SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 14, 2014, Pages 3014-3017

Synthesis and evaluation of N-alkyl-9-aminoacridines with antibacterial activity

(6) Benoit, Adam R a Schiaffo, Charles a Salomon, Christine E b Goodell, John R c Hiasa, Hiroshi a Ferguson, David M a,b

a UNIVERSITY OF MINNESOTA (United States)

b UNIVERSITY OF MINNESOTA (United States)

c ILLINOIS STATE UNIVERSITY (United States)

Author keywords

Acridines; Amphiphiles; Antimicrobials; Drug design; Intercalation; MRSA; SAR; Synthesis; Topoisomerase

Indexed keywords

ACRIDINE; ALKYL GROUP; AMINOACRIDINE DERIVATIVE; ANTIBIOTIC AGENT; CARBON; DNA TOPOISOMERASE; N ALKYL 9 AMINOACRIDINE DERIVATIVE; PLASMID DNA; QUATERNARY AMMONIUM DERIVATIVE; UNCLASSIFIED DRUG; ANTIINFECTIVE AGENT; METICILLIN;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIAL CELL; BACTERIAL MEMBRANE; BACTERIAL STRAIN; CELL MEMBRANE; DRUG SCREENING; DRUG SYNTHESIS; ENZYME INHIBITION; INTERCALATION COMPLEX; METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS; METHICILLIN SUSCEPTIBLE STAPHYLOCOCCUS AUREUS; NONHUMAN; STRUCTURE ACTIVITY RELATION; CHEMICAL STRUCTURE; CHEMISTRY; DOSE RESPONSE; DRUG EFFECTS; MICROBIAL SENSITIVITY TEST; STAPHYLOCOCCUS AUREUS; SYNTHESIS;

METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS; STAPHYLOCOCCUS AUREUS;

AMINOACRIDINES; ANTI-BACTERIAL AGENTS; DOSE-RESPONSE RELATIONSHIP, DRUG; METHICILLIN; MICROBIAL SENSITIVITY TESTS; MOLECULAR STRUCTURE; STAPHYLOCOCCUS AUREUS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84902551850 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2014.05.037 Document Type: Article

Times cited : (29)

References (33)

1
- 77951620048
- F.R. DeLeo, M. Otto, B.N. Kreiswirth, and H.F. Chambers Lancet 375 2010 1557
- (2010) Lancet , vol.375 , pp. 1557
- Deleo, F.R.¹ Otto, M.² Kreiswirth, B.N.³ Chambers, H.F.⁴

2
- 79751474565
- S.D. Kobayashi, and F.R. DeLeo Nat. Med. 17 2011 168
- (2011) Nat. Med. , vol.17 , pp. 168
- Kobayashi, S.D.¹ Deleo, F.R.²

3
- 72849182077
- M. Barber J. Clin. Pathol. 14 1961 385
- (1961) J. Clin. Pathol. , vol.14 , pp. 385
- Barber, M.¹

4
- 33747343208
- G.J. Moran, A. Krishnadasan, R.J. Gorwitz, G.E. Fosheim, L.K. McDougal, R.B. Carey, and D.A. Talan N. Eng. J. Med. 355 2006 666
- (2006) N. Eng. J. Med. , vol.355 , pp. 666
- Moran, G.J.¹ Krishnadasan, A.² Gorwitz, R.J.³ Fosheim, G.E.⁴ McDougal, L.K.⁵ Carey, R.B.⁶ Talan, D.A.⁷

5
- 35349019173
- R.M. Klevens, M.A. Morrison, J. Nadle, S. Petit, K. Gershrnan, S. Ray, L.H. Harrison, R. Lynfield, G. Dumyati, J.M. Townes, A.S. Craig, E.R. Zell, G.E. Fosheim, L.K. McDougal, R.B. Carey, and S.K. Fridkin J. Am. Med. Assoc. 298 2007 1763
- (2007) J. Am. Med. Assoc. , vol.298 , pp. 1763
- Klevens, R.M.¹ Morrison, M.A.² Nadle, J.³ Petit, S.⁴ Gershrnan, K.⁵ Ray, S.⁶ Harrison, L.H.⁷ Lynfield, R.⁸ Dumyati, G.⁹ Townes, J.M.¹⁰ Craig, A.S.¹¹ Zell, E.R.¹² Fosheim, G.E.¹³ McDougal, L.K.¹⁴ Carey, R.B.¹⁵ Fridkin, S.K.¹⁶

6
- 20144386837
- S.K. Fridkin, J.C. Hageman, M. Morrison, L.T. Sanza, K. Como-Sabtti, J.A. Jernigan, K. Harriman, L.H. Harrison, R. Lynfield, and M.M. Farley N. Eng. J. Med. 352 2005 1436
- (2005) N. Eng. J. Med. , vol.352 , pp. 1436
- Fridkin, S.K.¹ Hageman, J.C.² Morrison, M.³ Sanza, L.T.⁴ Como-Sabtti, K.⁵ Jernigan, J.A.⁶ Harriman, K.⁷ Harrison, L.H.⁸ Lynfield, R.⁹ Farley, M.M.¹⁰

7
- 69249083586
- H.F. Chambers, and F.R. Deleo Nat. Rev. Microbiol. 7 2009 629
- (2009) Nat. Rev. Microbiol. , vol.7 , pp. 629
- Chambers, H.F.¹ Deleo, F.R.²

8
- 84869472086
- R. Reynolds, R. Hope, M. Warner, A.P. MacGowan, D.M. Livermore, and M.J. Ellington J. Antimicrob. Chemother. 67 2012 2912
- (2012) J. Antimicrob. Chemother. , vol.67 , pp. 2912
- Reynolds, R.¹ Hope, R.² Warner, M.³ Macgowan, A.P.⁴ Livermore, D.M.⁵ Ellington, M.J.⁶

9
- 84855484682
- I.M. Gould, M.Z. David, S. Esposito, J. Garau, G. Lina, T. Mazzei, and G. Peters Int. J. Antimicrob. Agents 39 2012 96
- (2012) Int. J. Antimicrob. Agents , vol.39 , pp. 96
- Gould, I.M.¹ David, M.Z.² Esposito, S.³ Garau, J.⁴ Lina, G.⁵ Mazzei, T.⁶ Peters, G.⁷

10
- 84861361413
- P.O. Hernandez, S. Lema, S.K. Tyring, and N. Mendoza Infect. Drug Resist. 5 2012 23
- (2012) Infect. Drug Resist. , vol.5 , pp. 23
- Hernandez, P.O.¹ Lema, S.² Tyring, S.K.³ Mendoza, N.⁴

11
- 79951821210
- C. Liu, A. Bayer, S.E. Cosgrove, R.S. Daum, S.K. Fridkin, R.J. Gorwitz, S.L. Kaplan, A.W. Karchmer, D.P. Levine, B.E. Murray, J.M. Rybak, D.A. Talan, and H.F. Chambers Clin. Infect. Dis. 52 2011 285
- (2011) Clin. Infect. Dis. , vol.52 , pp. 285
- Liu, C.¹ Bayer, A.² Cosgrove, S.E.³ Daum, R.S.⁴ Fridkin, S.K.⁵ Gorwitz, R.J.⁶ Kaplan, S.L.⁷ Karchmer, A.W.⁸ Levine, D.P.⁹ Murray, B.E.¹⁰ Rybak, J.M.¹¹ Talan, D.A.¹² Chambers, H.F.¹³

12
- 0035177432
- M. Wainwright J. Antimicrob. Chemother. 47 2001 1
- (2001) J. Antimicrob. Chemother. , vol.47 , pp. 1
- Wainwright, M.¹

13
- 77958468563
- A. Albert, S.D. Rubbo, and M.I. Burvill Br. J. Exp. Pathol. 30 1949 159
- (1949) Br. J. Exp. Pathol. , vol.30 , pp. 159
- Albert, A.¹ Rubbo, S.D.² Burvill, M.I.³

14
- 0001521730
- A. Albert, S.D. Rubbo, R.J. Goldacre, M.E. Davey, and J.D. Stone Br. J. Exp. Pathol. 26 1945 160
- (1945) Br. J. Exp. Pathol. , vol.26 , pp. 160
- Albert, A.¹ Rubbo, S.D.² Goldacre, R.J.³ Davey, M.E.⁴ Stone, J.D.⁵

15
- 0001877793
- L.S. Lerman Proc. Natl. Acad. Sci. 49 1963 94
- (1963) Proc. Natl. Acad. Sci. , vol.49 , pp. 94
- Lerman, L.S.¹

16
- 0032190252
- K.N. Kreuzer Biochim. Biophys. Acta 1400 1998 339
- (1998) Biochim. Biophys. Acta , vol.1400 , pp. 339
- Kreuzer, K.N.¹

17
- 33745601106
- J.R. Goodell, A.A. Madhok, H. Hiasa, and D.M. Ferguson Bioorg. Med. Chem. 14 2006 5467
- (2006) Bioorg. Med. Chem. , vol.14 , pp. 5467
- Goodell, J.R.¹ Madhok, A.A.² Hiasa, H.³ Ferguson, D.M.⁴

18
- 38349194792
- J.R. Goodell, A.V. Ougolkov, H. Hiasa, H. Kaur, R. Remmel, D.D. Billadeau, and D.M. Ferguson J. Med. Chem. 51 2008 179
- (2008) J. Med. Chem. , vol.51 , pp. 179
- Goodell, J.R.¹ Ougolkov, A.V.² Hiasa, H.³ Kaur, H.⁴ Remmel, R.⁵ Billadeau, D.D.⁶ Ferguson, D.M.⁷

19
- 58149159553
- L.M. Oppegard, A.V. Ougolkov, D.N. Luchini, R.A. Schoon, J.R. Goodell, H. Kaur, D.D. Billadeau, D.M. Ferguson, and H. Hiasa Eur. J. Pharmacol. 602 2009 223
- (2009) Eur. J. Pharmacol. , vol.602 , pp. 223
- Oppegard, L.M.¹ Ougolkov, A.V.² Luchini, D.N.³ Schoon, R.A.⁴ Goodell, J.R.⁵ Kaur, H.⁶ Billadeau, D.D.⁷ Ferguson, D.M.⁸ Hiasa, H.⁹

20
- 44649137331
- A. Kommreddy, M.S. Bowsher, M.R. Gunna, K. Botha, and T.K. Vinod Tetrahedron Lett. 49 2008 4378
- (2008) Tetrahedron Lett. , vol.49 , pp. 4378
- Kommreddy, A.¹ Bowsher, M.S.² Gunna, M.R.³ Botha, K.⁴ Vinod, T.K.⁵

21
- 2942604523
- R. Csuk, A. Barthel, and C. Raschke Tetrahedron 60 2004 5737
- (2004) Tetrahedron , vol.60 , pp. 5737
- Csuk, R.¹ Barthel, A.² Raschke, C.³

22
- 34547610513
- S.H. Watterson, P. Chen, Y. Zhao, H.H. Gu, T.G.M. Dhar, Z. Xiao, S.K. Ballentine, Z. Shen, C.A. Fleener, K.A. Rouleau, M. Obermeier, Z. Yang, K.W. McIntyre, D.J. Shuster, M. Witmer, D. Dambach, S. Chao, A. Mathur, B.-C. Chen, J.C. Barrish, J.A. Robl, R. Townsend, and E.J. Iwanowicz J. Med. Chem. 50 2007 3730
- (2007) J. Med. Chem. , vol.50 , pp. 3730
- Watterson, S.H.¹ Chen, P.² Zhao, Y.³ Gu, H.H.⁴ Dhar, T.G.M.⁵ Xiao, Z.⁶ Ballentine, S.K.⁷ Shen, Z.⁸ Fleener, C.A.⁹ Rouleau, K.A.¹⁰ Obermeier, M.¹¹ Yang, Z.¹² McIntyre, K.W.¹³ Shuster, D.J.¹⁴ Witmer, M.¹⁵ Dambach, D.¹⁶ Chao, S.¹⁷ Mathur, A.¹⁸ Chen, B.-C.¹⁹ Barrish, J.C.²⁰ more..

23
- 0023634678
- A.M. Galy, J.P. Galy, J. Barbe, and D. Sharples Arzneim.-Forsch. 37 1987 1095
- (1987) Arzneim.-Forsch. , vol.37 , pp. 1095
- Galy, A.M.¹ Galy, J.P.² Barbe, J.³ Sharples, D.⁴

24
- 78549238235
- Ö.V. Rúnarsson, J. Holappa, C. Malainer, H. Steinsson, M. Hjalmarsdóttir, T. Nevalainen, and M. Másson Eur. Polym. J. 46 2010 1251
- (2010) Eur. Polym. J. , vol.46 , pp. 1251
- Rúnarsson, Ö.V.¹ Holappa, J.² Malainer, C.³ Steinsson, H.⁴ Hjalmarsdóttir, M.⁵ Nevalainen, T.⁶ Másson, M.⁷

25
- 77957329669
- B. Findlay, G.G. Zhanel, and F. Schweizer Antimicrob. Agents Chemother. 54 2010 4049
- (2010) Antimicrob. Agents Chemother. , vol.54 , pp. 4049
- Findlay, B.¹ Zhanel, G.G.² Schweizer, F.³

26
- 84865476398
- J. Hoque, P. Akkapeddi, V. Yarlagadda, D.S.S.M. Uppu, P. Kumar, and J. Haldar Langmuir 28 2012 12225
- (2012) Langmuir , vol.28 , pp. 12225
- Hoque, J.¹ Akkapeddi, P.² Yarlagadda, V.³ Uppu, D.S.S.M.⁴ Kumar, P.⁵ Haldar, J.⁶

27
- 0004299767
- 2nd ed. Edward Arnold London
- A. Albert The Acridines: Their Preparation, Physical, Chemical and Biological Properties and Uses 2nd ed. 1966 Edward Arnold London
- (1966) The Acridines: Their Preparation, Physical, Chemical and Biological Properties and Uses
- Albert, A.¹

28
- 37049158074
- A. Albert, and R. Goldacre J. Chem. Soc. 1946 706
- (1946) J. Chem. Soc. , pp. 706
- Albert, A.¹ Goldacre, R.²

29
- 0031005930
- Z. Oren, J. Hong, and Y. Shai J. Biol. Chem. 272 1997 14643
- (1997) J. Biol. Chem. , vol.272 , pp. 14643
- Oren, Z.¹ Hong, J.² Shai, Y.³

30
- 0032926818
- G. McDonnell, and A.D. Russell Clin. Microbiol. Rev. 12 1999 147
- (1999) Clin. Microbiol. Rev. , vol.12 , pp. 147
- McDonnell, G.¹ Russell, A.D.²

31
- 78650293305
- J.G. Hurdle, A.J. O'Neill, I. Chopra, and R.E. Lee Nat. Rev. Microbiol. 9 2011 62
- (2011) Nat. Rev. Microbiol. , vol.9 , pp. 62
- Hurdle, J.G.¹ O'Neill, A.J.² Chopra, I.³ Lee, R.E.⁴

32
- 33845903833
- D.J. Payne, M.N. Gwynn, D.J. Holmes, and D.L. Pompliano Nat. Rev. Drug Disc. 6 2007 29
- (2007) Nat. Rev. Drug Disc. , vol.6 , pp. 29
- Payne, D.J.¹ Gwynn, M.N.² Holmes, D.J.³ Pompliano, D.L.⁴

33
- 84875731528
- H. Zou, J.-J. Koh, J. Li, S. Qiu, T.T. Aung, H. Lin, A.L. Tan, C. Verma, D.T.H. Tan, H.S.O. Chan, P. Sarawathi, D. Cao, S. Liu, and R.W. Beuerman J. Med. Chem. 56 2013 2359
- (2013) J. Med. Chem. , vol.56 , pp. 2359
- Zou, H.¹ Koh, J.-J.² Li, J.³ Qiu, S.⁴ Aung, T.T.⁵ Lin, H.⁶ Tan, A.L.⁷ Verma, C.⁸ Tan, D.T.H.⁹ Chan, H.S.O.¹⁰ Sarawathi, P.¹¹ Cao, D.¹² Liu, S.¹³ Beuerman, R.W.¹⁴

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.