Hybrid dopamine uptake blocker-serotonin releaser ligands: A new twist on transporter-focused therapeutics

ACS Medicinal Chemistry Letters

Volumn 5, Issue 6, 2014, Pages 623-627

  Blough, Bruce E ^a   Landavazo, Antonio ^a   Partilla, John S ^b   Baumann, Michael H ^b   Decker, Ann M ^a   Page, Kevin M ^a   Rothman, Richard B ^b  

^a RTI INTERNATIONAL   (United States)

^b NATIONAL INSTITUTE ON DRUG ABUSE   (United States)

Author keywords

cocaine; Dopamine uptake inhibitors; methamphetamine; serotonin receptor; serotonin releasers

Indexed keywords

DOPAMINE TRANSPORTER; DOPAMINE UPTAKE INHIBITOR; LIGAND; NORADRENALIN TRANSPORTER; PLASMA MEMBRANE NEUROTRANSMITTER TRANSPORTER; PROPIOPHENONE DERIVATIVE; SEROTONIN;

ANIMAL TISSUE; ARTICLE; BRAIN; BRAIN SYNAPTOSOME; DOPAMINE UPTAKE; DRUG SYNTHESIS; HYBRID; IC 50; NONHUMAN; PRIORITY JOURNAL; RAT; SUBSTITUTION REACTION;

EID: 84902513198     PISSN: None     EISSN: 19485875     Source Type: Journal    
DOI: 10.1021/ml500113s     Document Type: Article

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