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Volumn 4, Issue 1, 2013, Pages 41-49

Impact of voglibose on the pharmacokinetics of dapagliflozin in japanese patients with type 2 diabetes

Author keywords

Dapagliflozin; drug drug interaction; Pharmacokinetics; Sodium glucose cotransporter 2 inhibitor; Type 2 diabetes; Voglibose

Indexed keywords

C PEPTIDE; DAPAGLIFLOZIN; GLIMEPIRIDE; GLUCOSE; GLUCURONOSYLTRANSFERASE 1A9; HEMOGLOBIN A1C; METFORMIN; PIOGLITAZONE; SITAGLIPTIN; SODIUM GLUCOSE COTRANSPORTER 2; VOGLIBOSE;

EID: 84891871893     PISSN: 18696953     EISSN: 18696961     Source Type: Journal    
DOI: 10.1007/s13300-012-0016-5     Document Type: Article
Times cited : (15)

References (28)
  • 1
    • 79959936188 scopus 로고    scopus 로고
    • National, regional, and global trends in fasting plasma glucose and diabetes prevalence since 1980: Systematic analysis of health examination surveys and epidemiological studies with 370 country-years and 2.7 million participants
    • Danaei G, Finucane MM, Lu Y, et al. National, regional, and global trends in fasting plasma glucose and diabetes prevalence since 1980: systematic analysis of health examination surveys and epidemiological studies with 370 country-years and 2.7 million participants. Lancet. 2011;378:31-40.
    • (2011) Lancet , vol.378 , pp. 31-40
    • Danaei, G.1    Finucane, M.M.2    Lu, Y.3
  • 2
    • 84899893355 scopus 로고    scopus 로고
    • The Japan Diabetes Society Accessed 25 Apr 2012
    • The Japan Diabetes Society. Introduction to the Japan Diabetes Society. http://www.jds.or.jp/e/about_jds/message.html. Accessed 25 Apr 2012.
    • Introduction to the Japan Diabetes Society
  • 4
    • 0026581055 scopus 로고
    • Antiobesity and antidiabetic actions of a new potent disaccharidase inhibitor in genetically obesediabetic mice, KKA(y
    • Odaka H, Shino A, Ikeda H, Matsuo T. Antiobesity and antidiabetic actions of a new potent disaccharidase inhibitor in genetically obesediabetic mice, KKA(y). J Nutr Sci Vitaminol (Tokyo). 1992;38:27-37.
    • (1992) J Nutr Sci Vitaminol (Tokyo) , vol.38 , pp. 27-37
    • Odaka, H.1    Shino, A.2    Ikeda, H.3    Matsuo, T.4
  • 5
    • 9844269569 scopus 로고    scopus 로고
    • The alphaglucosidase inhibitor voglibose (AO-128) does not change pharmacodynamics or pharmacokinetics of warfarin
    • Fuder H, Kleist P, Birkel M, et al. The alphaglucosidase inhibitor voglibose (AO-128) does not change pharmacodynamics or pharmacokinetics of warfarin. Eur J Clin Pharmacol. 1997;53:153-7.
    • (1997) Eur J Clin Pharmacol , vol.53 , pp. 153-157
    • Fuder, H.1    Kleist, P.2    Birkel, M.3
  • 6
    • 0028784208 scopus 로고
    • Voglibose (AO-128) is an efficient alpha-glucosidase inhibitor and mobilizes the endogenous GLP-1 reserve
    • Goke B, Fuder H, Wieckhorst G, et al. Voglibose (AO-128) is an efficient alpha-glucosidase inhibitor and mobilizes the endogenous GLP-1 reserve. Digestion. 1995;56:493-501.
    • (1995) Digestion , vol.56 , pp. 493-501
    • Goke, B.1    Fuder, H.2    Wieckhorst, G.3
  • 7
    • 0022455206 scopus 로고
    • Synthesis and alpha-D-glucosidase inhibitory activity of N-substituted valiolamine derivatives as potential oral antidiabetic agents
    • Horii S, Fukase H, Matsuo T, Kameda Y, Asano N, Matsui K. Synthesis and alpha-D-glucosidase inhibitory activity of N-substituted valiolamine derivatives as potential oral antidiabetic agents. J Med Chem. 1986;29:1038-46.
    • (1986) J Med Chem , vol.29 , pp. 1038-1046
    • Horii, S.1    Fukase, H.2    Matsuo, T.3    Kameda, Y.4    Asano, N.5    Matsui, K.6
  • 8
    • 77954242599 scopus 로고    scopus 로고
    • SGLT2 inhibition-a novel strategy for diabetes treatment
    • Chao EC, Henry RR. SGLT2 inhibition-a novel strategy for diabetes treatment. Nat Rev Drug Discov. 2010;9:551-9.
    • (2010) Nat Rev Drug Discov , vol.9 , pp. 551-559
    • Chao, E.C.1    Henry, R.R.2
  • 9
    • 41649087328 scopus 로고    scopus 로고
    • Discovery of dapagliflozin: A potent, selective renal sodiumdependent glucose cotransporter 2 (SGLT2) inhibitor for the treatment of type 2 diabetes
    • Meng W, Ellsworth BA, Nirschl AA, et al. Discovery of dapagliflozin: a potent, selective renal sodiumdependent glucose cotransporter 2 (SGLT2) inhibitor for the treatment of type 2 diabetes. J Med Chem. 2008;51:1145-9.
    • (2008) J Med Chem , vol.51 , pp. 1145-1149
    • Meng, W.1    Ellsworth, B.A.2    Nirschl, A.A.3
  • 10
    • 77956921439 scopus 로고    scopus 로고
    • Dapagliflozin monotherapy in type 2 diabetic patients with inadequate glycemic control by diet and exercise: A randomized, double-blind, placebocontrolled, phase III trial
    • Ferrannini E, Ramos SJ, Salsali A, Tang W, List JF. Dapagliflozin monotherapy in type 2 diabetic patients with inadequate glycemic control by diet and exercise: a randomized, double-blind, placebocontrolled, phase III trial. Diabetes Care. 2010;33:2217-24.
    • (2010) Diabetes Care , vol.33 , pp. 2217-2224
    • Ferrannini, E.1    Ramos, S.J.2    Salsali, A.3    Tang, W.4    List, J.F.5
  • 11
    • 84876322398 scopus 로고    scopus 로고
    • Dapagliflozin, metformin-XR, or both together as initial therapy for T2DM [abstract
    • A84. Abstract 307-OR
    • Henry R, Murray A, Marmolejo MH, Hennicken D, Ptaszynska A, List JF. Dapagliflozin, metformin-XR, or both together as initial therapy for T2DM [abstract]. Diabetes. 2011;60:A84. Abstract 307-OR.
    • (2011) Diabetes , vol.60
    • Henry, R.1    Murray, A.2    Marmolejo, M.H.3    Hennicken, D.4    Ptaszynska, A.5    List, J.F.6
  • 12
    • 77953857048 scopus 로고    scopus 로고
    • Effect of dapagliflozin in patients with type 2 diabetes who have inadequate glycaemic control with metformin: A randomised, double-blind, placebo-controlled trial
    • Bailey CJ, Gross JL, Pieters A, Bastien A, List JF. Effect of dapagliflozin in patients with type 2 diabetes who have inadequate glycaemic control with metformin: a randomised, double-blind, placebo-controlled trial. Lancet. 2010;375:2223-33.
    • (2010) Lancet , vol.375 , pp. 2223-2233
    • Bailey, C.J.1    Gross, J.L.2    Pieters, A.3    Bastien, A.4    List, J.F.5
  • 13
    • 84861030350 scopus 로고    scopus 로고
    • Long-term efficacy of dapagliflozin as addon to metformin (MET) in T2DM inadequately controlled with metformin alone [abstract
    • A271, Abstract 988-P
    • Bailey CJ, Gross JL, Yadav M, Iqbal N, Mansfield TA, List JF. Long-term efficacy of dapagliflozin as addon to metformin (MET) in T2DM inadequately controlled with metformin alone [abstract]. Diabetes. 2011;60:A271. Abstract 988-P.
    • (2011) Diabetes , vol.60
    • Bailey, C.J.1    Gross, J.L.2    Yadav, M.3    Iqbal, N.4    Mansfield, T.A.5    List, J.F.6
  • 14
    • 84875206602 scopus 로고    scopus 로고
    • Dapagliflozin as add-on therapy to sitagliptin with or without metformin: A randomized, double-blind, placebocontrolled study
    • A275, Abstract 1071-P
    • Jabbour S, Hardy E, Sugg J, Parikh S. Dapagliflozin as add-on therapy to sitagliptin with or without metformin: a randomized, double-blind, placebocontrolled study. Diabetes. 2012;61:A275. Abstract 1071-P.
    • (2012) Diabetes , vol.61
    • Jabbour, S.1    Hardy, E.2    Sugg, J.3    Parikh, S.4
  • 15
    • 80155124676 scopus 로고    scopus 로고
    • Dapagliflozin versus glipizide as add-on therapy in patients with type 2 diabetes who have inadequate glycemic control with metformin: A randomized, 52-week, double-blind, active-controlled noninferiority trial
    • Nauck MA, Del PS, Meier JJ, et al. Dapagliflozin versus glipizide as add-on therapy in patients with type 2 diabetes who have inadequate glycemic control with metformin: a randomized, 52-week, double-blind, active-controlled noninferiority trial. Diabetes Care. 2011;34:2015-22.
    • (2011) Diabetes Care , vol.34 , pp. 2015-2022
    • Nauck, M.A.1    Del, P.S.2    Meier, J.J.3
  • 16
    • 84862875221 scopus 로고    scopus 로고
    • Effects of dapagliflozin, a sodium-glucose cotransporter-2 inhibitor, on hemoglobin A1c, body weight, and hypoglycemia risk in patients with type 2 diabetes inadequately controlled on pioglitazone monotherapy
    • Rosenstock J, Vico M, Wei L, Salsali A, List JF. Effects of dapagliflozin, a sodium-glucose cotransporter-2 inhibitor, on hemoglobin A1c, body weight, and hypoglycemia risk in patients with type 2 diabetes inadequately controlled on pioglitazone monotherapy. Diabetes Care. 2012;35:1473-8.
    • (2012) Diabetes Care , vol.35 , pp. 1473-1478
    • Rosenstock, J.1    Vico, M.2    Wei, L.3    Salsali, A.4    List, J.F.5
  • 17
    • 79952731806 scopus 로고    scopus 로고
    • Efficacy and safety of dapagliflozin in patients with type 2 diabetes mellitus and inadequate glycaemic control on glimepiride monotherapy [abstract
    • S347. Abstract 870
    • Strojek K, Hruba V, Elze M, Langkilde A, Parikh S. Efficacy and safety of dapagliflozin in patients with type 2 diabetes mellitus and inadequate glycaemic control on glimepiride monotherapy [abstract]. Diabetologia. 2010;53:S347. Abstract 870.
    • (2010) Diabetologia , vol.53
    • Strojek, K.1    Hruba, V.2    Elze, M.3    Langkilde, A.4    Parikh, S.5
  • 18
    • 0030881247 scopus 로고    scopus 로고
    • Comparison of the effects of acarbose and voglibose in healthy subjects
    • Kageyama S, Nakamichi N, Sekino H, Nakano S. Comparison of the effects of acarbose and voglibose in healthy subjects. Clin Ther. 1997;19:720-9.
    • (1997) Clin Ther , vol.19 , pp. 720-729
    • Kageyama, S.1    Nakamichi, N.2    Sekino, H.3    Nakano, S.4
  • 19
    • 84876586956 scopus 로고    scopus 로고
    • Reduction in postprandial glucose with dapagliflozin in type 2 diabetes [abstract
    • A303. Abstract 1104-P
    • Salsali A, Hruba V, Ying L, et al. Reduction in postprandial glucose with dapagliflozin in type 2 diabetes [abstract]. Diabetes. 2011;60:A303. Abstract 1104-P.
    • (2011) Diabetes , vol.60
    • Salsali, A.1    Hruba, V.2    Ying, L.3
  • 20
    • 79951897566 scopus 로고    scopus 로고
    • Pharmacokinetics and pharmacodynamics of dapagliflozin, a novel selective inhibitor of sodium-glucose co-transporter type 2, in Japanese subjects without and with type 2 diabetes mellitus
    • Kasichayanula S, Chang M, Hasegawa M, et al. Pharmacokinetics and pharmacodynamics of dapagliflozin, a novel selective inhibitor of sodium-glucose co-transporter type 2, in Japanese subjects without and with type 2 diabetes mellitus. Diabetes Obes Metab. 2011;13:357-65.
    • (2011) Diabetes Obes Metab , vol.13 , pp. 357-365
    • Kasichayanula, S.1    Chang, M.2    Hasegawa, M.3
  • 21
    • 67349275999 scopus 로고    scopus 로고
    • Dapagliflozin, a novel, selective SGLT2 inhibitor, improved glycemic control over 2 weeks in patients with type 2 diabetes mellitus
    • Komoroski B, Vachharajani N, Feng Y, Li L, Kornhauser D, Pfister M. Dapagliflozin, a novel, selective SGLT2 inhibitor, improved glycemic control over 2 weeks in patients with type 2 diabetes mellitus. Clin Pharmacol Ther. 2009;85:513-9.
    • (2009) Clin Pharmacol Ther , vol.85 , pp. 513-519
    • Komoroski, B.1    Vachharajani, N.2    Feng, Y.3    Li, L.4    Kornhauser, D.5    Pfister, M.6
  • 22
    • 67349180574 scopus 로고    scopus 로고
    • Dapagliflozin, a novel SGLT2 inhibitor, induces dose-dependent glucosuria in healthy subjects
    • Komoroski B, Vachharajani N, Boulton D, et al. Dapagliflozin, a novel SGLT2 inhibitor, induces dose-dependent glucosuria in healthy subjects. Clin Pharmacol Ther. 2009;85:520-6.
    • (2009) Clin Pharmacol Ther , vol.85 , pp. 520-526
    • Komoroski, B.1    Vachharajani, N.2    Boulton, D.3
  • 23
    • 76749111151 scopus 로고    scopus 로고
    • In vitro characterization and pharmacokinetics of dapagliflozin (BMS-512148), a potent sodiumglucose cotransporter type II inhibitor, in animals and humans
    • Obermeier M, Yao M, Khanna A, et al. In vitro characterization and pharmacokinetics of dapagliflozin (BMS-512148), a potent sodiumglucose cotransporter type II inhibitor, in animals and humans. Drug Metab Dispos. 2010;38:405-14.
    • (2010) Drug Metab Dispos , vol.38 , pp. 405-414
    • Obermeier, M.1    Yao, M.2    Khanna, A.3
  • 24
    • 78649715079 scopus 로고    scopus 로고
    • Lack of pharmacokinetic interaction between dapagliflozin, a novel SGLT2 inhibitor, and metformin, pioglitazone, glimepiride, or sitagliptin in healthy subjects
    • Kasichayanula S, Liu X, Shyu WC, et al. Lack of pharmacokinetic interaction between dapagliflozin, a novel SGLT2 inhibitor, and metformin, pioglitazone, glimepiride, or sitagliptin in healthy subjects. Diabetes Obes Metab. 2011;13:47-54.
    • (2011) Diabetes Obes Metab , vol.13 , pp. 47-54
    • Kasichayanula, S.1    Liu, X.2    Shyu, W.C.3
  • 25
    • 84863297468 scopus 로고    scopus 로고
    • Lack of pharmacokinetic interactions between dapagliflozin and simvastatin, valsartan, warfarin, or digoxin
    • Kasichayanula S, Chang M, Liu X, et al. Lack of pharmacokinetic interactions between dapagliflozin and simvastatin, valsartan, warfarin, or digoxin. Adv Ther. 2012;29:163-77.
    • (2012) Adv Ther , vol.29 , pp. 163-177
    • Kasichayanula, S.1    Chang, M.2    Liu, X.3
  • 28
    • 0027787882 scopus 로고
    • Effect of an alpha-glucosidase inhibitor on intestinal fermentation and faecal lipids in diabetic patients
    • Nakamura T, Takebe K, Kudoh K, et al. Effect of an alpha-glucosidase inhibitor on intestinal fermentation and faecal lipids in diabetic patients. J Int Med Res. 1993;21:257-67.
    • (1993) J Int Med Res , vol.21 , pp. 257-267
    • Nakamura, T.1    Takebe, K.2    Kudoh, K.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.