1,4-Diazepines

Comprehensive Heterocyclic Chemistry II: A Review of the Literature 1982-1995

Volumn 9, Issue , 1996, Pages 151-182

  Tucker, Howard ^a   Le Count, David J ^b  

^a ASTRAZENECA   (United Kingdom)

^b NONE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

DIAZEPINES;

EID: 84944049079     PISSN: None     EISSN: None     Source Type: Book    
DOI: 10.1016/B978-008096518-5.00214-8     Document Type: Chapter

References (120)

1. G. Schwarzenbach K. Lutz Helv Chim. Acta 23 1940 1139
2. J.A. Barltrop II C.G. Richards D.M. Russell G. Ryback J. Chem. Soc. 1959 1192
3. S.C. Bell S.J. Childress J. Org. Chem. 27 1962 1691
4. C.S. Hofmann S.R. Safir J. Org. Chem. 27 1962 3565
5. S. Cbell C. Gochman S.J. Childress J. Org. Chem. 28 1963 3010
6. S.C. Bell S.J. Childress J. Org. Chem. 29 1964 506
7. H.A. Staab F. Vögtle Chem. Ber. 98 1965 2701
8. H.A. Staab C. Wünsche Chem. Ber. 98 1965 3479
9. P. Linscheid J.-M. Lehn Bull. Soc. Chim. Fr. 1967 992
10. W. Sadée J. Med. Chem. 13 1970 475
11. Y. Okamoto T. Ueda J. Chem. Soc., Chem. Comm. 1973 367
12. D. Lloyd R.K. Mackie H. McNab D.R. Marshall J. Chem. Soc., Perkin Trans. 2 1973 1729
13. L. Sternbach F. Sancilio J. Blount J. Med. Chem. 17 1974 374
14. R.H. Begland D.R. Hartter F.N. Jones D.J. Sam W. Sheppard O. Webster F. Weigert J. Org. Chem. 39 1974 2341
15. P. Levillain M. Bertucat B. Perrot Eur. J. Med. Chem. 10 1975 433
16. D. Lloyd H. McNab D.R. Marshall J. Chem. Soc., Perkin Trans. 1 1975 1260
17. P. Nedenskov M. Mandrup Acta Chem. Scand. Ser. B 31 1977 701
18. T. Blair G. Webb J. Med. Chem. 20 1977 1206
19. L.V. Pribega V.I. Avramenko Z.F. Solomko A.M. Sipyagin Chem. Heterocycl. Compd. (Engl. Transl.) 1978 1270
20. S.P. Singh S.S. Parmar S.A. Farnum V.I. Stenberg J. Heterocycl. Chem. 15 1978 1083
21. H. Natsugari K. Meguro Y. Kuwada Chem. Pharm. Bull. 27 1979 2608
22. H. Natsugari Y. Kuwada Chem. Pharm. Bull. 27 1979 2618
23. T. Kovac M. Oklobdzija V. Sunjić F. Kaifez J. Heterocycl. Chem. 16 1979 1449
24. R.W. Luceck W.A. Garland W. Dairman Fed. Proc. 38 1979 541
25. M. Majchrzak A. Kotelko R. Guryn Pol. J. Chem. 53 1979 2135
26. H.-G. Schecker G. Zinner Arch. Pharm. (Weinheim, Ger.) 313 1980 926
27. R. Haran J.P. Tuchagues J. Heterocycl. Chem. 17 1980 1483
28. K. Kovar D. Linden Arch. Pharm. (Weinheim, Ger.) 314 1981 186
29. B. Unterhalt Arch. Pharm. (Weinheim, Ger.) 314 1981 733
30. T. Mukai T. Kumagai Y. Yamashita Heterocycles 15 1981 1569
31. E. Decorte R. Toso A. Sega V. Sunjić Z. Ružić-Toroš B. Kojic-Prodić N. Bresciani-Pahor G. Nardin L. Randaccio Helv. Chim. Acta 64 1981 1145
32. D. Lloyd K.S. Tucker D.R. Marshall J. Chem. Soc., Perkin Trans. 1 1981 726
33. R. Isaksson T. Liljefors J. Chem. Soc., Perkin Trans. 2 1981 1344
34. L. Capuano K. Gärtner J. Heterocycl. Chem. 18 1981 1341
35. J.R. Wolfe B.E. Reitter Y.P. Sachdeva J. Org. Chem. 46 1981 3945
36. A. Patra A.K. Mukhopadhyay A.K. Mitra A.K. Acharyya Org. Magn. Reson. 15 1981 99
37. I. Ueda M. Matsuo K. Taniguchi Chem. Pharm. Bull. 30 1982 1141
38. I. Ueda T. Watanabe M. Matsuo K. Taniguchi Chem. Pharm. Bull. 30 1982 1473
39. T. Watanabe M. Matsuo K. Taniguchi I. Ueda Chem. Pharm. Bull. 30 1982 1477
40. J.P. Freeman D.J. Duchamp C.G. Chidester G. Slomp J. Szmuszkovicz M. Raban J. Am. Chem. Soc. 104 1982 1380
41. D. Lloyd A. Cuthbertson C. Glidewell J. Chem. Res. (S) 1982 80
42. F. Hollywood Z.U. Khan E.F.C. Scriven R.K. Smalley H. Suschitzky R. Hull J. Chem. Soc., Perkin Trans. 1 1982 431
43. K. Kostka M. Owczarek Pol. J. Chem. 56 1982 1605
44. K. Kostka M. Owczarek Pol. J. Chem. 56 1982 83
45. T. Gunda C. Enebäck Acta Chem. Scand. Ser. B 37 1983 75
46. L. Crombie R.C.F. Jones S. Osborne A.R. Mat-Zin J. Chem. Soc., Chem. Commun. 1983 959
47. H. Quast H.M. Seidenspinner J. Stawitz Liebigs Ann. Chem. 1983 1207
48. H. Quast H.M. Seidenspinner J. Stawitz Liebigs Ann. Chem. 1983 1230
49. T.A. Hamor I.L. Martin G.P. Ellis G.B. West Progress in Medicinal Chemistry vol. 20 1983 Elsevier Science Publishers Amsterdam
50. T.A. Scahill S.L. Smith Org. Magn. Reson. 21 1983 621
51. A. Lin J. Hoch Arzneim.-Forsch. 34 1984 640
52. J. Lehmann G. Kraft Arch. Pharm. (Weinheim, Ger.) 317 1984 595
53. H. Quast W. Von der Saal Chem. Ber. 117 1984 1591
54. J.T. Sharp 1st edn. Comp. Heterocycl. Chem. 7 1984 593
55. H. Sawanishi K. Tajima M. Osada T. Tsuchiya Chem. Pharm. Bull. 32 1984 4694
56. S.R. Boyer G. Fitchett J.H. Wasley G. Zaunius J. Heterocycl. Chem. 21 1984 833
57. G. Loew J. Nienow M. Poulsen Mol. Pharmacol. 26 1984 19
58. S. Kasprzyk R. Kolinski Pol. J. Chem. 58 1984 721
59. J. Kurita K. Iwata H. Sakai T. Tsuchiya Chem. Pharm. Bull. 33 1985 4572
60. Y. Ohba I. Matsukura Y. Fukazawa T. Nishiwaki Heterocycles 23 1985 287
61. D. Obrecht B. Scholl H. Heimgartner Helv. Chim. Acta 68 1985 465
62. T. Nishio T. Tokunaga Y. Omote J. Heterocycl. Chem. 22 1985 405
63. T.A. Scahill S.L. Smith Magn. Reson. Chem. 23 1985 280
64. P.L. Southwick C.H. Chou T.E. Fink J.R. Kirchner Synthesis 1985 339
65. S.R. Salman S.T. Hamdi K.Y. Ahmed Can. J. Spectrosc. 31 1986 127
66. A. Calsy J. King D. Lloyd C. Reichardt M. Struthers Liebigs Ann. Chem. 1986 1387
67. C.Y. Fiakpui E.E. Knaus Can. J. Chem. 65 1987 1158
68. H. Sawanishi K. Tajima T. Tsuchiya Chem. Pharm. Bull. 35 1987 1179
69. J. Kurita K. Iwata T. Tsuchiya Chem. Pharm. Bull. 35 1987 3166 Chem. Abstr. 108 1988 167 439
70. H. Sawanishi K. Tajima T. Tsuchiya Chem. Pharm. Bull. 35 1987 3175
71. H. Sashida A. Fujii T. Tsuchiya Chem. Pharm. Bull. 35 1987 3182
72. H. Sashida A. Fujii T. Tsuchiya Chem. Pharm. Bull. 35 1987 4110
73. L. Bonsignore S. Cabiddu G. Loy D. Secci Heterocycles 26 1987 1619
74. J. Kurita T. Yoneda N. Kakusawa T. Tsuchiya Heterocycles 26 1987 3085
75. M. Bock R. DiPardo B. Evans K. Rittle D. Veber R. Freidinger J. Hirshfield J.P. Springer J. Org. Chem. 52 1987 3232
76. C.V. Ratnam P.S. Reddy G. Mohiuddin Magn. Reson. Chem. 25 1987 642
77. K. Kostka M. Owczarek Pol. J. Chem. 61 1987 103
78. O.P. Goel U. Krolls Synthesis 1987 162
79. T. Fujii T. Saito T. Fujisawa Heterocycles 27 1988 1163
80. C. Betschart B. Schmidt D. Seebach Helv. Chim. Acta 71 1988 1999
81. Y.K. Srivastava S. Singh B.L. Verma Natl. Acad. Sci. Lett. (India) 11 1988 387
82. M. Andreocci C. Cauletti K.-D. Schleinitz U. Hess Spectrochim. Acta, Part A 44A 1988 1079
83. U. Schëllkopf J. Mittendorf Angew. Chem., Int. Ed. Engl. 101 1989 613
84. M.C. Aversa P. Bonaccorsi P. Giannetto D.A. Leigh J. Heterocycl. Chem. 26 1989 1619
85. M.G. Bock R.M. DiPardo B.E. Evans K.E. Rittle W.L. Whitter D.F. Veber P.S. Anderson R.M. Freidinger J. Med. Chem. 32 1989 13
86. J.T. Sharp M.F. Ansell Rodd’s Chemistry of Carbon Compounds 1989 Elsevier Amsterdam 201 suppl. to vol. IV, part K
87. J. Kurita T. Yoneda N. Kakusawa T. Tsuchiya Chem. Pharm. Bull. 38 1990 2911
88. T. Tsuchiya H. Sashida M. Kaname Chem. Pharm. Bull. 38 1990 2919
89. K. Matsumoto H. Minatogawa M. Toda M. Munakata Heterocycles 31 1990 1217
90. N.W. Gilman P. Rosen J.V. Earley C. Cook L.J. Todaro J. Am. Chem. Soc. 112 1990 3969
91. J.R. Ascenso M.A. Santos J.J. Frausto da Silva M. Candida T.A. Vaz M.G.B. Drew J. Chem. Soc., Perkin Trans. 2 1990 2211
92. M. Block R. DiPardo B. Evans K. Rittle W. Whotter D. Veber R. Freidinger R. Chang T. Chen V. Lotti J. Med. Chem. 33 1990 450
93. V. Merluzzi K.D. Hargrave M. Labadia K. Grozinger M. Skoog J.C. Wu C.-K. Shih K. Eckner S. Hattox J. Adams A.S. Rosenthal R. Faanes R.J. Eckner R.A. Koup J.L. Sullivan Science 250 1990 1411
94. L.D. Basanagoudar C.S. Mahajanshetti S.B. Dambal Indian J. Chem., Sect. B 30B 1991 1018
95. A. Hasnaoui A. Baouid J.P. Lavergne J. Heterocycl. Chem. 28 1991 73
96. M. Kukla H. Breslin C. Diamond P. Grous C. Ho M. Miranda J. Rodgers R. Sherrill E. De Clerq R. Pauwels K. Andries L. Moens M. Janssen P. Janssen J. Med. Chem. 34 1991 3187
97. T. Shono N. Kise E. Shirakawa H. Matsumoto E. Okazaki J. Org. Chem. 56 1991 3063
98. R.I. Fryer A. Walser E.C. Taylor The Chemistry of Heterocyclic Compounds vol. 50 1991 Interscience New York 1
99. M.-C. Hsu A.D. Schutt M. Holly L.W. Slice M.I. Sherman D.D. Richman M.J. Potash D.J. Volsky Science 254 1991 1799
100. J.Y. Mérour J.Y. Coadou Tetrahedron Lett. 32 1991 2469
101. B.A. Bunin J. Ellman J. Am. Chem. Soc. 114 1992 10 997
102. C. Betschart L.S. Hegedus J. Am. Chem. Soc. 114 1992 5010
103. F. Povazanec B. Decroix J. Morel J. Heterocycl. Chem. 29 1992 1507
104. A. Padwa D.N. Kline S.S. Murphree P.E. Yeske J. Org. Chem. 57 1992 298
105. J. Messinger V. Buss J. Org. Chem. 57 1992 3320
106. K.A. Parker C.A. Coburn J. Org. Chem. 57 1992 97
107. J. Barluenga M. Tomas A. Ballesteros J. Kong Synthesis 1992 106
108. D. Lloyd H. McNab A.R. Katritzky Adv. Heterocycl. Chem. 56 1993 1
109. M. Chambers S. Hobbs S. Fletcher V. Matassa P. Mitchell A. Watt R. Baker S. Freedman S. Patel A. Smith Bioorg. Med. Chem. Lett. 3 1993 1919
110. M. Chammache E.M. Essassi R. Zniber Bull. Soc. Chim. Belg. 102 1993 89
111. J. Barluenga C.R. Perez J. Gonzalez J. Joglar F.L. Ortiz S. Fustero Bull. Soc. Chim. Fr. 130 1993 566
112. J. Barluenga M. Tomás A. Ballesteros J.S. Kong S. Garcia-Granda A. Aguirre J. Chem. Soc., Chem. Commun. 1993 217
113. S. Hamdi K. Ahmed Can. J. Spectrosc. 38 1993 82
114. A. Benalil A. Guerin B. Carboni M. Vaultier J. Chem. Soc., Perkin Trans. 1 1993 1061
115. R.I. Fryer J.C. Pinto R.B. Upasani J. Heterocycl. Chem. 30 1993 945
116. M. Akssira M. Boumzebra H. Kasmi A. Dahdouh M. Roumestant P. Viallefont Synth. Commun. 23 1993 2265
117. G.A. Showell S. Bourrain J.G. Neduvelil S.R. Fletcher R. Baker A.P. Watt A.E. Fletcher S.B. Freedman J.A. Kemp G.R. Marshall S. Patel A.J. Smith V.G. Matassa J. Med. Chem. 37 1994 719
118. S. Bourrain G. Showell Synthesis 1994 505
119. M. Akssira M. Boumzebra H. Kasmi A. Dahdouh Tetrahedron 50 1994 9051
120. R.R. Webb II P.C. Barker M. Baier M.G. Reynolds K.D. Robarge B.K. Blackburn M.H. Tischler K.J. Weese Tetrahedron Lett. 35 1994 2113