Development of a Manufacturing Route to Avibactam, a β-Lactamase Inhibitor

Organic Process Research and Development

Volumn 20, Issue 10, 2016, Pages 1799-1805

  Ball, Matthew ^a   Boyd, Alistair ^a   Ensor, Gareth J ^a   Evans, Matthew ^a   Golden, Michael ^a   Linke, Simon R ^a   Milne, David ^a   Murphy, Rebecca ^a   Telford, Alex ^a   Kalyan, Yuriy ^b   Lawton, Graham R ^b   Racha, Saibaba ^b   Ronsheim, Melanie ^b   Zhou, Shao Hong ^b  

^a ASTRAZENECA   (United Kingdom)

^b FOREST RESEARCH INSTITUTE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

COST EFFECTIVENESS; UREA;

COMMERCIAL PROCESS; COST EFFECTIVE; DEBENZYLATION; ENVIRONMENTAL FOOTPRINTS; LACTAMASES; PROCESS DEVELOPMENT; PROTECTING GROUP; SULFATION REACTION;

MANUFACTURE;

EID: 84992215916     PISSN: 10836160     EISSN: 1520586X     Source Type: Journal    
DOI: 10.1021/acs.oprd.6b00268     Document Type: Article

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