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Volumn 58, Issue 11, 2017, Pages 1743-1748

In vivo quantification of ERb expression by pharmacokinetic modeling: Studies with18F-FHNP PET

Author keywords

Estrogen receptors; Oncology; PET; Pharmacokinetics; Quantification

Indexed keywords

2 FLUORO 6 (6 HYDROXYNAPHTHALEN 2 YL)PYRIDIN 3 OL F 18; ESTRADIOL; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; GENISTEIN; TRACER; UNCLASSIFIED DRUG; 2-FLUORO-6-(6-HYDROXYNAPHTHALEN-2-YL)PYRIDIN-3-OL; NAPHTHOL DERIVATIVE; PYRIDINE DERIVATIVE; RADIOPHARMACEUTICAL AGENT;

EID: 85032839103     PISSN: 01615505     EISSN: 2159662X     Source Type: Journal    
DOI: 10.2967/jnumed.117.192666     Document Type: Article
Times cited : (7)

References (18)
  • 2
    • 46749108373 scopus 로고    scopus 로고
    • ERb in breast cancer: Onlooker, passive player, or active protector?
    • Fox EM, Davis RJ, Shupnik MA. ERb in breast cancer: onlooker, passive player, or active protector? Steroids. 2008;73:1039–1051.
    • (2008) Steroids , vol.73 , pp. 1039-1051
    • Fox, E.M.1    Davis, R.J.2    Shupnik, M.A.3
  • 3
    • 84879474652 scopus 로고    scopus 로고
    • Expression of both estrogen receptor-beta 1 (ER-b) and its co-regulator steroid receptor RNA activator protein (SRAP) are predictive for benefit from tamoxifen therapy in patients with estrogen receptor-alpha (ER-a)negative early breast cancer (EBC)
    • Yan Y, Li X, Blanchard A, et al. Expression of both estrogen receptor-beta 1 (ER-b) and its co-regulator steroid receptor RNA activator protein (SRAP) are predictive for benefit from tamoxifen therapy in patients with estrogen receptor-alpha (ER-a)negative early breast cancer (EBC). Ann Oncol. 2013;24:1986–1993.
    • (2013) Ann Oncol , vol.24 , pp. 1986-1993
    • Yan, Y.1    Li, X.2    Blanchard, A.3
  • 4
    • 33847147996 scopus 로고    scopus 로고
    • The combination of letrozole and trastu-zumab as first or second-line biological therapy produces durable responses in a subset of HER2 positive and ER positive advanced breast cancers
    • Marcom PK, Isaacs C, Harris L, et al. The combination of letrozole and trastu-zumab as first or second-line biological therapy produces durable responses in a subset of HER2 positive and ER positive advanced breast cancers. Breast Cancer Res Treat. 2007;102:43–49.
    • (2007) Breast Cancer Res Treat , vol.102 , pp. 43-49
    • Marcom, P.K.1    Isaacs, C.2    Harris, L.3
  • 5
    • 34548537574 scopus 로고    scopus 로고
    • A phase II placebo-controlled trial of neo-adjuvant anastrozole alone or with gefitinib in early breast cancer
    • Smith IE, Walsh G, Skene A, et al. A phase II placebo-controlled trial of neo-adjuvant anastrozole alone or with gefitinib in early breast cancer. J Clin Oncol. 2007;25:3816–3822.
    • (2007) J Clin Oncol , vol.25 , pp. 3816-3822
    • Smith, I.E.1    Walsh, G.2    Skene, A.3
  • 6
    • 84856790756 scopus 로고    scopus 로고
    • PET imaging of estrogen receptors as a diagnostic tool for breast cancer patients presenting with a clinical dilemma
    • van Kruchten M, Glaudemans AWJM, de Vries EFJ, et al. PET imaging of estrogen receptors as a diagnostic tool for breast cancer patients presenting with a clinical dilemma. J Nucl Med. 2012;53:182–190.
    • (2012) J Nucl Med , vol.53 , pp. 182-190
    • Van Kruchten, M.1    Awjm, G.2    De Vries, E.F.J.3
  • 7
    • 51649084814 scopus 로고    scopus 로고
    • Intratumoral estrogens and estrogen receptors in human non-small cell lung carcinoma
    • Niikawa H, Suzuki T, Miki Y, et al. Intratumoral estrogens and estrogen receptors in human non-small cell lung carcinoma. Clin Cancer Res. 2008;14:4417–4426.
    • (2008) Clin Cancer Res , vol.14 , pp. 4417-4426
    • Niikawa, H.1    Suzuki, T.2    Miki, Y.3
  • 8
    • 84984620735 scopus 로고    scopus 로고
    • Synchronous multiple lung adenocarci-nomas: Estrogen concentration in peripheral lung
    • Ikeda K, Shiraishi K, Yoshida A, et al. Synchronous multiple lung adenocarci-nomas: estrogen concentration in peripheral lung. PLoS One. 2016;11:e0160910.
    • (2016) Plos One , vol.11 , pp. e0160910
    • Ikeda, K.1    Shiraishi, K.2    Yoshida, A.3
  • 9
    • 85017094856 scopus 로고    scopus 로고
    • Synthesis and evaluation of the new estrogen receptor b selective radioligand [18F]FHNP: Comparison with [18F]FES
    • Antunes IF, van Waarde A, Dierckx RA, de Vries EGE, Hospers GAP, de Vries EF. Synthesis and evaluation of the new estrogen receptor b selective radioligand [18F]FHNP: comparison with [18F]FES. J Nucl Med. 2017;58:554–559.
    • (2017) J Nucl Med , vol.58 , pp. 554-559
    • Antunes, I.F.1    Van Waarde, A.2    Dierckx, R.A.3    De Vries, E.G.E.4    Hospers, G.A.P.5    De Vries, E.F.6
  • 10
    • 84899473276 scopus 로고    scopus 로고
    • In vivo imaging of brain estrogen receptors in rats: A 16a-18F-fluoro-17b-estradiol PET study
    • Khayum MA, de Vries EFJ, Glaudemans AWJM, Dierckx RAJO, Doorduin J. In vivo imaging of brain estrogen receptors in rats: a 16a-18F-fluoro-17b-estradiol PET study. J Nucl Med. 2014;55:481–487.
    • (2014) J Nucl Med , vol.55 , pp. 481-487
    • Khayum, M.A.1    De Vries, E.F.J.2    Awjm, G.3    Rajo, D.4    Doorduin, J.5
  • 11
    • 0020956774 scopus 로고
    • Graphical evaluation of blood-to-brain transfer constants from multiple-time uptake data
    • Patlak CS, Blasberg RG, Fenstermacher JD. Graphical evaluation of blood-to-brain transfer constants from multiple-time uptake data. J Cereb Blood Flow Metab. 1983;3:1–7.
    • (1983) J Cereb Blood Flow Metab , vol.3 , pp. 1-7
    • Patlak, C.S.1    Blasberg, R.G.2    Fenstermacher, J.D.3
  • 12
    • 35648967028 scopus 로고    scopus 로고
    • Choosing the optimal fit function: Comparison of the Akaike information criterion and the F-test
    • Glatting G, Kletting P, Reske SN, Hohl K, Ring C. Choosing the optimal fit function: comparison of the Akaike information criterion and the F-test. Med Phys. 2007;34:4285–4292.
    • (2007) Med Phys , vol.34 , pp. 4285-4292
    • Glatting, G.1    Kletting, P.2    Reske, S.N.3    Hohl, K.4    Ring, C.5
  • 13
    • 85012247397 scopus 로고    scopus 로고
    • High estrogen receptor b expression is prognostic among adjuvant chemotherapy–treated patients: Results from a population-based breast cancer cohort
    • Elebro K, Borgquist S, Rosendahl AH, et al. High estrogen receptor b expression is prognostic among adjuvant chemotherapy–treated patients: results from a population-based breast cancer cohort. Clin Cancer Res. 2017;23:766–777.
    • (2017) Clin Cancer Res , vol.23 , pp. 766-777
    • Elebro, K.1    Borgquist, S.2    Rosendahl, A.H.3
  • 14
    • 26444610710 scopus 로고    scopus 로고
    • Synthesis of an estrogen receptor b-selective radioligand: 5-[18F]fluoro-(2R*,3S*)-2,3-bis(4-hydroxyphenyl)pentanenitrile and comparison of in vivo distribution with 16a-[18F]fluoro-17b-estradiol
    • Yoo J, Dence CS, Sharp TL, Katzenellenbogen JA, Welch MJ. Synthesis of an estrogen receptor b-selective radioligand: 5-[18F]fluoro-(2R*,3S*)-2,3-bis(4-hydroxyphenyl)pentanenitrile and comparison of in vivo distribution with 16a-[18F]fluoro-17b-estradiol. J Med Chem. 2005;48:6366–6378.
    • (2005) J Med Chem , vol.48 , pp. 6366-6378
    • Yoo, J.1    Dence, C.S.2    Sharp, T.L.3    Katzenellenbogen, J.A.4    Welch, M.J.5
  • 15
    • 84867855209 scopus 로고    scopus 로고
    • Synthesis and biological evaluation of two agents for imaging estrogen receptor b by positron emission tomography: Challenges in PET imaging of a low abundance target
    • Lee JH, Peters O, Lehmann L, et al. Synthesis and biological evaluation of two agents for imaging estrogen receptor b by positron emission tomography: challenges in PET imaging of a low abundance target. Nucl Med Biol. 2012;39:1105–1116.
    • (2012) Nucl Med Biol , vol.39 , pp. 1105-1116
    • Lee, J.H.1    Peters, O.2    Lehmann, L.3
  • 16
    • 0033233297 scopus 로고    scopus 로고
    • Interactions of 16a-[18F]-fluoroestradiol (FES) with sex steroid binding protein (SBP)
    • Tewson TJ, Mankoff DA, Peterson LM, Woo I, Petra P. Interactions of 16a-[18F]-fluoroestradiol (FES) with sex steroid binding protein (SBP). Nucl Med Biol. 1999;26:905–913.
    • (1999) Nucl Med Biol. , vol.26 , pp. 905-913
    • Tewson, T.J.1    Mankoff, D.A.2    Peterson, L.M.3    Woo, I.4    Petra, P.5
  • 17
    • 75749116783 scopus 로고    scopus 로고
    • Pharmacokinetic assessment of the uptake of 16b-18F-fuoro-5a-dihydrotestosterone (FDHT) in prostate tumors as measured by PET
    • Beattie BJ, Smith-Jones PM, Jhanwar YS, et al. Pharmacokinetic assessment of the uptake of 16b-18F-fuoro-5a-dihydrotestosterone (FDHT) in prostate tumors as measured by PET. J Nucl Med. 2010;51:183–192.
    • (2010) J Nucl Med , vol.51 , pp. 183-192
    • Beattie, B.J.1    Smith-Jones, P.M.2    Jhanwar, Y.S.3
  • 18
    • 0030786893 scopus 로고    scopus 로고
    • Analysis of blood clearance and labeled metabolites for the estrogen receptor tracer [F-18]-16 alpha-fluoroestradiol (FES)
    • Mankoff DA, Tewson TJ, Eary JF. Analysis of blood clearance and labeled metabolites for the estrogen receptor tracer [F-18]-16 alpha-fluoroestradiol (FES). Nucl Med Biol. 1997;24:341–348.
    • (1997) Nucl Med Biol , vol.24 , pp. 341-348
    • Mankoff, D.A.1    Tewson, T.J.2    Eary, J.F.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.