Optimization of pyrrolidinone based HIV protease inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 1, 2005, Pages 81-84

  Sherrill, Ronald G ^a   Andrews, C Webster ^a   Bock, William J ^a   Davis Ward, Ronda G ^a   Furfine, Eric S ^a   Hazen, Richard J ^a   Rutkowske, Randy D ^a   Spaltenstein, Andrew ^a   Wright, Lois L ^a  

^a GLAXOSMITHKLINE   (United States)

Author keywords

HIV protease inhibitors

Indexed keywords

2 PYRROLIDONE DERIVATIVE; AMPRENAVIR; PROTEINASE INHIBITOR;

ALKYLATION; ANTIVIRAL ACTIVITY; ARTICLE; HIGHLY ACTIVE ANTIRETROVIRAL THERAPY; HYDROGENATION; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; REDUCTION; X RAY DIFFRACTION;

HIV PROTEASE INHIBITORS; MODELS, MOLECULAR; PYRROLIDINONES;

EID: 9644252787     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.10.029     Document Type: Article

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