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Volumn 22, Issue 17, 2016, Pages 4280-4282

Targeting androgen receptor aberrations in castration-resistant prostate cancer

Author keywords

[No Author keywords available]

Indexed keywords

ABIRATERONE ACETATE; ANDROGEN RECEPTOR; ANTINEOPLASTIC AGENT; ENZALUTAMIDE; EPI 506; UNCLASSIFIED DRUG; ANDROGEN RECEPTOR ANTAGONIST;

EID: 84988645712     PISSN: 10780432     EISSN: 15573265     Source Type: Journal    
DOI: 10.1158/1078-0432.CCR-16-1137     Document Type: Article
Times cited : (16)

References (12)
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    • Targeting androgen receptor activation function-1 with EPI to overcome resistance mechanisms in castration-resistant prostate cancer
    • Yang YC, Banuelos CA, Mawji NR, Wang J, Kato M, Haile S, et al. Targeting androgen receptor activation function-1 with EPI to overcome resistance mechanisms in castration-resistant prostate cancer. Clin Cancer Res 2016;22:4466-77.
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    • Yang, Y.C.1    Banuelos, C.A.2    Mawji, N.R.3    Wang, J.4    Kato, M.5    Haile, S.6
  • 2
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    • Targeting the androgen receptor pathway in castration-resistant prostate cancer: Progresses and prospects
    • Ferraldeschi R, Welti J, Luo J, Attard G, de Bono JS. Targeting the androgen receptor pathway in castration-resistant prostate cancer: progresses and prospects. Oncogene 2015;34:1745-57.
    • (2015) Oncogene , vol.34 , pp. 1745-1757
    • Ferraldeschi, R.1    Welti, J.2    Luo, J.3    Attard, G.4    De Bono, J.S.5
  • 3
    • 84964588123 scopus 로고    scopus 로고
    • Analytical validation and clinical qualification of a new immunohistochemical assay for androgen receptor splice variant-7 protein expression in metastatic castration-resistant prostate cancer
    • Apr Epub ahead of print
    • Welti J, Rodrigues DN, Sharp A, Sun S, Lorente D, Riisnaes R, et al. Analytical validation and clinical qualification of a new immunohistochemical assay for androgen receptor splice variant-7 protein expression in metastatic castration-resistant prostate cancer. Eur Urol 2016 Apr 22. [Epub ahead of print].
    • (2016) Eur Urol , vol.22
    • Welti, J.1    Rodrigues, D.N.2    Sharp, A.3    Sun, S.4    Lorente, D.5    Riisnaes, R.6
  • 5
    • 84942860161 scopus 로고    scopus 로고
    • Androgen receptor splice variants dimerize to transactivate target genes
    • Xu D, Zhan Y, Qi Y, Cao B, Bai S, Xu W, et al. Androgen receptor splice variants dimerize to transactivate target genes. Cancer Res 2015;75:3663-71.
    • (2015) Cancer Res , vol.75 , pp. 3663-3671
    • Xu, D.1    Zhan, Y.2    Qi, Y.3    Cao, B.4    Bai, S.5    Xu, W.6
  • 6
    • 84963813308 scopus 로고    scopus 로고
    • BET bromodomain inhibitors enhance efficacy and disrupt resistance to AR antagonists in the treatment of prostate cancer
    • Asangani IA, Wilder-Romans K, Dommeti VL, Krishnamurthy PM, Apel IJ, Escara-Wilke J, et al. BET bromodomain inhibitors enhance efficacy and disrupt resistance to AR antagonists in the treatment of prostate cancer. Mol Cancer Res 2016;14:324-31.
    • (2016) Mol Cancer Res , vol.14 , pp. 324-331
    • Asangani, I.A.1    Wilder-Romans, K.2    Dommeti, V.L.3    Krishnamurthy, P.M.4    Apel, I.J.5    Escara-Wilke, J.6
  • 7
    • 84969627173 scopus 로고    scopus 로고
    • Second-generation HSP90 inhibitor onalespib blocks mRNA splicing of androgen receptor variant 7 in prostate cancer cells
    • Ferraldeschi R, Welti J, Powers MV, Yuan W, Smyth T, Seed G, et al. Second-generation HSP90 inhibitor onalespib blocks mRNA splicing of androgen receptor variant 7 in prostate cancer cells. Cancer Res 2016;76: 2731-42.
    • (2016) Cancer Res , vol.76 , pp. 2731-2742
    • Ferraldeschi, R.1    Welti, J.2    Powers, M.V.3    Yuan, W.4    Smyth, T.5    Seed, G.6
  • 8
    • 84966591443 scopus 로고    scopus 로고
    • TAS3681: New class of androgen receptor antagonist with androgen receptor downregulating activity
    • abstr 266
    • Minamiguchi K, Seki M, Aoyagi H, Kajiwara D, Mori T, Masuko N, et al. TAS3681: new class of androgen receptor antagonist with androgen receptor downregulating activity. J Clin Oncol 33, 2015 (suppl 7; abstr 266).
    • (2015) J Clin Oncol , vol.33
    • Minamiguchi, K.1    Seki, M.2    Aoyagi, H.3    Kajiwara, D.4    Mori, T.5    Masuko, N.6
  • 9
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    • Structural characterization of the native NH2-terminal transactivation domain of the human androgen receptor: A collapsed disordered conformation underlies structural plasticity and protein-induced folding
    • Lavery DN, McEwan IJ. Structural characterization of the native NH2-terminal transactivation domain of the human androgen receptor: a collapsed disordered conformation underlies structural plasticity and protein-induced folding. Biochemistry 2008;47:3360-9.
    • (2008) Biochemistry , vol.47 , pp. 3360-3369
    • Lavery, D.N.1    McEwan, I.J.2
  • 11
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    • EPI-001 is a selective peroxisome proliferator-activated receptorgamma modulator with inhibitory effects on androgen receptor expression and activity in prostate cancer
    • Brand LJ, Olson ME, Ravindranathan P, Guo H, Kempema AM, Andrews TE, et al. EPI-001 is a selective peroxisome proliferator-activated receptorgamma modulator with inhibitory effects on androgen receptor expression and activity in prostate cancer. Oncotarget 2015;6:3811-24.
    • (2015) Oncotarget , vol.6 , pp. 3811-3824
    • Brand, L.J.1    Olson, M.E.2    Ravindranathan, P.3    Guo, H.4    Kempema, A.M.5    Andrews, T.E.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.