메뉴 건너뛰기




Volumn 201, Issue , 2014, Pages 197-205

Crizotinib

Author keywords

[No Author keywords available]

Indexed keywords

5 (2,6 DICHLOROBENZYLSULFONYL) 3 [3,5 DIMETHYL 4 [2 (1 PYRROLIDINYLMETHYL) 1 PYRROLIDINYLCARBONYL] 1H PYRROL 2 YLMETHYLENE] 1,3 DIHYDRO 2H INDOL 2 ONE; ANAPLASTIC LYMPHOMA KINASE; BIOLOGICAL MARKER; CRIZOTINIB; EPIDERMAL GROWTH FACTOR RECEPTOR; KETOCONAZOLE; MIDAZOLAM; REACTIVE OXYGEN METABOLITE; RIFAMPICIN; SCATTER FACTOR RECEPTOR; ANTINEOPLASTIC AGENT; EML4 ALK FUSION PROTEIN, HUMAN; EML4-ALK FUSION PROTEIN, HUMAN; ONCOPROTEIN; PROTEIN KINASE INHIBITOR; PYRAZOLE DERIVATIVE; PYRIDINE DERIVATIVE;

EID: 84906927012     PISSN: 00800015     EISSN: 21976767     Source Type: Book Series    
DOI: 10.1007/978-3-642-54490-3_11     Document Type: Article
Times cited : (28)

References (29)
  • 1
    • 84866934606 scopus 로고    scopus 로고
    • Activity and safety of crizotinib in patients with ALK-positive non-small-cell lung cancer: Updated results from a phase 1 study
    • Camidge DR, Bang YJ, Kwak EL, Iafrate AJ, Varella-Garcia M, Fox SB et al (2012) Activity and safety of crizotinib in patients with ALK-positive non-small-cell lung cancer: updated results from a phase 1 study. Lancet Oncol 13(10):1011-1019
    • (2012) Lancet Oncol , vol.13 , Issue.10 , pp. 1011-1019
    • Camidge, D.R.1    Bang, Y.J.2    Kwak, E.L.3    Iafrate, A.J.4    Varella-Garcia, M.5    Fox, S.B.6
  • 2
    • 78049426513 scopus 로고    scopus 로고
    • EML4-ALK mutations in lung cancer that confer resistance to ALK inhibitors
    • Choi YL, Soda M, Yamashita Y, Ueno T, Takashima J, Nakajima T et al (2010) EML4-ALK mutations in lung cancer that confer resistance to ALK inhibitors. N Engl J Med 363(18):1734-1739
    • (2010) N Engl J Med , vol.363 , Issue.18 , pp. 1734-1739
    • Choi, Y.L.1    Soda, M.2    Yamashita, Y.3    Ueno, T.4    Takashima, J.5    Nakajima, T.6
  • 3
    • 37549059613 scopus 로고    scopus 로고
    • Cytoreductive antitumor activity of PF-2341066, a novel inhibitor of anaplastic lymphoma kinase and c-Met, in experimental models of anaplastic large-cell lymphoma
    • Christensen JG, Zou HY, Arango ME, Li Q, Lee JH, McDonnell SR et al (2007) Cytoreductive antitumor activity of PF-2341066, a novel inhibitor of anaplastic lymphoma kinase and c-Met, in experimental models of anaplastic large-cell lymphoma. Mol Cancer Ther 6(12):3314-3322
    • (2007) Mol Cancer Ther , vol.6 , Issue.12 , pp. 3314-3322
    • Christensen, J.G.1    Zou, H.Y.2    Arango, M.E.3    Li, Q.4    Lee, J.H.5    McDonnell, S.R.6
  • 4
    • 84875889772 scopus 로고    scopus 로고
    • Aberrant activation of ROS1 represents a new molecular defect in chronic myelomonocytic leukemia
    • Cilloni D, Carturan S, Bracco E, Campia V, Rosso V, Torti D et al (2013) Aberrant activation of ROS1 represents a new molecular defect in chronic myelomonocytic leukemia. Leuk Res 37(5):520-530
    • (2013) Leuk Res , vol.37 , Issue.5 , pp. 520-530
    • Cilloni, D.1    Carturan, S.2    Bracco, E.3    Campia, V.4    Rosso, V.5    Torti, D.6
  • 5
    • 79957487193 scopus 로고    scopus 로고
    • CSF concentration of the anaplastic lymphoma kinase inhibitor crizotinib
    • Costa DB, Kobayashi S, Pandya SS, Yeo WL, Shen Z, Tan W et al (2011) CSF concentration of the anaplastic lymphoma kinase inhibitor crizotinib. J Clin Oncol 29(15):e443-e445
    • (2011) J Clin Oncol , vol.29 , Issue.15
    • Costa, D.B.1    Kobayashi, S.2    Pandya, S.S.3    Yeo, W.L.4    Shen, Z.5    Tan, W.6
  • 6
    • 80052806086 scopus 로고    scopus 로고
    • Structure based drug design of crizotinib (PF-02341066), a potent and selective dual inhibitor of mesenchymalepithelial transition factor (c-MET) kinase and anaplastic lymphoma kinase (ALK)
    • Cui JJ, Tran-Dube M, Shen H, Nambu M, Kung PP, Pairish M et al (2011) Structure based drug design of crizotinib (PF-02341066), a potent and selective dual inhibitor of mesenchymalepithelial transition factor (c-MET) kinase and anaplastic lymphoma kinase (ALK). J Med Chem 54(18):6342-6363
    • (2011) J Med Chem , vol.54 , Issue.18 , pp. 6342-6363
    • Cui, J.J.1    Tran-Dube, M.2    Shen, H.3    Nambu, M.4    Kung, P.P.5    Pairish, M.6
  • 7
    • 84055193418 scopus 로고    scopus 로고
    • Crizotinib: In locally advanced or metastatic non-small cell lung cancer
    • Curran MP (2012) Crizotinib: in locally advanced or metastatic non-small cell lung cancer. Drugs 72(1):99-107
    • (2012) Drugs , vol.72 , Issue.1 , pp. 99-107
    • Curran, M.P.1
  • 11
    • 84876666653 scopus 로고    scopus 로고
    • Identification of ROS1 rearrangement in gastric adenocarcinoma
    • Lee J, Lee SE, Kang SY, Do IG, Lee S, Ha SY et al (2013) Identification of ROS1 rearrangement in gastric adenocarcinoma. Cancer 119(9):1627-1635
    • (2013) Cancer , vol.119 , Issue.9 , pp. 1627-1635
    • Lee, J.1    Lee, S.E.2    Kang, S.Y.3    Do, I.G.4    Lee, S.5    Ha, S.Y.6
  • 12
    • 84861152766 scopus 로고    scopus 로고
    • Promising therapeutic targets in neuroblastoma
    • Matthay KK, George RE, Yu AL (2012) Promising therapeutic targets in neuroblastoma. Clin Cancer Res 18(10):2740-2753
    • (2012) Clin Cancer Res , vol.18 , Issue.10 , pp. 2740-2753
    • Matthay, K.K.1    George, R.E.2    Yu, A.L.3
  • 13
    • 84863786449 scopus 로고    scopus 로고
    • Antitumor action of the MET tyrosine kinase inhibitor crizotinib (PF-02341066) in gastric cancer positive for MET amplification
    • Okamoto W, Okamoto I, Arao T, Kuwata K, Hatashita E, Yamaguchi H et al (2012) Antitumor action of the MET tyrosine kinase inhibitor crizotinib (PF-02341066) in gastric cancer positive for MET amplification. Mol Cancer Ther 11(7):1557-1564
    • (2012) Mol Cancer Ther , vol.11 , Issue.7 , pp. 1557-1564
    • Okamoto, W.1    Okamoto, I.2    Arao, T.3    Kuwata, K.4    Hatashita, E.5    Yamaguchi, H.6
  • 14
    • 84872329681 scopus 로고    scopus 로고
    • Use of targeted therapy for refractory ALK-positive anaplastic large cell lymphoma as a bridging strategy prior to allogeneic transplantation
    • Ordemann R, Stohlmacher J, Beuthien-Baumann B, Platzek I, van den Hoff J, Kroschinsky F et al (2013) Use of targeted therapy for refractory ALK-positive anaplastic large cell lymphoma as a bridging strategy prior to allogeneic transplantation. Ann Hematol 92(1):125-127
    • (2013) Ann Hematol , vol.92 , Issue.1 , pp. 125-127
    • Ordemann, R.1    Stohlmacher, J.2    Beuthien-Baumann, B.3    Platzek, I.4    Van Den Hoff, J.5    Kroschinsky, F.6
  • 15
    • 79955458487 scopus 로고    scopus 로고
    • Activity of crizotinib (PF02341066), a dual mesenchymal-epithelial transition (MET) and anaplastic lymphoma kinase (ALK) inhibitor, in a non-small cell lung cancer patient with de novo MET amplification
    • Ou SH, Kwak EL, Siwak-Tapp C, Dy J, Bergethon K, Clark JW et al (2011) Activity of crizotinib (PF02341066), a dual mesenchymal-epithelial transition (MET) and anaplastic lymphoma kinase (ALK) inhibitor, in a non-small cell lung cancer patient with de novo MET amplification. J Thorac Oncol 6(5):942-946
    • (2011) J Thorac Oncol , vol.6 , Issue.5 , pp. 942-946
    • Ou, S.H.1    Kwak, E.L.2    Siwak-Tapp, C.3    Dy, J.4    Bergethon, K.5    Clark, J.W.6
  • 16
    • 84883451574 scopus 로고    scopus 로고
    • Efficacy and safety of crizotinib in patients with advanced ROS1-rearranged non-small cll lung cancer (NSCLC)
    • Ou SH, Bang YJ, Camidge DR, Riely G (2013) Efficacy and safety of crizotinib in patients with advanced ROS1-rearranged non-small cll lung cancer (NSCLC). J Clin Oncol 31:8032
    • (2013) J Clin Oncol , vol.31
    • Ou, S.H.1    Bang, Y.J.2    Camidge, D.R.3    Riely, G.4
  • 17
    • 84863784502 scopus 로고    scopus 로고
    • Immunohistochemical screening for anaplastic lymphoma kinase (ALK) rearrangement in advanced non-small cell lung cancer patients
    • Park HS, Lee JK, Kim DW, Kulig K, Kim TM, Lee SH et al (2012) Immunohistochemical screening for anaplastic lymphoma kinase (ALK) rearrangement in advanced non-small cell lung cancer patients. Lung Cancer 77(2):288-292
    • (2012) Lung Cancer , vol.77 , Issue.2 , pp. 288-292
    • Park, H.S.1    Lee, J.K.2    Kim, D.W.3    Kulig, K.4    Kim, T.M.5    Lee, S.H.6
  • 18
    • 79952767398 scopus 로고    scopus 로고
    • Crizotinib, a small-molecule dual inhibitor of the c-Met and ALK receptor tyrosine kinases
    • Rodig SJ, Shapiro GI (2010) Crizotinib, a small-molecule dual inhibitor of the c-Met and ALK receptor tyrosine kinases. Curr Opin Invest Drugs 11(12):1477-1490
    • (2010) Curr Opin Invest Drugs , vol.11 , Issue.12 , pp. 1477-1490
    • Rodig, S.J.1    Shapiro, G.I.2
  • 19
    • 84940992905 scopus 로고    scopus 로고
    • Visual effects in anaplastic lymphoma kinase (ALK)-positive advanced non-small cell lung cancer (NSCLC) treated with crizotinib
    • Salgia R, Solomon B, Shaw AT, Camidge DR (2011) Visual effects in anaplastic lymphoma kinase (ALK)-positive advanced non-small cell lung cancer (NSCLC) treated with crizotinib. J Clin Oncol 30:7596
    • (2011) J Clin Oncol , vol.30
    • Salgia, R.1    Solomon, B.2    Shaw, A.T.3    Camidge, D.R.4
  • 20
    • 78649475696 scopus 로고    scopus 로고
    • The neuroblastoma-associated F1174L ALK mutation causes resistance to an ALK kinase inhibitor in ALK-translocated cancers
    • Sasaki T, Okuda K, Zheng W, Butrynski J, Capelletti M, Wang L et al (2010) The neuroblastoma-associated F1174L ALK mutation causes resistance to an ALK kinase inhibitor in ALK-translocated cancers. Cancer Res 70(24):10038-10043
    • (2010) Cancer Res , vol.70 , Issue.24 , pp. 10038-10043
    • Sasaki, T.1    Okuda, K.2    Zheng, W.3    Butrynski, J.4    Capelletti, M.5    Wang, L.6
  • 21
    • 80053386829 scopus 로고    scopus 로고
    • Effect of crizotinib on overall survival in patients with advanced non-small-cell lung cancer harbouring ALK gene rearrangement: A retrospective analysis
    • Shaw AT, Yeap BY, Solomon BJ, Riely GJ, Gainor J, Engelman JA et al (2011) Effect of crizotinib on overall survival in patients with advanced non-small-cell lung cancer harbouring ALK gene rearrangement: a retrospective analysis. Lancet Oncol 12(11):1004-1012
    • (2011) Lancet Oncol , vol.12 , Issue.11 , pp. 1004-1012
    • Shaw, A.T.1    Yeap, B.Y.2    Solomon, B.J.3    Riely, G.J.4    Gainor, J.5    Engelman, J.A.6
  • 22
    • 84879071011 scopus 로고    scopus 로고
    • Crizotinib versus Chemotherapy in advanced ALK-positive lung cancer
    • Shaw AT, Kim DW, Nakagawa K, Seto T, Crino L, Ahn MJ et al (2013a) Crizotinib versus Chemotherapy in advanced ALK-positive lung cancer. N Engl J Med 368:2385-2394
    • (2013) N Engl J Med , vol.368 , pp. 2385-2394
    • Shaw, A.T.1    Kim, D.W.2    Nakagawa, K.3    Seto, T.4    Crino, L.5    Ahn, M.J.6
  • 23
    • 84884993118 scopus 로고    scopus 로고
    • Clinical activity of the ALK inhibitor LDK378 in advanced, ALK-positive NSCLC
    • abstr 8010
    • Shaw AT, Mehra R, Kim DW, Felip E (2013b) Clinical activity of the ALK inhibitor LDK378 in advanced, ALK-positive NSCLC. J Clin Oncol 31(suppl), abstr 8010. 2013
    • (2013) J Clin Oncol , vol.31
    • Shaw, A.T.1    Mehra, R.2    Kim, D.W.3    Felip, E.4
  • 24
    • 84876354373 scopus 로고    scopus 로고
    • Clinical impact of continued Crizotinib administration after isolated central nervous system progression in patients with lung cancer positive for ALK rearrangement
    • Takeda M, Okamoto I, Nakagawa K (2013) Clinical impact of continued Crizotinib administration after isolated central nervous system progression in patients with lung cancer positive for ALK rearrangement. J Thorac Oncol 8(5):654-657
    • (2013) J Thorac Oncol , vol.8 , Issue.5 , pp. 654-657
    • Takeda, M.1    Okamoto, I.2    Nakagawa, K.3
  • 25
    • 80052969848 scopus 로고    scopus 로고
    • MET tyrosine kinase inhibitor crizotinib (PF-02341066) shows differential antitumor effects in nonsmall cell lung cancer according to MET alterations
    • Tanizaki J, Okamoto I, Okamoto K, Takezawa K, Kuwata K, Yamaguchi H et al (2011) MET tyrosine kinase inhibitor crizotinib (PF-02341066) shows differential antitumor effects in nonsmall cell lung cancer according to MET alterations. J Thorac Oncol 6(10):1624-1631
    • (2011) J Thorac Oncol , vol.6 , Issue.10 , pp. 1624-1631
    • Tanizaki, J.1    Okamoto, I.2    Okamoto, K.3    Takezawa, K.4    Kuwata, K.5    Yamaguchi, H.6
  • 26
    • 84862129436 scopus 로고    scopus 로고
    • Anaplastic lymphoma kinase-directed therapy in inflammatory myofibroblastic tumors
    • Tothova Z, Wagner AJ (2012) Anaplastic lymphoma kinase-directed therapy in inflammatory myofibroblastic tumors. Curr Opin Oncol 24(4):409-413
    • (2012) Curr Opin Oncol , vol.24 , Issue.4 , pp. 409-413
    • Tothova, Z.1    Wagner, A.J.2
  • 27
    • 84941006956 scopus 로고    scopus 로고
    • Xalkori (crizotinib) prescribing information. Pfizer Inc
    • Xalkori (crizotinib) prescribing information. Pfizer Inc. 2012
    • (2012)
  • 28
    • 84862846839 scopus 로고    scopus 로고
    • Preclinical rationale for use of the clinically available multitargeted tyrosine kinase inhibitor crizotinib in ROS1- translocated lung cancer
    • Yasuda H, de Figueiredo-Pontes LL, Kobayashi S, Costa DB (2012) Preclinical rationale for use of the clinically available multitargeted tyrosine kinase inhibitor crizotinib in ROS1- translocated lung cancer. J Thorac Oncol 7(7):1086-1090
    • (2012) J Thorac Oncol , vol.7 , Issue.7 , pp. 1086-1090
    • Yasuda, H.1    De Figueiredo-Pontes, L.L.2    Kobayashi, S.3    Costa, D.B.4
  • 29
    • 34249324494 scopus 로고    scopus 로고
    • An orally available small-molecule inhibitor of c-Met, PF-2341066, exhibits cytoreductive antitumor efficacy through antiproliferative and antiangiogenic mechanisms
    • Zou HY, Li Q, Lee JH, Arango ME, McDonnell SR, Yamazaki S et al (2007) An orally available small-molecule inhibitor of c-Met, PF-2341066, exhibits cytoreductive antitumor efficacy through antiproliferative and antiangiogenic mechanisms. Cancer Res 67(9):4408-4417
    • (2007) Cancer Res , vol.67 , Issue.9 , pp. 4408-4417
    • Zou, H.Y.1    Li, Q.2    Lee, J.H.3    Arango, M.E.4    McDonnell, S.R.5    Yamazaki, S.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.