Condensation of 2-amino-5-chlorobenzoxazole with α-bromoketones: A mechanistic study

Heterocycles

Volumn 45, Issue 11, 1997, Pages 2239-2246

  Roy, Patrick J ^a   Landry, Kerri ^a   Leblanc, Yves ^a   Li, Chun ^a   Tsou, Nancy ^b  

^a MERCK FROSST CENTRE FOR THERAPEUTIC RESEARCH   (Canada)

^b MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0000634382     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/com-97-7861     Document Type: Article

References (9)

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2. J. P. Paolini in 'Chemistry of Heterocyclic Compounds,' Vol. 30, ed. by A. Wiessberger and E. C. Taylor, John Wiley and Sons, Inc., New York, 1977, p. 11.
3. Crystallographic details to be submitted for publication in Acta Crystallographica C (N. Tsou, R. Ball, P. Roy, and Y. Leblanc)
4. L. M. Werbel and M.L. Zamora, J. Heterocycl. Chem., 1965, 2, 287.
5. 18O
6. 18O
7. H. Bredereck, F. Effenberger, F. Marquez, and K. Ockewitz, Chem. Ber., 1960, 93, 2083.
8. J. Y. Gauthier, C. K. Lau, P. Roy, M. Thérien, and Z. Wang, US Patent 5,552,422 (1996) (Chem. Abstr.,1996, 125, 195659b).
9. Y. Leblanc, J. Y. Gauthier, D. Ethier, J. Guay, J. Mancini, D. Riendeau, P. Tagari, P. Vickers, E. Wong, and P. Prasit, Biorg. Med. Chem. Lett., 1995, 5, 2123.