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Angewandte Chemie - International Edition

Volumn 54, Issue 20, 2015, Pages 6057-6061

Identification of covalent bromodomain binders through DNA display of small moleculeS

(8) Daguer, Jean Pierre a Zambaldo, Claudio a Abegg, Daniel a Barluenga, Sofia a Tallant, Cynthia b Müller, Susanne b Adibekian, Alexander a Winssinger, Nicolas a,b

a UNIVERSITY OF GENEVA (Switzerland)

b UNIVERSITY OF OXFORD (United Kingdom)

Author keywords

activity based proteomic profiling; bromodomains; covalent inhibitors; microarrays

Indexed keywords

AMINO ACIDS; CELL DEATH; MICROARRAYS; MOBILE SECURITY; PATHOLOGY;

BROMODOMAINS; CELLULAR GROWTH; COVALENT BINDING; CYSTEINE RESIDUES; PROTEOMIC ANALYSIS; PROTEOMIC PROFILING; SMALL MOLECULES; TRANSCRIPTIONAL PROGRAM;

MOLECULES;

CYSTEINE; DNA; ETACRYNIC ACID; MOLECULAR LIBRARY; MOLECULAR PROBE;

BINDING SITE; CHEMICAL STRUCTURE; CHEMISTRY; DRUG EFFECTS; GENETIC EPIGENESIS; HUMAN; MOLECULAR LIBRARY; MOLECULAR PROBE; PHARMACOLOGY; PROTEIN TERTIARY STRUCTURE; PROTEOMICS;

BINDING SITES; CYSTEINE; DNA; EPIGENESIS, GENETIC; ETHACRYNIC ACID; HUMANS; MODELS, MOLECULAR; MOLECULAR PROBES; MOLECULAR STRUCTURE; PROTEIN STRUCTURE, TERTIARY; PROTEOMICS; SMALL MOLECULE LIBRARIES;

EID: 84928889206 PISSN: 14337851 EISSN: 15213773 Source Type: Journal
DOI: 10.1002/anie.201412276 Document Type: Article

Times cited : (53)

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