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MedChemComm

Volumn 5, Issue 2, 2014, Pages 180-185

Fragment growing to retain or alter the selectivity of anchored kinase hinge-binding fragments

(5) Allen, Charlotte E a Welford, Amanda J a Matthews, Thomas P a Caldwell, John J a Collins, Ian a

a INSTITUTE OF CANCER RESEARCH (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ANCHORED KINASE HINGE BINDING FRAGMENT; CHECKPOINT KINASE 1; PROTEIN KINASE; PROTEIN KINASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL MODIFICATION; CONCENTRATION RESPONSE; CONTROLLED STUDY; CRYSTALLOGRAPHY; DRUG POTENCY; DRUG SCREENING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; DRUG TARGETING; IC 50; INHIBITION KINETICS; PRIORITY JOURNAL;

EID: 84893306189 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c3md00308f Document Type: Article

Times cited : (6)

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