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Volumn 143, Issue 1, 2015, Pages 147-155
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A multi-parameter in vitro screen in human stem cell-derived cardiomyocytes identifies ponatinib-induced structural and functional cardiac toxicity
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IQVIA
(United States)
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Author keywords
ABL inhibitors; cardiac toxicity; human stem cell derived cardiomyocytes; in vitro toxicity testing; targeted oncology agents
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Indexed keywords
ANTINEOPLASTIC AGENT;
IMIDAZOLE DERIVATIVE;
PONATINIB;
PROTEIN KINASE INHIBITOR;
PYRIDAZINE DERIVATIVE;
TROPONIN;
ACTIN FILAMENT;
CELL DEATH;
CELL DIFFERENTIATION;
CELL LINE;
CHEMICALLY INDUCED;
DOSE RESPONSE;
DRUG EFFECTS;
HEART DISEASE;
HEART MITOCHONDRION;
HEART MUSCLE CELL;
HEART RATE;
HUMAN;
METABOLISM;
OXIDATIVE STRESS;
PATHOLOGY;
PATHOPHYSIOLOGY;
PLURIPOTENT STEM CELL;
PROCEDURES;
RISK ASSESSMENT;
SIGNAL TRANSDUCTION;
TIME;
TOXICITY TESTING;
ACTIN CYTOSKELETON;
ANTINEOPLASTIC AGENTS;
CELL DEATH;
CELL DIFFERENTIATION;
CELL LINE;
DOSE-RESPONSE RELATIONSHIP, DRUG;
HEART DISEASES;
HEART RATE;
HUMANS;
IMIDAZOLES;
INDUCED PLURIPOTENT STEM CELLS;
MITOCHONDRIA, HEART;
MYOCYTES, CARDIAC;
OXIDATIVE STRESS;
PROTEIN KINASE INHIBITORS;
PYRIDAZINES;
RISK ASSESSMENT;
SIGNAL TRANSDUCTION;
TIME FACTORS;
TOXICITY TESTS;
TROPONIN;
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EID: 84947787375
PISSN: None
EISSN: 10960929
Source Type: Journal
DOI: 10.1093/toxsci/kfu215 Document Type: Article |
Times cited : (63)
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References (0)
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