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Volumn 75, Issue 17, 2015, Pages 2045-2049

Evogliptin: First Global Approval

Author keywords

[No Author keywords available]

Indexed keywords

EVOGLIPTIN; HEMOGLOBIN A1C; 4-(3-AMINO-4-(2,4,5-TRIFLUOROPHENYL)BUTANOYL)-3-(TERT-BUTOXYMETHYL)PIPERAZIN-2-ONE; DIPEPTIDYL PEPTIDASE IV INHIBITOR; PIPERAZINE DERIVATIVE;

EID: 84946907635     PISSN: 00126667     EISSN: 11791950     Source Type: Journal    
DOI: 10.1007/s40265-015-0496-5     Document Type: Article
Times cited : (35)

References (17)
  • 1
    • 29944436303 scopus 로고    scopus 로고
    • International Diabetes Federation Accessed 12 Oct 2015
    • International Diabetes Federation. Global guideline for type 2 diabetes. 2012. http://www.idf.org/sites/default/files/IDF-Guideline-for-Type-2-Diabetes.pdf. Accessed 12 Oct 2015.
    • (2012) Global Guideline for Type 2 Diabetes
  • 3
    • 84946935774 scopus 로고    scopus 로고
    • PipelineReview.com Accessed 13 Oct 2015
    • PipelineReview.com. Dong-A ST's DPP4 inhibitor, SUGANON, got approved for type 2 diabetes in Korea. 2015. http://www.pipelinereview.com/index.php/2015100259148/Small-Molecules/Dong-A-STs-DPP4-inhibitor-SUGANON-got-approved-for-type-2-diabetes-in-Korea.html. Accessed 13 Oct 2015.
    • (2015) Dong-A ST's DPP4 Inhibitor, SUGANON, Got Approved for Type 2 Diabetes in Korea
  • 4
    • 84946935775 scopus 로고    scopus 로고
    • Dong-A ST Accessed 13 Oct 2015
    • Dong-A ST. 2Q 2015 Performance Results. 2015. http://en.donga-st.com/B05.da?method=IRResourceList. Accessed 13 Oct 2015.
    • (2015) 2Q 2015 Performance Results
  • 5
    • 84946913153 scopus 로고    scopus 로고
    • Dong-A ST. Accessed 13 Oct 2015
    • Dong-A ST. 2014 Annual report. 2015. http://en.donga-st.com/Pass.da?viewPath=/b05/IRReport. Accessed 13 Oct 2015.
    • (2015) 2014 Annual Report
  • 6
    • 84946935776 scopus 로고    scopus 로고
    • Dong-A ST Accessed 13 Oct 2015
    • Dong-A ST. 1Q 2015 Performance results. 2015. http://en.donga-st.com/B05.da?method=IRResourceList. Accessed 13 Oct 2015.
    • (2015) 1Q 2015 Performance Results
  • 8
    • 79957865337 scopus 로고    scopus 로고
    • Discovery of DA-1229: A potent, long acting dipeptidyl peptidase-4 inhibitor for the treatment of type 2 diabetes
    • 1:CAS:528:DC%2BC3MXntFKht78%3D 21570283
    • Kim HJ, Kwak WY, Min JP, et al. Discovery of DA-1229: a potent, long acting dipeptidyl peptidase-4 inhibitor for the treatment of type 2 diabetes. Bioorg Med Chem Lett. 2011;21(12):3809-12.
    • (2011) Bioorg Med Chem Lett. , vol.21 , Issue.12 , pp. 3809-3812
    • Kim, H.J.1    Kwak, W.Y.2    Min, J.P.3
  • 9
    • 84941558262 scopus 로고    scopus 로고
    • Clinical pharmacology of dipeptidyl peptidase 4 inhibitors indicated for the treatment of type 2 diabetes mellitus
    • 1:CAS:528:DC%2BC2MXhsV2ltbjE 26173919
    • Chen XW, He ZX, Zhou ZW, et al. Clinical pharmacology of dipeptidyl peptidase 4 inhibitors indicated for the treatment of type 2 diabetes mellitus. Clin Exp Pharmacol Physiol. 2015;42(10):999-1024.
    • (2015) Clin Exp Pharmacol Physiol. , vol.42 , Issue.10 , pp. 999-1024
    • Chen, X.W.1    He, Z.X.2    Zhou, Z.W.3
  • 10
    • 84655170276 scopus 로고    scopus 로고
    • DA-1229, a novel and potent DPP4 inhibitor, improves insulin resistance and delays the onset of diabetes
    • 1:CAS:528:DC%2BC3MXhs1Oms7zJ 22056373
    • Kim M-K, Chae YN, Kim HD, et al. DA-1229, a novel and potent DPP4 inhibitor, improves insulin resistance and delays the onset of diabetes. Life Sci. 2012;90(1):21-9.
    • (2012) Life Sci. , vol.90 , Issue.1 , pp. 21-29
    • Kim, M.-K.1    Chae, Y.N.2    Kim, H.D.3
  • 11
    • 84908077770 scopus 로고    scopus 로고
    • Multiple-dose pharmacokinetics and pharmacodynamics of evogliptin (DA-1229), a novel dipeptidyl peptidase IV inhibitor, in healthy volunteers
    • 4199987 1:CAS:528:DC%2BC2MXisFWls78%3D 25336915
    • Gu N, Park MK, Kim TE, et al. Multiple-dose pharmacokinetics and pharmacodynamics of evogliptin (DA-1229), a novel dipeptidyl peptidase IV inhibitor, in healthy volunteers. Drug Des Devel Ther. 2014;8:1709-21.
    • (2014) Drug des Devel Ther. , vol.8 , pp. 1709-1721
    • Gu, N.1    Park, M.K.2    Kim, T.E.3
  • 12
    • 78650584379 scopus 로고    scopus 로고
    • A novel dipeptidyl peptidase IV inhibitor DA-1229 ameliorates streptozotocin-induced diabetes by increasing beta-cell replication and neogenesis
    • 1:CAS:528:DC%2BC3cXhs1Wkur3M 21093089
    • Cho JM, Jang HW, Cheon H, et al. A novel dipeptidyl peptidase IV inhibitor DA-1229 ameliorates streptozotocin-induced diabetes by increasing beta-cell replication and neogenesis. Diabetes Res Clin Pract. 2011;91(1):72-9.
    • (2011) Diabetes Res Clin Pract. , vol.91 , Issue.1 , pp. 72-79
    • Cho, J.M.1    Jang, H.W.2    Cheon, H.3
  • 13
    • 84866179930 scopus 로고    scopus 로고
    • Evaluation of the pharmacokinetics, food effect, pharmacodynamics, and tolerability of DA-1229, a dipeptidyl peptidase IV inhibitor, in healthy volunteers: First-in-human study
    • 1:CAS:528:DC%2BC38XhtlOisr7K 22943970
    • Kim TE, Lim KS, Park MK, et al. Evaluation of the pharmacokinetics, food effect, pharmacodynamics, and tolerability of DA-1229, a dipeptidyl peptidase IV inhibitor, in healthy volunteers: first-in-human study. Clin Ther. 2012;34(9):1986-98.
    • (2012) Clin Ther. , vol.34 , Issue.9 , pp. 1986-1998
    • Kim, T.E.1    Lim, K.S.2    Park, M.K.3
  • 14
    • 84946906905 scopus 로고    scopus 로고
    • Metabolism and excretion of [14C]evogliptin, a DPP-4 inhibitor, in rats [abstract no. P323]
    • Park KJ, Shim HJ. Metabolism and excretion of [14C]evogliptin, a DPP-4 inhibitor, in rats [abstract no. P323]. Drug Metab Rev. 2014;45(Suppl 1):195.
    • (2014) Drug Metab Rev. , vol.45 , pp. 195
    • Park, K.J.1    Shim, H.J.2
  • 16
    • 84924287356 scopus 로고    scopus 로고
    • A randomized, double-blind, placebo-controlled, phase II clinical trial to investigate the efficacy and safety of oral DA-1229 in patients with type 2 diabetes mellitus who have inadequate glycaemic control with diet and exercise
    • 1:CAS:528:DC%2BC2MXjvFyntLw%3D 25362864
    • Jung CH, Park CY, Ahn KJ, et al. A randomized, double-blind, placebo-controlled, phase II clinical trial to investigate the efficacy and safety of oral DA-1229 in patients with type 2 diabetes mellitus who have inadequate glycaemic control with diet and exercise. Diabetes Metab Res Rev. 2015;31(3):295-306.
    • (2015) Diabetes Metab Res Rev. , vol.31 , Issue.3 , pp. 295-306
    • Jung, C.H.1    Park, C.Y.2    Ahn, K.J.3
  • 17
    • 84946935779 scopus 로고    scopus 로고
    • Dong-A ST Accessed 20 Oct 2015
    • Dong-A ST. 4Q 2014 performance results. 2015. http://en.donga-st.com/B05.da?method=IRResourceList. Accessed 20 Oct 2015.
    • (2015) 4Q 2014 Performance Results


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.