Effects of benznidazole: Cyclodextrin complexes on the drug bioavailability upon oral administration to rats

International Journal of Biological Macromolecules

Volumn 62, Issue , 2013, Pages 543-548

  Leonardi, D ^a,b   Bombardiere, M E ^b   Salomon, C J ^a  

^a UNIVERSIDAD NACIONAL DE ROSARIO   (Argentina)

^b Facultad de Ciencias Naturales e Instituto M Lillo   (Argentina)

Author keywords

Benznidazole; Bioavailability; Chagas' disease; Complexation; Cyclodextrins; Dissolution rate

Indexed keywords

BENZNIDAZOLE; BETA CYCLODEXTRIN; CYCLODEXTRIN; METHYL BETA CYCLODEXTRIN;

ANIMAL CELL; ANIMAL EXPERIMENT; AREA UNDER THE CURVE; ARTICLE; COMPLEX FORMATION; CONTROLLED STUDY; DIFFERENTIAL SCANNING CALORIMETRY; DRUG BIOAVAILABILITY; DRUG BLOOD LEVEL; DRUG SOLUBILITY; MALE; NONHUMAN; RAT; SCANNING ELECTRON MICROSCOPY; SINGLE DRUG DOSE; STOICHIOMETRY; WISTAR RAT; X RAY DIFFRACTION;

RATTUS;

BENZNIDAZOLE; BIOAVAILABILITY; CHAGAS' DISEASE; COMPLEXATION; CYCLODEXTRINS; DISSOLUTION RATE;

ADMINISTRATION, ORAL; ANIMALS; BIOLOGICAL AVAILABILITY; CALORIMETRY, DIFFERENTIAL SCANNING; CYCLODEXTRINS; KINETICS; MALE; NITROIMIDAZOLES; RATS; SOLUBILITY; THERMOGRAVIMETRY; X-RAY DIFFRACTION;

EID: 84886869861     PISSN: 01418130     EISSN: 18790003     Source Type: Journal    
DOI: 10.1016/j.ijbiomac.2013.10.007     Document Type: Article

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