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Bioorganic and Medicinal Chemistry

Volumn 22, Issue 4, 2014, Pages 1383-1393

Synthesis and biological evaluation of all eight stereoisomers of DPP-IV inhibitor saxagliptin

(6) Dong, Jizhe a Gong, Yanchun a Liu, Jun a Chen, Xiangfeng b Wen, Xiaoan a Sun, Hongbin a

a CHINA PHARMACEUTICAL UNIVERSITY (China)

b Jiangsu Aosaikang Pharmaceutical Co Ltd (China)

Author keywords

Configuration activity relationship; DPP IV inhibitors; Saxagliptin; Stereoisomers; Synthesis

Indexed keywords

CONFIGURATION-ACTIVITY RELATIONSHIP; DPP-IV INHIBITORS; SAXAGLIPTIN; STEREOISOMERS; SYNTHESIS;

ADAMANTANE; BINDING SITES; CATALYTIC DOMAIN; DIPEPTIDES; DIPEPTIDYL PEPTIDASE 4; DIPEPTIDYL-PEPTIDASE IV INHIBITORS; ENZYME ACTIVATION; MOLECULAR DOCKING SIMULATION; PROTEIN BINDING; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84893800923 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2013.12.061 Document Type: Article

Times cited : (7)

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