Labeling of (S)-des-4-amino-3-[125I]iodozacopride (DAIZAC), a high-affinity radioligand for the 5-HT-3 receptor

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 38, Issue 11, 1996, Pages 955-961

  Mason, N Scott ^a   Hewlett, William A ^a   Ebert, Michael H ^a   Schmidt, Dennis E ^a   De Paulis, Tomas ^a  

^a VANDERBILT UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

5 HT 3 receptors; Iododestannylation; Radioligands; 125I Iodobenzamides

Indexed keywords

CHLORINE COMPOUNDS; AMIDES; SODIUM COMPOUNDS;

5-HT-3 RECEPTOR; BENZAMIDES; CHLORAMINE-T; HIGH AFFINITY; IODODESTANNYLATION; LABELINGS; METHOXY; RADIOLIGANDS; TRIBUTYL TIN; [125I]IODOBENZAMIDE;

SODIUM COMPOUNDS; CHLORINE COMPOUNDS;

5 CHLORO 3 IODO 2 METHOXY N (1 AZABICYCLO[2.2.2]OCT 3 YL)BENZAMIDE; BENZAMIDE DERIVATIVE; IODINE 125; SEROTONIN 3 RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BRAIN; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; ISOTOPE LABELING; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; RAT; RECEPTOR DENSITY;

ANIMALIA;

EID: 85078686099     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(sici)1099-1344(199611)38:11<955::aid-jlcr912>3.0.co;2-%23     Document Type: Article

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