Effect of the hydrophobic nature of triacetyl-β-cyclodextrin on the complexation with nicardipine hydrochloride: Physicochemical and dissolution properties of the kneaded and spray-dried complexes

Chemical and Pharmaceutical Bulletin

Volumn 50, Issue 12, 2002, Pages 1597-1602

  Fernandes, Catarina Marques ^a   Veiga, Francisco José Baptista ^a  

^a UNIVERSITY OF COIMBRA   (Portugal)

Author keywords

Kneading; Nicardipine; Spray drying; Sustained release; Triacetyl cyclodextrin

Indexed keywords

CYCLODEXTRIN DERIVATIVE; NICARDIPINE; TRIACETYL BETA CYCLODEXTRIN; UNCLASSIFIED DRUG; BETA CYCLODEXTRIN DERIVATIVE; CYCLODEXTRIN; TRIACETYL-BETA-CYCLODEXTRIN;

ACIDITY; ARTICLE; COMPARATIVE STUDY; COMPLEX FORMATION; DIFFERENTIAL SCANNING CALORIMETRY; DRUG EFFECT; DRUG SOLUBILITY; HYDROPHOBICITY; IN VITRO STUDY; INFRARED SPECTROSCOPY; INTESTINE FLUID; MODEL; PHARMACEUTICAL ENGINEERING; PHYSICAL CHEMISTRY; SCANNING ELECTRON MICROSCOPY; SOLID STATE; SPRAY DRYING; STATISTICAL SIGNIFICANCE; STOMACH PH; SUSTAINED DRUG RELEASE; TECHNIQUE; UNITED STATES; X RAY DIFFRACTION; CHEMISTRY; DELAYED RELEASE FORMULATION; DRUG FORMULATION; METHODOLOGY; PH; SOLUBILITY; SURFACE PROPERTY;

BETA-CYCLODEXTRINS; CALORIMETRY, DIFFERENTIAL SCANNING; CYCLODEXTRINS; DELAYED-ACTION PREPARATIONS; DRUG COMPOUNDING; HYDROGEN-ION CONCENTRATION; HYDROPHOBICITY; MICROSCOPY, ELECTRON, SCANNING; NICARDIPINE; SOLUBILITY; SPECTROSCOPY, FOURIER TRANSFORM INFRARED; SURFACE PROPERTIES; X-RAY DIFFRACTION;

EID: 0000566128     PISSN: 00092363     EISSN: 13475223     Source Type: Journal    
DOI: 10.1248/cpb.50.1597     Document Type: Article

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