Solid-phase synthesis of NH-1,2,3-triazoles using 4,4′- bismethoxybenzhydryl azide

Synlett

Volumn 25, Issue 13, 2014, Pages 1891-1895

  Cohrt, A Emil ^a   Le Quement, Sebastian T ^a   Nielsen, Thomas E ^a,b  

^a TECHNICAL UNIVERSITY OF DENMARK   (Denmark)

^b NANYANG TECHNOLOGICAL UNIVERSITY   (Singapore)

Author keywords

azide; click chemistry; cross coupling; N H 1,2,3 triazoles; solid phase synthesis

Indexed keywords

1,2,3 TRIAZOLE DERIVATIVE; 4,4' BISMETHOXYBENZHYDRYL AZIDE; ALKYNE DERIVATIVE; AZIDE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL STRUCTURE; CYCLOADDITION; DEPROTECTION REACTION; REACTION ANALYSIS; SOLID PHASE SYNTHESIS; STOICHIOMETRY;

EID: 84905498883     PISSN: 09365214     EISSN: 14372096     Source Type: Journal    
DOI: 10.1055/s-0034-1378228     Document Type: Article

References (15)

1. Fray M. J., Bull D. J., Carr C. L., Gautier E. C. L, Mowbray C. E., Stobie A. J. Med. Chem.: 2001; 44 1951
2. Komeda S., Lutz M., Spek A. L., Chikuma M., Reedijk J. Inorg. Chem.: 2000; 39 4230
3. Dimroth O., Fester G. Ber. Dtsch. Chem. Ges.: 1910; 43 2219
4. Hartzel L. W., Benson F. R. J. Am. Chem. Soc.: 1954; 76 667
5. Tanaka Y., Velen S. R., Miller S. I. Tetrahedron: 1973; 29 3271
6. Tanaka Y., Miller S. I. J. Org. Chem.: 1973; 38 2708
7. Woerner F. P., Reimlinger H. Chem. Ber.: 1970; 103 1908
8. Tornoe C. W., Christensen C., Meldal M. J. Org. Chem.: 2002; 67 3057
9. Rostovtsev V. V., Green L. G., Fokin V. V., Sharpless K. B. Angew. Chem. Int. Ed.: 2002; 41 2596
10. Negishi E.-I, Kotora M., Xu C. J. Org. Chem.: 1997; 62 8957
11. Sonogashira K., Tohda Y., Hagihara N. Tetrahedron Lett.: 1975; 4467
12. King A. O., Okukado N., Negishi E.-I. J. Chem. Soc., Chem. Commun.: 1977; 683
13. Dieck H. A., Heck F. R. J. Organomet. Chem.: 1975; 93 259
14. Sheehan J. C., Robinson C. A. J. Am. Chem. Soc.: 1949; 71 1436
15. Ikeda Y., Kawahara S.-I, Taki M., Kuno A., Hasegawa T., Taira K. Protein Eng.: 2003; 16 699