Pyridazines and their Benzo Derivatives

Comprehensive Heterocyclic Chemistry II: A Review of the Literature 1982-1995

Volumn 6, Issue , 1996, Pages 1-91

  Coates, William J ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

PYRIDAZINE;

EID: 84944056338     PISSN: None     EISSN: None     Source Type: Book    
DOI: 10.1016/B978-008096518-5.00117-9     Document Type: Chapter

References (321)

1. J.S. Morley J. Chem. Soc. 1951 1971
2. P.C. Coad R.A. Coad S. Clough J. Hyepock R. Salisbury C. Wilkins J. Org. Chem. 28 1963 218
3. R. Schonbeck E. Kloimstein Monatsh. Chem. 99 1968 15
4. G. Bachmann (BASF); Br. Pat. 1 168 291 (1969) ( Chem. Abstr. , 1970, 72 , 31 824).
5. J.A. Elvidge J.A. Pickett J. Chem. Soc., Perkin Trans. 1 1972 1483
6. G.M. Singerman Chem. Heterocycl. Compd. 27 1973 1
7. N.R. Patel Chem. Heterocycl. Comp. 27 1973 323
8. M. Tisler B. Stanovnik Chem. Heterocycl. Comp. 28 1973 1
9. S. Alazawe J.A. Elvidge J. Chem. Soc., Perkin Trans. 1 1974 696
10. P.H. Lacy D.C.C. Smith J. Chem. Soc., Perkin Trans. 1 1975 419
11. J.W. Barton Adv. Heterocycl. Chem. 24 1979 151
12. J.J. Bourguignon C.G. Wermuth J. Org. Chem. 46 1981 4889
13. C.A. Panetta A.S. Dixit Synthesis 1981 59
14. V.V. Mezheritskii D.M. Elisevich G.N. Dorofeenko Zh. Org. Khim. 17 1981 2444 Chem. Abstr. 96 1982 104 (167)
15. A. Katoh C. Kashima Y. Omote Heterocycles 19 1982 2283
16. H. Hara H.C. van der Plas J. Heterocycl. Chem. 19 1982 1285
17. C.H. Womack L.M. Martin G.E. Martin K. Smith J. Heterocycl. Chem. 19 1982 1447
18. H. Hiranuma S.I. Miller J. Org. Chem. 47 1982 5083
19. S. Tokita K. Hiruta S. Ishikawa K. Kitahara H. Nishi Synthesis 1982 854
20. B.J. Hussey R.A.W. Johnstone I.D. Entwistle Tetrahedron 38 1982 3775
21. D.M. Elisevich V.V. Mezheritskii G.N. Dorofeenko Zh. Org. Khim. 18 1982 415 Chem. Abstr. 96 1982 181 (227)
22. O. Schneider M. Hanack Angew. Chem., Int. Ed. Engl. 22 1983 784
23. G. Heinisch I. Kirchner I. Kurzmann G. Loetsch R. Waglechner Arch. Pharm. (Weinheim, Ger.) 316 1983 508
24. Y. Ikemi K. Matsumoto T. Uchida Heterocycles 20 1983 1009
25. P. Matyus E. Kasztreiner G. Szilagyi M. Soti P. Sohar Heterocycles 20 1983 2225
26. A. Krbavcic L. Povse B. Stanovnik Heterocycles 20 1983 2347
27. C.B. Rao P.V.N. Raju R. Flammang A. Maquestiau J. Elguero Heterocycles 20 1983 2385
28. L. Ceraulo L. Lamartina O. Migliara S. Petruso V. Sprio Heterocycles 20 1983 551
29. A. Amer H. Zimmer J. Heterocycl. Chem. 20 1983 1231
30. A. Counotte-Potman H.C. van der Plas J. Heterocycl. Chem. 20 1983 1259
31. I. Sircar J. Heterocycl. Chem. 20 1983 1473
32. C.O. Okafor R.N. Castle J. Heterocycl. Chem. 20 1983 199
33. D.V. Bautista G. Bullock F.W. Hartstock L.K. Thompson J. Heterocycl. Chem. 20 1983 345
34. D.J. Katz D.S. Wise L.B. Townsend J. Heterocycl. Chem. 20 1983 369
35. J. Baker W. Hedges J.W. Timberlake L.M. Trefonas J. Heterocycl. Chem. 20 1983 855
36. D.R. Carver T.D. Greenwood J.S. Hubbard A.P. Komin Y.P. Sachdeva J.F. Wolfe J. Org. Chem. 48 1983 1180
37. K. Jug J. Org. Chem. 48 1983 1344
38. I. Maeba K. Iwata F. Usami H. Furukawa J. Org. Chem. 48 1983 2998
39. H. Hiranuma S.I. Miller J. Org. Chem. 48 1983 3096
40. D.J. Katz D.S. Wise L.B. Townsend J. Org. Chem. 48 1983 3765
41. L. Lepage Y. Lepage Synthesis 1983 1018
42. A. Ohsawa T. Kawaguchi H. Igeta Synthesis 1983 1037
43. T. Sakamoto M. Shiraiwa Y. Kondo H. Yamanaka Synthesis 1983 312
44. C. Joliveau C.G. Wermuth Tetrahedron 39 1983 2295
45. M. Tisler B. Stanovnik 1st edn. Comp. Heterocycl. Chem. 3B 1984 1
46. G. Heinisch G. Loetsch Heterocycles 22 1984 1395
47. B. Stanovnik O. Bajt B. Belcic B. Koren M. Prhavc A. Stimac M. Tisler Heterocycles 22 1984 1545
48. B. Singh Heterocycles 22 1984 1801
49. D. Konwar D. Prajapati J.S. Sandhu T. Kametani T. Honda Heterocycles 22 1984 2483
50. K. Kaji H. Nagashima H. Oda Heterocycles 22 1984 675
51. K. Kaji H. Nagashima Y. Ohta K. Tabashi H. Oda J. Heterocycl. Chem. 21 1984 1249
52. N.P. Peet J. Heterocycl. Chem. 21 1984 1389
53. G. Heinisch R. Waglechner J. Heterocycl. Chem. 21 1984 1727
54. G. Allmaier G. Heinisch J. Heterocycl. Chem. 21 1984 435
55. R.P. Gagnier M.J. Halat B.A. Otter J. Heterocycl. Chem. 21 1984 481
56. W.D. Jones Jr. J.M. Kane A.D. Sill J. Heterocycl. Chem. 21 1984 889
57. S.F. Nelsen J. Org. Chem. 49 1984 1891
58. D.L. Boger R.S. Coleman J. Org. Chem. 49 1984 2240
59. V. Bakthavachalam M. D’Alarcao N.J. Leonard J. Org. Chem. 49 1984 289
60. D.L. Boger R.S. Coleman J.S. Panek D. Yohannes J. Org. Chem. 49 1984 4405
61. G. Heinisch R. Waglechner Monatsh. Chem. 115 1984 1171
62. L. Stefaniak J.D. Roberts M. Witanowski G.A. Webb Org. Magn. Reson. 22 1984 201
63. T. Sakamoto Y. Kondo M. Shiraiwa H. Yamanaka Synthesis 1984 245
64. S. Podergajs B. Stanovnik M. Tisler Synthesis 1984 263
65. I. Reichelt H.U. Reissig Synthesis 1984 786
66. M.F. El-Zohry M.I. Younes S.A. Metwally Synthesis 1984 972
67. K.K. Sharma K.B.G. Torssell Tetrahedron 40 1984 1085
68. M.F. Ismail F.A. El-Bassiouny H.A. Younes Tetrahedron 40 1984 2983
69. F.A. Neugebauer S. Kuhnhaeuser Angew. Chem., Int. Ed. Engl. 24 1985 596
70. D. Binder C.R. Noe K. Baumann J.M.F. Wildburger Arch. Pharm. (Weinheim, Ger.) 318 1985 243
71. T. Higashino M. Takemoto K. Tanji C. Iijima E. Hayashi Chem. Pharm. Bull. 33 1985 4193
72. A. M. Roe, W. J. Coates, R. A. Slater, S. P. Breukelman and G. D. Meakins (SKandF Labs); Eur. Pat. 138 344 (1985) ( Chem. Abstr. , 1985, 103 , 141 993).
73. K. Kamata O. Tsuge Heterocycles 23 1985 1675
74. F.D. Popp J. Kant Heterocycles 23 1985 2193
75. K. Makino G. Sakata Heterocycles 23 1985 2603
76. N. Haider G. Heinisch Heterocycles 23 1985 2651
77. A.T.M. Marcelis H.C. van der Plas Heterocycles 23 1985 683
78. S.P. Breukelman G.D. Meakins A.M. Roe J. Chem. Soc., Perkin Trans. 1 1985 1627
79. J. Kant F.D. Popp B.C. Uff J. Heterocycl. Chem. 22 1985 1065
80. W. Dostal G. Heinisch J. Heterocycl. Chem. 22 1985 1543
81. A. Camparini F. Ponticelli P. Tedeschi J. Heterocycl. Chem. 22 1985 1561
82. J. Taoufik J.M. Couquelet J.D. Couquelet P. Tronche J. Heterocycl. Chem. 22 1985 1615
83. J.P. Montheard J.C. Dubois J. Heterocycl. Chem. 22 1985 719
84. C. Kashima A. Katoh M. Fukasawa Y. Omote J. Heterocycl. Chem. 22 1985 927
85. D.W. Boykin P. Balakrishnan A.L. Baumstark J. Heterocycl. Chem. 22 1985 981
86. V.L. Styles R.W. Morrison Jr. J. Org. Chem. 50 1985 346
87. S.F. Nelsen N.P. Yumibe J. Org. Chem. 50 1985 4749
88. E. Fos J. Vilarrasa J. Fernández J. Org. Chem. 50 1985 4894
89. W. Adam A. Berkessel K. Hildenbrand E.M. Peters K. Peters H.G. von Schnering J. Org. Chem. 50 1985 4899
90. T. Sheradsky R. Moshenberg J. Org. Chem. 50 1985 5604
91. V. Konecny S. Kovac S. Varkonda Chem. Papers 39 1985 513
92. S.L. Spassov I.A. Atanassova M.A. Haimova Magn. Reson. Chem. 23 1985 795
93. L. Campayo B. Jimenez T. Manzano P. Navarro Synthesis 1985 197
94. G. Heinisch G. Loetsch Tetrahedron 41 1985 1199
95. M. Dietrich J. Heinze H. Fischer F.A. Neugebauer Angew. Chem., Int. Ed. Engl. 25 1986 1021
96. M.C. Gomez-Gil V. Gomez-Parra F. Sanchez T. Torres Arch. Pharm. (Weinheim, Ger.) 319 1986 60
97. E. Sato M. Hasebe Y. Kanaoka Chem. Pharm. Bull. 34 1986 3061
98. P.G. Tsoungas Gazz. Chim. Ital. 116 1986 405
99. K. Kamata O. Tsuge Heterocycles 24 1986 3059
100. V. Dal Piaz G. Ciciani S. Chimichi Heterocycles 24 1986 3143
101. W. Dostal G. Heinisch Heterocycles 24 1986 793
102. H. Maehr C.M. Liu N.J. Pallerini J. Smallheer L. Todaro T.H. Williams J.F. Blount J. Antibiot. 39 1986 17
103. S. Kaban J. Heterocycl. Chem. 23 1986 13
104. E.W. Badger W.H. Moos J. Heterocycl. Chem. 23 1986 1515
105. H. Heydt P. Eisenbarth K. Feith M. Regitz J. Heterocycl. Chem. 23 1986 385
106. K. Kamata O. Tsuge J. Heterocycl. Chem. 23 1986 557
107. H. Tondys H.C. van der Plas J. Heterocycl. Chem. 23 1986 621
108. G. Heinisch W. Holzer G.A.M. Nawwar J. Heterocycl. Chem. 23 1986 93
109. I.A. Shaikh F. Johnson A.P. Grollman J. Med. Chem. 29 1986 1329
110. T. Minami T. Chikugo T. Hanamoto J. Org. Chem. 51 1986 2210
111. T. Sheradsky R. Moshenberg J. Org. Chem. 51 1986 3123
112. D.L. Boger R.S. Coleman J. Org. Chem. 51 1986 3250
113. D.R. Andrews D.H.R. Barton R.H. Hesse M.M. Pechet J. Org. Chem. 51 1986 4819
114. C.W. Bird Tetrahedron 42 1986 89
115. G. Seitz R. Hoferichter R. Mohr Angew. Chem., Int. Ed. Engl. 26 1987 332
116. H. Yamazaki H. Harada K. Matsuzaki K. Yoshioka M. Takase E. Ohki Chem. Pharm. Bull. 35 1987 2243
117. H. Nagashima K. Ukai H. Oda Y. Masaki K. Kaji Chem. Pharm. Bull. 35 1987 350
118. H. Nagashima H. Oda J. Hida K. Kaji Chem. Pharm. Bull. 35 1987 421
119. F. Gomez Contreras M. Lora-Tamayo A.M. Sanz Heterocycles 25 1987 193
120. H. Nagashima H. Oda T. Hayakawa K. Kaji Heterocycles 26 1987 1
121. H. Zimmer A. Amer Heterocycles 26 1987 1177
122. A. Amer N. Rashed M.M. Abdel Rahman H. Zimmer Heterocycles 26 1987 1277
123. A. Amer K. Weisz H. Zimmer Heterocycles 26 1987 1853
124. E.S.H. El Ashry Y. El Kilany A. Amer Heterocycles 26 1987 2101
125. A. Ohsawa T. Itoh H. Igeta Heterocycles 26 1987 2677
126. D.R. Borthakur D. Prajapati J.S. Sandhu Heterocycles 26 1987 337
127. G. Heinisch G. Loetsch Heterocycles 26 1987 731
128. H. Matsuyama M. Kobayashi H.H. Wasserman Heterocycles 26 1987 85
129. R.L. Zey J. Heterocycl. Chem. 24 1987 1261
130. S. Sueur M. Lagrenee F. Abraham C. Bremard J. Heterocycl. Chem. 24 1987 1285
131. H.M.F. Allah R. Soliman J. Heterocycl. Chem. 24 1987 1745
132. M.S. Akhtar V.L. Sharma A.P. Bhaduri J. Heterocycl. Chem. 24 1987 23
133. E.S.H. El-Ashry A. Amer G.H. Labib M.M. Abdel Rahman A.M. El-Massry J. Heterocycl. Chem. 24 1987 63
134. W.B. Smith J. Heterocycl. Chem. 24 1987 745
135. D.W. Robertson N.D. Jones J.H. Krushinski G.D. Pollock J.K. Swartzendruber J.S. Hayes J. Med. Chem. 30 1987 623
136. T. Sheradsky R. Moshenberg J. Org. Chem. 52 1987 101
137. G. Lunn J. Org. Chem. 52 1987 1043
138. M. Balogh P. Laszlo K. Simon J. Org. Chem. 52 1987 2026
139. A. Hosomi S. Hayashi K. Hoashi S. Kohra Y. Tominaga J. Org. Chem. 52 1987 4423
140. M.S. Baird H.H. Hussain Tetrahedron 43 1987 215
141. T.H. Fisher J.C. Crook S. Chang Tetrahedron 43 1987 2443
142. U. Gruseck M. Heuschmann Tetrahedron Lett. 28 1987 6027
143. G. Scheffler J. Engel B. Kutscher W.S. Sheldrick P. Bell Arch. Pharm. (Weinheim, Ger.) 321 1988 205
144. G. Seitz R. Hoferichter Arch. Pharm. (Weinheim, Ger.) 321 1988 889
145. T. Miyamoto J. Matsumoto Chem. Pharm. Bull. 36 1988 1321
146. C. Rubat P. Coudert J. Couquelet P. Bastide J. Bastide Chem. Pharm. Bull. 36 1988 1558
147. H. Sawanishi S. Saito T. Tsuchiya Chem. Pharm. Bull. 36 1988 4240
148. C. Rubat P. Coudert P. Bastide P. Tronche Chem. Pharm. Bull. 36 1988 5000
149. F. Farina V. Martin M. Romanach F. Sanchez Heterocycles 27 1988 1431
150. E. Sato M. Hasebe Y. Kanaoka Heterocycles 27 1988 1665
151. Y. Tominaga Y. Ichihara A. Hosomi Heterocycles 27 1988 2345
152. R. Grote Y. Chen A. Zeeck Z. Chen H. Zaehner P. Mischnick-Luebbecke W.A. Koenig J. Antibiot. 41 1988 595
153. T.A. Smitka J.B. Deeter A.H. Hunt F.P. Mertz R.M. Ellis L.D. Boeck R.C. Yao J. Antibiot. 41 1988 726
154. R.G. Sutherland A.S. Abd El Aziz A. Piorko U.S. Gill C.C. Lee J. Heterocycl. Chem. 25 1988 1107
155. N. Haider G. Heinisch D. Lassnigg J. Heterocycl. Chem. 25 1988 119
156. P. Matyus G. Szilagyi E. Kasztreiner G. Rabloczky P. Sohar J. Heterocycl. Chem. 25 1988 1535
157. C.B. Ziegler Jr. N.A. Kuck S.M. Harris Y. Lin J. Heterocycl. Chem. 25 1988 1543
158. P.H. Olesen T. Kappe J. Becher J. Heterocycl. Chem. 25 1988 1719
159. J.W. Lyga J. Heterocycl. Chem. 25 1988 1757
160. P. Coudert J. Couquelet P. Tronche J. Heterocycl. Chem. 25 1988 799
161. A.T.M. Marcelis H. Tondijs H.C. van der Plas J. Heterocycl. Chem. 25 1988 831
162. R.L. Zey J. Heterocycl. Chem. 25 1988 847
163. J. Ezquerra J. Alvarez-Builla J. Heterocycl. Chem. 25 1988 917
164. D.L. Boger S.M. Sakya J. Org. Chem. 53 1988 1415
165. Z. Hou Y. Fujiwara H. Taniguchi J. Org. Chem. 53 1988 3118
166. C.F. Wilcox Jr. K.R. Lassila S. Kang J. Org. Chem. 53 1988 4333
167. R.E. Hackler B.A. Dreikorn G.W. Johnson D.L. Varie J. Org. Chem. 53 1988 5704
168. Y. Mugnier E. Laviron J. Org. Chem. 53 1988 5781
169. J.G. Samaritoni Org. Prep. Proceed. Int. 20 1988 117
170. L.W. Singh H. Ila H. Junjappa Synthesis 1988 89
171. M. Gebauer G. Heinisch G. Lotsch Tetrahedron 44 1988 2449
172. F. Effenberger J. Koenig Tetrahedron 44 1988 3281
173. P.G. Baraldi A. Barco S. Benetti S. Manfredini G.P. Pollini D. Simoni V. Zanirato Tetrahedron 44 1988 6451
174. G. Seitz R. Hoferichter R. Mohr Arch. Pharm. (Weinheim, Ger.) 322 1989 415
175. J. Nakayama T. Konishi A. Ishii M. Hoshino Bull. Chem. Soc. Jpn. 62 1989 2608
176. T. Miyamoto J. Matsumoto Chem. Pharm. Bull. 37 1989 93
177. M.J.S. Dewar A.J. Holder Heterocycles 28 1989 1135
178. F. Gomez Contreras M. Lora-Tamayo A.M. Sanz Heterocycles 28 1989 791
179. W.J. Coates A. McKillop Heterocycles 29 1989 1077
180. D. Villemin D. Goussu Heterocycles 29 1989 1255
181. J. Easmon G. Heinisch W. Holzer Heterocycles 29 1989 1399
182. V. Dal Piaz G. Ciciani M.P. Giovannoni G. Turco Heterocycles 29 1989 1595
183. P. Matyus N. Makk E. Kasztreiner G. Jerkovich Heterocycles 29 1989 67
184. G. Heinisch T. Huber C. Langer W. Goessler G. Kollenz J. Heterocycl. Chem. 26 1989 1009
185. M.D. Taylor K.R. Anderson E.W. Badger J. Heterocycl. Chem. 26 1989 1353
186. R.L. Zey G. Richter H. Randa J. Heterocycl. Chem. 26 1989 1437
187. C. Yaroslavsky P. Bracha R. Glaser J. Heterocycl. Chem. 26 1989 1649
188. B.D. Schober G. Megyeri T. Kappe J. Heterocycl. Chem. 26 1989 169
189. G. Heinisch T. Huber J. Heterocycl. Chem. 26 1989 1787
190. T.N. Srinivasan P.B. Sattur K.R. Rao A.S.B. Prasad E.D. Jemmis J. Heterocycl. Chem. 26 1989 553
191. P.Y. Boamah N. Haider G. Heinisch J. Heterocycl. Chem. 26 1989 933
192. P. Hughes J. Clardy J. Org. Chem. 54 1989 3260
193. K. Ohe S. Uemura N. Sugita H. Masuda T. Taga J. Org. Chem. 54 1989 4169
194. J.E. Oliver R.M. Waters W.R. Lusby J. Org. Chem. 54 1989 4970
195. O. Mo M. Yanez J. Elguero J. Mol. Struct. 60 1989 17
196. U.G. Wagner C. Kratky T. Kappe Monatsh. Chem. 120 1989 329
197. D.J. Pettibone Endocrinology (Baltimore) 125 1989 217
198. V. Dal Piaz G. Ciciani G. Turco Synthesis 1989 213
199. T. Kappe A. Pfaffenschlager W. Stadlbauer Synthesis 1989 666
200. A. Csampai K. Kormendy P. Sohar F. Ruff Tetrahedron 45 1989 5539
201. E. Sato Y. Ikeda Y. Kanaoka Chem. Pharm. Bull. 38 1990 1205
202. K. Sasamoto Y. Ohkura Chem. Pharm. Bull. 38 1990 1323
203. I. Takeuchi Y. Hamada K. Hatano Y. Kurono T. Yashiro Chem. Pharm. Bull. 38 1990 1504
204. T. Itoh M. Okada K. Nagata K. Yamaguchi A. Ohsawa Chem. Pharm. Bull. 38 1990 2108
205. H. Sawanishi S. Saito T. Tsuchiya Chem. Pharm. Bull. 38 1990 2992
206. C. Rubat P. Coudert B. Refouvelet P. Tronche P. Bastide J. Bastide Chem. Pharm. Bull. 38 1990 3009
207. E. Oishi N. Taido K. Iwamoto A. Miyashita T. Higashino Chem. Pharm. Bull. 38 1990 3268
208. H. Arakawa J. Ishida M. Yamaguchi M. Nakamura Chem. Pharm. Bull. 38 1990 3491
209. H. Yamazaki H. Harada K. Matsuzaki K. Yoshioka M. Takase E. Ohki Chem. Pharm. Bull. 38 1990 45
210. J. Kurita N. Kakusawa S. Yasuike T. Tsuchiya Heterocycles 31 1990 1937
211. E. Ravina C. Teran L. Santana N. Garcia I. Estevez Heterocycles 31 1990 1967
212. B. Singh G.Y. Lesher Heterocycles 31 1990 2163
213. H. Yamanaka S. Ohba Heterocycles 31 1990 895
214. P. Friedman K.F. Ferris Int. J. Quantum Chem., Quantum Chem. Symp. 24 1990 843
215. J. Nakayama R. Hasemi J. Am. Chem. Soc. 112 1990 5654
216. J. Nakayama A. Hirashima J. Am. Chem. Soc. 112 1990 7648
217. M. Nakagawa Y. Hayakawa K. Furihata H. Seto J. Antibiot. 43 1990 477
218. E. Licandro S. Maiorana A. Papagni D. Tarallo A.M.Z. Slawin D.J. Williams J. Heterocycl. Chem. 27 1990 1103
219. I. Perhauc C. Zheng J. Heterocycl. Chem. 27 1990 1313
220. A. Turck N. Plé L. Mojovic G. Quéguiner J. Heterocycl. Chem. 27 1990 1377
221. N. Haider G. Heinisch G. Kemetmueller J. Heterocycl. Chem. 27 1990 1645
222. M.M. Curzu G.A. Pinna D. Barlocco G. Cignarella J. Heterocycl. Chem. 27 1990 205
223. R.L. Zey M.L. Gross G.S. Groenewold J. Heterocycl. Chem. 27 1990 209
224. M.J. Kornet J. Heterocycl. Chem. 27 1990 2125
225. B.D. Schober G. Megyeri T. Kappe J. Heterocycl. Chem. 27 1990 471
226. J.P. Vors J. Heterocycl. Chem. 27 1990 579
227. B. Chantegrel C. Deshayes B. Pujol J. Zhong J. Heterocycl. Chem. 27 1990 927
228. W. J. Coates, H. D, Prain, M. L. Reeves and B. H. Warrington; 1990, 33 , 1735.
229. M.G. Bock R.M. Dipardo P.D. Williams D.J. Pettibone B.V. Clineschmidt R.G. Ball D.F. Veber R.M. Freidinger J. Med. Chem. 33 1990 2321
230. S.C. Benson J.L. Gross J.K. Snyder J. Org. Chem. 55 1990 3257
231. R.J. Mattson C.P. Sloan J. Org. Chem. 55 1990 3410
232. W.J. Coates A. MeKillop J. Org. Chem. 55 1990 5418
233. A.R. Katritzky V. Feygelman G. Musumarra P. Barczynski M. Szafran J. Prakt. Chem. 332 1990 853
234. A.R. Katritzky V. Feygelman G. Musumarra P. Barczynski M. Szafran J. Prakt. Chem. 332 1990 870
235. B.D. Schober T. Kappe Monatsh. Chem. 121 1990 565
236. G. Heinisch H. Frank G.P. Ellis G.G. West Progress in Medicinal Chemistry 1990 Elsevier Amsterdam
237. Y. Kamitori M. Hojo R. Masuda K. Kawasaki S. Takata J. Ida Synthesis 1990 467
238. A. Stimac B. Stanovnik M. Tisler L. Golic Tetrahedron 46 1990 6915
239. T.V. Lee A.J. Leigh C.B. Chapleo Tetrahedron 46 1990 921
240. G. Maier F. Fletcher H.O. Kalinowski R. Boese Angew. Chem., Int. Ed. Engl. 30 1991 1484
241. E. Ravina C. Teran N.G. Dominguez C.F. Masaguer J. Gil-Longo F. Orallo J.M. Calleja Arch. Pharm. (Weinheim, Ger.) 324 1991 455
242. G. Heinisch W. Holzer Can. J. Chem. 69 1991 972
243. Y. Eguchi Y. Sato S. Sekizaki M. Ishikawa Chem. Pharm. Bull. 39 1991 2009
244. K. Sasamoto Y. Ohkura Chem. Pharm. Bull. 39 1991 411
245. V. Dal Piaz G. Ciciani M.P. Giovannoni Heterocycles 32 1991 1173
246. T. Sakamoto N. Funami Y. Kondo H. Yamanaka Heterocycles 32 1991 1387
247. O.D. Hensens J. Antibiot. 44 1991 249
248. J.P. Vors J. Heterocycl. Chem. 28 1991 1043
249. M. Hahn G. Heinisch W. Holzer H. Schwarz J. Heterocycl. Chem. 28 1991 1189
250. S.Y. Choi S.G. Lee Y.J. Yoon J. Heterocycl. Chem. 28 1991 1235
251. B. Jelen A. Stimac B. Stanovnik M. Tisler J. Heterocycl. Chem. 28 1991 369
252. S.Y. Choi S.C. Shin Y.J. Yoon J. Heterocycl. Chem. 28 1991 385
253. A. Stimac B. Stanovnik M. Tisler J. Heterocycl. Chem. 28 1991 417
254. J.G. Samaritoni G. Babbitt J. Heterocycl. Chem. 28 1991 583
255. B.L. Mylari W.J. Zembrowski J. Org. Chem. 56 1991 2587
256. T. Brinck J.S. Murray P. Politzer R.E. Carter J. Org. Chem. 56 1991 2934
257. R.E. Johnson J. Org. Chem. 56 1991 5218
258. H.E. Katz M.L. Schilling J. Org. Chem. 56 1991 5318
259. F. Gavina A.M. Costero M.R. Andreu M.D. Ayet J. Org. Chem. 56 1991 5417
260. C.H. Weidner F.M. Michaels D.J. Beltman C.J. Montgomery D.H. Wadsworth B.T. Briggs M.L. Picone J. Org. Chem. 56 1991 5594
261. N. Haider Tetrahedron 47 1991 3959
262. A. Csampai K. Kormendy F. Ruff Tetrahedron 47 1991 4457
263. S.J. Clarke T.L. Gilchrist A. Lemos T.G. Roberts Tetrahedron 47 1991 5615
264. H. Uno S. Okada H. Suzuki Tetrahedron 47 1991 6231
265. N. Haider G. Heinisch J. Moshuber Tetrahedron 47 1991 8573
266. G. Maier F. Fleischer Tetrahedron Lett. 32 1991 57
267. N. Haider G. Heinisch J. Moshuber Arch. Pharm. (Weinheim, Ger.) 325 1992 119
268. K. Goerlitzer M. Boemeke Arch. Pharm. (Weinheim, Ger.) 325 1992 13
269. S. Ito K. Yamaguchi Y. Komoda Chem. Pharm. Bull. 40 1992 3327
270. C. Yamagami N. Takao Chem. Pharm. Bull. 40 1992 925
271. A. Miyashita T. Kawashima C. Iijima T. Higashino Heterocycles 33 1992 211
272. Y. Uchibori M. Umeno H. Yoshioka Heterocycles 34 1992 1507
273. S. Konno M. Sagi F. Siga H. Yamanaka Heterocycles 34 1992 225
274. T. Ogita A. Sato R. Enokita K. Susuki M. Ishii T. Negishi T. Okazaki K. Tamaki K. Tanzawa J. Antibiot. 45 1992 1723
275. K. Tanzawa M. Ishii T. Ogita K. Shimada J. Antibiot. 45 1992 1733
276. A.E. Mourad D.S. Wise L.B. Townsend J. Heterocycl. Chem. 29 1992 1583
277. S. Mataka O. Misumi W.H. Lin M. Tashiro K. Takahashi A. Torii J. Heterocycl. Chem. 29 1992 87
278. N. Klempier A. De Raadt H. Griengl G. Heinisch J. Heterocycl. Chem. 29 1992 93
279. J.E. Gready P.M. Hatton S. Sternhell J. Heterocycl. Chem. 29 1992 935
280. A. Melikian G. Schlewer J.-P. Chambon C.G. Wermuth J. Med. Chem. 35 1992 4092
281. K.B. Sharpless J. Org. Chem. 57 1992 2768
282. D.S. Perlow J.M. Erb N.P. Gould R.D. Tung R.M. Freidinger P.D. Williams D.F. Veber J. Org. Chem. 57 1992 4394
283. H. Tsukube H. Minatogawa M. Munakata M. Toda K. Matsumoto J. Org. Chem. 57 1992 542
284. G. Heinisch H. Kopelent-Frank G.P. Ellis D.K. Luscombe Progress in Medicinal Chemistry 1992 Elsevier Amsterdam
285. A. Csampai O. Farkas Tetrahedron 48 1992 1507
286. C.W. Bird Tetrahedron 48 1992 335
287. K. Kikuchi T. Nagano H. Hayakawa Y. Hirata M. Hirobe Anal. Chem. 65 1993 1794
288. R. Hoferichter U. Reimers G. Seitz Arch. Pharm. (Weinheim, Ger.) 326 1993 29
289. A. Kuno H. Sakai Y. Sugiyama H. Takasugi Chem. Pharm. Bull. 41 1993 156
290. W.J. Coates A. McKillop Heterocycles 35 1993 1313
291. M. Takahashi H. Kotashima T. Saitoh Heterocycles 35 1993 909
292. K.J. Hwang K.H. Park Heterocycles 36 1993 219
293. E. Zara-Kaczian P. Matyus Heterocycles 36 1993 519
294. P. Matyus K. Czako A. Behr I. Varga B. Podanyi M. von Arnim P. Varkonyi Heterocycles 36 1993 785
295. H. Durr R. Schwarz C. Andreis I. Willner J. Am. Chem. Soc. 115 1993 12 362
296. E.J. Corey M.C. Noe J. Am. Chem. Soc. 115 1993 12 579
297. E.J. Corey M.C. Noe S. Sarshar J. Am. Chem. Soc. 115 1993 3828
298. K. Sugawara S. Toda T. Moriyama M. Konishi T. Oki J. Antibiot. 46 1993 928
299. A.E. Mourad D.S. Wise L.B. Townsend J. Heterocycl. Chem. 30 1993 1365
300. S.G. Hegde C.R. Jones J. Heterocycl. Chem. 30 1993 1501
301. A.P. Krapcho M.J. Maresch A.L. Helgason K.E. Rosner M.P. Hacker J. Heterocycl. Chem. 30 1993 1597
302. S. Shilcrat I. Lantos M. McGuire L. Pridgeon L. Davis D. Eggleston D. Staiger L. Webb J. Heterocycl. Chem. 30 1993 1663
303. G. Heinisch T. Langer J. Heterocycl. Chem. 30 1993 1685
304. P.S. Ray J. Boute C.A. Webster M.J. Manning J. Heterocycl. Chem. 30 1993 45
305. J.P. Chupp C.R. Jones M.L. Dahl J. Heterocycl. Chem. 30 1993 789
306. W. Amberg Y.L. Bennani R.K. Chadha G.A. Crispino W.D. Davis J. Hartung K.S. Jeong Y. Ogino T. Shibata K.B. Sharpless J. Org. Chem. 58 1993 844
307. S.E. Galembeck N.B. da Costa Jr. M.N. Ramos B.de.B. Neto J. Mol. Struct. 101 1993 97
308. W.J. Coates A. McKillop Synthesis 1993 334
309. P.N.W. Baxter J.-M. Lehn J. Fischer M.-T. Youinou Angew. Chem., Int. Ed. Engl. 33 1994 2284
310. D. Toussaint J. Suffert C.G. Wermuth Heterocycles 38 1994 1273
311. P. Matyus K. Fuji K. Tanaka Heterocycles 38 1994 1957
312. G. Heinisch B. Matuszczak K. Mereiter Heterocycles 38 1994 2081
313. H.C. Kolb P.G. Andersson K.B. Sharpless J. Am. Chem. Soc. 116 1994 1278
314. I. Henderson K.B. Sharpless C.-H. Wong J. Am. Chem. Soc. 116 1994 558
315. Z.-M. Wang H.C. Kolb K.B. Sharpless J. Org. Chem. 59 1994 5104
316. W.J. Coates S.T. Flynn Z.-X. Guo A. McKillop poster P-7 presented at the 4th Int. Symp. on the Chemistry and Pharmacology of Pyridazines 1994 Bled Slovenia
317. T. Kappe Acta Chim. Slovenica 41 1994 219
318. G. Cignarella D. Barlocco J. Heterocycl. Chem. 32 1995 79
319. M. Kocevar P. Mihorko S. Polanc J. Org. Chem. 60 1995 1466
320. H. Zimmer A.R. Safwat D. Ho A. Amer M. Badawi J. Org. Chem. 60 1995 1908
321. N. Plé A. Turck K. Couture G. Quéguiner J. Org. Chem. 60 1995 3781