Screening HIV-1 fusion inhibitors based on capillary electrophoresis head-end microreactor targeting to the core structure of gp41

Journal of Pharmaceutical and Biomedical Analysis

Volumn 120, Issue , 2016, Pages 153-157

  Liu, Lihong ^a   Xu, Xiaoying ^a   Liu, Yanhui ^b   Zhang, Xuanxuan ^a   Li, Lin ^a   Jia, Zhimin ^a  

^a SOUTHERN MEDICAL UNIVERSITY   (China)

^b People's Hospital of Jinzhou   (China)

Author keywords

Gp41; HIV 1 inhibitors; Microreactor; Six helix bundles; Traditional Chinese medicines

Indexed keywords

ANTIVIRUS AGENT; BUFFER; GLYCOPROTEIN GP 41; HUMAN IMMUNODEFICIENCY VIRUS FUSION INHIBITOR; PHERETIMA ASPERGILLUM EXTRACT; UNCLASSIFIED DRUG; CHEMOKINE RECEPTOR CCR5 ANTAGONIST; GP41 PROTEIN, HUMAN IMMUNODEFICIENCY VIRUS 1; HERBACEOUS AGENT;

ANTIVIRAL ACTIVITY; ARTICLE; BIOREACTOR; CAPILLARY ELECTROPHORESIS; CHINESE MEDICINE; DRUG SCREENING; DRUG SYNTHESIS; HUMAN IMMUNODEFICIENCY VIRUS 1; MICROANALYSIS; MICROREACTOR; NONHUMAN; PHERETIMA; PHERETIMA ASPERGILLUM; PRIORITY JOURNAL; REACTOR DESIGN; ANTAGONISTS AND INHIBITORS; CHEMISTRY; DOSE RESPONSE; DRUG DELIVERY SYSTEM; DRUG EFFECTS; HUMAN; PHYSIOLOGY; PRECLINICAL STUDY; PROCEDURES;

CCR5 RECEPTOR ANTAGONISTS; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DELIVERY SYSTEMS; DRUG EVALUATION, PRECLINICAL; DRUGS, CHINESE HERBAL; ELECTROPHORESIS, CAPILLARY; HIV ENVELOPE PROTEIN GP41; HIV-1; HUMANS;

EID: 84951752605     PISSN: 07317085     EISSN: 1873264X     Source Type: Journal    
DOI: 10.1016/j.jpba.2015.12.021     Document Type: Article

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