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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 22, 2013, Pages 6052-6059

Synthesis and structure-activity relationships of phenyl-substituted coumarins with anti-tubercular activity that target FadD32

(7) Kawate, Tomohiko a,b,c Iwase, Noriaki a Shimizu, Motohisa a Stanley, Sarah A a,b,c Wellington, Samantha a,c Kazyanskaya, Edward a Hung, Deborah T a,b,c

a BROAD INSTITUTE OF MIT AND HARVARD (United States)

b MASSACHUSETTS GENERAL HOSPITAL (United States)

c HARVARD MEDICAL SCHOOL (United States)

Author keywords

Coumarin; Inhibitor; Mycobacterium tuberculosis; Structure activity relationship (SAR)

Indexed keywords

6 ARYL 5,7 DIMETHYL 4 PHENYL COUMARIN; ANILINE DERIVATIVE; BROMINE DERIVATIVE; CARBOXYLIC ACID DERIVATIVE; COUMARIN DERIVATIVE; ISONIAZID; MORPHOLINE DERIVATIVE; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIBIOTIC RESISTANCE; ARTICLE; BACTERIAL STRAIN; CONTROLLED STUDY; CYCLIZATION; DRUG CONCENTRATION; DRUG POTENCY; DRUG SYNTHESIS; DRUG TARGETING; HIGH THROUGHPUT SCREENING; HYDROPHILICITY; IC 90; MOUSE; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; PHYSICAL CHEMISTRY; STRUCTURE ACTIVITY RELATION; SUZUKI REACTION; TUBERCULOSIS;

MYCOBACTERIUM TUBERCULOSIS;

COUMARIN; INHIBITOR; MYCOBACTERIUM TUBERCULOSIS; STRUCTURE-ACTIVITY RELATIONSHIP (SAR);

ANIMALS; ANTITUBERCULAR AGENTS; COUMARINS; CRYSTALLOGRAPHY, X-RAY; DISEASE MODELS, ANIMAL; HUMANS; MALE; MICE; MICE, INBRED BALB C; MICROBIAL SENSITIVITY TESTS; MOLECULAR CONFORMATION; MYCOBACTERIUM TUBERCULOSIS; STRUCTURE-ACTIVITY RELATIONSHIP; TUBERCULOSIS;

EID: 84885957426 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.09.035 Document Type: Article

Times cited : (60)

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