Organoiodine (III) mediated synthesis of 3-aryl/hetryl-5,7-dimethyl-1,2,4- triazolo[4,3-a]pyrimidines as antibacterial agents

European Journal of Medicinal Chemistry

Volumn 39, Issue 12, 2004, Pages 1073-1077

  Prakash, Om ^a   Bhardwaj, Vikas ^a   Kumar, Ravi ^a   Tyagi, Parikshit ^a   Aneja, Kamal R ^a  

^a KURUKSHETRA UNIVERSITY   (India)

Author keywords

Antibacterial activity; Iodobenzene diacetate; Triazolopyrimidines

Indexed keywords

3 (3',4' DIMETHOXYPHENYL) 5,7 DIMETHYL 1,2,4 TRIAZOLO[4,3 A]PYRIMIDINE; 3 (4' PYRIDYL) 5,7 DIMETHYL 1,2,4 TRIAZOLO[4,3 A]PYRIMIDINE; AMPICILLIN; ANTIINFECTIVE AGENT; CHLORAMPHENICOL; CIPROFLOXACIN; PYRIMIDINE DERIVATIVE; STREPTOMYCIN; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACILLUS SUBTILIS; CONTROLLED STUDY; DRUG SYNTHESIS; ESCHERICHIA COLI; IN VITRO STUDY; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; OXIDATION; SALMONELLA TYPHI; STAPHYLOCOCCUS AUREUS;

ANTI-BACTERIAL AGENTS; BACILLUS SUBTILIS; CATALYSIS; ESCHERICHIA COLI; IODOBENZENES; PYRIMIDINES; SALMONELLA TYPHI; STAPHYLOCOCCUS AUREUS; TRIAZOLES;

EID: 9644265233     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejmech.2004.06.011     Document Type: Article

References (19)

1. Deshmukh A.A., Mody M.K., Ramalingam T., and Sattur P.B. Indian J. Chem. 23B 1984 793
2. Loye B., Musser J.H., Brown R.E., Jones H., Kahenan R., Huang Fu.Ch., Khandwala A., Sonnio-Goldman P., and Leibowitz M.J. J. Med. Chem. 28 1985 363
3. Hiremath S.P., Ullagaddi A., Shivaramayya K., and Purohit M.G. Indian J. Heterocycl. Chem. 3 1999 145
4. Gupta R., Gupta A.K., Paul S., and Kachroo P.L. Indian J. Chem. 37B 1998 1211
5. Moriarty R.M., Vaid R.K., and Koser G.F. Synlett. 1990 365 383
6. Prakash O., Saini N., and Sharma P.K. Heterocycles 38 1994 409
7. Prakash O. Aldrichimica Acta 28 1995 63 71
8. Varvoglis A. Hypervalent Iodine in Organic Synthesis 1997 Academic press London
9. Moriarty R.M., and Prakash O. Adv. Heterocycl. Chem. 69 1998 1
10. Ochiai M. Akibia K. Chemistry of Hypervalent Compounds 1999 VCH Publishers New York 359 387 (Chapter 13)
11. Koser G.F. Aldrichimica Acta 34 2002 89 102
12. Moriarty R.M., and Prakash O. Oxidation of phenolic compounds with organohypervalent iodine reagents Overman L.E. Organic Reactions 57 2001 John Wiley & Sons Inc 327 415
13. Zhdankin V.V., and Stang P.J. Chem. Rev. 102 2002 2523 2584
14. Prakash O., Batra H., Sharma V., and Singh S.P. Indian J. Chem. 37B 1998 583 584
15. Sadana A.K., Mirza Y., Aneja K.R., and Prakash O. Eur. J. Med. Chem. 38 2003 533 536
16. Prakash O., Kaur H., Batra H., Rani N., and Singh S.P. Synthetic Commun. 30 2000 417
17. Kosolapoff G.M., and Roy C.H. J. Org. Chem. 26 1961 1895
18. Fabbrini L. Guzz. Chim. Ital. 87 1957 1293 1302 (Univ. Florence)
19. Vanderhaeghe H., and Claesen M. Bull. Soc. Chim. Belg. 68 1959 30 46 (Univ. Louvain)