Synthesis of 6-[11C]methyl-m-tyrosine ([11C]6MemTyr) for dopamine synthesis imaging in living brain using PET

Bioorganic and Medicinal Chemistry

Volumn 23, Issue 4, 2015, Pages 729-734

  Kanazawa, Masakatsu ^a   Ohba, Hiroyuki ^a   Iwazaki, Aiko ^a   Kakiuchi, Takeharu ^a   Tsukada, Hideo ^a  

^a CENTRAL RESEARCH LABORATORY   (Japan)

Author keywords

6 11C methyl m tyrosine; Brain; Dopamine; 18F FDOPA PET

Indexed keywords

6 FLUORODOPA F 18; CARBON; CARBON METHYL M TYROSINE C 11; DOPAMINE; DRUG ANALYSIS; FLUORINE; LEVODOPA; METHYL-3-TYROSINE; METIROSINE; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG;

ANIMAL; ANIMAL EXPERIMENT; ARTICLE; BRAIN; CONTROLLED STUDY; CORPUS STRIATUM; DOPAMINE METABOLISM; HAPLORHINI; ISOTOPE LABELING; MACACA FASCICULARIS; MALE; METABOLISM; METHYLATION; MOLECULAR PROBE; NEUROIMAGING; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; PRESYNAPTIC MEMBRANE; PROCEDURES; RADIOCHEMISTRY; SCINTISCANNING; SYNTHESIS;

ANALYSIS; ANIMALS; BRAIN; CARBON RADIOISOTOPES; CHEMICAL SYNTHESIS; CORPUS STRIATUM; DOPAMINE; FLUORINE RADIOISOTOPES; LEVODOPA; MACACA FASCICULARIS; MALE; METABOLISM; METHODS; METHYLTYROSINES; POSITRON-EMISSION TOMOGRAPHY; RADIONUCLIDE IMAGING; RADIOPHARMACEUTICALS;

EID: 84964224990     PISSN: 09680896     EISSN: 14643391     Source Type: Journal    
DOI: 10.1016/j.bmc.2014.12.061     Document Type: Article

References (23)

1. A.J. Lees, J. Hardy, and T. Revesz Lancet. 373 2009 2055
2. D.J. Brooks J. Nucl. Med. 51 2010 596
3. V. Sossi, R. de La Fuente-Fernández, J.E. Holden, D.J. Doudet, J. McKenzie, A.J. Stoessl, and T.J. Ruth J. Cereb. Blood Flow Metab. 22 2002 232
4. H.C. Guldberg, and C.A. Marsden Pharmacol. Rev. 27 1975 135
5. J. Reith, S. Dyve, H. Kuwabara, M. Guttman, M. Diksic, and A. Gjedde J. Cereb. Blood Flow Metab. 10 1990 707
6. A. Luxen, M. Guillaume, W.P. Melega, V.W. Pike, O. Solin, and R. Wagner Int. J. Rad. Appl. Instrum. B 19 1992 149
7. C. Lemaire, P. Damhaut, A. Plenevaux, and D. Comar J. Nucl. Med. 35 1994 1996
8. C. Lemaire, S. Gillet, S. Guillouet, A. Plenevaux, J. Aerts, and A. Luxen Eur. J. Org. Chem. 2004 2004 2899
9. S. Jordan, J.L. Eberling, K.S. Bankiewicz, D. Rosenberg, P.G. Coxson, H.F. VanBrocklin, J.P. O'Neil, M.E. Emborg, and W.J. Jagust Brain Res. 750 1997 264
10. O.T. DeJesus Drug Dev. Res. 59 2003 249
11. H. Doi, I. Ban, A. Nonoyama, K. Sumi, C. Kuang, T. Hosoya, H. Tsukada, and M. Suzuki Chem. Eur. J. 15 2009 4165
12. G. Bartoli, M. Bosco, M. Locatelli, E. Marcantoni, P. Melchiorre, and L. Sambri Org. Lett. 7 2005 427
13. T. Ishiyama, M. Murata, and N. Miyaura J. Org. Chem. 60 1995 7508
14. M. Suzuki, H. Doi, M. Björkman, Y. Andersson, B. Långström, Y. Watanabe, and R. Noyori Chem. Eur. J. 3 1997 2039
15. M. Suzuki, K. Sumi, H. Koyama, T. Hosoya, M. Takashima-Hirano, and H. Doi Chem. Eur. J. 15 2009 12489
16. C.J. Endres, S. Swaminathan, O.T. DeJesus, M. Sievert, A.E. Ruoho, D. Murali, S.G. Rommelfanger, and J.E. Holden Life Sci. 60 1997 2399
17. H. Tsukada, K.J. Lindner, P. Hartvig, Y. Tani, J. Valtysson, P. Bjurling, T. Kihlberg, G. Westerberg, Y. Watanabe, and B. Långström Brain Res. 713 1996 92
18. H. Tsukada, N. Harada, S. Nishiyama, H. Ohba, and T. Kakiuchi J. Neurosci. 20 2000 7067
19. B. Långström, G. Antoni, P. Gullberg, C. Halldin, P. Malmborg, K. Någren, A. Rimland, and H. Svärd J. Nucl. Med. 28 1987 1037
20. W.P. Melega, J.M. Hoffman, A. Luxen, C.H. Nissenson, M.E. Phelps, and J.R. Barrio Life Sci. 47 1990 149
21. M. Watanabe, H. Okada, K. Shimizu, T. Omura, E. Yoshikawa, T. Kosugi, S. Mori, and T. Yamashita IEEE Trans. Nucl. Sci. 44 1997 1277
22. E.G. Jones, J.M. Stone, and H.J. Karten Ann. N.Y. Acad. Sci. 1225 2011 E147
23. C.S. Patlak, and R.G. Blasberg J. Cereb. Blood Flow Metab. 5 1985 584