; Bahsas, A. J. Org. Chem. 1987, 26, 5647. (h) Olsen, R. K. J. Org. Chem. 1970, 35, 1912. (i) Hansen, D. W.; Pilipauskas, D. J. Org. Chem. 1985, 50, 945. (j) Pine, S. H. J. Org. Chem. 1971, 36, 829. (k) Borch, R. F.; Hassid, A. I. J. Org. Chem. 1972, 37, 1673. (l) Coggins, J. R.; Benoiton, N. L. Can. J. Chem. 1971, 1, 1968.
- (1971) J. Org. Chem. , vol.36 , pp. 829
- Pine, S.H.¹

78
- 33947089510
- For some N-alkylation methods, see: (a) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906. (b) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911. (c) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 916. (d) Freidinger, R. M.; Hinkle, J. S.; Perlow, D. S.; Arison, B. H. J. Org. Chem. 1983, 48, 77. (e) McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915. (f) Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991,56, 5196. (g) Grieco, P. A.; Bahsas, A. J. Org. Chem. 1987, 26, 5647. (h) Olsen, R. K. J. Org. Chem. 1970, 35, 1912. (i) Hansen, D. W.; Pilipauskas, D. J. Org. Chem. 1985, 50, 945. (j) Pine, S. H. J. Org. Chem. 1971, 36, 829. (k) Borch, R. F.; Hassid, A. I. J. Org. Chem. 1972, 37, 1673. (l) Coggins, J. R.; Benoiton, N. L. Can. J. Chem. 1971, 1, 1968.
- (1972) J. Org. Chem. , vol.37 , pp. 1673
- Borch, R.F.¹ Hassid, A.I.²

79
- 0000524317
- For some N-alkylation methods, see: (a) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906. (b) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911. (c) Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 916. (d) Freidinger, R. M.; Hinkle, J. S.; Perlow, D. S.; Arison, B. H. J. Org. Chem. 1983, 48, 77. (e) McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915. (f) Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991,56, 5196. (g) Grieco, P. A.; Bahsas, A. J. Org. Chem. 1987, 26, 5647. (h) Olsen, R. K. J. Org. Chem. 1970, 35, 1912. (i) Hansen, D. W.; Pilipauskas, D. J. Org. Chem. 1985, 50, 945. (j) Pine, S. H. J. Org. Chem. 1971, 36, 829. (k) Borch, R. F.; Hassid, A. I. J. Org. Chem. 1972, 37, 1673. (l) Coggins, J. R.; Benoiton, N. L. Can. J. Chem. 1971, 1, 1968.
- (1971) Can. J. Chem. , vol.1 , pp. 1968
- Coggins, J.R.¹ Benoiton, N.L.²

80
- 0001605966
- McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 2555.
- (1973) Can. J. Chem. , vol.51 , pp. 2555
- McDermott, J.R.¹ Benoiton, N.L.²

81
- 0001023730
- McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 2562.
- (1973) Can. J. Chem. , vol.51 , pp. 2562
- McDermott, J.R.¹ Benoiton, N.L.²

82
- 85033311166
- For a detailed discussion, see the Segment Coupling section
- For a detailed discussion, see the Segment Coupling section.

83
- 0011169578
- Galpin, I. J.; Mohommed, A. K. A.; Patel, A. Tetrahedron 1988, 44, 1685.
- (1988) Tetrahedron , vol.44 , pp. 1685
- Galpin, I.J.¹ Mohommed, A.K.A.² Patel, A.³

84
- 37049105216
- Davies, J. S.; Mohammed, A. K. J. Chem. Soc. Perkin I 1981, 2982.
- (1981) J. Chem. Soc. Perkin I , pp. 2982
- Davies, J.S.¹ Mohammed, A.K.²

85
- 0026642114
- Frerot, E.; Coste, J.; Poncet, J.; Jouin, P.; Castro, B. Tetrahedron Lett. 1992, 33, 2815.
- (1992) Tetrahedron Lett. , vol.33 , pp. 2815
- Frerot, E.¹ Coste, J.² Poncet, J.³ Jouin, P.⁴ Castro, B.⁵

86
- 0017893016
- Rich, D. H.; Bhatnagar, P.; Mathiaparanam, P.; Grant, J. A.; Tam, J. P. J. Org. Chem. 1978, 43, 296.
- (1978) J. Org. Chem. , vol.43 , pp. 296
- Rich, D.H.¹ Bhatnagar, P.² Mathiaparanam, P.³ Grant, J.A.⁴ Tam, J.P.⁵

87
- 0015527159
- Khosla, M. C.; Smeby, R. R.; Bumpus, F. M. J. Am. Chem. Soc. 1972, 94, 4721.
- (1972) J. Am. Chem. Soc. , vol.94 , pp. 4721
- Khosla, M.C.¹ Smeby, R.R.² Bumpus, F.M.³

88
- 0015492764
- Gisin, B. F.; Merrifield, R. B. J. Am. Chem. Soc. 1972, 94, 3102.
- (1972) J. Am. Chem. Soc. , vol.94 , pp. 3102
- Gisin, B.F.¹ Merrifield, R.B.²

89
- 85004816680
- van der Auwera, C.; Anteunis, M. J. O. Int. J. Peptide Protein Res. 1988, 37, 186.
- (1988) Int. J. Peptide Protein Res. , vol.37 , pp. 186
- Van Der Auwera, C.¹ Anteunis, M.J.O.²

90
- 85004775257
- Anteunis, M. J. O.; Van Der Auwera, C. Int. J. Peptide Protein Res. 1988, 31, 301.
- (1988) Int. J. Peptide Protein Res. , vol.31 , pp. 301
- Anteunis, M.J.O.¹ Van Der Auwera, C.²

91
- 49549139072
- Castro, B.; Dormoy, J.-R.; Evin, G.; Selve, C. Tetrahedron Lett. 1975, 16, 1219.
- (1975) Tetrahedron Lett. , vol.16 , pp. 1219
- Castro, B.¹ Dormoy, J.-R.² Evin, G.³ Selve, C.⁴

92
- 0025868658
- Coste, J.; Frerot, E.; Jouin, P.; Castro, B. Tetrahedron Lett. 1991, 32, 1967.
- (1991) Tetrahedron Lett. , vol.32 , pp. 1967
- Coste, J.¹ Frerot, E.² Jouin, P.³ Castro, B.⁴

93
- 0346593093
- Gross, E., Meienhofer, J., Eds.; Academic Press: New York-London
- For studies on racemization in peptide synthesis, see: Kovacs, J. In The Peptides; Gross, E., Meienhofer, J., Eds.; Academic Press: New York-London, 1980; Vol. 2, p 485. Kemp, D. S. In The Peptides; Gross, E., Meienhofer, J., Eds.; Academic Press: New York-London, 1979; Vol. 1, p 315. Davies, J. S.; Mohammed, A. K. J. Chem. Soc. Perkin I 1981, 2982.
- (1980) The Peptides , vol.2 , pp. 485
- Kovacs, J.¹

94
- 0001587747
- Gross, E., Meienhofer, J., Eds.; Academic Press: New York-London
- For studies on racemization in peptide synthesis, see: Kovacs, J. In The Peptides; Gross, E., Meienhofer, J., Eds.; Academic Press: New York-London, 1980; Vol. 2, p 485. Kemp, D. S. In The Peptides; Gross, E., Meienhofer, J., Eds.; Academic Press: New York-London, 1979; Vol. 1, p 315. Davies, J. S.; Mohammed, A. K. J. Chem. Soc. Perkin I 1981, 2982.
- (1979) The Peptides , vol.1 , pp. 315
- Kemp, D.S.¹

95
- 37049105216
- For studies on racemization in peptide synthesis, see: Kovacs, J. In The Peptides; Gross, E., Meienhofer, J., Eds.; Academic Press: New York-London, 1980; Vol. 2, p 485. Kemp, D. S. In The Peptides; Gross, E., Meienhofer, J., Eds.; Academic Press: New York-London, 1979; Vol. 1, p 315. Davies, J. S.; Mohammed, A. K. J. Chem. Soc. Perkin I 1981, 2982.
- (1981) J. Chem. Soc. Perkin I , pp. 2982
- Davies, J.S.¹ Mohammed, A.K.²

96
- 85007985025
- Chang, C. F.; Myokei, R.; Sakurai, A.; Takahashi, N.; Tamura, S. Agric. Biol. Chem. 1969, 33, 1501.
- (1969) Agric. Biol. Chem. , vol.33 , pp. 1501
- Chang, C.F.¹ Myokei, R.² Sakurai, A.³ Takahashi, N.⁴ Tamura, S.⁵

97
- 0014475017
- Myokei, R.; Sakurai, A.; Chang, C. F.; Kodaira, Y.; Takahashi, N.; Tamura, S. Tetrahedron Lett. 1969, 9, 695.
- (1969) Tetrahedron Lett. , vol.9 , pp. 695
- Myokei, R.¹ Sakurai, A.² Chang, C.F.³ Kodaira, Y.⁴ Takahashi, N.⁵ Tamura, S.⁶

98
- 0021159751
- Dourtoglou, V.; Gross, B. Synthesis 1984, 572.
- (1984) Synthesis , pp. 572
- Dourtoglou, V.¹ Gross, B.²

99
- 0001001070
- Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 911.
- (1977) Can. J. Chem. , vol.55 , pp. 911
- Cheung, S.T.¹ Benoiton, N.L.²

100
- 33845377031
- Tung, R. D.; Rich, D. H. J. Am. Chem. Soc. 1985, 107, 4342.
- (1985) J. Am. Chem. Soc. , vol.107 , pp. 4342
- Tung, R.D.¹ Rich, D.H.²

101
- 85004721004
- Van der Auwera, C.; Anteunis, M. J. Int. J. Peptide Protein Res. 1987, 29, 574.
- (1987) Int. J. Peptide Protein Res. , vol.29 , pp. 574
- Van Der Auwera, C.¹ Anteunis, M.J.²

102
- 0024507836
- Jouin, P.; Poncet, J.; Dufour, M.-N.; Pantaloni, A.; Castro, B. J. Org. Chem. 1989, 54, 617.
- (1989) J. Org. Chem. , vol.54 , pp. 617
- Jouin, P.¹ Poncet, J.² Dufour, M.-N.³ Pantaloni, A.⁴ Castro, B.⁵

103
- 12044258245
- Carpino, L. A. J. Am. Chem. Soc. 1993, 115, 4397.
- (1993) J. Am. Chem. Soc. , vol.115 , pp. 4397
- Carpino, L.A.¹

104
- 37049086201
- Schmidt, U.; Griesser, H. J. Chem. Soc., Chem. Commun. 1993, 1461.
- (1993) J. Chem. Soc., Chem. Commun. , pp. 1461
- Schmidt, U.¹ Griesser, H.²

105
- 0025014627
- Coste, J.; Le-Nguyen, D.; Castro, B. Tetrahedron Lett. 1990, 31, 205.
- (1990) Tetrahedron Lett. , vol.31 , pp. 205
- Coste, J.¹ Le-Nguyen, D.² Castro, B.³

106
- 84988060670
- Anteunis, M. J. O.; Sharma, N. K. Bull. Soc. Chim. Belg. 1988, 97, 281.
- (1988) Bull. Soc. Chim. Belg. , vol.97 , pp. 281
- Anteunis, M.J.O.¹ Sharma, N.K.²

107
- 0027935320
- Angell, Y. M.; Garcia-Echeverria, C.; Rich, D. H. Tetrahedron Lett. 1994, 35, 5981.
- (1994) Tetrahedron Lett. , vol.35 , pp. 5981
- Angell, Y.M.¹ Garcia-Echeverria, C.² Rich, D.H.³

108
- 0025061710
- Colucci, W. J.; Tung, R. D.; Petri, J. A.; Rich, D. A. J. Org. Chem. 1990, 55, 2895.
- (1990) J. Org. Chem. , vol.55 , pp. 2895
- Colucci, W.J.¹ Tung, R.D.² Petri, J.A.³ Rich, D.A.⁴

109
- 0025819848
- Chu, K. S.; Negrete, G. R.; Konopelski, J. P. J. Org. Chem. 1991, 56, 5196.
- (1991) J. Org. Chem. , vol.56 , pp. 5196
- Chu, K.S.¹ Negrete, G.R.² Konopelski, J.P.³

110
- 0023759025
- Grieco, P. A.; Perez-Medrano, A. Tetrahedron Lett. 1988, 29, 4225.
- (1988) Tetrahedron Lett. , vol.29 , pp. 4225
- Grieco, P.A.¹ Perez-Medrano, A.²

111
- 0029144907
- Valentekovich, R. J.; Schreiber, S. L. J. Am. Chem. Soc. 1995, 117, 9069.
- (1995) J. Am. Chem. Soc. , vol.117 , pp. 9069
- Valentekovich, R.J.¹ Schreiber, S.L.²

112
- 33645672005
- White, J. D.; Amedio, J. C. J. Org. Chem. 1989, 54, 736.
- (1989) J. Org. Chem. , vol.54 , pp. 736
- White, J.D.¹ Amedio, J.C.²

113
- 37049102648
- Warnke, J. G.; Young, G. T. J. Chem. Soc., Perkin I 1980, 2797.
- (1980) J. Chem. Soc., Perkin I , pp. 2797
- Warnke, J.G.¹ Young, G.T.²

114
- 0023017976
- Tung, R. D.; Dhaon, M. K.; Rich, D. H. J. Org. Chem. 1986, 51, 3350.
- (1986) J. Org. Chem. , vol.51 , pp. 3350
- Tung, R.D.¹ Dhaon, M.K.² Rich, D.H.³

115
- 0011850124
- Diago-Meseguer, J.; Palomo-Col, A. L.; Fernandez-Lizarbe, J. R.; Zugaza-Bilbao, A. Synthesis 1980, 547.
- (1980) Synthesis , pp. 547
- Diago-Meseguer, J.¹ Palomo-Col, A.L.² Fernandez-Lizarbe, J.R.³ Zugaza-Bilbao, A.⁴

116
- 84989422133
- Van der Auwera, C.; Anteunis, M. J. Bull. Soc. Chim. Belg. 1986, 95, 203.
- (1986) Bull. Soc. Chim. Belg. , vol.95 , pp. 203
- Van Der Auwera, C.¹ Anteunis, M.J.²

117
- 85004733560
- Deber, C. M., Hruby, V. J., Kopple, K. D., Eds.; Pierce Chemical Co.: Rockford, IL
- Tung, R. D.; Rich, D. H. In Peptides: Structure and Function; Deber, C. M., Hruby, V. J., Kopple, K. D., Eds.; Pierce Chemical Co.: Rockford, IL, 1985; p 217.
- (1985) Peptides: Structure and Function , pp. 217
- Tung, R.D.¹ Rich, D.H.²

118
- 33845375891
- Carpino, L. A.; Cohen, B. J.; Stephens, K. E. J.; Sadat-Aalaee, S. Y.; Tien, J.-H.; Langridge, D. C. J. Org. Chem. 1986, 51, 3732.
- (1986) J. Org. Chem. , vol.51 , pp. 3732
- Carpino, L.A.¹ Cohen, B.J.² Stephens, K.E.J.³ Sadat-Aalaee, S.Y.⁴ Tien, J.-H.⁵ Langridge, D.C.⁶

119
- 84981962827
- Bechtolsheimer, H.-H.; Kunz, H. Angew Chem., Int. Ed. Engl. 1982, 21, 630.
- (1982) Angew Chem., Int. Ed. Engl. , vol.21 , pp. 630
- Bechtolsheimer, H.-H.¹ Kunz, H.²

120
- 84985216649
- Kunz, H.; Bechtolsheimer, H.-H. Liebigs Ann. Chem. 1982, 2068.
- (1982) Liebigs Ann. Chem. , pp. 2068
- Kunz, H.¹ Bechtolsheimer, H.-H.²

121
- 33751499095
- Carpino, L. A.; Chao, H. G.; Beyermann, M.; Bienert, M. J. Org. Chem. 1991, 2635.
- (1991) J. Org. Chem. , pp. 2635
- Carpino, L.A.¹ Chao, H.G.² Beyermann, M.³ Bienert, M.⁴

122
- 0028200949
- Sivanandaiah, K. M.; Suresh Babu, V. V.; Shankaramma, S. C. Int. J. Peptide Protein Res. 1994, 44, 24.
- (1994) Int. J. Peptide Protein Res. , vol.44 , pp. 24
- Sivanandaiah, K.M.¹ Suresh Babu, V.V.² Shankaramma, S.C.³

123
- 0023952266
- Galpin, I. J.; Mohammed, A. K. A.; Patel, A. Tetrahedron 1988, 44, 1783.
- (1988) Tetrahedron , vol.44 , pp. 1783
- Galpin, I.J.¹ Mohammed, A.K.A.² Patel, A.³

124
- 0003068305
- Castro, B.; Dormoy, J.-R. Tetrahedron Lett. 1973, 3243.
- (1973) Tetrahedron Lett. , pp. 3243
- Castro, B.¹ Dormoy, J.-R.²

125
- 0025057125
- Coste, J.; Dufour, M.-N.; Pantaloni, A.; Castro, B. Tetrahedron Lett. 1990, 31, 669.
- (1990) Tetrahedron Lett. , vol.31 , pp. 669
- Coste, J.¹ Dufour, M.-N.² Pantaloni, A.³ Castro, B.⁴

126
- 33845312505
- Carpino, L. A.; El-Faham, A.; Minor, C. A.; Albericio, F. J. Chem. Soc., Chem. Commun. 1994, 201.
- (1994) J. Chem. Soc., Chem. Commun. , pp. 201
- Carpino, L.A.¹ El-Faham, A.² Minor, C.A.³ Albericio, F.⁴

127
- 0028222937
- Carpino, L. A.; El-Faham, A.; Albericio, F. Tetrahedron Lett. 1994, 35, 2279.
- (1994) Tetrahedron Lett. , vol.35 , pp. 2279
- Carpino, L.A.¹ El-Faham, A.² Albericio, F.³

128
- 0028997484
- Carpino, L. A.; El-Faham, A. J. Org. Chem. 1995, 60, 3561.
- (1995) J. Org. Chem. , vol.60 , pp. 3561
- Carpino, L.A.¹ El-Faham, A.²

129
- 0029132233
- Kim, H.-O.; Gardner, B. G.; Kahn, M. Tetraherdon Lett. 1995, 36, 6013.
- (1995) Tetraherdon Lett. , vol.36 , pp. 6013
- Kim, H.-O.¹ Gardner, B.G.² Kahn, M.³

130
- 0024495619
- Hamada, Y.; Kondo, Y.; Shibata, M.; Shioiri, T. J. Am. Chem. Soc. 1989, 111, 669.
- (1989) J. Am. Chem. Soc. , vol.111 , pp. 669
- Hamada, Y.¹ Kondo, Y.² Shibata, M.³ Shioiri, T.⁴

131
- 0023939819
- Schmidt, U.; Kroner, M.; Griesser, H. Tetrahedron Lett. 1988, 29, 3057.
- (1988) Tetrahedron Lett. , vol.29 , pp. 3057
- Schmidt, U.¹ Kroner, M.² Griesser, H.³

132
- 0001686304
- Rinehart, K. L.; Kishore, V.; Nagarajan, S.; Lake, R. J.; Gloer, J. B.; Bozich, F. A.; Li, K. M.; Maleczka, R. E., Jr. Todsen, W. L.; Munro, M. H. G.; Sullins, D. W.; Sakai, R. J. Am. Chem. Soc. 1987, 109, 6846.
- (1987) J. Am. Chem. Soc. , vol.109 , pp. 6846
- Rinehart, K.L.¹ Kishore, V.² Nagarajan, S.³ Lake, R.J.⁴ Gloer, J.B.⁵ Bozich, F.A.⁶ Li, K.M.⁷ Maleczka Jr., R.E.⁸ Todsen, W.L.⁹ Munro, M.H.G.¹⁰ Sullins, D.W.¹¹ Sakai, R.¹²

133
- 0021681704
- Rodriguez, M.; Goodman, M. J. Med. Chem. 1984, 27, 1668.
- (1984) J. Med. Chem. , vol.27 , pp. 1668
- Rodriguez, M.¹ Goodman, M.²

134
- 0028825390
- Sammes, P. G.; Weller, D. J. Synthesis 1995, 1205.
- (1995) J. Synthesis , pp. 1205
- Sammes, P.G.¹ Weller, D.²

135
- 0013086552
- Nagaraj, R.; Balaram, P. Heterocycles 1977, 7, 885.
- (1977) Heterocycles , vol.7 , pp. 885
- Nagaraj, R.¹ Balaram, P.²

136
- 0019805456
- Balasubramanian, T. M.; Kendrick, N. C. E.; Taylor, M.; Marshall, G. R.; Hall, J. E.; Vodyanoy, I.; Reusser, F. J. Am. Chem. Soc. 1981, 103, 6127.
- (1981) J. Am. Chem. Soc. , vol.103 , pp. 6127
- Balasubramanian, T.M.¹ Kendrick, N.C.E.² Taylor, M.³ Marshall, G.R.⁴ Hall, J.E.⁵ Vodyanoy, I.⁶ Reusser, F.⁷

137
- 4243938924
- Bruckner, H.; König, W. A.; Greiner, M.; Günther, J. Angew. Chem. 1979, 91, 508.
- (1979) Angew. Chem. , vol.91 , pp. 508
- Bruckner, H.¹ König, W.A.² Greiner, M.³ Günther, J.⁴

138
- 0001947018
- Leplawy, M. T.; Jones, D. S.; Kenner, G. W.; Sheppard, R. C. Tetrahedron 1960, 11, 39.
- (1960) Tetrahedron , vol.11 , pp. 39
- Leplawy, M.T.¹ Jones, D.S.² Kenner, G.W.³ Sheppard, R.C.⁴

139
- 0025319387
- Wipf, P.; Heimgartner, H. Helv. Chim. Acta 1990, 73, 13.
- (1990) Helv. Chim. Acta , vol.73 , pp. 13
- Wipf, P.¹ Heimgartner, H.²

140
- 0000523261
- Leibfritz, D.; Haupt, E.; Dubischar, N.; Lachmann, H.; Oekonomopulos, R.; Jung, G. Tetrahedron 1982, 38, 2165.
- (1982) Tetrahedron , vol.38 , pp. 2165
- Leibfritz, D.¹ Haupt, E.² Dubischar, N.³ Lachmann, H.⁴ Oekonomopulos, R.⁵ Jung, G.⁶

141
- 0018612455
- Oekonomopulos, R.; Jung, G. Liebigs Ann. Chem. 1979, 1151.
- (1979) Liebigs Ann. Chem. , pp. 1151
- Oekonomopulos, R.¹ Jung, G.²

142
- 85004882387
- Gorecka, A.; Leplawy, M.; Zabrocki, J.; Zwierzak, A. Synthesis 1978, 474.
- (1978) Synthesis , pp. 474
- Gorecka, A.¹ Leplawy, M.² Zabrocki, J.³ Zwierzak, A.⁴

143
- 84981903937
- Schmidt, U.; Dietsche, M. Angew. Chem. Int. Ed. Engl. 1982, 27, 143.
- (1982) Angew. Chem. Int. Ed. Engl. , vol.27 , pp. 143
- Schmidt, U.¹ Dietsche, M.²

144
- 84987505863
- Obrecht, D.; Heimgartner, H. Helv. Chim. Acta 1987, 70, 102.
- (1987) Helv. Chim. Acta , vol.70 , pp. 102
- Obrecht, D.¹ Heimgartner, H.²

145
- 0026010908
- Frerot, E.; Coste, J.; Pantaloni, A.; Dufour, M.-N.; Jouin, P. Tetrahedron 1991, 47, 259.
- (1991) Tetrahedron , vol.47 , pp. 259
- Frerot, E.¹ Coste, J.² Pantaloni, A.³ Dufour, M.-N.⁴ Jouin, P.⁵

146
- 0027481339
- Auvin-Guette, C.; Frérot, E.; Coste, J.; Rebuffat, S.; Jouin, P.; Bodo, B. Tetrahedron Lett. 1993, 34, 2481.
- (1993) Tetrahedron Lett. , vol.34 , pp. 2481
- Auvin-Guette, C.¹ Frérot, E.² Coste, J.³ Rebuffat, S.⁴ Jouin, P.⁵ Bodo, B.⁶

147
- 0026498006
- Walker, M. A.; Heathcock, C. H. J. Org. Chem. 1992, 57, 5566.
- (1992) J. Org. Chem. , vol.57 , pp. 5566
- Walker, M.A.¹ Heathcock, C.H.²

148
- 84987593553
- Wipf, P.; Heimgartner, H. Helv. Chim. Acta 1986, 69, 1153.
- (1986) Helv. Chim. Acta , vol.69 , pp. 1153
- Wipf, P.¹ Heimgartner, H.²

149
- 0030575426
- Barton, D. H.; Ferreira, J. A. Tetrahedron 1996, 52, 9367.
- (1996) Tetrahedron , vol.52 , pp. 9367
- Barton, D.H.¹ Ferreira, J.A.²

150
- 0000791684
- Saha, A. K.; Schultz, P.; Rapoport, H. J. Am. Chem. Soc. 1989, 111, 4857.
- (1989) J. Am. Chem. Soc. , vol.111 , pp. 4857
- Saha, A.K.¹ Schultz, P.² Rapoport, H.³

151
- 0026473072
- Spencer, J. R.; Antonenko, V. V.; Delaet, N. G. J.; Goodman, M. Int. J. Peptide Protein Res. 1992, 40, 282.
- (1992) Int. J. Peptide Protein Res. , vol.40 , pp. 282
- Spencer, J.R.¹ Antonenko, V.V.² Delaet, N.G.J.³ Goodman, M.⁴

152
- 0000528761
- Wenschuh, H.; Beyermann, M.; Krause, E.; Brudel, M.; Winter, R.; Schumann, M.; Carpino, L. A.; Bienert, M. J. Org. Chem. 1994, 59, 3275.
- (1994) J. Org. Chem. , vol.59 , pp. 3275
- Wenschuh, H.¹ Beyermann, M.² Krause, E.³ Brudel, M.⁴ Winter, R.⁵ Schumann, M.⁶ Carpino, L.A.⁷ Bienert, M.⁸

153
- 0012370877
- Kopple, K. D. J. Am. Chem. Soc. 1957, 79, 662.
- (1957) J. Am. Chem. Soc. , vol.79 , pp. 662
- Kopple, K.D.¹

154
- 0000589494
- Carpino, L. A.; Beyermann, M.; Wenschuh, H.; Bienert, M. Acc. Chem. Res. 1996, 29, 268.
- (1996) Acc. Chem. Res. , vol.29 , pp. 268
- Carpino, L.A.¹ Beyermann, M.² Wenschuh, H.³ Bienert, M.⁴

155
- 33751498929
- Carpino, L. A.; Mansour, E.-S. M. E.; Sadat-Aalaee, D. J. Org. Chem. 1991, 56, 2611.
- (1991) J. Org. Chem. , vol.56 , pp. 2611
- Carpino, L.A.¹ Mansour, E.-S.M.E.² Sadat-Aalaee, D.³

156
- 0025671995
- Carpino, L. A.; Sadat-Aalaee, D.; Chao, H. G.; DeSelms, R. H. J. Am. Chem. Soc. 1990, 112, 9651.
- (1990) J. Am. Chem. Soc. , vol.112 , pp. 9651
- Carpino, L.A.¹ Sadat-Aalaee, D.² Chao, H.G.³ DeSelms, R.H.⁴

157
- 37049076980
- Wenshuh, H.; Beyermann, M.; El-Faham, A.; Ghassemi, S.; Carpino, L. A. J. Chem. Soc., Chem. Commun. 1995, 669.
- (1995) J. Chem. Soc., Chem. Commun. , pp. 669
- Wenshuh, H.¹ Beyermann, M.² El-Faham, A.³ Ghassemi, S.⁴ Carpino, L.A.⁵

158
- 0001201464
- Rajeswari, S.; Jones, R. J.; Cava, M. P. Tetrahedron Lett. 1987, 28, 5099.
- (1987) Tetrahedron Lett. , vol.28 , pp. 5099
- Rajeswari, S.¹ Jones, R.J.² Cava, M.P.³

159
- 0027068161
- For efficient Fmoc amino acid fluoride-induced acylations of aromatic amines without BTSA activation, see: Bunin, B. A.; Ellman, J. A. J. Am. Chem. Soc. 1992, 114, 10997.
- (1992) J. Am. Chem. Soc. , vol.114 , pp. 10997
- Bunin, B.A.¹ Ellman, J.A.²

160
- 0027243640
- Wenschuh, H.; Beyermann, E.; Krause, E.; Carpino, L. A.; Bienert, M. Tetrahedron Lett. 1993, 34, 3733.
- (1993) Tetrahedron Lett. , vol.34 , pp. 3733
- Wenschuh, H.¹ Beyermann, E.² Krause, E.³ Carpino, L.A.⁴ Bienert, M.⁵

161
- 37049076980
- Wenschuh, H.; Beyermann, M.; El-Faham, A.; Chassemi, S.; Carpino, L. A.; Bienert, M. J. Chem. Soc., Chem. Commun. 1995, 669.
- (1995) J. Chem. Soc., Chem. Commun. , pp. 669
- Wenschuh, H.¹ Beyermann, M.² El-Faham, A.³ Chassemi, S.⁴ Carpino, L.A.⁵ Bienert, M.⁶

162
- 85015356069
- Olah, G. A. Synthesis 1973, 487.
- (1973) Synthesis , pp. 487
- Olah, G.A.¹

163
- 33846323284
- Kaduk, C.; Wenschuh, H.; Beyermann, M.; Forner, K.; Carpino, L. A.; Bienert, M. Lett. Peptide Sci. 1996, 2, 285.
- (1996) Lett. Peptide Sci. , vol.2 , pp. 285
- Kaduk, C.¹ Wenschuh, H.² Beyermann, M.³ Forner, K.⁴ Carpino, L.A.⁵ Bienert, M.⁶

164
- 0029109071
- Carpino, L. A.; El-Faham, A. J. Am. Chem. Soc. 1995, 117, 5401.
- (1995) J. Am. Chem. Soc. , vol.117 , pp. 5401
- Carpino, L.A.¹ El-Faham, A.²

165
- 0026645155
- Akaji, K.; Kuriyama, N.; Kimura, T.; Fujiwara, Y.; Kiso, Y. Tetrahedron Lett. 1992, 33, 3177.
- (1992) Tetrahedron Lett. , vol.33 , pp. 3177
- Akaji, K.¹ Kuriyama, N.² Kimura, T.³ Fujiwara, Y.⁴ Kiso, Y.⁵

166
- 0029891170
- Akaji, K.; Kuriyama, N.; Kiso, Y. J. Org. Chem. 1996, 61, 3350.
- (1996) J. Org. Chem. , vol.61 , pp. 3350
- Akaji, K.¹ Kuriyama, N.² Kiso, Y.³

167
- 0028298856
- Akaji, K.; Kuriyama, N.; Kiso, Y. Tetrahedron Lett. 1994, 35, 3315.
- (1994) Tetrahedron Lett. , vol.35 , pp. 3315
- Akaji, K.¹ Kuriyama, N.² Kiso, Y.³

168
- 0011402882
- Love, A. L.; Olsen, R. K. J. Org. Chem. 1972, 37, 3431.
- (1972) J. Org. Chem. , vol.37 , pp. 3431
- Love, A.L.¹ Olsen, R.K.²

169
- 0017308856
- Breitholle, E. G.; Stammer, C. H. J. Org. Chem. 1976, 41, 1344.
- (1976) J. Org. Chem. , vol.41 , pp. 1344
- Breitholle, E.G.¹ Stammer, C.H.²

170
- 0020445340
- Botes, D. P.; Viljoen, C. C.; Kruger, H.; Wessels, P. L.; Williams, D. H. Toxicon 1982, 20, 1037.
- (1982) Toxicon , vol.20 , pp. 1037
- Botes, D.P.¹ Viljoen, C.C.² Kruger, H.³ Wessels, P.L.⁴ Williams, D.H.⁵

171
- 0019982027
- Noda, K.; Gazis, D.; Gross, E. Int. J. Peptide Protein Res. 1982, 19, 413.
- (1982) Int. J. Peptide Protein Res. , vol.19 , pp. 413
- Noda, K.¹ Gazis, D.² Gross, E.³

172
- 0343480851
- Rich, D. H.; Tam, J.; Mathiaparanam, P.; Grant, J. A. Synthesis 1975, 402.
- (1975) Synthesis , pp. 402
- Rich, D.H.¹ Tam, J.² Mathiaparanam, P.³ Grant, J.A.⁴

173
- 0001023731
- McDermott, J. R.; Benoiton, N. L. Can. J. Chem. 1973, 51, 1915.
- (1973) Can. J. Chem. , vol.51 , pp. 1915
- McDermott, J.R.¹ Benoiton, N.L.²

174
- 0041080930
- Academic Press: New York-London
- Schröder, E.; Lübke, K. The Peptides; Academic Press: New York-London, 1965.
- (1965) The Peptides
- Schröder, E.¹ Lübke, K.²

175
- 0017783272
- Rich, D. H.; Tam, J. P. J. Org. Chem. 1977, 42, 3815.
- (1977) J. Org. Chem. , vol.42 , pp. 3815
- Rich, D.H.¹ Tam, J.P.²

176
- 0029959471
- Humphrey, J. M.; Aggen, J. B.; Chamberlin, A. R. J. Am. Chem. Soc. 1996, 118, 11759.
- (1996) J. Am. Chem. Soc. , vol.118 , pp. 11759
- Humphrey, J.M.¹ Aggen, J.B.² Chamberlin, A.R.³

177
- 55549083919
- Williams, M. W.; Young, G. T. J. Chem. Soc. 1963, 881.
- (1963) J. Chem. Soc. , pp. 881
- Williams, M.W.¹ Young, G.T.²

178
- 0026464897
- Poulos, C.; Ashton, C. P.; Green, J.; Ogunjobi, O. M.; Ramage, R.; Tsegenidis, T. Int. J. Peptide Protein Res. 1992, 40, 315.
- (1992) Int. J. Peptide Protein Res. , vol.40 , pp. 315
- Poulos, C.¹ Ashton, C.P.² Green, J.³ Ogunjobi, O.M.⁴ Ramage, R.⁵ Tsegenidis, T.⁶

179
- 0027373903
- For a review on solid-phase peptide synthesis, see: Lloyd-Williams, P.; Albericio, F.; Giralt, E. Tetrahedron 1993, 49, 11065.
- (1993) Tetrahedron , vol.49 , pp. 11065
- Lloyd-Williams, P.¹ Albericio, F.² Giralt, E.³

180
- 0031012514
- Akaji, K.; Tamai, Y.; Kiso, Y. Tetrahedron 1997, 53, 567.
- (1997) Tetrahedron , vol.53 , pp. 567
- Akaji, K.¹ Tamai, Y.² Kiso, Y.³

181
- 0021341035
- Wenger, R. M. Helv. Chim. Acta 1984, 67, 502.
- (1984) Helv. Chim. Acta , vol.67 , pp. 502
- Wenger, R.M.¹

182
- 0023831121
- Grieco, P. A.; Hon, Y. S.; Perez-Medrano, A. J. Am. Chem. Soc. 1988, 110, 1630.
- (1988) J. Am. Chem. Soc. , vol.110 , pp. 1630
- Grieco, P.A.¹ Hon, Y.S.² Perez-Medrano, A.³

183
- 33751158654
- Carpino, L. A.; El-Faham, A. J. Org. Chem. 1994, 59, 695.
- (1994) J. Org. Chem. , vol.59 , pp. 695
- Carpino, L.A.¹ El-Faham, A.²

184
- 0001271559
- Ho, G.-J.; Emerson, K. M.; Mathre, D. J.; Shuman, R. F.; Grabowski, E. J. J. J. Org. Chem. 1995, 60, 3569.
- (1995) J. Org. Chem. , vol.60 , pp. 3569
- Ho, G.-J.¹ Emerson, K.M.² Mathre, D.J.³ Shuman, R.F.⁴ Grabowski, E.J.J.⁵

185
- 0027244347
- Ehrlich, A.; Rothemund, S.; Brudel, M.; Beyermann, M.; Carpino, L. A.; Bienert, M. Tetrahedron Lett. 1993, 34, 4781.
- (1993) Tetrahedron Lett. , vol.34 , pp. 4781
- Ehrlich, A.¹ Rothemund, S.² Brudel, M.³ Beyermann, M.⁴ Carpino, L.A.⁵ Bienert, M.⁶

186
- 0001625501
- Kopple, K. D. J. Pharm. Sci. 1972, 61, 1345.
- (1972) J. Pharm. Sci. , vol.61 , pp. 1345
- Kopple, K.D.¹

187
- 0345263290
- Walter-de Gruyter: Berlin-New York
- Ovichinikov, Y.; Chipens, G.; Ivanov, V. In Peptides 1982; Walter-de Gruyter: Berlin-New York, 1983; p 1.
- (1983) Peptides 1982 , pp. 1
- Ovichinikov, Y.¹ Chipens, G.² Ivanov, V.³

188
- 0000477615
- Cavelier-Frontin, F.; Pépe, G.; Verducci, J.; Siri, D.; Jacquier, R. J. Am. Chem. Soc. 1992, 14, 8885.
- (1992) J. Am. Chem. Soc. , vol.14 , pp. 8885
- Cavelier-Frontin, F.¹ Pépe, G.² Verducci, J.³ Siri, D.⁴ Jacquier, R.⁵

189
- 8344231040
- Weber, E., Vögtle, F., Eds.; Springer-Verlag: Berlin Heidelberg
- Meng, Q.; Hesse, M. In Topics in Current Chemistry; Weber, E., Vögtle, F., Eds.; Springer-Verlag: Berlin Heidelberg, 1992; p 161.
- (1992) Topics in Current Chemistry , pp. 161
- Meng, Q.¹ Hesse, M.²

190
- 0030470879
- Ehrlich, A.; Heyne, H.-U.; Winter, R.; Beyermann, M.; Haber, H.; Carpino, L. A.; Bienert, M. J. Org. Chem. 1996, 61, 8831.
- (1996) J. Org. Chem. , vol.61 , pp. 8831
- Ehrlich, A.¹ Heyne, H.-U.² Winter, R.³ Beyermann, M.⁴ Haber, H.⁵ Carpino, L.A.⁶ Bienert, M.⁷

191
- 33845560832
- Brady, S. F.; Varga, S. L.; Freidinger, R. M.; Schwenk, D. A.; Mendlowski, M.; Holly, F. W.; Veber, D. F. J. Org. Chem. 1979, 44, 3101.
- (1979) J. Org. Chem. , vol.44 , pp. 3101
- Brady, S.F.¹ Varga, S.L.² Freidinger, R.M.³ Schwenk, D.A.⁴ Mendlowski, M.⁵ Holly, F.W.⁶ Veber, D.F.⁷

192
- 0022904036
- Edwards, J. V.; Lax, A. R.; Lillehoj, E. B.; Boudreaux, G. J. Int. J. Peptide Protein Res. 1986, 28, 603.
- (1986) Int. J. Peptide Protein Res. , vol.28 , pp. 603
- Edwards, J.V.¹ Lax, A.R.² Lillehoj, E.B.³ Boudreaux, G.J.⁴

193
- 0024546922
- Schmidt, U.; Beutler, U.; Lieberknecht, A. Angew. Chem., Int. Ed. Engl. 1989, 28, 333.
- (1989) Angew. Chem., Int. Ed. Engl. , vol.28 , pp. 333
- Schmidt, U.¹ Beutler, U.² Lieberknecht, A.³

194
- 84985520817
- Schmidt, U.; Lieberknecht, A.; Griesser, H.; Häusler, J. Angew. Chem., Int. Ed. Engl. 1981, 20, 281.
- (1981) Angew. Chem., Int. Ed. Engl. , vol.20 , pp. 281
- Schmidt, U.¹ Lieberknecht, A.² Griesser, H.³ Häusler, J.⁴

195
- 0021255704
- Schmidt, U.; Lieberknecht, A.; Griesser, H.; Bartkowiak, F. Angew. Chem., Int. Ed. Engl. 1984, 23, 318.
- (1984) Angew. Chem., Int. Ed. Engl. , vol.23 , pp. 318
- Schmidt, U.¹ Lieberknecht, A.² Griesser, H.³ Bartkowiak, F.⁴

196
- 0027218805
- Baldwin, J. E.; Adlington, R. M.; Godfrey, C. R.; Patel, V. K. Tetrahedron 1993, 49, 7837.
- (1993) Tetrahedron , vol.49 , pp. 7837
- Baldwin, J.E.¹ Adlington, R.M.² Godfrey, C.R.³ Patel, V.K.⁴

197
- 0029795991
- Tounton, J.; Collins, J. L.; Schreiber, S. L. J. Am. Chem. Soc. 1996, 118, 10412.
- (1996) J. Am. Chem. Soc. , vol.118 , pp. 10412
- Tounton, J.¹ Collins, J.L.² Schreiber, S.L.³

198
- 33845378280
- Boden, E. P.; Keck, G. E. J. Org. Chem. 1985, 50, 2394.
- (1985) J. Org. Chem. , vol.50 , pp. 2394
- Boden, E.P.¹ Keck, G.E.²

199
- 0027931069
- Ishiwata, H.; Sone, H.; Kigoshi, H.; Yamada, K. J. Org. Chem. 1994, 59, 4712.
- (1994) J. Org. Chem. , vol.59 , pp. 4712
- Ishiwata, H.¹ Sone, H.² Kigoshi, H.³ Yamada, K.⁴

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