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Volumn 56, Issue 18, 2013, Pages 7243-7259

Dihydrothiazolopyridone derivatives as a novel family of positive allosteric modulators of the metabotropic glutamate 5 (mGlu5) receptor

(25)  Bartolomé Nebreda, José Manuel a   Conde Ceide, Susana a   Delgado, Francisca a   Iturrino, Laura a   Pastor, Joaquín a   Pena, Miguel Ángel a   Trabanco, Andrés A a   Tresadern, Gary a   Wassvik, Carola M a   Stauffer, Shaun R b,c,d   Jadhav, Satyawan b   Gogi, Kiran b   Vinson, Paige N b   Noetzel, Meredith J b   Days, Emily b   Weaver, C David b   Lindsley, Craig W b,c,d   Niswender, Colleen M b,c   Jones, Carrie K b,c   Conn, P Jeffrey b,c   more..


Author keywords

[No Author keywords available]

Indexed keywords

2 (2 FLUOROPHENOXYMETHYL) 5 (4 FLUOROPHENYL) 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 2 (3 FLUOROPHENOXYMETHYL) 5 (4 FLUOROPHENYL) 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 2 (4 FLUOROPHENOXYMETHYL) 5 (4 FLUOROPHENYL) 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 2 PHENOXYMETHYL 5 (TETRAHYDROPYRAN 4 YLMETHYL) 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 2 PHENOXYMETHYL 5 PYRIDIN 2 YL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 2 PHENOXYMETHYL 5 PYRIDIN 3 YL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 2 PHENOXYMETHYL 5 PYRIDIN 4 YL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 2 PHENYLETHYNYL THIAZOLO[5,4 C]PYRIDIN 4 ONE 6,7 DIHYDRO 5H; 5 (2 METHOXYETHYL) 2 PHENOXYMETHYL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 5 (2,4 DIFLUOROPHENYL) 2 PHENOXYMETHYL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 5 (3 FLUOROPYRIDIN 2 YL) 2 PHENOXYMETHYL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 5 (4 FLUOROPHENYL) 2 PHENOXYMETHYL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 5 (5 FLUOROPYRIDIN 2 YL) 2 PHENOXYMETHYL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 5 CYCLOPROPYL 2 PHENOXYMETHYL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 5 CYCLOPROPYLMETHYL 2 PHENOXYMETHYL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 5 ETHYL 2 PHENOXYMETHYL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 5 ISOPROPYL 2 PHENOXYMETHYL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 5 METHYL 2 PHENOXYMETHYL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; 5 METHYL 2 PHENYLETHYNYL 6,7 DIHYDRO 5H THIAZOLO[5,4 C]PYRIDIN 4 ONE; DIHYDROTHIAZOLOPYRIDONE DERIVATIVE; METABOTROPIC RECEPTOR 5; METABOTROPIC RECEPTOR AGONIST; NEUROLEPTIC AGENT; PYRIDONE DERIVATIVE; UNCLASSIFIED DRUG; THIAZOLE DERIVATIVE;

EID: 84885000221     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm400650w     Document Type: Article
Times cited : (23)

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