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0028222149
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(a) Vacca, J. P.; Dorsey, B. D.; Schleif, W. A.; Levin, R. B.; McDaniel, S. L.; Darke, P. L.; Zugay, J.; Quintero, J. C.; Blahy, O. M.; Roth, E.; Sardana, V. V.; Schlabach, A. J.; Graham, P. I.; Condra, J. H.; Gotlib, L.; Holloway, M. K.; Lin, J.; Chen, I.-W.; Vastag, K.; Ostovic, D.; Anderson, P. S.; Emini, E. A.; Huff, J. R. Proc. Natl. Acad. Sci. USA, 1994, 91, 4096.
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Dorsey, B.D.2
Schleif, W.A.3
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Zugay, J.7
Quintero, J.C.8
Blahy, O.M.9
Roth, E.10
Sardana, V.V.11
Schlabach, A.J.12
Graham, P.I.13
Condra, J.H.14
Gotlib, L.15
Holloway, M.K.16
Lin, J.17
Chen, I.-W.18
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Ostovic, D.20
Anderson, P.S.21
Emini, E.A.22
Huff, J.R.23
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2
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0027969994
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(b) Vacca, J. P.; Dorsey, B. D.; Schleif, W. A.; Levin, R. B.; McDaniel, S. L.; Darke, P. L.; Zugay, J.; Quintero, J. C.; Blahy, O. M.; Roth, E.; Sardana, V. V.; Schlabach, A. J.; Graham, P. I.; Condra, J. H.; Gotlib, L.; Holloway, M. K.; Lin, J.; Chen, I.-W.; Vastag, K.; Ostovic, D.; Anderson, P. S.; Emini, E. A.; Huff, J. R. Idem., J. Med. Chem. 1994, 37, 3443, and references cited therein.
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Schleif, W.A.3
Levin, R.B.4
McDaniel, S.L.5
Darke, P.L.6
Zugay, J.7
Quintero, J.C.8
Blahy, O.M.9
Roth, E.10
Sardana, V.V.11
Schlabach, A.J.12
Graham, P.I.13
Condra, J.H.14
Gotlib, L.15
Holloway, M.K.16
Lin, J.17
Chen, I.-W.18
Vastag, K.19
Ostovic, D.20
Anderson, P.S.21
Emini, E.A.22
Huff, J.R.23
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3
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0030051486
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(a) Davies, I. W.; Senanayake, C. H.; Larsen, R. D.; Verhoeven, T. R.; Reider, P. J. Tetrahedron Lett. 1996, 37, 813.
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Davies, I.W.1
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(b) Hong, Y.; Gao, Y.; Nie, X.; Zepp, C. M. Tetrahedron Lett. 1994, 35, 6631.
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Hong, Y.1
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(c) Simone, B. D.; Savoia, D.; Tagliavini, E.; Umani-Ronchi, A. Tetrahedron: Asymmetry 1995, 6, 301.
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Simone, B.D.1
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8
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0028840495
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(c) Davies, I.W.; Senanayake, C. H.; Castonguay, L.; Larsen, R. D.; Verhoeven, T. R.; Reider, P. J. Tetrahedron Lett. 1995, 36, 7619.
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11
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0031005924
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Zheng, N.1
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Volante, R.P.4
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12
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0025910637
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Synthesis of cis-aminoindanol is seen in: (a) Didier, E.; Loubinoux, B.; Tombo, G. M. R.; Rihs, G. Tetrahedron 1991, 47, 4941.
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(1991)
Tetrahedron
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Didier, E.1
Loubinoux, B.2
Tombo, G.M.R.3
Rihs, G.4
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13
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0028147531
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(b) Askin, D.; Eng, K. K.; Rossen. K.; Purick, R. M.; Wells, K. M.; Volante, R. P.; Reider, P. J. Tetrahedron Lett. 1994, 35, 673.
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Askin, D.1
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Volante, R.P.6
Reider, P.J.7
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14
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0028787044
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(c) Senanayake, C. H.; DiMichele, Liu, J.; Fredenburgh, L. E.; Ryan, K. M.; Roberts, F. E.; Larsen, R. D.; Verhoeven, T. R.; Reider, P. J. Tetrahedron Lett. 1995, 36, 7615.
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Senanayake, C.H.1
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Larsen, R.D.6
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18
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0013573601
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JP Patent 96-228586
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Oda, Y.; Yuasa, M. JP Patent 96-228586, Chem. Abstr. 124 : 145646.
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Oda, Y.1
Yuasa, M.2
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20
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26844466833
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note
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Ee was determined by HPLC (DAICEL CHIRALCEL OB analytical column (0.46 mm, 25 cm)) analysis after conversion to the corresponding methyl ester using trimethylsilyldiazomethane.
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22
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0343009106
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(a) McClure, D. E.; Arison, B. H.; Jones, J. H.; Baldwin, J. J. J. Org. Chem. 1981, 46, 2431.
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McClure, D.E.1
Arison, B.H.2
Jones, J.H.3
Baldwin, J.J.4
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24
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0000059212
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(c) Nguy, N. M.; Chiu, I. -C.; Kohn, H. J. Org. Chem. 1987, 52, 1649.
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Nguy, N.M.1
Chiu, I.-C.2
Kohn, H.3
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25
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85088545676
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note
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D = -19 (c 1.0, MeOH).
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29
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85088547100
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note
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3 (65%) exhibit relatively good yield after 24 h.
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30
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85088546684
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note
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3): See ref 6.
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32
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85064667331
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3 in aqueous media is seen in (b) Kobayashi, S. Synlett 1994, 689, and references cited therein.
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(1994)
Synlett
, pp. 689
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Kobayashi, S.1
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33
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0012615648
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(a) Ishihara, K.; Kubota, M.; Kurihara, H.; Yamamoto, H. J. Org. Chem. 1996, 61, 4560.
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Ishihara, K.1
Kubota, M.2
Kurihara, H.3
Yamamoto, H.4
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34
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0029862760
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(b) Shull, B. K.; Sakai, T.; Koreeda, M. J. Am. Chem. Soc. 1996, 118, 11690.
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Shull, B.K.1
Sakai, T.2
Koreeda, M.3
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35
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85061411950
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(c) Yanada, R.; Negoro, N.; Bessho, K.; Yanada, K. Synlett, 1995, 1261.
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(1995)
Synlett
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Yanada, R.1
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Yanada, K.4
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36
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0002693163
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(d) Inanaga, J.; Yokoyama, Y.; Hanamoto, T. J. Chem. Soc., Chem. Commun. 1993, 1090, and references cited therein.
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Inanaga, J.1
Yokoyama, Y.2
Hanamoto, T.3
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37
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26844543218
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note
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The geometry of 9 was determined by NOE experiments after conversion to 2-acetoxy-1-acetoxyiminoindanone.
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38
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85088545997
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note
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Rs observed at a flow rate of 0.5 mL·min-1 were as follows: 14.7 min (R-form), 20.2 min (S-form). Analysis of Z-9 was performed by DAICEL CHIRALPAK AD analytical column (0.46 mm, 25 cm) with 14% 2-propanol in hexane as an eluent.
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39
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0029058104
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(a) Tillyer, R. D.; Boudreau, C.; Tschaen, D.; Dolling, U. -H.; Reider, P. J. Tetrahedron Lett. 1995, 36, 4337.
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Tetrahedron Lett.
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Tillyer, R.D.1
Boudreau, C.2
Tschaen, D.3
Dolling, U.-H.4
Reider, P.J.5
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41
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0014540187
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(c) Rimek, H. -J.; Yupraphat, T.; Zymalkowsky, F. Liebigs Ann. Chem. 1969, 725, 116.
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Liebigs Ann. Chem.
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Rimek, H.-J.1
Yupraphat, T.2
Zymalkowsky, F.3
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42
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26844500229
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(d) Ghosh, A. K.; McKee, S. P.; Sanders, W. M. Tetrahedron Lett. 1991, 32, 111.
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(1991)
Tetrahedron Lett.
, vol.32
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Ghosh, A.K.1
McKee, S.P.2
Sanders, W.M.3
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43
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0000212545
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(e) Desimoni, G.; Faita, G.; Mellerio, G.; Righetti, P. P.; Zanelli, C. Gazz. Chim. Ital. 1992, 122, 269.
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Gazz. Chim. Ital.
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Desimoni, G.1
Faita, G.2
Mellerio, G.3
Righetti, P.P.4
Zanelli, C.5
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44
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0007600557
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(f) Huebner, C. F.; Donoghue, E. M.; Novak, C. J.; Dorfman, L.; Wenkert, E. J. Org. Chem. 1970, 35, 1149.
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Huebner, C.F.1
Donoghue, E.M.2
Novak, C.J.3
Dorfman, L.4
Wenkert, E.5
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45
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26844554832
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JP Patent 95-242614
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(g) Oda, Y.; Yuasa, M. JP Patent 95-242614, Chem. Abstr. 124 : 55593.
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Chem. Abstr.
, vol.124
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-
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Oda, Y.1
Yuasa, M.2
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46
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85088546817
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note
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2, 82%, and 28%; Ir black, 89%, and 31%, and Rh black, 75%, and 33%.
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-
-
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47
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26844480594
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note
-
Even when the E- or Z-isomer was used respectively as a substrate, the ratio of cis and trans did not change, as might be expected on the basis of the isomerization experiment in an acidic solution.
-
-
-
-
48
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85088547169
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note
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4 aq. (pH 2).
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