CANCER RESEARCH;
DRUG BLOOD LEVEL;
DRUG CLEARANCE;
DRUG DISPOSITION;
DRUG UPTAKE;
LETTER;
MEDICAL LITERATURE;
NONHUMAN;
PHENOTYPE;
PRIORITY JOURNAL;
PUBLICATION;
ANIMAL;
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COMPARATIVE STUDY;
DBA MOUSE;
KNOCKOUT MOUSE;
MALE;
MOUSE;
PHYSIOLOGY;
Influence of polymorphic OATP1B-type carriers on the disposition of docetaxel
De Graan A-J, Lancaster CS, Obaidat A, Hagenbuch B, Elens L, Friberg LE, et al. Influence of polymorphic OATP1B-type carriers on the disposition of docetaxel. Clin Cancer Res 2012;18:4433-40.
Inhibition of OATP1B1 by tyrosine kinase inhibitors: In vitro-in vivo correlations
Hu S, Mathijssen RH, De Bruijn P, Baker SD, Sparreboom A. Inhibition of OATP1B1 by tyrosine kinase inhibitors: in vitro-in vivo correlations. Br J Cancer 2014;110:894-8.
Influence of drug formulation on OATP1B2-mediated transport of paclitaxel
Nieuweboer AJ, Hu S, Gui C, Hagenbuch B, Ghobadi Moghaddam-Helmantel I, Gibson AA, et al. Influence of drug formulation on OATP1B2-mediated transport of paclitaxel. Cancer Res 2014;74:3137-45.
Contribution of hepatic uptake transporters OATP1B1/OATP1B3 to the disposition of docetaxel
Washington, DC. Philadelphia PA: AACR
Lee HJ, Leake BF, Teft W, Kim RB, Ho RH. Contribution of hepatic uptake transporters OATP1B1/OATP1B3 to the disposition of docetaxel. In: Proceedings of the Annual Meeting of the American Association for Cancer Research; 2014; Washington, DC. Philadelphia (PA): AACR; 2006. 3682.
Human OATP1B1, OATP1B3 and OATP1A2 can mediate the in vivo uptake and clearance of docetaxel
Epub ahead of print
Iusuf D, Hendrix JJ, Van Esch A, Van De Steeg E, Wagenaar E, Rosing H, et al. Human OATP1B1, OATP1B3 and OATP1A2 can mediate the in vivo uptake and clearance of docetaxel. Int J Cancer 2014 [Epub ahead of print].
High impact of Oatp1a/1b transporters on in vivo disposition of the hydrophobic anticancer drug paclitaxel
Van De Steeg E, Van Esch A, Wagenaar E, Van Der Kruijssen CM, Van Tellingen O, Kenworthy KE, et al. High impact of Oatp1a/1b transporters on in vivo disposition of the hydrophobic anticancer drug paclitaxel. Clin Cancer Res 2011;17:294-301.
Influence of human OATP1B1, OATP1B3, and OATP1A2 on the pharmacokinetics of methotrexate and paclitaxel in humanized transgenic mice
Van De Steeg E, Van Esch A, Wagenaar E, Kenworthy KE, Schinkel AH. Influence of human OATP1B1, OATP1B3, and OATP1A2 on the pharmacokinetics of methotrexate and paclitaxel in humanized transgenic mice. Clin Cancer Res 2013;19:821-32.