Novel and efficient debenzylation of N-benzyltetrazole derivatives with the rosenmund catalyst

Synthesis (Germany)

Volumn 46, Issue 23, 2014, Pages 3249-3255

  Seki, Masahiko ^a  

^a API Corporation   (Japan)

Author keywords

cleavage; heterocycles; hydrogen transfer; palladium; protecting groups

Indexed keywords

PALLADIUM;

AMMONIUM FORMATE; ANGIOTENSIN II; CATALYTIC TRANSFER HYDROGENATION; CLEAVAGE; FUNCTIONALIZED SUBSTRATES; HETEROCYCLES; HYDROGEN TRANSFER; PROTECTING GROUP;

CATALYSTS;

1 BENZYL 5 PHENYL 1H TETRAZOLE; BARIUM SULFATE; CANDESARTAN HEXETIL; IRBESARTAN; LOSARTAN; N BENZYLCANDESARTAN CILEXETIL; N BENZYLIRBESARTAN; N BENZYLLOSARTAN; N BENZYLTETRAZOLE DERIVATIVE; N BENZYLVALSARTAN BENZYL ESTER; PALLADIUM; TETRAZOLE DERIVATIVE; UNCLASSIFIED DRUG; VALSARTAN;

ARTICLE; CATALYST; DEBENZYLATION; DEPROTECTION REACTION; DRUG STRUCTURE; DRUG SYNTHESIS; HYDROGENATION; REACTION ANALYSIS; ROSENMUND CATALYST;

EID: 85027938253     PISSN: 00397881     EISSN: 1437210X     Source Type: Journal    
DOI: 10.1055/s-0034-1378585     Document Type: Article

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