Benzimidazole CB2 agonists: Design, synthesis and SAR

Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 4, 2014, Pages 1218-1221

  Nanda, Kausik K ^a   Henze, Darrell A ^a   Della Penna, Kimberly ^a   Desai, Reshma ^a   Leitl, Michael ^a   Lemaire, Wei ^a   White, Rebecca B ^a   Yeh, Suzie ^a   Brouillette, Janine N ^a   Hartman, George D ^a   Bilodeau, Mark T ^a   Trotter, B Wesley ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

Benzimidazole; Cannabinoid 2 receptor; CB2 agonist

Indexed keywords

BENZIMIDAZOLE; CANNABINOID 2 RECEPTOR; CB2 AGONIST;

BENZIMIDAZOLES; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DESIGN; HUMANS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; RECEPTOR, CANNABINOID, CB2; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84893758848     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2013.12.068     Document Type: Article

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