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Volumn 49, Issue 4, 2013, Pages 614-623

Pharmaceutical salts: A summary on doses of salt formers from the Orange Book

Author keywords

Counter ions; Drug development; Pharmaceutical salts; Salt screening; Salt selection; Toxicology

Indexed keywords

ACETIC ACID; AMLODIPINE BESYLATE; ATRACURIUM BESILATE; BENZOIC ACID; BROMIDE; CARBONIC ACID; CASPOFUNGIN; CITRIC ACID; DESMOPRESSIN ACETATE; DEXTROPROPOXYPHENE NAPSILATE; EMBONIC ACID; FUMARIC ACID; GLUCOHEPTONIC ACID; GLUCONIC ACID; GLUCURONIC ACID; HIPPURIC ACID; INORGANIC SALT; IODIDE; ISETHIONIC ACID; LACTIC ACID; LACTOBIONIC ACID; LITHIUM CARBONATE; MALEIC ACID; MALIC ACID; MESORIDAZINE BESYLATE; MESYLIC ACID; NITRATE; OXALIC ACID; PYRIDOSTIGMINE; SULFATE;

EID: 84879478391     PISSN: 09280987     EISSN: 18790720     Source Type: Journal    
DOI: 10.1016/j.ejps.2013.05.026     Document Type: Review
Times cited : (78)

References (21)
  • 4
    • 77953314802 scopus 로고    scopus 로고
    • European Medicines Agency, Press Release 20th September, London. EMEA/H/C/164/Z/109
    • European Medicines Agency, Press Release 20th September 2007, CHMP Assessment Report for Viracept, London. EMEA/H/C/164/Z/109.
    • (2007) CHMP Assessment Report for Viracept
  • 6
    • 85030409880 scopus 로고    scopus 로고
    • FDA Orange Book. (assessed 28.12.12)
    • FDA Orange Book. (assessed 28.12.12).
  • 7
    • 0005248386 scopus 로고    scopus 로고
    • FDAa. Maximum Recommended Therapeutic Dose (MRTD) Database (assessed 28.12.12)
    • FDAa, 2012. US Food and Drug Administration, Maximum Recommended Therapeutic Dose (MRTD) Database, (assessed 28.12.12).
    • (2012) US Food and Drug Administration
  • 8
    • 84885046002 scopus 로고    scopus 로고
    • FDA. 05/04/2011-FDA-FAQs on KI (assessed 5.05.13)
    • FDA, 2013. , 05/04/2011-FDA-FAQs on KI (assessed 5.05.13).
    • (2013)
  • 9
    • 0023032232 scopus 로고
    • Salt selection for basic drugs
    • DOI 10.1016/0378-5173(86)90055-4
    • Gould, P.L., 1986. Salt selection for basic drugs. Int. J. Pharm. 33, 201-217. (Pubitemid 17197805)
    • (1986) International Journal of Pharmaceutics , vol.33 , Issue.1-3 , pp. 201-217
    • Gould, P.L.1
  • 10
    • 84885053312 scopus 로고    scopus 로고
    • Institute of Medicine. from the Institute of Medicine of the National Academies: (assessed 5.05.13)
    • Institute of Medicine, 2013. Dietary reference intakes: water, potassium, sodium, chloride, and sulfate, from the Institute of Medicine of the National Academies: , (assessed 5.05.13).
    • (2013) Dietary Reference Intakes: Water, Potassium, Sodium, Chloride, and Sulfate
  • 13
    • 37349115571 scopus 로고    scopus 로고
    • Trends in active pharmaceutical ingredient salt selection based on analysis of the orange book database
    • DOI 10.1021/jm701032y
    • Paulekuhn, S., Dressman, J.B., Saal, C., 2007. Trends in active pharmaceutical ingredient salt selection based on analysis of the orange book database. J. Med. Chem. 50, 6665-6672. (Pubitemid 350309103)
    • (2007) Journal of Medicinal Chemistry , vol.50 , Issue.26 , pp. 6665-6672
    • Paulekuhn, G.S.1    Dressman, J.B.2    Saal, C.3
  • 14
    • 84885033046 scopus 로고    scopus 로고
    • Biological effects of the api salt form
    • In: Stahl, P.H., Wermuth, C.G. (Eds.). VHCA, Verlag Helvetica Chimica Acta, Zürich and Wiley-VCH, Weinheim
    • Pfannkuch, F., Rettig, H., Stahl, P.H., 2011. Biological effects of the API salt form. In: Stahl, P.H., Wermuth, C.G. (Eds.), Handbook of Pharmaceutical Salts. VHCA, Verlag Helvetica Chimica Acta, Zürich and Wiley-VCH, Weinheim, pp. 125-146.
    • (2011) Handbook of Pharmaceutical Salts , pp. 125-146
    • Pfannkuch, F.1    Rettig, H.2    Stahl, P.H.3
  • 15
    • 82255162786 scopus 로고    scopus 로고
    • A survey of top 200 drugs-inconsistent practice of drug strength expression for drugs containing salt forms
    • Prohotsky, D.L., Zhao, F., 2012. A survey of top 200 drugs-inconsistent practice of drug strength expression for drugs containing salt forms. J. Pharm. Sci. 10, 1-6.
    • (2012) J. Pharm. Sci. , vol.10 , pp. 1-6
    • Prohotsky, D.L.1    Zhao, F.2
  • 18
    • 84867525603 scopus 로고    scopus 로고
    • Non-clinical toxicological considerations of pharmaceutical salt selection
    • Thackaberry, E.A., 2012. Non-clinical toxicological considerations of pharmaceutical salt selection. Exp. Opin. Drug Metab. Toxicol. 8, 1419-1433.
    • (2012) Exp. Opin. Drug Metab. Toxicol. , vol.8 , pp. 1419-1433
    • Thackaberry, E.A.1
  • 21
    • 84885056838 scopus 로고    scopus 로고
    • US Pharmacopeia 35. (assessed 14.01.12)
    • US Pharmacopeia 35, 2012. Amikacin Sulfate. (assessed 14.01.12).
    • (2012) Amikacin Sulfate


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.