-
1
-
-
84884193767
-
-
Nassar, A. F.; Hollenberg, P. F.; Scatina, J. Eds., John: Hoboken
-
King, R. S. In Drug Metabolism Handbook: Concepts and Applications; Nassar, A. F.; Hollenberg, P. F.; Scatina, J. Eds., John: Hoboken, 2009, pp 3-38.
-
(2009)
Drug Metabolism Handbook: Concepts and Applications
, pp. 3-38
-
-
King, R.S.1
-
2
-
-
84884186615
-
-
Vogel, H.; Hock F.; Maas, J.; Mayer, D. Eds.; Springer: Berlin, Heidelberg, New York
-
Dudda, A.; Kürzel, G.-U. In Drug Discovery and Evaluation Safety and Pharmacokinetic Assays; Vogel, H.; Hock F.; Maas, J.; Mayer, D. Eds.; Springer: Berlin, Heidelberg, New York, 2006, pp 151-193.
-
(2006)
Drug Discovery and Evaluation Safety and Pharmacokinetic Assays
, pp. 151-193
-
-
Dudda, A.1
Kürzel, G.-U.2
-
3
-
-
18644385994
-
-
Baillie, T. A.; Cayen, M. N.; Fouda, H.; Gerson, R. J.; Green, J. D.; Grossman, S. J.; Klunk, L. J.; LeBlanc, B.; Perkins, D. G.; Shipley, L. A.; Toxicol. Appl. Pharmacol. 2002, 182, 188.
-
(2002)
Toxicol. Appl. Pharmacol.
, vol.182
, pp. 188
-
-
Baillie, T.A.1
Cayen, M.N.2
Fouda, H.3
Gerson, R.J.4
Green, J.D.5
Grossman, S.J.6
Klunk, L.J.7
LeBlanc, B.8
Perkins, D.G.9
Shipley, L.A.10
-
4
-
-
0037306174
-
-
Shipkova, M.; Armstrong, V. W.; Oellerich, M.; Wieland, E. Ther. Drug. Monit. 2003, 25, 1.
-
(2003)
Ther. Drug. Monit.
, vol.25
, pp. 1
-
-
Shipkova, M.1
Armstrong, V.W.2
Oellerich, M.3
Wieland, E.4
-
15
-
-
70350243185
-
-
Walker, D.; Brady, J.; Dalvie, D.; Davis, J.; Dowty, M.; Duncan, J. N.; Nedderman, A.; Obach, R. S.; Wright P. Chem. Res. Toxicol. 2009, 22, 1653.
-
(2009)
Chem. Res. Toxicol.
, vol.22
, pp. 1653
-
-
Walker, D.1
Brady, J.2
Dalvie, D.3
Davis, J.4
Dowty, M.5
Duncan, J.N.6
Nedderman, A.7
Obach, R.S.8
Wright, P.9
-
18
-
-
76749135296
-
-
Drǎgon, C.-A.; Buchheit, D.; Bischoff, D.; Ebener, T.; Bureik, M. Drug Metab. Dispos. 2010, 38, 509.
-
(2010)
Drug Metab. Dispos.
, vol.38
, pp. 509
-
-
Drǎgon, C.-A.1
Buchheit, D.2
Bischoff, D.3
Ebener, T.4
Bureik, M.5
-
19
-
-
79952470677
-
-
Zöllner, A.; Buchheit, D.; Mayer, M. R.; Maurer, H. H.; Peters, F. T.; Bureik, M. Bioanalysis 2010, 2, 1277.
-
(2010)
Bioanalysis
, vol.2
, pp. 1277
-
-
Zöllner, A.1
Buchheit, D.2
Mayer, M.R.3
Maurer, H.H.4
Peters, F.T.5
Bureik, M.6
-
20
-
-
0032054655
-
-
For review of glucuronidation methods and the preparation of the most common glucuronate glycosyl donors see
-
For review of glucuronidation methods and the preparation of the most common glucuronate glycosyl donors see Stachulski, A. V.; G. Jenkins, G. Natural Product Reports 1998, 173.
-
(1998)
Natural Product Reports
, pp. 173
-
-
Stachulski, A.V.1
G Jenkins, G.2
-
21
-
-
78649495086
-
-
Regan, S. I.; Maggs, J. I.; Hammond, T. G.; Lambert, C.; Williams, D. P.; Park, B. K. Biopharm. Drug. Dispos. 2010, 31, 367.
-
(2010)
Biopharm. Drug. Dispos.
, vol.31
, pp. 367
-
-
Regan, S.I.1
Maggs, J.I.2
Hammond, T.G.3
Lambert, C.4
Williams, D.P.5
Park, B.K.6
-
22
-
-
0442282104
-
-
Vanderhoeven, S. J.; Lindon, J. C.; Troke, J.; Tranter, G. E.; Wilson, I. D.; Nicholson, J. K. Xenobiotica, 2004, 34, 73.
-
(2004)
Xenobiotica
, vol.34
, pp. 73
-
-
Vanderhoeven, S.J.1
Lindon, J.C.2
Troke, J.3
Tranter, G.E.4
Wilson, I.D.5
Nicholson, J.K.6
-
27
-
-
84926516035
-
-
(a) Becker, R.; Barua, A. B.; Olson, J. A. Biochem. J. 1996, 25, 212.
-
(1996)
Biochem. J.
, vol.25
, pp. 212
-
-
Becker, R.1
Barua, A.B.2
Olson, J.A.3
-
29
-
-
0026623080
-
-
Panfil, I.; Lehman, P. A.; Zimniak, P.; Ernst, B.; Franz, T.; Lester, R.; Radominska, A. Biochim. Biophys. Act. 1992, 1126, 221.
-
(1992)
Biochim. Biophys. Act.
, vol.1126
, pp. 221
-
-
Panfil, I.1
Lehman, P.A.2
Zimniak, P.3
Ernst, B.4
Franz, T.5
Lester, R.6
Radominska, A.7
-
30
-
-
0000287232
-
-
(b) Smith III, A. B.; Hale, K. J.; Rivero, R. A. Tetrahedron Lett. 1986, 27, 5813.
-
(1986)
Tetrahedron Lett.
, vol.27
, pp. 5813
-
-
Smith III, A.B.1
Hale, K.J.2
Rivero, R.A.3
-
33
-
-
0000165272
-
-
De Mesmaker, A.; Hoffmann, P.; Ernst, B. Tetrahedron Lett. 1989, 30, 3773.
-
(1989)
Tetrahedron Lett.
, vol.30
, pp. 3773
-
-
De Mesmaker, A.1
Hoffmann, P.2
Ernst, B.3
-
35
-
-
0031550869
-
-
(a) Juteau, H.; Gareau, Y.; Labelle, M. Tetrahedron Lett. 1997, 38, 1481.
-
(1997)
Tetrahedron Lett.
, vol.38
, pp. 1481
-
-
Juteau, H.1
Gareau, Y.2
Labelle, M.3
-
36
-
-
2442635266
-
-
(b) Kenny, J. R.; Maggs, J. L.; Meng, X.; Sinnott, D.; Clarke, S. E.; Park, B. K.; Stachulski, A. V. J. Med. Chem. 2004, 47, 2816.
-
(2004)
J. Med. Chem.
, vol.47
, pp. 2816
-
-
Kenny, J.R.1
Maggs, J.L.2
Meng, X.3
Sinnott, D.4
Clarke, S.E.5
Park, B.K.6
Stachulski, A.V.7
-
37
-
-
29844439969
-
-
Perrie, J. A.; Harding, J. R.; Holt, D. W.; Johnston, A.; Meath, P.; Stachulski, A. V. Org. Lett. 2005, 7, 2591.
-
(2005)
Org. Lett.
, vol.7
, pp. 2591
-
-
Perrie, J.A.1
Harding, J.R.2
Holt, D.W.3
Johnston, A.4
Meath, P.5
Stachulski, A.V.6
-
38
-
-
0025907617
-
-
Smith III, A. B.; Rivero, R. A.; Hale, K. J.; Vaccaro, H. A. J. Am. Chem. Soc. 1991, 113, 2092.
-
(1991)
J. Am. Chem. Soc.
, vol.113
, pp. 2092
-
-
Smith III, A.B.1
Rivero, R.A.2
Hale, K.J.3
Vaccaro, H.A.4
-
40
-
-
3543016262
-
-
(b) Biesalski, H.-K.; Doepner, G.; Kunz, H.; Paust, J.; Liebigs. Ann. 1995, 717.
-
(1995)
Liebigs. Ann.
, pp. 717
-
-
Biesalski, H.-K.1
Doepner, G.2
Kunz, H.3
Paust, J.4
-
42
-
-
0026603303
-
-
see also (b)
-
see also (b) Kunz, H.; Kullmann, R.; Werning, P.; Zimmer, J. Tetrahedron Lett. 1992, 33, 1969.
-
(1992)
Tetrahedron Lett.
, vol.33
, pp. 1969
-
-
Kunz, H.1
Kullmann, R.2
Werning, P.3
Zimmer, J.4
-
43
-
-
84884194985
-
-
Boisnard S., Sanofi, Chilly-Mazarin, personal note
-
Boisnard S., Sanofi, Chilly-Mazarin, personal note.
-
-
-
-
45
-
-
0022400351
-
-
(b) Rachmel, A.; Hazelton, G. A.; Yergey, A. L.; Liberato, D. I. Drug. Metab. Dispos. 1985, 13, 705.
-
(1985)
Drug. Metab. Dispos.
, vol.13
, pp. 705
-
-
Rachmel, A.1
Hazelton, G.A.2
Yergey, A.L.3
Liberato, D.I.4
-
46
-
-
0030914234
-
-
Vogt, P. F.; Hansel, J.-G.; Miller, M. J. Tetrahedron Lett. 1991, 38, 2803.
-
(1991)
Tetrahedron Lett.
, vol.38
, pp. 2803
-
-
Vogt, P.F.1
Hansel, J.-G.2
Miller, M.J.3
-
47
-
-
0034714490
-
-
(a) Malkinson, J. P.; Falconer, R. A.; Toth, I. J. Org. Chem. 2000, 65, 5249.
-
(2000)
J. Org. Chem.
, vol.65
, pp. 5249
-
-
Malkinson, J.P.1
Falconer, R.A.2
Toth, I.3
-
48
-
-
85030285764
-
-
(b) Fiandor, J.; Garcias-Lopez, M. T.; De Las Heras, F. G.; Mendez-Gastrillon, P. P. Synthesis, 1985, 1121.
-
(1985)
Synthesis
, pp. 1121
-
-
Fiandor, J.1
Garcias-Lopez, M.T.2
De Las Heras, F.G.3
Mendez-Gastrillon, P.P.4
-
50
-
-
0035969919
-
-
(b) Agostan K.; Dobo, A.; Rako, J.; Keregyarto, J.; Szurmai, Z. Carbohydrate Res. 2001, 330, 183.
-
(2001)
Carbohydrate Res.
, vol.330
, pp. 183
-
-
Agostan, K.1
Dobo, A.2
Rako, J.3
Keregyarto, J.4
Szurmai, Z.5
-
51
-
-
84989499447
-
-
Seebach, D.; Hungerbühler, E.; Naef, R.; Schnurrenberger, P.; Weidmann, B.; Zuger, M.; Synthesis, 1982, 138.
-
(1982)
Synthesis
, pp. 138
-
-
Seebach, D.1
Hungerbühler, E.2
Naef, R.3
Schnurrenberger, P.4
Weidmann, B.5
Zuger, M.6
-
53
-
-
0033535445
-
-
Suzuki, T.; Mabuchi, K.; Fukazawa, N. Bioorg. Med Chem. Lett. 1999, 9, 659.
-
(1999)
Bioorg. Med Chem. Lett.
, vol.9
, pp. 659
-
-
Suzuki, T.1
Mabuchi, K.2
Fukazawa, N.3
-
61
-
-
0037467684
-
-
Iyer, S. S,; Rele, S. M.; Baskaran, S.; Chaikof, E. L. Tetrahedron 2003, 59, 631.
-
(2003)
Tetrahedron
, vol.59
, pp. 631
-
-
Iyer, S.S.1
Rele, S.M.2
Baskaran, S.3
Chaikof, E.L.4
-
62
-
-
0033578705
-
-
Deng, S.; Yu, B.; Xie, J.; Hui, Y. J. Org. Chem. 1999, 64, 7265.
-
(1999)
J. Org. Chem.
, vol.64
, pp. 7265
-
-
Deng, S.1
Yu, B.2
Xie, J.3
Hui, Y.4
-
63
-
-
84884174905
-
-
note
-
Methyl 1-bromo-1-deoxy-2,3,4-tri-O-acetyl- α-D-glucopyranuronate 2b was purchased from Fluka, the corresponding benzoyl and pivaloyl derivatives were prepared in three steps from D-glucuronolactone according to Ref. 34.
-
-
-
-
64
-
-
33947461023
-
-
Bollenback, G. N.; Long, J. W.; Benjamin, D. G.; Lindquist, J. A. J. Am. Chem. Soc. 1955, 77, 3310.
-
(1955)
J. Am. Chem. Soc.
, vol.77
, pp. 3310
-
-
Bollenback, G.N.1
Long, J.W.2
Benjamin, D.G.3
Lindquist, J.A.4
-
65
-
-
84884170230
-
-
Ed. L. Lash, Human Press: Totowa, New Jersey
-
(a) Falany, C.S. In Methods in Pharmacology and Toxicology, Drug Metabolism and Transport: Molecular Methods and Mechanisms, 2005, Ed. L. Lash, Human Press: Totowa, New Jersey, 342-375.
-
(2005)
Methods in Pharmacology and Toxicology, Drug Metabolism and Transport: Molecular Methods and Mechanisms
, pp. 342-375
-
-
Falany, C.S.1
-
68
-
-
0026731582
-
-
(b) Shinkawa, T.; Nakajima, H.; Nishijima, K.; Yamasaki, F.; Kato, K.; Ohzawa, N.; Mizota, M. Eur. J. Pharm. 1992, 219, 217.
-
(1992)
Eur. J. Pharm.
, vol.219
, pp. 217
-
-
Shinkawa, T.1
Nakajima, H.2
Nishijima, K.3
Yamasaki, F.4
Kato, K.5
Ohzawa, N.6
Mizota, M.7
-
70
-
-
78650679122
-
-
Varadi, A.; Gergely, A.; Beni, S.; Jankovics, P.; Noszal, B.; Hosztafi, S. Eur. J. Pharm. Sci. 2011, 42, 65.
-
(2011)
Eur. J. Pharm. Sci.
, vol.42
, pp. 65
-
-
Varadi, A.1
Gergely, A.2
Beni, S.3
Jankovics, P.4
Noszal, B.5
Hosztafi, S.6
-
71
-
-
4043159234
-
-
Ishizaki, M.; Yamada, M.; Watanabe, S.; Hoshino, O.; Nishitani, K.; Hayashida, M.; Tanaka, A.; Hara, H. Tetrahedron 2004, 60, 7973.
-
(2004)
Tetrahedron
, vol.60
, pp. 7973
-
-
Ishizaki, M.1
Yamada, M.2
Watanabe, S.3
Hoshino, O.4
Nishitani, K.5
Hayashida, M.6
Tanaka, A.7
Hara, H.8
-
72
-
-
0028225658
-
-
Beugelmans, R.; Bourdet, S.; Bigot, A.; Zhu, J. Tetrahedron Lett. 1994, 35, 4349.
-
(1994)
Tetrahedron Lett.
, vol.35
, pp. 4349
-
-
Beugelmans, R.1
Bourdet, S.2
Bigot, A.3
Zhu, J.4
-
73
-
-
84884183049
-
-
WO0105764, US6465490
-
Bernotas, R.; Brown, P.; Emmons, G.; King, C.-H. WO0105764, US6465490.
-
-
-
Bernotas, R.1
Brown, P.2
Emmons, G.3
King, C.-H.4
-
75
-
-
27844601627
-
-
(b) Marek, G. J.; Martin-Ruiz, R. A. A.; Artigas, F. Neuropsychopharmacology 2005, 30, 2205.
-
(2005)
Neuropsychopharmacology
, vol.30
, pp. 2205
-
-
Marek, G.J.1
Martin-Ruiz, R.A.A.2
Artigas, F.3
-
76
-
-
48149115938
-
-
(c) Teegarden, B.R.; Al Shamma, H.; Xiong, Y. Curr. Top. Med. Chem. 2008, 8, 969.
-
(2008)
Curr. Top. Med. Chem.
, vol.8
, pp. 969
-
-
Teegarden, B.R.1
Al Shamma, H.2
Xiong, Y.3
-
78
-
-
26444539668
-
-
Gilar, M.; Olivova, P.; Daly, A. E.; Gebler, J. C. Anal. Chem. 2005, 77, 6426.
-
(2005)
Anal. Chem.
, vol.77
, pp. 6426
-
-
Gilar, M.1
Olivova, P.2
Daly, A.E.3
Gebler, J.C.4
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