1,2,5-Thiadiazoles

Comprehensive Heterocyclic Chemistry II: A Review of the Literature 1982-1995

Volumn 4, Issue , 1996, Pages 355-377

  Shinkai, Ichiro ^a   Reider, Paul J ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

5]THIADIAZOLE;

EID: 84944034756     PISSN: None     EISSN: None     Source Type: Book    
DOI: 10.1016/B978-008096518-5.00087-3     Document Type: Chapter

References (208)

1. D. Shew Diss. Abstr. 20 1959 1593
2. L.M. Weinstock Diss. Abstr. 19 1959 3136
3. W.R. Sherman R.C. Elderfield Heterocyclic Compounds vol. 7 1961 Wiley New York 579 chap. 7
4. V.G. Pesin A.M. Khaletskii V.A. Sergeev J. Gen. Chem. USSR (Engl. Transl.) 33 1963 1714
5. S.F. Mason Phys. Methods Heterocycl. Chem. 2 1963 61
6. J.M. Ross W.C. Smith J. Am. Chem. Soc. 86 1964 2861
7. V. Bertini P. Pino Angew. Chem., Int. Ed. Engl. 4 1965 239
8. N.P. Buu-Hoî P. Jacquignon M. Mangane J. Chem. Soc., Chem. Commun. 1965 624
9. C.W. Haigh M.H. Palmer B. Semple J. Chem. Soc. 1965 6004
10. B. Šoptrajanov G.E. Ewing Spectrochim. Acta 22 1966 1417
11. H. Beecken Chem. Ber. 100 1967 2170
12. I.W. Stapelton Diss. Abstr. Int. B 27 1967 4330
13. V. Bertini A. De Munno Gazz. Chim. Ital. 97 1967 1614
14. V. Bertini Gazz. Chim. Ital. 97 1967 1870
15. E. Benedetti G. Sbrana V. Bertini Gazz. Chim, Ital. 97 1967 379
16. N.M. Atherton J.N. Ockwell R. Dietz J. Chem. Soc. (A) 1967 771
17. D.M. Mulvey L.M. Weinstock J. Heterocycl. Chem. 4 1967 445
18. L.M. Weinstock P. Davis B. Handelsman R. Tull J. Org. Chem. 32 1967 2823
19. E.I. Fedin Z.V. Todres L.S. Efros Khim. Geterotsikl. Soedin. 1967 297
20. S.P. Solodovnikov Z.V. Todres Khim. Geterotsikl. Soedin. 1967 811
21. L.M. Weinstock P.J. Pollack Adv. Heterocycl. Chem. 9 1968 107
22. W. Wucherpfenning Chem. Ber. 101 1968 371
23. T. Naito J. Okumura K. Kasai Chem. Pharm. Bull. 16 1968 544
24. G. Tuchtehagen K. Ruehlmann Justus Liebigs Ann. Chem. 711 1968 174
25. V.G. Pesin Chem. Heterocycl. Compd. (Engl. Transl.) 5 1969 180
26. V.G. Pesin V.A. Sergeev Chem. Heterocycl. Compd. (Engl. Transl.) 5 1969 53
27. M. Kamiya S. Katayama Y. Akahori Chem. Pharm. Bull. 17 1969 1821
28. N.K. Ray P.T. Narasimhan Indian J. Chem. 7 1969 97
29. J.D. Bowler R.H. Schlessinger J. Am. Chem. Soc. 91 1969 6891
30. V.G. Pesin Khim. Geterotsikl. Soedin. 1969 235
31. L. Braier P.V. Petrovskii Z.V. Todres E.I. Fedin Khim. Geterotsikl. Soedin. 1969 62
32. M. Carmack I.W. Stapleton R.Y. Wen Org. Prep. Proceed. Int. 1 1969 255
33. F.L. Tobiason J.H. Goldstein Spectrochim. Acta, Part A 25 1969 1027
34. H.H. Hoerhold H. Eibisch Tetrahedron 25 1969 4277
35. G. Kresze H. Grill Tetrahedron Lett. 10 1969 4117
36. D. Dal Monte E. Sandri W. Cere Ann. Chim. (Rome) 60 1970 801
37. M. Kamiya Y. Akahori Bull. Chem. Soc. Jpn. 43 1970 268
38. A. G. Oesterreichische Stickstoffwerke; Br. Pat. 1 190 359 (1970).
39. R.G. Micetich Can. J. Chem. 48 1970 2006
40. A. Lawson R.B. Tinkler Chem. Rev. 70 1970 593
41. K. Pilgram M. Zupan R. Skiles J. Heterocycl. Chem. 7 1970 629
42. K. Pilgram J. Org. Chem. 35 1970 1165
43. V.G. Pesin Russ. Chem. Rev. (Engl. Transl.) 39 1970 923
44. G.H. Harts K.B. De Roos C.A. Salemink Recl. Trav. Chim. Pays-Bas 89 1970 5
45. J. Marn B. Stanovnik M. Tisler Croat Chem. Acta 43 1971 101 Chem. Abstr. 75 1971 98 523
46. V. Bertini A. De Munno Gazz. Chim. Ital. 101 1971 259
47. D.L. Forster T.L. Gilchrist C.W. Rees J. Chem. Soc. (C) 1971 993
48. D. Pichler R.N. Castle J. Heterocycl. Chem. 8 1971 441
49. C.W. Bird C.K. Wong Tetrahedron Lett. 12 1971 2143
50. A.W. Richardson Can. J. Chem. 50 1972 627
51. A.R. Katritzky Y. Takeuchi J. Chem. Soc., Perkin Trans. 2 1972 1682
52. E.F. Elslager N.F. Haley J. Heterocycl. Chem. 9 1972 1109
53. K.T. Potts R. Armbruster J. Heterocycl. Chem. 9 1972 651
54. J.E. Oliver S.C. Chang R.T. Brown J.B. Stokes A.B. Borkovec J. Med. Chem. 15 1972 315
55. R.W. Begland D.R. Hartter J. Org. Chem. 37 1972 4136
56. M. Haake H. Fode B. Eichenauer Justus Liebigs Ann. Chem. 759 1972 107
57. C.L. Khetrapal A.V. Patankar Mol. Cryst. Liq. Cryst. 15 1972 367
58. D.E. Horning J.M. Muchowski Can. J. Chem. 51 1973 2349
59. A.W. Richardson Can. J. Chem. 51 1975 680
60. A. Matsumoto M. Yoshida O. Simamura Bull. Chem. Soc. Jpn. 47 1974 1493
61. K. Pilgram J. Heterocycl. Chem. 11 1974 835
62. R.W. Begland D.R. Hartter D.S. Donald A. Cairncross W.A. Sheppard J. Org. Chem. 39 1974 1235
63. G.W.H. Cheeseman C.J. Turner Org. Magn. Reson. 6 1974 430
64. G. Ege E. Beisiegel Synthesis 1974 22
65. A.S. Angeloni D. Dal Monte S. Pollicino E. Sandri G. Scapini Tetrahedron 30 1974 3839
66. C.L. Pedersen J. Møller Acta Chem. Scand., Ser. B 29 1975 483
67. F.C.V. Larsson S.O. Lawesson I. Jardine R.I. Reed Acta Chem. Scand., Ser. B 29 1975 622
68. V.V. Dovlatyan R.S. Mirzoyan Arm. Khim. Zh. 28 1975 412 Chem. Abstr. 83 1975 206 174
69. Y.C. Tong J. Heterocycl. Chem. 12 1975 451
70. A.P. Komin M. Carmack J. Heterocycl. Chem. 12 1975 829
71. R.Y. Wen A.P. Komin R.W. Street M. Carmack J. Org. Chem. 40 1975 2743
72. A.P. Komin R.W. Street M. Carmack J. Org. Chem. 40 1975 2749
73. R. Appel J.R. Lundehn E. Lassmann Chem. Ber. 109 1976 2442
74. F.S. Mikhailitsyn A.F. Bekhli Chem. Heterocycl. Compd. (Engl. Transl.) 12 1976 61
75. D.R. Jones C.H. Wang D.H. Christensen O.F. Nielson J. Chem. Phys. 64 1976 4475
76. A.P. Komin M. Carmack J. Heterocycl. Chem. 13 1976 13
77. L.M. Weinstock D.M. Mulvey R. Tull J. Org. Chem. 41 1976 3121
78. R. Appel J.R. Lundehn Chem. Ber. 110 1977 3205
79. T. Honma Y. Tada Heterocycles 6 1977 1985
80. M. Tashiro S. Matake K. Takahashi Heterocycles 6 1977 933
81. D.H.R. Barton W.A. Bubb J. Chem. Soc., Perkin Trans. 1 1977 916
82. C.A. Veracini A. De Munno V. Bertini M. Longeri G. Chidichimo J. Chem. Soc., Perkin Trans. 2 1977 561
83. J.A. Deyrup H.L. Gingrich J. Org. Chem. 42 1977 1015
84. C.L. Pedersen C. Lohse M. Poliakoff Acta Chem. Scand., Ser. B 32 1978 625
85. M. Preiss Chem. Ber. 111 1978 1915
86. P.C. Belanger Can. J. Chem. 56 1978 722
87. T. Uno K. Takagi M. Tomoeda Chem. Pharm. Bull. 26 1978 3896
88. G.H. Hartman S.E. Biffar L.M. Weinstock R. Tull J. Org. Chem. 43 1978 960
89. I.D. Entwistle T. Gilkerson R.A.W. Johnstone R.P. Telford Tetrahedron 34 1978 213
90. L. Capuano G. Urhahn A. Willmes Chem. Ber. 112 1979 1012
91. O. Glemser J.M. Shreeve Inorg. Chem. 18 1979 213
92. S. Mataka K. Takahashi S. Ishii M. Tashiro J. Chem. Soc., Perkin Trans. 1 1979 2905
93. S. Mataka K. Takahashi Y. Yamada M. Tashiro J. Heterocycl. Chem. 16 1979 1009
94. J.D. Warren V.J. Lee R.B. Angier J. Heterocycl. Chem. 16 1979 1617
95. R.B. Meyer Jr. E.B. Skibo J. Med. Chem. 22 1979 944
96. J. Rokach P. Hamel Y. Girard G. Reader J. Org. Chem. 44 1979 1118
97. H. Buchwald K. Ruehlmann J. Organomet. Chem. 166 1979 25
98. S. Mataka A. Hosoki K. Takahashi M. Tashiro Synthesis 1979 524
99. S. Mataka K. Takahashi M. Tashiro Synthesis 1979 687
100. T. Uno K. Takagi M. Tomoeda Chem. Pharm. Bull. 28 1980 1909
101. S. Mataka A. Hosoki K. Takahashi M. Tashiro J. Heterocycl. Chem. 17 1980 1681
102. B. Danylec M. Davis J. Heterocycl. Chem. 17 1980 537
103. R. Beckert R. Mayer J. Prakt. Chem. 322 1980 273
104. V.L. Savel’ev O.S. Artamonova T.G. Afanas’eva V.A. Zagorevskii Khim. Geterotsikl. Soedin. 1980 853 Chem. Abstr. 93 1980 186 256
105. S. Mataka T. Takahashi M. Tashiro Y. Tsuda Synthesis 1980 842
106. V. Bertini F. Lucchesini A. De Munno Tetrahedron 36 1980 1245
107. S. Karady J.S. Amato D. Dortmund L.M. Weinstock Heterocycles 16 1981 1561
108. P.S. Rao V. Veeranagaiah Indian J. Chem., Sect. B 20 1981 111
109. K. Masuda J. Adachi K. Nomura J. Chem. Soc., Perkin Trans. 1 1981 1033
110. D.L. Boger C.E. Brotherton J. Heterocycl. Chem. 18 1981 1247
111. K.T. Potts R.D. Cody R.J. Dennis J. Org. Chem. 46 1981 4065
112. K.S. Sharma S. Kumari R.P. Singh Synthesis 1981 316
113. M. Geisel R. Mews Chem. Ber. 115 1982 2135
114. M.R. Bryce P. Hanson J.M. Vernon J. Chem. Soc., Chem. Commun. 1982 299
115. K.S. Sharma R.P. Singh Indian J. Chem., Sect. B 21 1982 65
116. J.S. Amato S. Karady R.A. Reamer H.B. Schlegel J.P. Springer L.M. Weinstock J. Am. Chem. Soc. 104 1982 1375
117. W.J. Spillane J. Chem. Res. (S) 3 1982 84
118. P.E. Marecki J.N. Wemple G.P. Butke J. Heterocycl. Chem. 19 1982 1247
119. S. Mataka K. Takahashi T. Imura M. Tashiro J. Heterocycl. Chem. 19 1982 1481
120. W.C. Lumma Jr. J. Med. Chem. 25 1982 207
121. A.A. Algieri G.M. Luke R.T. Standridge M. Brown R.A. Partyka R.R. Crenshaw J. Med. Chem. 25 1982 210
122. S. Mataka A. Hosoki K. Takahashi M. Tashiro Synthesis 11 1982 976
123. D.M. Goldish B.W. Axom H.W. Moore Heterocycles 20 1983 187
124. S. Mataka K. Takahashi M. Tashiro Heterocycles 20 1983 2047
125. W. Sliwa A. Thomas Heterocycles 20 1983 71
126. A.H. Cowley S.K. Mehrotra H.W. Roesky Inorg. Chem. 22 1983 2095
127. A. Bhattacharyya A.A. Bhattacharyya Indian J. Chem., Sect. B 22 1983 802
128. G.G. Furin A.I. Rezvukhin M.A. Fedotov G.G. Yakobson J. Fluorine Chem. 22 1983 231
129. A.M. Pietruszkiewicz J.J. Baldwin W.A. Bolhofer J.M. Hoffman W.C. Lumma J. Heterocycl. Chem. 20 1983 821
130. A.O.K. Nieminen L.H.J. Lajunen T. Holster L. Hietaniemi H. Nupponen Acta Chem. Scand., Ser. B 38 1984 67
131. C. Dainty D.W. Bruce D.J. Cole-Hamilton P. Camilleri J. Chem. Soc., Chem. Commun. 1984 1324
132. S.T.A.K. Daley C.W. Rees D.J. Williams J. Chem. Soc., Chem. Commun. 1984 57
133. L.M. Weinstock I. Shinkai 1st edn. Comp. Heterocycl. Chem. 6 1984 513
134. H. Natsugari R.R. Whittle S.M. Weinreb J. Am. Chem. Soc. 106 1984 7867
135. M.R. Bryce J. Chem. Soc., Perkin Trans. 1 1984 2591
136. P.O. Burke S.D. McDermott T.J. Hannigan W.J. Spillane J. Chem. Soc., Perkin Trans. 2 1984 1851
137. S. Mataka M. Kurisu K. Takahashi M. Tashiro J. Heterocycl. Chem. 21 1984 1157
138. L. Stefaniak J.D. Roberts M. Witanowski G.A. Webb Org. Magn. Reson. 22 1984 215
139. S. Mataka K. Takahashi S. Shiwaku M. Tashiro J. Chem. Res. (S) 11 1985 346
140. S. Mataka K. Takahashi M. Tashiro J. Heterocycl. Chem. 22 1985 1497
141. S. Mataka K. Takahashi M. Tashiro Org. Prep. Proced. Int. 17 1985 152
142. C.W. Bird Tetrahedron 41 1985 1409
143. S. Karady J.S. Amato R.A. Reamer L.M. Weinstock Tetrahedron Lett. 26 1985 6155
144. S. Karady J.S. Amato R.A. Reamer L.M. Weinstock Heterocycles 24 1986 1193
145. A. De Munno V. Bertini N. Picci Heterocycles 24 1986 1131
146. K.S. Sharma R.P. Singh S. Kumari Indian J. Chem., Sect. B 25 1986 271
147. V.J. Arán A.G. Bielsa J.R. Ruiz M. Stud J. Chem. Soc., Perkin Trans. 1 1986 643
148. T. Hatta S. Mataka M. Tashiro J. Heterocycl. Chem. 23 1986 813
149. R. Neidlein D. Knecht Chem. Ber. 120 1987 1593
150. P.J. Dunn C.W. Rees J. Chem. Soc., Chem. Commun. 1987 59
151. H. Natsugari E. Turos S.M. Weinreb R.J. Cvetovich Heterocycles 25 1987 19
152. P.J. Dunn C.W. Rees J. Chem. Soc, Perkin Trans. 1 1987 1579
153. V.J. Arán J.R. Ruiz M. Stud J. Chem. Soc., Perkin Trans. 1 5 1987 955
154. Y. Yamashita K. Saito T. Suzuki C. Kabuto T. Mukai T. Miyashi Angew. Chem., Int. Ed. Engl. 27 1988 434
155. K. Takahashi H. Eguchi S. Shiwaku T. Hatta E. Kyoya T. Yonemitsu S. Mataka M. Tashiro J. Chem. Soc., Perkin Trans. 1 1988 1869
156. M.R. Bryce T.A. Dransfield K.A. Kandeel J.M. Vernon J. Chem. Soc., Perkin Trans. 1 1988 2141
157. E. Turos M. Parvez R.S. Garigipati S.M. Weinreb J. Org. Chem. 53 1988 1116
158. I.A. Belen’kaya Khim. Geterotsikl. Soedin. 1988 114
159. V.L. Savel’ev O.L. Samsonova V.S. Troitskaya V.G. Vinokurov V.P. Moscow L.D. Smirnov Khim. Geterotsikl. Soedin. 1988 977
160. V.J. Arán J.R. Ruiz E. Dávila I. Alkorta M. Stud Liebigs Ann. Chem. 1988 337
161. J.E. Swiger R.T. Standridge T.A. Montzka J.D. Matiskella K.A. Pittman J. Label Comp. Radio. 25 1988 1035
162. S. Mataka H. Eguchi K. Takahashi T. Hatta M. Tashiro Bull. Chem. Soc. Jpn. 62 1989 3127
163. O.E. Desvard M.F. Rozas M.V. Mirifico Collect. Czech. Chem. Commun. 54 1989 2176
164. J.N. Robinson D.J. Cole-Hamilton P. Camilleri C. Dainty V. Maxwell J. Chem. Soc., Faraday Trans. 1 85 1989 3385
165. P.J. Dunn C.W. Rees J. Chem. Soc., Perkin Trans. 1 1989 2485
166. J.M. Klunder T. Onami K.B. Sharpless J. Org. Chem. 54 1989 1295
167. C.-H. Lee J.D. Korp J. Kohn J. Org. Chem. 54 1989 3077
168. G.W. Muller G.E. DuBois J. Org. Chem. 54 1989 4471
169. J.W. Timberlake W.J. Ray Jr. E.D. Stevens C.L. Klein J. Org. Chem. 54 1989 5824
170. M. Herberhold A.F. Hill J. Organomet. Chem. 377 1989 151
171. I. Alkorta V.J. Arán E. Dávila J.R. Ruiz M. Stud Liebigs Ann. Chem. 1989 1135
172. J.T. Ralph Synth. Commun. 19 1989 1381
173. Y. Yamashita J. Eguchi T. Suzuki C. Kabuto T. Miyashi S. Tanaka Angew. Chem., Int. Ed. Engl. 29 1990 643
174. K. Yamaguchi A. Ohsawa C. Kawabata Acta Crystallogr., Sect. C 46 1990 1749
175. J. Kivikoski J. Valkonen E. Pohjala Acta Crystallogr., Sect. C 46 1990 2431
176. N.W. Alcock A.F. Hill M.S. Roe J. Chem. Soc., Dalton Trans. 1990 1737
177. A.V. Zibarev A.O. Miller J. Fluorine Chem. 50 1990 359
178. T. Hatta S. Mataka M. Tashiro K. Numano S. Tanimoto A. Torii J. Heterocycl. Chem. 27 1990 1861
179. A.R. Katritzky P. Barczynski J. Prakt. Chem. 332 1990 885
180. O.M. Fugaeva A.V. Zibarev I.K. Korobeinicheva G.G. Furin J. Mol. Struct. 218 1990 169
181. K. Praefcke B. Kohne F. Korinth Liebigs Ann. Chem. 1990 203
182. K. Takahashi S. Mataka Y. Ikezaki M. Tashiro Senryo to Yakuhin 35 1990 207
183. S. Mataka K. Takahashi Y. Ikezaki T. Hatta A. Torii M. Tashiro Bull. Chem. Soc. Jpn. 64 1991 68
184. I. Bennett J. Antibiot. 44 1991 331
185. T. Hatta S. Mataka M. Tashiro H. Suzuki K. Numano J. Heterocycl. Chem. 28 1991 289
186. T. Hatta S. Mataka M. Tashiro K. Numano H. Suzuki A. Torii J. Heterocycl. Chem. 28 1991 55
187. W.T. Smith Jr. J.M. Patterson A.C. Kovelesky J. Heterocycl. Chem. 28 1991 813
188. A. Alberti M. Benaglia J. Organomet. Chem. 401 1991 13
189. A. Lork G. Gard M. Hare R. Mews W.D. Stohrer R. Winter J. Chem. Soc., Chem. Commun. 1992 898
190. S. Mataka Y. Ikezaki K. Takahashi A. Torii M. Tashiro Heterocycles 33 1992 791
191. S. Mignani C. Gueremy J.L. Malleron A. Truchon J.F. Peyronel J.P. Bastart Heterocycles 34 1992 907
192. M. Matsuoka A. Iwamoto N. Furukawa T. Kitao J. Heterocycl. Chem. 29 1992 439
193. I. Rozas J. Phys. Org. Chem. 5 1992 74
194. C.-H. Lee S.Y. Jin C.Y. Lee B.Y. Chung Bull. Korean Chem. Soc. 13 1992 8
195. G. Dewynter J.-L. Montero Comp. Rend. Acad. Sci. Ser. II 315 1992 1675
196. D.J. Milner Synth. Commun. 22 1992 73
197. W.H.W. Lunn J.K. Shadle Tetrahedron 48 1992 8615
198. K.H. Ahn D.J. Yoo J.S. Kim Tetrahedron Lett. 33 1992 6661
199. E.I. Ivanov A.A. Yavolovskii E.A. Kuklenko R.Y. Ivanova Zh. Org. Khim. 28 1992 422
200. K. Kim J. Cho J. Chem. Soc., Perkin Trans. 1 1993 2345
201. M.V. Mirifico J.A. Caram E.J. Vasini J.E. Sicre J. Phys. Org. Chem. 6 1993 341
202. Y.A. Simonov A.A. Dvorkin E.I. Ivanov A.A. Jawolovskii E.A. Kuklenko Zh. Strukt. Khim. 34 1993 169
203. J.L. Castro V.G. Matassa Tetrahedron Lett. 34 1993 4705
204. L.N. Markovskii T.N. Dubinina G.G. Barashenkov E.A. Romanenko Y.G. Shermolovich Zh. Org. Khim. 29 1993 491
205. E.H. Mørkved H. Kjøsen S.M. Neset Acta Chem. Scand. 48 1994 372
206. K. Kim J. Cho Heterocycles 38 1994 1859
207. J.L. Castro V.G. Matassa J. Org. Chem. 59 1994 2289
208. W. Kozminski J. Jazwinski L. Stefaniak G.A. Webb J. Mol. Struct. 323 1994 177