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Volumn 37, Issue 2, 1996, Pages 307-311

In vivo labeling of angiotensin II receptors with a carbon-11-labeled selective nonpeptide antagonist

Author keywords

angiotensin II receptors; carbon 11 L 159,884; PET

Indexed keywords

1 (4 DIMETHYLAMINO 3 METHYLBENZYL) 5 DIPHENYLACETYL 4,5,6,7 TETRAHYDRO 1H IMIDAZO[4,5 C]PYRIDINE 6 CARBOXYLIC ACID; 2 BUTYL 4 CHLORO 1 [[2' (1H TETRAZOL 5 YL) 4 BIPHENYLYL]METHYL] 5 IMIDAZOLECARBOXYLIC ACID; ANGIOTENSIN 2 RECEPTOR ANTAGONIST; CARBON 11; DL PROPANOLOL; L 159689; L 159884; L 159913; L 162914; N [[4' [(2 ETHYL 5,7 DIMETHYL 3H IMIDAZO[4,5 B]PYRIDIN 3 YL)METHYL] 2 BIPHENYLYL]SULFONYL]BENZAMIDE; PRAZOSIN; PROPRANOLOL; UNCLASSIFIED DRUG; YOHIMBINE;

EID: 9344245114     PISSN: 01615505     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (19)

References (40)
  • 1
    • 0001601599 scopus 로고
    • The renin-angiotensin-aldosterone system for normal regulation of blood pressure and sodium and potassium homeostasis
    • Laragh JH, Brenner BM, eds New York. Raven Press
    • Sealey JE, Laragh JH. The renin-angiotensin-aldosterone system for normal regulation of blood pressure and sodium and potassium homeostasis. In. Laragh JH, Brenner BM, eds Hypertension pathophysiology, diagnosis and management New York. Raven Press; 1990:1287-1317.
    • (1990) Hypertension Pathophysiology, Diagnosis and Management , pp. 1287-1317
    • Sealey, J.E.1    Laragh, J.H.2
  • 2
  • 3
    • 0002463701 scopus 로고
    • Mechanisms of angiotensin action on vascular smooth muscle, the adrenal and the kidney
    • Laragh JH, Brenner BM, eds New York: Raven Press
    • Marsden PA, Brenner BM, Ballermann BJ Mechanisms of angiotensin action on vascular smooth muscle, the adrenal and the kidney. In: Laragh JH, Brenner BM, eds Hypertension pathophysiology, diagnosis and management. New York: Raven Press; 1990 1247-1272
    • (1990) Hypertension Pathophysiology, Diagnosis and Management , pp. 1247-1272
    • Marsden, P.A.1    Brenner, B.M.2    Ballermann, B.J.3
  • 4
    • 0027208070 scopus 로고
    • Angiotensin II receptors and angiotensin II receptor antagonists
    • Timmermans PB, Wong PC, Chiu AT, et al Angiotensin II receptors and angiotensin II receptor antagonists Pharmacol Rev 1993,45:205-251
    • (1993) Pharmacol Rev , vol.45 , pp. 205-251
    • Timmermans, P.B.1    Wong, P.C.2    Chiu, A.T.3
  • 5
    • 0026082048 scopus 로고
    • Angiotensin II receptors in the rat lung are of the AII-1 subtype
    • Entzeroth M, Hadamovsky S. Angiotensin II receptors in the rat lung are of the AII-1 subtype Eur J Pharmacol 1991;206:237-241.
    • (1991) Eur J Pharmacol , vol.206 , pp. 237-241
    • Entzeroth, M.1    Hadamovsky, S.2
  • 6
    • 0016166636 scopus 로고
    • Stimulation and inhibition of aldosterone biosynthesis in vitro by angiotensin II and analogs
    • Peach MJ, Chiu AT. Stimulation and inhibition of aldosterone biosynthesis in vitro by angiotensin II and analogs. Circ Res 1974;1(suppl 1):34-35.
    • (1974) Circ Res , vol.1 , Issue.1 SUPPL. , pp. 34-35
    • Peach, M.J.1    Chiu, A.T.2
  • 7
    • 0026516486 scopus 로고
    • The discovery of DuP 753, a potent, orally active nonpeptide angiotensin II receptor antagonist
    • Duncia JV, Carini DJ, Chiu AT, et al. The discovery of DuP 753, a potent, orally active nonpeptide angiotensin II receptor antagonist. Med Res Rev 1992;12:149-191.
    • (1992) Med Res Rev , vol.12 , pp. 149-191
    • Duncia, J.V.1    Carini, D.J.2    Chiu, A.T.3
  • 8
    • 0026335409 scopus 로고
    • Synthesis and structure-activity relationships of a novel series of non-peptide angiotensin II receptor binding inhibitors specific for the AT2 subtype
    • Blankley CJ, Hodges JC, Klutchko SR, et al Synthesis and structure-activity relationships of a novel series of non-peptide angiotensin II receptor binding inhibitors specific for the AT2 subtype. J Med Chem 1991;34:3248-3260.
    • (1991) J Med Chem , vol.34 , pp. 3248-3260
    • Blankley, C.J.1    Hodges, J.C.2    Klutchko, S.R.3
  • 9
    • 0008901702 scopus 로고
    • Selective ligands reveal subtypes of angiotensin receptors in rat vasculatures and brain
    • Chang RS, Lotti VJ. Selective ligands reveal subtypes of angiotensin receptors in rat vasculatures and brain [Abstract] Pharmacologist 1989;31.150.
    • (1989) Pharmacologist , vol.31 , pp. 150
    • Chang, R.S.1    Lotti, V.J.2
  • 11
    • 0024421343 scopus 로고
    • Preliminary biochemical characterization of two angiotensin II receptor subtypes
    • Whitebread S, Mele M, Kamber B, de Gasparo M Preliminary biochemical characterization of two angiotensin II receptor subtypes Biochem Biophys Res Commun 1989;163 284-291.
    • (1989) Biochem Biophys Res Commun , vol.163 , pp. 284-291
    • Whitebread, S.1    Mele, M.2    Kamber, B.3    De Gasparo, M.4
  • 12
    • 0025214101 scopus 로고
    • Two distinct angiotensin II receptor binding sites in rat adrenal revealed by new selective nonpeptide ligands
    • Chang RS, Lotti VJ. Two distinct angiotensin II receptor binding sites in rat adrenal revealed by new selective nonpeptide ligands. Mol Pharmacol 1990,37:347-351.
    • (1990) Mol Pharmacol , vol.37 , pp. 347-351
    • Chang, R.S.1    Lotti, V.J.2
  • 13
    • 0025086862 scopus 로고
    • Nonpeptide angiotensin II receptor antagonists XI. Pharmacology of EXP3174, an active metabolite of DuP 753, an orally active antihypertensive agent
    • Wong PC, Price WA, Chiu AT, et al Nonpeptide angiotensin II receptor antagonists XI. Pharmacology of EXP3174, an active metabolite of DuP 753, an orally active antihypertensive agent. J Pharmacol Exp Ther 1990,255:211-217
    • (1990) J Pharmacol Exp Ther , vol.255 , pp. 211-217
    • Wong, P.C.1    Price, W.A.2    Chiu, A.T.3
  • 14
    • 0025906857 scopus 로고
    • Nomenclature for angiotensin receptors. A report of the Nomenclature Committee of the Council for High Blood Pressure Research
    • Bumpus FM, Catt KJ, Chiu AT, et al. Nomenclature for angiotensin receptors. A report of the Nomenclature Committee of the Council for High Blood Pressure Research. Hypertension 1991.17 720-721
    • (1991) Hypertension , vol.17 , pp. 720-721
    • Bumpus, F.M.1    Catt, K.J.2    Chiu, A.T.3
  • 17
    • 0005179353 scopus 로고
    • Analysis of receptor binding data
    • Cincinnati, OH: Society for Neuroscience
    • Bylund DB Analysis of receptor binding data In: Receptor binding techniques. Cincinnati, OH: Society for Neuroscience: 1980;70-79.
    • (1980) Receptor Binding Techniques , pp. 70-79
    • Bylund, D.B.1
  • 18
    • 0026616797 scopus 로고
    • 125I]RT1-55 to dopamine transporters: Pharmacology and regional distribution with autoradiography
    • 125I]RT1-55 to dopamine transporters: pharmacology and regional distribution with autoradiography. Synapse 1992;12:37-46.
    • (1992) Synapse , vol.12 , pp. 37-46
    • Cline, E.J.1    Scheffel, U.2    Boja, J.W.3
  • 19
    • 0028847531 scopus 로고
    • In vivo receptor occupancy of the angiotensin II receptor by nonpeptide antagonists: Relationship to in vitro affinities and in vivo pharmacological potency
    • Beauchamp HT, Chang RSL, Siegl PKS, and Gibson RE In vivo receptor occupancy of the angiotensin II receptor by nonpeptide antagonists: relationship to in vitro affinities and in vivo pharmacological potency. J Pharmacol Exp Ther 1995; 272:612-618.
    • (1995) J Pharmacol Exp Ther , vol.272 , pp. 612-618
    • Beauchamp, H.T.1    Chang, R.S.L.2    Siegl, P.K.S.3    Gibson, R.E.4
  • 23
    • 0025756064 scopus 로고
    • Cloning and expression of a complementary DNA encoding a bovine adrenal angiotensin II type-1 receptor
    • Sasaki K, Yamano Y, Bardhan S, et al. Cloning and expression of a complementary DNA encoding a bovine adrenal angiotensin II type-1 receptor. Nature 1991;351:230-233.
    • (1991) Nature , vol.351 , pp. 230-233
    • Sasaki, K.1    Yamano, Y.2    Bardhan, S.3
  • 24
    • 85013562768 scopus 로고
    • Angiotensin receptor assay and charaterization
    • Conn PM, ed. San Diego: Academic Press
    • McQueen J, Semple PF Angiotensin receptor assay and charaterization In: Conn PM, ed. Methods in neurosci. San Diego: Academic Press; 1991:312-330.
    • (1991) Methods in Neurosci , pp. 312-330
    • McQueen, J.1    Semple, P.F.2
  • 25
    • 0026690935 scopus 로고
    • In vitro pharmacology of L-158,809, a new highly potent and selective angiotensin II receptor antagonist
    • Chang RS, Siegl PK, Clineschmidt BV, et al. In vitro pharmacology of L-158,809, a new highly potent and selective angiotensin II receptor antagonist J Pharmacol Exp Ther 1992;262:133-138.
    • (1992) J Pharmacol Exp Ther , vol.262 , pp. 133-138
    • Chang, R.S.1    Siegl, P.K.2    Clineschmidt, B.V.3
  • 26
    • 0026645647 scopus 로고
    • In vivo pharmacology of L-158,809, a new highly potent and selective nonpeptide angiotensin II receptor antagonist
    • Siegl PK, Chang RS, Mantlo NB et al. In vivo pharmacology of L-158,809, a new highly potent and selective nonpeptide angiotensin II receptor antagonist. J Pharmacol Exp Ther 1992;262:139-144
    • (1992) J Pharmacol Exp Ther , vol.262 , pp. 139-144
    • Siegl, P.K.1    Chang, R.S.2    Mantlo, N.B.3
  • 28
    • 0025297396 scopus 로고
    • Mendelsohn FA in vitro autoradiographic localization of binding to angiotensin receptors in the rat heart
    • Allen AM, Yamada H. Mendelsohn FA In vitro autoradiographic localization of binding to angiotensin receptors in the rat heart Jnt J Cardiol 1990;28 25-33
    • (1990) Jnt J Cardiol , vol.28 , pp. 25-33
    • Allen, A.M.1    Yamada, H.2
  • 29
    • 0025965281 scopus 로고
    • Regional distribution of the two subtypes of angiotensin II receptor in rat brain using selective nonpeptide antagonists
    • Leung KH, Smith RD, Timmermans PB, Chiu AT. Regional distribution of the two subtypes of angiotensin II receptor in rat brain using selective nonpeptide antagonists Neurosci Lett 1991;123:95-98.
    • (1991) Neurosci Lett , vol.123 , pp. 95-98
    • Leung, K.H.1    Smith, R.D.2    Timmermans, P.B.3    Chiu, A.T.4
  • 30
    • 0025013075 scopus 로고
    • Evidence for the presence of angiotensin II-type 1 receptors in brain
    • Wamsley JK, Herblin WF, Alburges ME, Hunt M. Evidence for the presence of angiotensin II-type 1 receptors in brain Brain Res Bull 1990,25.397-400
    • (1990) Brain Res Bull , vol.25 , pp. 397-400
    • Wamsley, J.K.1    Herblin, W.F.2    Alburges, M.E.3    Hunt, M.4
  • 31
    • 0026597875 scopus 로고
    • Mapping of angiotensin II receptor subtype heterogeneity in rat brain
    • Song K, Allen AM, Paxinos G, Mendelsohn FA Mapping of angiotensin II receptor subtype heterogeneity in rat brain J Comp Neurol 1992;316 467-484
    • (1992) J Comp Neurol , vol.316 , pp. 467-484
    • Song, K.1    Allen, A.M.2    Paxinos, G.3    Mendelsohn, F.A.4
  • 33
    • 0026046501 scopus 로고
    • Identification of angiotensin II receptor subtypes in human brain
    • Barnes JM, Barber PC, Barnes NM Identification of angiotensin II receptor subtypes in human brain Neuroreport 1991;2 605-608.
    • (1991) Neuroreport , vol.2 , pp. 605-608
    • Barnes, J.M.1    Barber, P.C.2    Barnes, N.M.3
  • 34
    • 0025195614 scopus 로고
    • Subclasses of angiotensin II binding sites and their functional significance
    • Dudley DT, Panek RL, Major TC, et al Subclasses of angiotensin II binding sites and their functional significance. Mol Pharmacol 1990;38.370-377
    • (1990) Mol Pharmacol , vol.38 , pp. 370-377
    • Dudley, D.T.1    Panek, R.L.2    Major, T.C.3
  • 35
    • 0025018306 scopus 로고
    • Biochemical characterization of two angiotensin II receptor subtypes in the rat
    • de Gasparo M, Whitebread S, Mele M, et al. Biochemical characterization of two angiotensin II receptor subtypes in the rat. J Cardiovasc Pharmacol 1990;16(suppl 4):S31-S35.
    • (1990) J Cardiovasc Pharmacol , vol.16 , Issue.4 SUPPL.
    • Gasparo, M.1    Whitebread, S.2    Mele, M.3
  • 36
    • 9344224629 scopus 로고
    • Compartmental modeling of an angiotensin II/AT1 receptor imaging agent: Carbon-11 L-159,884
    • Kao PF, Szabo Z, Dannals RF, et al Compartmental modeling of an angiotensin II/AT1 receptor imaging agent: carbon-11 L-159,884 [Abstract]. J Nucl Med 1994; 35:137P
    • (1994) J Nucl Med , vol.35
    • Kao, P.F.1    Szabo, Z.2    Dannals, R.F.3
  • 37
    • 0027129793 scopus 로고
    • Analysis of the evolution of angiotensin II type 1 receptor gene in mammals (mouse, rat, bovine and human)
    • Yoshida H, Kakuchi J, Guo DF, et al. Analysis of the evolution of angiotensin II type 1 receptor gene in mammals (mouse, rat, bovine and human). Biochem Biophys Res Commun 1992;186:1042-1049.
    • (1992) Biochem Biophys Res Commun , vol.186 , pp. 1042-1049
    • Yoshida, H.1    Kakuchi, J.2    Guo, D.F.3
  • 38
  • 39
    • 0026751991 scopus 로고
    • Angiotensin II type-1 receptor subtype cDNAs: Differential tissue expression and hormonal regulation
    • Kakar SS, Sellers JC, Devor DC, Musgrove LC, Neill JD. Angiotensin II type-1 receptor subtype cDNAs: differential tissue expression and hormonal regulation Biochem Biophys Res Commun 1992.183:1090-1096.
    • (1992) Biochem Biophys Res Commun , vol.183 , pp. 1090-1096
    • Kakar, S.S.1    Sellers, J.C.2    Devor, D.C.3    Musgrove, L.C.4    Neill, J.D.5
  • 40
    • 0026756696 scopus 로고
    • Cloning and expression of a novel angiotensin II receptor subtype
    • Sandberg K, Ji H, Clark AJ, Shapira H, Catt KJ. Cloning and expression of a novel angiotensin II receptor subtype. J Biol Chem 1992,267.9455-9458
    • (1992) J Biol Chem , vol.267 , pp. 9455-9458
    • Sandberg, K.1    Ji, H.2    Clark, A.J.3    Shapira, H.4    Catt, K.J.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.